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Receptor 5-HT

Receptor 5-HT

Os receptores 5-HT, também conhecidos como receptores de serotonina, são um grupo de receptores acoplados à proteína G (GPCRs) que mediam os efeitos da serotonina, um neurotransmissor envolvido na regulação do humor, ansiedade, sono, apetite e outros processos fisiológicos. Esses receptores são divididos em vários subtipos, cada um com funções e propriedades farmacológicas distintas. Moduladores de receptores 5-HT são amplamente estudados por seus papéis no tratamento da depressão, distúrbios de ansiedade e outras condições neuropsiquiátricas. Na CymitQuimica, oferecemos uma variedade de moduladores de receptores 5-HT de alta qualidade para apoiar sua pesquisa em neurofarmacologia, transtornos do humor e sinalização GPCR.

Foram encontrados 940 produtos de "Receptor 5-HT"

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  • TG6-10-1

    CAS:
    <p>TG6-10-1 is an EP2 antagonist.</p>
    Fórmula:C23H23F3N2O4
    Pureza:99.66% - ≥95%
    Cor e Forma:Solid
    Peso molecular:448.43
  • Puerarin

    CAS:
    <p>Puerarin (Kakonein), also known as Kakonein, is a member of the class of compounds known as isoflavonoid C-glycosides. It is a 5-HT2C receptor antagonist.</p>
    Fórmula:C21H20O9
    Pureza:98.90% - 99.21%
    Cor e Forma:Yellow Brown Fine Powder
    Peso molecular:416.38
  • Rotigotine Hydrochloride

    CAS:
    <p>Rotigotine HCl, D3-preferential dopamine agonist, is 50x stronger than quinpirole in anti-Parkinson's efficacy.</p>
    Fórmula:C19H26ClNOS
    Pureza:99.53% - 99.56%
    Cor e Forma:Almost White To White Crystalline Powder
    Peso molecular:351.93
  • Rotigotine-

    CAS:
    <p>Rotigotine (N-0923) is a non-ergot dopamine receptor agonist used in the therapy of Parkinson disease and restless leg syndrome.</p>
    Fórmula:C19H25NOS
    Pureza:98.08% - 99.59%
    Cor e Forma:Solid
    Peso molecular:315.47
  • MK 212 hydrochloride

    CAS:
    <p>MK 212 hydrochloride is a 5-HT2C receptor agonist</p>
    Fórmula:C8H11ClN4·HCl
    Pureza:99.88%
    Cor e Forma:Solid
    Peso molecular:235.12
  • Metadoxine

    CAS:
    <p>Metadoxine (Metadoxil) is a neurotransmitter stimulant.</p>
    Fórmula:C8H11NO3·C5H7NO3
    Pureza:99.19%
    Cor e Forma:Off-White Powder
    Peso molecular:298.29
  • Intepirdine

    CAS:
    <p>Intepirdine (GSK-742457) is a highly selective 5-HT6 receptor antagonist, used in trials studying the treatment of Alzheimer's Disease.</p>
    Fórmula:C19H19N3O2S
    Pureza:98% - 98.63%
    Cor e Forma:Solid
    Peso molecular:353.44
  • Mosapride Citrate

    CAS:
    <p>Mosapride Citrate (TAK-370 citrate), a gastroprokinetic agent, utilizes as a selective 5HT4 agonist.</p>
    Fórmula:C21H25ClFN3O3·C6H8O7
    Pureza:99.70%
    Cor e Forma:White Powder
    Peso molecular:614.02
  • GSK163090

    CAS:
    <p>GSK163090 is a specific and orally active 5-HT1A/B/D receptor antagonist (pKis: 9.4/8.5/9.7, and 6.3/6.7 for 5-HT1A/B/D, and dopamine D2/D3).</p>
    Fórmula:C25H29N5O
    Pureza:99.2%
    Cor e Forma:Solid
    Peso molecular:415.53
  • Tianeptine

    CAS:
    <p>Tianeptine (Tianeptine sodium) 是一种选择性5-HT 摄取促进剂,具有抗抑郁、抗焦虑和神经保护作用,可用于缓解疼痛的研究。</p>
    Fórmula:C21H25ClN2O4S
    Pureza:99.04%
    Cor e Forma:Solid
    Peso molecular:436.95
  • Niaprazine

    CAS:
    <p>Niaprazine is a histamine H1-receptor antagonist with marked sedative properties.</p>
    Fórmula:C20H25FN4O
    Pureza:99.56%
    Cor e Forma:Solid
    Peso molecular:356.44
  • BRL-15572 dihydrochloride

    CAS:
    <p>BRL-15572 dihydrochloride: 5-HT1D antagonist, pKi 7.9, also binds 5-HT1A/2B, 60x selective over 5-HT1B.</p>
    Fórmula:C25H27ClN2O·2HCl
    Pureza:99.74%
    Cor e Forma:Solid
    Peso molecular:479.87
  • Dolasetron Mesylate hydrate

    CAS:
    <p>Dolasetron Mesylate hydrate blocks 5HT3 to prevent chemo and radiotherapy nausea.</p>
    Fórmula:C20H26N2O7S
    Pureza:99.86% - 99.9%
    Cor e Forma:Solid
    Peso molecular:438.49
  • PRX-08066

    CAS:
    <p>PRX-08066 is a selective 5-hydroxytryptamine receptor 2B (5-HT2BR, IC50= 3.4 nM) antagonist that induces selective vasodilation of pulmonary arteries.</p>
    Fórmula:C19H17ClFN5S
    Pureza:97.79% - 98.07%
    Cor e Forma:Solid
    Peso molecular:401.89
  • Ipsapirone hydrochloride

    CAS:
    <p>Ipsapirone, a pyrimidinylpiperazine ligand, is potent and specific for 5-HT1A receptors and has potential therapeutic use in affective disorders.</p>
    Fórmula:C19H24ClN5O3S
    Cor e Forma:Solid
    Peso molecular:437.94
  • Donitriptan Mesylate

    CAS:
    <p>Donitriptan Mesylate, a 5-HT1B/1D agonist, is used potentially for the treatment of migraines.</p>
    Fórmula:C24H29N5O5S
    Cor e Forma:Solid
    Peso molecular:499.58
  • Melitracen

    CAS:
    <p>Melitracen is a tricyclic antidepressant.</p>
    Fórmula:C21H25N
    Cor e Forma:Solid
    Peso molecular:291.43
  • Abaperidone Hydrochloride

    CAS:
    <p>Abaperidone Hydrochloride is an atypical antipsychotic, potently binging to5-HT2 receptors and D2 receptors.</p>
    Fórmula:C25H26ClFN2O5
    Cor e Forma:Solid
    Peso molecular:488.94
  • Melperone

    CAS:
    <p>Melperone, a butyrophenone tranquillizer, caused bradycardia in vivo and in vitro.</p>
    Fórmula:C16H22FNO
    Pureza:98.84%
    Cor e Forma:Solid
    Peso molecular:263.35
  • Cannabigerol

    CAS:
    <p>Cannabigerol is a high affinity α±2-adrenergic receptor agonist, moderate affinity 5-HT1A receptor antagonist, and low affinity CB1 receptor antagonist ; also</p>
    Fórmula:C21H32O2
    Pureza:99.59% - 99.92%
    Cor e Forma:Solid
    Peso molecular:316.48
  • Temanogrel

    CAS:
    <p>Temanogrel (APD791) is a highly selective antagonist of the 5-HT2A receptor (Ki: 4.9 nM).</p>
    Fórmula:C24H28N4O4
    Pureza:99.24%
    Cor e Forma:Solid
    Peso molecular:436.5
  • 2'-O-Methylisoliquiritigenin

    CAS:
    <p>2'-O-Methylisoliquiritigenin, a compound synthesized by enzymes specifically induced in NR.2'-O-Methylisoliquiritigenin, isolated from the Arachis species, up-</p>
    Fórmula:C16H14O4
    Pureza:98.75%
    Cor e Forma:Solid
    Peso molecular:270.28
  • Alprenolol hydrochloride

    CAS:
    <p>Alprenolol hydrochloride is a non-selective blocker of beta, and also is a antagonist of5-HT1A receptor.</p>
    Fórmula:C15H24ClNO2
    Pureza:99.79%
    Cor e Forma:Solid
    Peso molecular:285.81
  • idalopirdine

    CAS:
    <p>Idalopirdine (Lu AE58054), a selective 5-HT6 receptor antagonist( Ki : 0.83 nM),as a treatment for Alzheimer's disease.</p>
    Fórmula:C20H19F5N2O
    Pureza:99.73%
    Cor e Forma:Solid
    Peso molecular:398.37
  • Nuciferine

    CAS:
    <p>Nuciferine ((-)-Nuciferine) is an alkaloid found within the plants Nymphaea caerulea and Nelumbo nucifera.</p>
    Fórmula:C19H21NO2
    Pureza:98.76% - 99.79%
    Cor e Forma:Solid
    Peso molecular:295.38
  • Naratriptan

    CAS:
    <p>Naratriptan is a selective agonist of 5-HT1 receptor and is is used for the treatment of migraine headaches.</p>
    Fórmula:C17H25N3O2S
    Pureza:99.08%
    Cor e Forma:Solid
    Peso molecular:335.47
  • Methiothepin mesylate

    CAS:
    <p>Methiothepin mesylate (Metitepine mesylate) is a potent and non-selective 5-HT2 receptor antagonist, used as an antipsychotic.</p>
    Fórmula:C21H28N2O3S3
    Pureza:98% - 99.92%
    Cor e Forma:Solid
    Peso molecular:452.65
  • Rotundine

    CAS:
    <p>Rotundine (Gindarine) (L-tetrahydropalmatine, L-THP) is a selective dopamine D1 receptor antagonist with IC50 of 166 nM.</p>
    Fórmula:C21H25NO4
    Pureza:99.8% - 99.91%
    Cor e Forma:Off-White Solid
    Peso molecular:355.43
  • BMY 7378 dihydrochloride

    CAS:
    <p>BMY 7378 dihydrochloride (BMY7378 HCl) , α1D-adrenergic receptor antagonist, is a weak partial agonist/antagonist of 5-HT1A receptor.</p>
    Fórmula:C22H33Cl2N3O3
    Pureza:97.32% - 99.08%
    Cor e Forma:Solid
    Peso molecular:458.42
  • F-15599

    CAS:
    <p>F-15599 is a highly selective G-protein biased 5-HT1A receptor agonist(Ki : 3.4 nM).</p>
    Fórmula:C19H21ClF2N4O
    Pureza:98.72%
    Cor e Forma:Solid
    Peso molecular:394.85
  • Pirenperone

    CAS:
    <p>Pirenperone is a putative 5-HT2 receptor antagonist with the central antiserotonergic and antidopaminergic action.</p>
    Fórmula:C23H24FN3O2
    Pureza:99.2%
    Cor e Forma:Solid
    Peso molecular:393.45
  • 7-Amino-4-(trifluoromethyl)coumarin

    CAS:
    <p>7-Amino-4-(trifluoromethyl)coumarin (Coumarin 151) is a 5-Hydroxytryptamine Receptor Subtype 1E (HTR1E) antagonist.</p>
    Fórmula:C10H6F3NO2
    Pureza:97.31% - 97.84%
    Cor e Forma:Yellow Powder
    Peso molecular:229.16
  • Cariprazine

    CAS:
    <p>Cariprazine (RGH-188) is a novel antipsychotic drug candidate that exhibits high affinity for the D3 (Ki=0.085 nM) and D2 (Ki=0.49 nM) receptors, and moderate</p>
    Fórmula:C21H32Cl2N4O
    Pureza:99.68% - 99.87%
    Cor e Forma:Solid
    Peso molecular:427.41
  • Almotriptan Malate

    CAS:
    <p>Almotriptan Malate (PNU180638), a selective 5-HT1B/1D receptor agonist, is used in the therapy of Migraine attacks in adults.</p>
    Fórmula:C17H25N3O2S·C4H6O5
    Pureza:99.95%
    Cor e Forma:Pale Yellow Solid
    Peso molecular:469.55
  • Escitalopram Oxalate

    CAS:
    <p>Escitalopram Oxalate ((S)-(+)Citalopram oxalate) is a selective serotonin (5-HT) reuptake inhibitor (SSRI) with Ki of 0.89 nM.</p>
    Fórmula:C22H23FN2O5
    Pureza:97.39% - 99.73%
    Cor e Forma:White Solid
    Peso molecular:414.43
  • Serotonin hydrochloride

    CAS:
    <p>Serotonin hydrochloride (Serotonin HCl) is an endogenous 5-HT receptor agonist, a monoamine neurotransmitter in the CNS, and a catechol O-methyltransferase (</p>
    Fórmula:C10H13ClN2O
    Pureza:98.05% - 99.93%
    Cor e Forma:White To Cream Powder
    Peso molecular:212.676
  • Azaphen

    CAS:
    <p>Azaphen (Pipofezin hydrochloride) is the reuptake of serotonin inhibitor.with antidepressant action and has sedative effects, suggesting antihistamine activity.</p>
    Fórmula:C16H21Cl2N5O
    Pureza:97.62%
    Cor e Forma:Solid
    Peso molecular:370.28
  • Piboserod

    CAS:
    <p>Piboserod (SB-207266) (SB 207266) is a selective 5-HT(4) receptor antagonist.</p>
    Fórmula:C22H31N3O2
    Pureza:97.21% - 99.49%
    Cor e Forma:Solid
    Peso molecular:369.5
  • Perospirone

    CAS:
    <p>Perospirone (Lullan) is an antagonist of serotonin 5HT2A receptors and dopamine D2 receptors.</p>
    Fórmula:C23H30N4O2S
    Pureza:99.23%
    Cor e Forma:White Powder
    Peso molecular:426.57
  • SB399885

    CAS:
    <p>SB399885 is a potent, brain-penetrant, oral SR-6 antagonist with 200-fold selectivity for SR-6 receptors.</p>
    Fórmula:C18H21Cl2N3O4S
    Pureza:98.94%
    Cor e Forma:Solid
    Peso molecular:446.35
  • LY334370

    CAS:
    <p>LY334370 is a selective 5-HT1F receptor agonist with a Ki of 1.6 nM</p>
    Fórmula:C21H22FN3O
    Pureza:99.32%
    Cor e Forma:Solid
    Peso molecular:351.42
  • Sevoflurane

    CAS:
    <p>Sevoflurane (Fluoromethyl), a noncompetitive inhibitor of 5-HT3 receptor, acts as a low-soluble inhalation anesthetics.</p>
    Fórmula:C4H3F7O
    Pureza:98%
    Cor e Forma:Less Oil Colorless Oil
    Peso molecular:200.05
  • Geissoschizine methyl ether

    CAS:
    <p>Geissoschizine methyl ether: an alkaloid from Uncaria hook, key in Yokukansan, impacts mood and social behavior enhancing serotonin activity.</p>
    Fórmula:C22H26N2O3
    Pureza:99.24% - 99.68%
    Cor e Forma:Solid
    Peso molecular:366.45
  • Ansofaxine hydrochloride

    CAS:
    <p>Ansofaxine hydrochloride (LY03005) is a serotonin-norepinephrine-dopamine reuptake inhibitor (IC50s: 723, 763 and 491 nM, respectively).</p>
    Fórmula:C24H32ClNO3
    Pureza:99.57% - 99.77%
    Cor e Forma:Solid
    Peso molecular:417.97
  • Tropisetron

    CAS:
    <p>Tropisetron (ICS 205-930) is an α7-nicotinic receptor agonist and 5-HT3 receptor antagonist with Kis of 6.9 nM and 5.3 nM, respectively.</p>
    Fórmula:C17H20N2O2
    Pureza:99.68%
    Cor e Forma:White Solid
    Peso molecular:284.35
  • Nelotanserin

    CAS:
    <p>Nelotanserin (APD125): strong 5-HT2A inverse agonist (IC50: 1.7 nM), moderate 5-HT2C (79 nM), weak 5-HT2B (791 nM).</p>
    Fórmula:C18H15BrF2N4O2
    Pureza:98.42% - 99.88%
    Cor e Forma:Solid
    Peso molecular:437.24
  • Amitriptyline

    CAS:
    <p>Amitriptyline: a tricyclic antidepressant used for depression and neuropathic pain.</p>
    Fórmula:C20H23N
    Pureza:98.24% - 99.64%
    Cor e Forma:Crystals Solid
    Peso molecular:277.4
  • Brexpiprazole HCl

    CAS:
    <p>Brexpiprazole HCl (OPC 34712 dihydrochloride) is a new antipsychotic drug.</p>
    Fórmula:C25H27N3O2S·xHCl
    Pureza:99.05%
    Cor e Forma:Solid
    Peso molecular:433.6
  • Sarpogrelate hydrochloride

    CAS:
    <p>Sarpogrelate hydrochloride (MCI-9042), a 5-HT2 antagonist with high affinity (Ki=8.39nM), is used as an anti-platelet for PAD, improving vascular function.</p>
    Fórmula:C24H32ClNO6
    Pureza:99.73%
    Cor e Forma:Colorless Liquid
    Peso molecular:465.97
  • Lurasidone hydrochloride

    CAS:
    <p>Lurasidone HCl: Atypical antipsychotic, treats schizophrenia &amp; bipolar, affects dopamine, serotonin &amp; adrenergic receptors.</p>
    Fórmula:C28H36N4O2S·HCl
    Pureza:99.51%
    Cor e Forma:Solid
    Peso molecular:529.14
  • PRX-07034 hydrochloride

    CAS:
    <p>PRX-07034 hydrochloride is a selective antagonist of 5-HT6 receptor. It has cognition and memory-enhancing properties and decreases body weight in rodents.</p>
    Fórmula:C21H29Cl2N3O4S
    Pureza:98.5%
    Cor e Forma:Solid
    Peso molecular:490.44
  • Clozapine N-Oxide

    CAS:
    <p>View and buy CLOZAPINE N-OXIDE from TargetMol.Clozapine N-oxide is a major metabolite of clozapine also known as DREADDs, technology to modulate synthetic receptors in vivo.Cited in 2 publications.</p>
    Fórmula:C18H19ClN4O
    Pureza:98.43% - 99.94%
    Cor e Forma:Solid
    Peso molecular:342.82
  • Nemifitide acetate(173240-15-8 free base)


    <p>Nemifitide acetate, synthetic 5-amino acid antidepressant, has quick effect, mimics MIF.</p>
    Fórmula:C35H47FN10O8
    Pureza:97.97%
    Cor e Forma:Solid
    Peso molecular:754.85
  • Cinitapride

    CAS:
    <p>Cinitapride (Blaston) treats acid reflux and gastric issues, targeting 5-HT2, 5-HT1, and 5-HT4 receptors.</p>
    Fórmula:C21H30N4O4
    Pureza:99.52%
    Cor e Forma:Solid
    Peso molecular:402.49
  • Pergolide mesylate

    CAS:
    <p>Pergolide mesylate (LY127809), a dopamine agonist for Parkinson's and hyperprolactinemia, was withdrawn for heart valve risk.</p>
    Fórmula:C20H30N2O3S2
    Pureza:99.70%
    Cor e Forma:White To Off-White Solid
    Peso molecular:410.59
  • Dasotraline hydrochloride

    CAS:
    <p>Dasotraline hydrochloride, a dopamine, norepinephrine, and serotonin reuptake inhibitor with IC50s: 4, 6, 11 nM.</p>
    Fórmula:C16H16Cl3N
    Pureza:98.92% - 99.6%
    Cor e Forma:Solid
    Peso molecular:328.66
  • L-745870 trihydrochloride

    CAS:
    <p>L-745870 trihydrochloride is a highly potent and selective D4 dopamine receptor antagonist.</p>
    Fórmula:C18H22Cl4N4
    Pureza:97.52%
    Cor e Forma:Solid
    Peso molecular:436.21
  • 5-Benzyloxygramine

    CAS:
    <p>5-Benzyloxygramine blocks the Dopamin receptors and antagonizes the effects of 5-HT on the rat uterus and the rabbit ear.</p>
    Fórmula:C18H20N2O
    Pureza:99.13%
    Cor e Forma:Solid
    Peso molecular:280.36
  • N-Desmethylclozapine

    CAS:
    <p>N-Desmethylclozapine: 5-HT2C antagonist (IC50: 7.1 nM), dopamine D4 antagonist, δ-opioid agonist.</p>
    Fórmula:C17H17ClN4
    Pureza:97.25% - 99.83%
    Cor e Forma:Yellow Crystalline Solid
    Peso molecular:312.8
  • NGB 2904

    CAS:
    <p>NGB 2904 is a potent and selective antagonist of dopamine D3 receptor. NGB2904 potently antagonizes mitogenesis stimulated by quinpirole (IC50 = 6.8 nM).</p>
    Fórmula:C28H29Cl2N3O
    Pureza:98.79%
    Cor e Forma:Solid
    Peso molecular:494.46
  • Chlorprothixene

    CAS:
    <p>Chlorprothixene (Truxal) is a typical antipsychotic drug of the thioxanthene class, which was the first of the series to be synthesized.</p>
    Fórmula:C18H18ClNS
    Pureza:98.77% - 99.756%
    Cor e Forma:Pale Yellow Crystals Solid
    Peso molecular:315.86
  • Piperacetazine

    CAS:
    <p>Piperacetazine (Piperacetazinum), an antipsychotic prodrug, is used forschizophrenia.</p>
    Fórmula:C24H30N2O2S
    Pureza:99.9% - 99.92%
    Cor e Forma:Solid
    Peso molecular:410.57
  • Loxapine

    CAS:
    <p>Loxapine, a dibenzoxazepine antipsychotic, treats schizophrenia by blocking D2/D4 and serotonin receptors. Related to clozapine.</p>
    Fórmula:C18H18ClN3O
    Pureza:99.88%
    Cor e Forma:Pale Yellowish Crystals From Petroleum Ether Solid
    Peso molecular:327.81
  • Brexpiprazole

    CAS:
    <p>Brexpiprazole (OPC-34712) is a partial agonist of human 5-hydroxytryptamine (5-HT) 5-HT1A and dopamine D2 receptors.</p>
    Fórmula:C25H27N3O2S
    Pureza:99.06% - 99.96%
    Cor e Forma:Solid
    Peso molecular:433.57
  • Jatrorrhizine

    CAS:
    <p>Jatrorrhizine (neprotin) is a protoberberine alkaloid isolated from Enantia chlorantha (Annonaceae) and other species.</p>
    Fórmula:C20H20NO4
    Pureza:97.18% - 99.06%
    Cor e Forma:Solid
    Peso molecular:338.38
  • Urapidil

    CAS:
    <p>Urapidil (Ebrantil), a sympatholytic antihypertensive drug, acts as a 5-HT1A receptor agonist and as an α1-adrenoceptor antagonist.</p>
    Fórmula:C20H29N5O3
    Pureza:99.85% - >99.99%
    Cor e Forma:Solid
    Peso molecular:387.48
  • RS-127445 hydrochloride

    CAS:
    <p>RS-127445 hydrochloride (MT 500) is a selective, high affinity, orally bioavailable 5-HT2B receptor antagonist(pKi : 9.5).</p>
    Fórmula:C17H17ClFN3
    Pureza:99.48%
    Cor e Forma:Solid
    Peso molecular:317.79
  • Zacopride hydrochloride

    CAS:
    <p>Zacopride is a highly potent 5-HT3 receptor antagonist (Kd = 0.38 nM) and 5-HT4 receptor agonist (Ki = 373 nM). It also is a selective IK1 channel agonist.</p>
    Fórmula:C15H20ClN3O2·HCl
    Pureza:98.32%
    Cor e Forma:Solid
    Peso molecular:346.26
  • 8-Hydroxy-DPAT hydrobromide

    CAS:
    <p>8-Hydroxy-DPAT hydrobromide (8-OH-DPAT hydrobromide) (8-OH-DPAT hydrobromide) is a potent and selective 5-HT1A agonist with a pIC50 of 8.19.</p>
    Fórmula:C16H26BrNO
    Pureza:98.90% - 99.09%
    Cor e Forma:Solid
    Peso molecular:328.29
  • SB-203186 hydrochloride

    CAS:
    <p>SB 203186 hydrochloride is a potent 5-HT4 receptor antagonist</p>
    Fórmula:C16H20N2O2·HCl
    Pureza:99.64%
    Cor e Forma:Solid
    Peso molecular:308.81
  • Myristicin

    CAS:
    <p>Myristicin is a natural spice extract with antibacterial, anti-inflammatory, and hepatoprotective properties, and can induce apoptosis.</p>
    Fórmula:C11H12O3
    Pureza:99.828%
    Cor e Forma:Liquid
    Peso molecular:192.21
  • Hypidone hydrochloride

    CAS:
    <p>Hypidone hydrochloride (YL0919) is a novel antidepressant candidate with dual activity as a 5-HT1A receptor agonist and a selective serotonin reuptake inhibitor</p>
    Fórmula:C18H23ClN2O2
    Pureza:99.82% - 99.93%
    Cor e Forma:Solid
    Peso molecular:334.84
  • Vortioxetine

    CAS:
    <p>Vortioxetine (Lu AA 21004) is a serotonergic antidepressant used for major depression disorders.</p>
    Fórmula:C18H22N2S
    Pureza:99.34% - 99.34%
    Cor e Forma:Solid
    Peso molecular:298.45
  • BRL 54443

    CAS:
    <p>BRL 54443 is a potent 5-HT1E/1F receptor agonist (pKi values are 8.7 and 8.9 respectively).</p>
    Fórmula:C14H18N2O
    Pureza:98.07%
    Cor e Forma:Solid
    Peso molecular:230.31
  • 6-fluoro-DL-Tryptophan

    CAS:
    <p>6-fluoro-DL-Tryptophan is an inhibitor of serotonin (5-HT) synthesis.</p>
    Fórmula:C11H11FN2O2
    Pureza:99.25%
    Cor e Forma:Off-White Powder
    Peso molecular:222.22
  • Serotonin

    CAS:
    <p>Serotonin (5-hydroxytryptamine) is a monoamine neurotransmitter in the CNS and an endogenous 5-HT receptor agonist. High-Quality, Low-Cost!</p>
    Fórmula:C10H12N2O
    Pureza:97.47% - 99.92%
    Cor e Forma:Solid
    Peso molecular:176.22
  • NAN-190 hydrobromide

    CAS:
    <p>NAN-190 hydrobromide is an antagonist of serotonin receptor 5-HT.</p>
    Fórmula:C23H28BrN3O3
    Pureza:95.20%
    Cor e Forma:Solid
    Peso molecular:474.39
  • Perospirone hydrochloride

    CAS:
    <p>Perospirone hydrochloride (Perospirone HCl) is an atypical antipsychotic agent for the treatment of schizophrenia.</p>
    Fórmula:C23H31ClN4O2S
    Pureza:99.37%
    Cor e Forma:White Solid
    Peso molecular:463
  • 3-AQC

    CAS:
    <p>3-AQC is a competitive antagonist of 5-HT3.</p>
    Fórmula:C20H21N5O4
    Pureza:99.45%
    Cor e Forma:Solid
    Peso molecular:395.41
  • AVN-101

    CAS:
    <p>AVN-101 is a very potent 5-HT7 receptor antagonist.Cost-effective and quality-assured.</p>
    Fórmula:C21H25ClN2
    Pureza:99.61%
    Cor e Forma:Solid
    Peso molecular:340.89
  • SCH-23390 hydrochloride

    CAS:
    <p>SCH-23390 hydrochloride (R-(+)-SCH23390 hydrochloride) is an effective dopamine receptor antagonist, and for the D1(Ki=0.2 nM) and D5(Ki=0.3 nM).</p>
    Fórmula:C17H19Cl2NO
    Pureza:98% - 99.83%
    Cor e Forma:Solid
    Peso molecular:324.24
  • Mosapride

    CAS:
    <p>Mosapride (AS-4370) is a selective 5HT4 agonist</p>
    Fórmula:C21H25ClFN3O3
    Pureza:99.56%
    Cor e Forma:White To Off-White Crystalline Solid
    Peso molecular:421.89
  • Tianeptine sodium salt

    CAS:
    <p>Tianeptine sodium salt 是一种选择性5-HT 摄取促进剂,具有抗抑郁、抗焦虑和神经保护作用,可用于缓解疼痛的研究。</p>
    Fórmula:C21H24ClN2NaO4S
    Pureza:99.82%
    Cor e Forma:Solid
    Peso molecular:458.93
  • Vilazodone Hydrochloride

    CAS:
    <p>Vilazodone Hydrochloride (EMD 68843) , a partial agonist of 5-HT1A receptors and specific serotonin reuptake inhibitor (SSRI), is utilized in treating of the</p>
    Fórmula:C26H27N5O2·HCl
    Pureza:99.56% - >99.99%
    Cor e Forma:Solid
    Peso molecular:477.99
  • Xaliproden hydrochloride

    CAS:
    <p>Xaliproden is a compound that mimics the effects of nerve growth factor and is also a serotonin 5-HT1A receptor agonist.</p>
    Fórmula:C24H23ClF3N
    Pureza:99.99%
    Cor e Forma:Solid
    Peso molecular:417.89
  • lumateperone Tosylate

    CAS:
    <p>lumateperone Tosylate (ITI-007) is a 5-HT2A receptor antagonist, a partial agonist of presynaptic D2 receptors and an antagonist of postsynaptic D2 receptors.</p>
    Fórmula:C31H36FN3O4S
    Pureza:95.83% - 99.95%
    Cor e Forma:Solid
    Peso molecular:565.7
  • Cerlapirdine

    CAS:
    <p>Cerlapirdine (PF-05212365), a 5-HT6 receptor antagonist, is in trials for Alzheimer's and schizophrenia cognition issues.</p>
    Fórmula:C22H23N3O3S
    Pureza:98.77%
    Cor e Forma:Solid
    Peso molecular:409.5
  • Cariprazine hydrochloride

    CAS:
    <p>Cariprazine hydrochloride (RGH188 hydrochloride) is an antipsychotic drug, is a D3 and D2 receptor partial agonist((Ki of 0.085 nM and 0.49 nM, respectively)</p>
    Fórmula:C21H33Cl3N4O
    Pureza:99.78% - >99.99%
    Cor e Forma:Solid
    Peso molecular:463.87
  • Lerisetron

    CAS:
    <p>Lerisetron is an antagonist of serotonin type 3 (5-HT3) receptor, with antiemetic activity.</p>
    Fórmula:C18H20N4
    Pureza:99.15% - 99.82%
    Cor e Forma:Solid
    Peso molecular:292.38
  • Indophagolin

    CAS:
    <p>Indophagolin: autophagy inhibitor, IC50 140 nM; blocks P2X4, P2X1, P2X3 receptors, IC50s 2.71, 2.40, 3.49 μM.</p>
    Fórmula:C19H15BrClF3N2O3S
    Pureza:99.76%
    Cor e Forma:Solid
    Peso molecular:523.75
  • Amperozide

    CAS:
    <p>Amperozide (FG 5606), an atypical antipsychotic, antagonizes 5-HT2A and modulates dopamine activity for schizophrenia treatment.</p>
    Fórmula:C23H29F2N3O
    Pureza:99.68%
    Cor e Forma:Solid
    Peso molecular:401.49
  • Metoclopramide hydrochloride hydrate

    CAS:
    <p>Metoclopramide hydrochloride hydrate (Metoclopramide monohydrochloride monohydrate) is a dopamine D2 antagonist that is a drug used for digestive dysfunction.</p>
    Fórmula:C14H25Cl2N3O3
    Pureza:99.33%
    Cor e Forma:Solid
    Peso molecular:354.27
  • Eltoprazine hydrochloride

    CAS:
    <p>Eltoprazine hydrochloride (DU 28853 hydrochloride) is a partial agonist at serotonin 5-HT1A, 5-HT1B, and 5-HT2B receptors (Ki value of 40, 52, and 81 nM,</p>
    Fórmula:C12H17ClN2O2
    Pureza:99.35%
    Cor e Forma:Solid
    Peso molecular:256.73
  • Vortioxetine hydrobromide

    CAS:
    <p>Vortioxetine hydrobromide (Lu AA21004 hydrobromide) is a serotonin (5-HT) modulator and stimulator (SMS), inhibits 5-HT1A/1B/3A/7 receptor and SERT (IC50: 15/33</p>
    Fórmula:C18H22N2S·HBr
    Pureza:98.85% - 99.98%
    Cor e Forma:Solid
    Peso molecular:379.36
  • Azaphen dihydrochloride monohydrate

    CAS:
    <p>Azaphen dihydrochloride monohydrate is a 5-hydroxytryptamine reabsorption inhibitor with antidepressant activity and can be used to study neurological diseases.</p>
    Fórmula:C16H23Cl2N5O2
    Pureza:99.85%
    Cor e Forma:Solid
    Peso molecular:388.29
  • RS-67333

    CAS:
    <p>RS-67333 is a partial agonist of 5-HT4R with neuroprotective effects.</p>
    Fórmula:C19H29ClN2O2
    Pureza:99.24%
    Cor e Forma:Solid
    Peso molecular:352.9
  • SB 243213

    CAS:
    <p>SB 243213 is a 5-HT2C receptor antagonist with anxiolytic and antidepressant activity used in schizophrenia and movement disorders.</p>
    Fórmula:C22H19F3N4O2
    Pureza:98.78% - 99.86%
    Cor e Forma:Solid
    Peso molecular:428.41
  • (S)-Mirtazapine

    CAS:
    <p>(S)-Mirtazapine ((S)-Org3770) is a 5-HT2 receptor antagonist with pro-nociceptive effects that can be used to study depression.</p>
    Fórmula:C17H19N3
    Pureza:99.37%
    Cor e Forma:Solid
    Peso molecular:265.35
  • Renzapride

    CAS:
    <p>Renzapride (BRL 24924) is a mixed 5-hydroxytryptamine type 4 (5-HT4) agonist and 5-HT3 receptor antagonist used in the study of irritable bowel syndrome.</p>
    Fórmula:C16H22ClN3O2
    Pureza:98.97% - 99.09%
    Cor e Forma:Solid
    Peso molecular:323.82
  • Ketanserin tartrate

    CAS:
    <p>Ketanserin tartrate (KJK-945 tartrate) is a 5-HT2A receptor and α1-adrenergic receptor antagonist for the study of systemic sclerosis.</p>
    Fórmula:C26H28FN3O9
    Pureza:99.68%
    Cor e Forma:Solid
    Peso molecular:545.51