Receptor GABA
Os receptores de GABA são os principais receptores de neurotransmissores inibitórios no sistema nervoso central, desempenhando um papel crítico na regulação da excitabilidade neuronal e na manutenção do equilíbrio entre excitação e inibição. A disfunção dos receptores de GABA está implicada em vários distúrbios neurológicos e psiquiátricos, incluindo epilepsia, ansiedade e depressão. Na CymitQuimica, oferecemos uma ampla gama de moduladores de receptores de GABA para apoiar sua pesquisa em neurobiologia, saúde mental e desenvolvimento terapêutico.
Foram encontrados 365 produtos de "Receptor GABA"
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ZK 93426 hydrochloride
CAS:benzodiazepine receptor antagonist,competitiveFórmula:C18H21ClN2O3Pureza:98%Cor e Forma:SolidPeso molecular:348.82TP003
CAS:<p>TP003 is a novel non-selective GABAA receptor benzodiazepine site agonist with affinity for α1β2gam2, α2β3gam2, α3β3gam2, α5β2gam2, EC50 of 20.3, 10.6, 3.24, 5.</p>Fórmula:C23H16F3N3OPureza:99.17%Cor e Forma:SolidPeso molecular:407.39BGT1-IN-1
CAS:BGT1-IN-1 (compound 9) is an effective inhibitor of BGT1, demonstrating IC50 values of 13.9 µM for hBGT1 and 58.3 µM for GAT3. It exhibits no cytotoxic effects and possesses neuroprotective activity.Fórmula:C6H9NO2Cor e Forma:SolidPeso molecular:127.14Cyproflanilide
CAS:Cyproflanilide is a GABAR antagonist that exhibits high activity against a variety of pests, including those from the Lepidoptera, Coleoptera, and Thysanoptera orders.Fórmula:C28H17BrF12N2O2Cor e Forma:SolidPeso molecular:721.33Thiomuscimol hydrobromide
CAS:Thiomuscimol hydrobromide is an agonist of GABAA receptor.Fórmula:C4H6N2OSPureza:98%Cor e Forma:SolidPeso molecular:130.17Fletazepam
CAS:Fletazepam, a benzodiazepine derivative, exhibits sedative, anti-anxiety, and muscle-relaxant properties. It is utilized in neurological research.Fórmula:C17H13ClF4N2Cor e Forma:SolidPeso molecular:356.74(-)-Bicuculline methobromide
CAS:(-)-Bicuculline methobromide is a potent antagonist of GABAA receptor .Fórmula:C21H20BrNO6Cor e Forma:WhitePeso molecular:462.29Alfadolone acetate
CAS:Alfadolone acetate is a gamma-aminobutyric acid (GABA) receptor agonist.Fórmula:C23H34O5Cor e Forma:SolidPeso molecular:390.512-AEMP TFA
CAS:2-AEMP TFA is a potent and rapidly acting antagonist of GABA(A)-ρ1 receptors. 2-AEMP is an analog of GABA.Fórmula:C3H10NO3PPureza:98%Cor e Forma:SolidPeso molecular:139.0913-Methylglutaconic acid
CAS:3-Methylglutaconic acid, a primary metabolite accumulating in 3-Methylglutaconic aciduria (MGTA), induces lipid and protein oxidation, while diminishing non-enzymatic antioxidant defenses in cerebral cortex supernatants, thereby promoting oxidative stress in the cerebral cortex. This compound is utilized in research concerning brain damage diseases [1].Fórmula:C6H8O4Pureza:98%Cor e Forma:SolidPeso molecular:144.13CGP 44532
CAS:CGP 44532 a GABAB receptor agonist.Fórmula:C4H12NO3PPureza:98%Cor e Forma:SolidPeso molecular:153.12Pipequaline
CAS:Pipequaline (PK-8165) is an anticonflict & anticonvulsant quinoline derivative. It is an anxiolytic drug that was never marketed. It possesses a novel chemical structure that is not closely related to other drugs of this type. The drug has a similar pharmacological profile to the benzodiazepine family of drugs, but with mainly anxiolytic properties and very little sedative, amnestic or anticonvulsant effects, and so is classified as a nonbenzodiazepine anxiolytic.Fórmula:C22H24N2Pureza:98%Cor e Forma:SolidPeso molecular:316.44Ref: TM-T4655
Produto descontinuadoPazinaclone
CAS:Pazinaclone is a non-benzodiazepine (GABAA) partial agonist with sedative and anxiolytic activity.Fórmula:C25H23ClN4O4Pureza:97.79% - 98.65%Cor e Forma:SolidPeso molecular:478.93Xilmenolone
CAS:<p>Xilmenolone acts as a positive allosteric modulator of the GABA_A receptor [1].</p>Fórmula:C26H37N3O2Pureza:98%Cor e Forma:SolidPeso molecular:423.59Ref: TM-T78670
Produto descontinuadoCGP 56999A
CAS:CGP 56999A is a GABA(B) receptor antagonist; it boosts BDNF and reduces dopamine loss in rat striatum.Fórmula:C19H30NO5PPureza:98%Cor e Forma:SolidPeso molecular:383.42
