Tansportador
As proteínas transportadoras estão envolvidas no movimento de moléculas através das membranas celulares, desempenhando papéis vitais na captação de nutrientes, eliminação de resíduos e resistência a medicamentos. Inibidores de proteínas transportadoras são usados para estudar a função dessas proteínas em vários processos fisiológicos e patológicos, incluindo distúrbios metabólicos, câncer e liberação de medicamentos. Ao modular a atividade dos transportadores, os pesquisadores podem obter insights sobre os mecanismos de transporte celular e desenvolver novas estratégias terapêuticas. Na CymitQuimica, oferecemos uma gama de inibidores de transportadores para apoiar sua pesquisa em farmacologia, biologia celular e regulação metabólica.
Foram encontrados 48 produtos para "Tansportador".
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EAAT2 activator 1
CAS:EAAT2 activator 1 (3-[(2-Chloro-6-fluorobenzyl)thio]-6-pyridin-2-ylpyridazine) is a thiopyridazine derivative that has been found to increase EAAT2 proteinFórmula:C16H11ClFN3SPureza:98.86%Cor e Forma:Yellow SolidPeso molecular:331.795Indican
CAS:Indican (Indoxyl-β-D-glucoside) is a natural protective compound that is used to protect the liver.Fórmula:C14H17NO6Pureza:99.78% - 99.92%Cor e Forma:Yellow SolidPeso molecular:295.2879Nefazodone hydrochloride
CAS:Nefazodone hydrochloride (Serzone) is a serotoninergic modulating antidepressant that is used in therapy of depression, aggressive behavior and panic disorder.Fórmula:C25H33Cl2N5O2Pureza:99% - 99.86%Cor e Forma:SolidPeso molecular:506.47Vorolanib
CAS:Vorolanib (X-82) is an orally active VEGFR/PDGFR dual inhibitor.Fórmula:C23H26FN5O3Pureza:97.35%Cor e Forma:SolidPeso molecular:439.4826KL-11743
CAS:KL-11743 blocks glucose metabolism, collapses NADH, and increases aspartate, shifting cells to oxidative phosphorylation.Fórmula:C30H30N6O3Pureza:98.46% - 99.57%Cor e Forma:SolidPeso molecular:522.5976UCPH-101
CAS:UCPH-101 is an inhibitor of excitatory amino acid transporter subtype 1 (EAAT1) with an IC50 of 0.66 μM.Fórmula:C27H22N2O3Pureza:98.58%Cor e Forma:White SolidPeso molecular:422.48AHN 1-055 hydrochloride
CAS:AHN 1-055 hydrochloride (3α-Bis-(4-fluorophenyl) Methoxytropane hydrochloride) is an inhibitor of dopamine transporter (DAT) and dopamine uptake(IC50 = 71 nM).Fórmula:C21H24ClF2NOPureza:99.89%Cor e Forma:SolidPeso molecular:379.87Nitrobenzylthioinosine
CAS:Nitrobenzylthioinosine (NBMPR) is an inhibitor of ENT1 transporter that binds to ENT1 transporter with high affinity.Fórmula:C17H17N5O6SPureza:99.69% - 99.74%Cor e Forma:White SolidPeso molecular:419.41WAY-213613
CAS:WAY-213613: Potent GLT-1/EAAT2 inhibitor (IC50: 85 nM), selective over EAAT1/EAAT3; inactive at glutamate receptors.Fórmula:C16H13BrF2N2O4Pureza:98%Cor e Forma:SolidPeso molecular:415.19Tormentic acid
CAS:Tormentic acid is a natural product. It has anticancer, anti-inflammatory, anti-atherogenic , anti-allodynic, and hepatoprotective properties,Fórmula:C30H48O5Pureza:97.02% - 99.86%Cor e Forma:SolidPeso molecular:488.6991BAY-876
CAS:BAY-876 is a selective and orally GLUT1 inhibitor. BAY-876 inhibits glycolytic metabolism and exhibits antitumor activity. Cost-effective and quality-assured.Fórmula:C24H16F4N6O2Pureza:98.61% - 99.78%Cor e Forma:White SolidPeso molecular:496.4165Dotinurad
CAS:Dotinurad ((3,5-dichloro-4-hydroxyphenyl)(1,1-dioxidobenzo[d]thiazol-3(2H)-yl)methanone) is a potent agent of uricosuric (IC50: 3.6 μM for uric acid).Fórmula:C14H9Cl2NO4SPureza:97.43% - 98.04%Cor e Forma:SolidPeso molecular:358.197CTPI-2
CAS:CTPI-2 inhibits SLC25A1 (KD: 3.5 μM), glycolysis, PPARγ, GLUT4, has anti-tumor effects, and combats NASH and diet-induced obesity.Fórmula:C13H9ClN2O6SPureza:97.23%Cor e Forma:SolidPeso molecular:356.738Valbenazine
CAS:Valbenazine (NBI-98854), a highly selective vesicular monoamine transporter 2(VMAT2) inhibitor, is approved for the treatment of tardive dyskinesia.Fórmula:C24H38N2O4Pureza:97.58%Cor e Forma:SolidPeso molecular:418.5695Hemicholinium 3
CAS:Hemicholinium 3 is a potent and selective choline uptake blocker.Fórmula:C24H34Br2N2O4Pureza:98% - 99.95%Cor e Forma:White SolidPeso molecular:574.346Clodronate disodium tetrahydrate
CAS:Clodronate disodium tetrahydrate (Clastoban) inhibits bone resorption and soft tissue calcification.Fórmula:CH10Cl2Na2O10P2Pureza:98%Cor e Forma:SolidPeso molecular:360.917TCID
CAS:TCID (UCH-L3 Inhibitor)(IC50=0.6 μM) is a DUB inhibitor of ubiquitin C-terminal hydrolase L3. It has the 125-fold selectivity to L1.Fórmula:C9H2Cl4O2Pureza:98.87% - 99.34%Cor e Forma:SolidPeso molecular:283.923WZB117
CAS:WZB117 inhibits GLUT1; IC50 ~10μM slows A549 lung & MCF7 breast cancer cell growth.Fórmula:C20H13FO6Pureza:99.03% - 99.18%Cor e Forma:White SolidPeso molecular:368.312DL-TBOA
CAS:DL-TBOA is an inhibitor of excitatory amino acid transporter proteins, inhibiting excitatory amino acid transporter protein 1 (EAAT1), EAAT2, and EAAT3.Fórmula:C11H13NO5Pureza:99.60%Cor e Forma:SolidPeso molecular:239.22DA-023
CAS:DA-023 (Compound 4) acts as a selective positive allosteric modulator (PAM) of EAAT2, exhibiting an EC 50 value of 1 nM [1].Fórmula:C20H25N7Cor e Forma:SolidPeso molecular:363.46
