Receptor GABA
Os receptores de GABA são os principais receptores de neurotransmissores inibitórios no sistema nervoso central, desempenhando um papel crítico na regulação da excitabilidade neuronal e na manutenção do equilíbrio entre excitação e inibição. A disfunção dos receptores de GABA está implicada em vários distúrbios neurológicos e psiquiátricos, incluindo epilepsia, ansiedade e depressão. Na CymitQuimica, oferecemos uma ampla gama de moduladores de receptores de GABA para apoiar sua pesquisa em neurobiologia, saúde mental e desenvolvimento terapêutico.
Foram encontrados 372 produtos de "Receptor GABA"
Ordenar por
Pureza (%)
0
100
|
0
|
50
|
90
|
95
|
100
TG41
CAS:TG41 is a GABAA receptors positive modulator.Fórmula:C18H13BrCl2N2O2Pureza:98%Cor e Forma:SolidPeso molecular:440.12Etbicyphat
CAS:Etbicyphat: potent GABA(A) antagonist, induces epileptiform activity, binds to GABA/benzodiazepine receptors.Fórmula:C6H11O4PCor e Forma:SolidPeso molecular:178.12TCS 1105
CAS:TCS 1105 is a GABAA BZR ligand, blocking Sema3A and altering mouse anxiety, aggression, and social dominance.Fórmula:C17H13FN2O2Pureza:99.75%Cor e Forma:SolidPeso molecular:296.3Pipazethate
CAS:Pipipyrazine is a nonnarcotic oral cough suppressant, cough suppressant.Fórmula:C21H25N3O3SCor e Forma:SolidPeso molecular:399.51NNC052090
CAS:NNC052090 inhibits GABA uptake, favoring hBGT-1 (Ki=1.4μM), affects α1/D2 receptors (IC50=266/1632nM).Fórmula:C27H30N2O2Cor e Forma:SolidPeso molecular:414.54RU 33965
CAS:RU 33965, a 3-cyclopropyl carbonyl imidazobenzodiazepine, act as a low-efficacy benzodiazepine receptor inverse agonist.Fórmula:C16H15N3O2Pureza:98%Cor e Forma:SolidPeso molecular:281.31ZAPA sulfate
CAS:GABAA receptors agonistFórmula:C4H8N2O6S2Pureza:98%Cor e Forma:SolidPeso molecular:244.25ZK93423
CAS:ZK93423: potent benzodiazepine agonist, IC50=1nM, non-selective, Ki=4.1-6nM for α1-α5 GABAA subunits.Fórmula:C23H22N2O4Cor e Forma:SolidPeso molecular:390.43NCS-382
CAS:γ-Hydroxybutyric acid antagonistFórmula:C13H14O3Pureza:98%Cor e Forma:SolidPeso molecular:218.25GABAA receptor modulator-2
CAS:Compound 20: Selective, oral α5-GABAAR inhibitor, Ki: 4.1 nM. High stability, CNS safe.Fórmula:C22H22FN3O5SCor e Forma:SolidPeso molecular:459.49Carburazepam
CAS:Carburazepam is a derivate of benzodiazepines. Benzodiazepines are a class of psychoactive drugs.Fórmula:C17H16ClN3O2Pureza:98%Cor e Forma:SolidPeso molecular:329.78UMB68 sodium
CAS:UMB-68 is a GHB receptor ligand with no affinity (IC(50) >100 microM) at GABA(A) or GABA(B) receptors.Fórmula:C6H12NaO3Cor e Forma:SolidPeso molecular:155.149β-CCB
CAS:benzodiazepine receptor ligandFórmula:C16H16N2O2Pureza:98%Cor e Forma:SolidPeso molecular:268.31GABAA receptor agent 8
CAS:Compound 5e, a GABAA receptor modulator, shows potent anticonvulsant effects with low neurotoxicity for epilepsy research.Fórmula:C19H16N4OCor e Forma:SolidPeso molecular:316.36Pregabalin arenacarbil
CAS:Pregabalin arenacarbil is a gabamimetic.Fórmula:C15H27NO6Cor e Forma:SolidPeso molecular:317.38CGP 36216 hydrochloride
CAS:CGP 36216 hydrochloride is a potent and selective antagonist of GABAB receptors (IC50: 43 μM).Fórmula:C5H14NO2PPureza:98%Cor e Forma:SolidPeso molecular:151.14(+)-Nipecotic acid
CAS:(+)-Nipecotic acid ((+)-β-Homoproline) is a specific inhibitor of GABA transport and uptake, capable of activating GABAA receptors.Fórmula:C6H11NO2Pureza:99.38%Cor e Forma:SolidPeso molecular:129.16Tracazolate hydrochloride
CAS:Tracazolate hydrochloride (Tracazolate (hydrochloride)) is a modulator of the GABAA receptor with anxiolytic and anticonvulsant activity.Fórmula:C16H25ClN4O2Pureza:99.52%Cor e Forma:SolidPeso molecular:340.85GABA-AT-IN-1
CAS:GABA-AT-IN-1 (Compound 6) is an inhibitor of γ-aminobutyric acid transaminase (GABA-AT) that crosses the blood-brain barrier.Fórmula:C23H18N2O6Cor e Forma:SolidPeso molecular:418.4(S)-SNAP5114
CAS:(S)-SNAP5114 is a selective inhibitor of GABA transport with IC50s of 5 μM for hGAT-3 and 21 μM for rGAT-2. (S)-SNAP5114 has anticonvulsant properties.Fórmula:C30H35NO6Pureza:98.20%Cor e Forma:SolidPeso molecular:505.6Ref: TM-T16831
5mg49,00€1mL*10mM (DMSO)49,00€10mg73,00€25mg152,00€50mg213,00€100mg309,00€200mg423,00€Radequinil
CAS:Radequinil is a benzodiazepine receptor partial inverse agonist. Rade quinil binds to GABA(-) and GABA(+) ligand (Kis: 5.15 and 6.11 nM, respectively).Fórmula:C18H14N4O3Pureza:98%Cor e Forma:SolidPeso molecular:334.333α,21-Dihydroxy-5α-pregnan-20-one
CAS:3α,21-Dihydroxy-5α-pregnan-20-one (5alpha-THDOC) is a GABAA modulator that can be used in the study of Alzheimer's-like neurological diseases.Fórmula:C21H34O3Pureza:98.00%Cor e Forma:SolidPeso molecular:334.49Phaclofen
CAS:GABAB antagonistFórmula:C9H13ClNO3PPureza:99.32%Cor e Forma:White SolidPeso molecular:249.63CCD-3693
CAS:CCD-3693 is a gamma-aminobutyric acid (GABA) receptor agonist.Fórmula:C21H31F3O2Pureza:98%Cor e Forma:SolidPeso molecular:372.46HZ166
CAS:HZ-166 is a positive GABAA receptor modulator and a GABAA receptor subtype-selective benzodiazepine site ligand.Fórmula:C21H16N4O2Pureza:98%Cor e Forma:SolidPeso molecular:356.38Chlormethiazole edisylate
CAS:Chlormethiazole edisylate is a positive allosteric modulator of the GABAA receptor. Chlormethiazole edisylate is a sedative and hypnotic.Fórmula:C8H14ClNO6S3Pureza:98%Cor e Forma:SolidPeso molecular:351.85COR628
CAS:COR628 is the GABA(B) receptor positive allosteric modulator.Fórmula:C16H23NO3SCor e Forma:SolidPeso molecular:309.42trans-4-Hydroxycrotonic acid
CAS:trans-4-Hydroxycrotonic acid (T-HCA) is a selective and competitive ligand for the γ-hydroxybutyric acid (GHB) binding site.Fórmula:C4H6O3Pureza:99.19%Cor e Forma:SolidPeso molecular:102.09LY 81067
CAS:LY 81067, a new anticonvulsant, prevents PTZ- and picrotoxin-induced seizures in mice via picrotoxin site interaction.Fórmula:C22H24N4OCor e Forma:SolidPeso molecular:360.45COR627
CAS:COR627 is the GABA receptor positive allosteric modulator.Fórmula:C20H27NO3SPureza:98%Cor e Forma:SolidPeso molecular:361.5CPP-115
CAS:CPP-115 is a GABA-aminotransferase inhibitor and a high-affinity vigabatrin analogue.Fórmula:C7H9F2NO2Cor e Forma:SolidPeso molecular:177.15JY-XHe-053
CAS:JY-XHe-053 is a selective modulator of GABAA receptors.Fórmula:C22H16FN3O2Pureza:98%Cor e Forma:SolidPeso molecular:373.38HIE-124
CAS:HIE-124 is a central cervous system active anticonvulsant and ultra-short acting hypnotic.Fórmula:C10H12N2O3SPureza:98%Cor e Forma:SolidPeso molecular:240.28Suclofenide
CAS:Suclofenide: a benzenesulfonamide anticonvulsant, effective in mouse seizure models, with side effects like lethargy and diarrhea.Fórmula:C16H13ClN2O4SPureza:98%Cor e Forma:SolidPeso molecular:364.8(S)-Baclofen
CAS:(S)-Baclofen may treat hyperacusis and tinnitus by reducing auditory pathway excitation.Fórmula:C10H12ClNO2Pureza:98%Cor e Forma:SolidPeso molecular:213.66Suriclone
CAS:Suriclone (RP 31264), a cyclic pyrrolidone for anxiety, modulates GABA-A receptors without major sedation.Fórmula:C20H20ClN5O3S2Pureza:99.21% - 99.73%Cor e Forma:SolidPeso molecular:477.99Ru-32514
CAS:Ru-32514 is a benzodiazepine receptor agonist.Fórmula:C18H17N3O2Pureza:99.21%Cor e Forma:SolidPeso molecular:307.35Divaplon
CAS:Divaplon is a GABA receptor agonist (IC50: 0.056 µM) that displays non-sedating anxiolytic behavioral characteristics in a rat model of anxiety.Fórmula:C17H17N3O2Pureza:97.44% - 98.25%Cor e Forma:SolidPeso molecular:295.34DMCM hydrochloride
CAS:DMCM hydrochloride is a non-selective fully inverse agonist of benzodiazepine.Fórmula:C17H19ClN2O4Pureza:99.56%Cor e Forma:SolidPeso molecular:350.8Ref: TM-T11061
1mg34,00€2mg50,00€5mg80,00€1mL*10mM (DMSO)88,00€10mg105,00€25mg236,00€50mg439,00€100mg620,00€Sarmazenil
CAS:Sarmazenil (Ro 15-3505) is a partial inverse agonist at the benzodiazepine receptor and is used in the study of chronic hepatic encephalopathy.Fórmula:C15H14ClN3O3Pureza:99.46%Cor e Forma:SolidPeso molecular:319.74Muscimol HBr
CAS:Muscimol HBr (Agarin HBr) is an agonist of GABAA receptor.Fórmula:C4H7BrN2O2Pureza:98.13%Cor e Forma:Off-White PowderPeso molecular:195.01Ref: TM-T20657
1mg113,00€2mg169,00€1mL*10mM (DMSO)205,00€5mg240,00€10mg385,00€25mg622,00€50mg898,00€100mg1.198,00€500mg2.422,00€DSP-0565
CAS:DSP-0565 is a broad-spectrum anti-epileptic with a high safety margin and effectiveness in several convulsant models.Fórmula:C14H12FNOPureza:99.51% - 99.56%Cor e Forma:SolidPeso molecular:229.25Ref: TM-T11106
1mg109,00€2mg163,00€1mL*10mM (DMSO)208,00€5mg241,00€10mg354,00€25mg532,00€50mg745,00€100mg1.018,00€500mg2.035,00€ELB-139
CAS:ELB-139 is a GABA A receptor agonist. ELB139 increases 5-HT in the striatum and prefrontal cortex of rats.Fórmula:C14H16ClN3OPureza:>99.99%Cor e Forma:SolidPeso molecular:277.75Lirequinil
CAS:Lirequinil (Ro 41-3696) is a small molecule GABAA receptor agonist used to study neurological disorders.Fórmula:C26H25ClN2O3Pureza:98.54%Cor e Forma:SolidPeso molecular:448.94L-838417
CAS:L-838417 is a GABAA receptor subtype-selective benzodiazepine site-selective ligand and GABAA receptor-positive modulator used in the study of anxiety disordersFórmula:C19H19F2N7OPureza:98.12% - 99.70%Cor e Forma:SolidPeso molecular:399.4NNC 05-711
CAS:NNC 05-711 (NO-711 hydrochloride) is a potent and selective inhibitor of GAT-1 (GABA transporter 1), exerting anticonvulsant and analgesic effects.Fórmula:C21H23ClN2O3Pureza:99.92%Cor e Forma:SolidPeso molecular:386.87Riluzole hydrochloride
CAS:Riluzole hydrochloride, an anticonvulsant Na+ channel blocker, inhibits GABA uptake (IC50: 43 µM).Fórmula:C8H6ClF3N2OSPureza:99.76%Cor e Forma:SolidPeso molecular:270.66Panadiplon
CAS:Panadiplon (FG 10571) is a selective gamma-aminobutyric acid receptor agonist and partial agonist of 5GABAA, a benzodiazepine receptor, used in the treatment ofFórmula:C18H17N5O2Pureza:98.30% - 98.94%Cor e Forma:SolidPeso molecular:335.36
