
Receptor 5-HT
Os receptores 5-HT, também conhecidos como receptores de serotonina, são um grupo de receptores acoplados à proteína G (GPCRs) que mediam os efeitos da serotonina, um neurotransmissor envolvido na regulação do humor, ansiedade, sono, apetite e outros processos fisiológicos. Esses receptores são divididos em vários subtipos, cada um com funções e propriedades farmacológicas distintas. Moduladores de receptores 5-HT são amplamente estudados por seus papéis no tratamento da depressão, distúrbios de ansiedade e outras condições neuropsiquiátricas. Na CymitQuimica, oferecemos uma variedade de moduladores de receptores 5-HT de alta qualidade para apoiar sua pesquisa em neurofarmacologia, transtornos do humor e sinalização GPCR.
Foram encontrados 940 produtos de "Receptor 5-HT"
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TG6-10-1
CAS:<p>TG6-10-1 is an EP2 antagonist.</p>Fórmula:C23H23F3N2O4Pureza:99.66% - ≥95%Cor e Forma:SolidPeso molecular:448.43Puerarin
CAS:<p>Puerarin (Kakonein), also known as Kakonein, is a member of the class of compounds known as isoflavonoid C-glycosides. It is a 5-HT2C receptor antagonist.</p>Fórmula:C21H20O9Pureza:98.90% - 99.21%Cor e Forma:Yellow Brown Fine PowderPeso molecular:416.38Rotigotine Hydrochloride
CAS:<p>Rotigotine HCl, D3-preferential dopamine agonist, is 50x stronger than quinpirole in anti-Parkinson's efficacy.</p>Fórmula:C19H26ClNOSPureza:99.53% - 99.56%Cor e Forma:Almost White To White Crystalline PowderPeso molecular:351.93Rotigotine-
CAS:<p>Rotigotine (N-0923) is a non-ergot dopamine receptor agonist used in the therapy of Parkinson disease and restless leg syndrome.</p>Fórmula:C19H25NOSPureza:98.08% - 99.59%Cor e Forma:SolidPeso molecular:315.47MK 212 hydrochloride
CAS:<p>MK 212 hydrochloride is a 5-HT2C receptor agonist</p>Fórmula:C8H11ClN4·HClPureza:99.88%Cor e Forma:SolidPeso molecular:235.12Metadoxine
CAS:<p>Metadoxine (Metadoxil) is a neurotransmitter stimulant.</p>Fórmula:C8H11NO3·C5H7NO3Pureza:99.19%Cor e Forma:Off-White PowderPeso molecular:298.29Intepirdine
CAS:<p>Intepirdine (GSK-742457) is a highly selective 5-HT6 receptor antagonist, used in trials studying the treatment of Alzheimer's Disease.</p>Fórmula:C19H19N3O2SPureza:98% - 98.63%Cor e Forma:SolidPeso molecular:353.44Mosapride Citrate
CAS:<p>Mosapride Citrate (TAK-370 citrate), a gastroprokinetic agent, utilizes as a selective 5HT4 agonist.</p>Fórmula:C21H25ClFN3O3·C6H8O7Pureza:99.70%Cor e Forma:White PowderPeso molecular:614.02GSK163090
CAS:<p>GSK163090 is a specific and orally active 5-HT1A/B/D receptor antagonist (pKis: 9.4/8.5/9.7, and 6.3/6.7 for 5-HT1A/B/D, and dopamine D2/D3).</p>Fórmula:C25H29N5OPureza:99.2%Cor e Forma:SolidPeso molecular:415.53Tianeptine
CAS:<p>Tianeptine (Tianeptine sodium) 是一种选择性5-HT 摄取促进剂,具有抗抑郁、抗焦虑和神经保护作用,可用于缓解疼痛的研究。</p>Fórmula:C21H25ClN2O4SPureza:99.04%Cor e Forma:SolidPeso molecular:436.95Niaprazine
CAS:<p>Niaprazine is a histamine H1-receptor antagonist with marked sedative properties.</p>Fórmula:C20H25FN4OPureza:99.56%Cor e Forma:SolidPeso molecular:356.44BRL-15572 dihydrochloride
CAS:<p>BRL-15572 dihydrochloride: 5-HT1D antagonist, pKi 7.9, also binds 5-HT1A/2B, 60x selective over 5-HT1B.</p>Fórmula:C25H27ClN2O·2HClPureza:99.74%Cor e Forma:SolidPeso molecular:479.87Dolasetron Mesylate hydrate
CAS:<p>Dolasetron Mesylate hydrate blocks 5HT3 to prevent chemo and radiotherapy nausea.</p>Fórmula:C20H26N2O7SPureza:99.86% - 99.9%Cor e Forma:SolidPeso molecular:438.49PRX-08066
CAS:<p>PRX-08066 is a selective 5-hydroxytryptamine receptor 2B (5-HT2BR, IC50= 3.4 nM) antagonist that induces selective vasodilation of pulmonary arteries.</p>Fórmula:C19H17ClFN5SPureza:97.79% - 98.07%Cor e Forma:SolidPeso molecular:401.89Ipsapirone hydrochloride
CAS:<p>Ipsapirone, a pyrimidinylpiperazine ligand, is potent and specific for 5-HT1A receptors and has potential therapeutic use in affective disorders.</p>Fórmula:C19H24ClN5O3SCor e Forma:SolidPeso molecular:437.94Donitriptan Mesylate
CAS:<p>Donitriptan Mesylate, a 5-HT1B/1D agonist, is used potentially for the treatment of migraines.</p>Fórmula:C24H29N5O5SCor e Forma:SolidPeso molecular:499.58Melitracen
CAS:<p>Melitracen is a tricyclic antidepressant.</p>Fórmula:C21H25NCor e Forma:SolidPeso molecular:291.43Abaperidone Hydrochloride
CAS:<p>Abaperidone Hydrochloride is an atypical antipsychotic, potently binging to5-HT2 receptors and D2 receptors.</p>Fórmula:C25H26ClFN2O5Cor e Forma:SolidPeso molecular:488.94Melperone
CAS:<p>Melperone, a butyrophenone tranquillizer, caused bradycardia in vivo and in vitro.</p>Fórmula:C16H22FNOPureza:98.84%Cor e Forma:SolidPeso molecular:263.35Cannabigerol
CAS:<p>Cannabigerol is a high affinity α±2-adrenergic receptor agonist, moderate affinity 5-HT1A receptor antagonist, and low affinity CB1 receptor antagonist ; also</p>Fórmula:C21H32O2Pureza:99.59% - 99.92%Cor e Forma:SolidPeso molecular:316.48Temanogrel
CAS:<p>Temanogrel (APD791) is a highly selective antagonist of the 5-HT2A receptor (Ki: 4.9 nM).</p>Fórmula:C24H28N4O4Pureza:99.24%Cor e Forma:SolidPeso molecular:436.52'-O-Methylisoliquiritigenin
CAS:<p>2'-O-Methylisoliquiritigenin, a compound synthesized by enzymes specifically induced in NR.2'-O-Methylisoliquiritigenin, isolated from the Arachis species, up-</p>Fórmula:C16H14O4Pureza:98.75%Cor e Forma:SolidPeso molecular:270.28Alprenolol hydrochloride
CAS:<p>Alprenolol hydrochloride is a non-selective blocker of beta, and also is a antagonist of5-HT1A receptor.</p>Fórmula:C15H24ClNO2Pureza:99.79%Cor e Forma:SolidPeso molecular:285.81idalopirdine
CAS:<p>Idalopirdine (Lu AE58054), a selective 5-HT6 receptor antagonist( Ki : 0.83 nM),as a treatment for Alzheimer's disease.</p>Fórmula:C20H19F5N2OPureza:99.73%Cor e Forma:SolidPeso molecular:398.37Nuciferine
CAS:<p>Nuciferine ((-)-Nuciferine) is an alkaloid found within the plants Nymphaea caerulea and Nelumbo nucifera.</p>Fórmula:C19H21NO2Pureza:98.76% - 99.79%Cor e Forma:SolidPeso molecular:295.38Naratriptan
CAS:<p>Naratriptan is a selective agonist of 5-HT1 receptor and is is used for the treatment of migraine headaches.</p>Fórmula:C17H25N3O2SPureza:99.08%Cor e Forma:SolidPeso molecular:335.47Methiothepin mesylate
CAS:<p>Methiothepin mesylate (Metitepine mesylate) is a potent and non-selective 5-HT2 receptor antagonist, used as an antipsychotic.</p>Fórmula:C21H28N2O3S3Pureza:98% - 99.92%Cor e Forma:SolidPeso molecular:452.65Rotundine
CAS:<p>Rotundine (Gindarine) (L-tetrahydropalmatine, L-THP) is a selective dopamine D1 receptor antagonist with IC50 of 166 nM.</p>Fórmula:C21H25NO4Pureza:99.8% - 99.91%Cor e Forma:Off-White SolidPeso molecular:355.43BMY 7378 dihydrochloride
CAS:<p>BMY 7378 dihydrochloride (BMY7378 HCl) , α1D-adrenergic receptor antagonist, is a weak partial agonist/antagonist of 5-HT1A receptor.</p>Fórmula:C22H33Cl2N3O3Pureza:97.32% - 99.08%Cor e Forma:SolidPeso molecular:458.42F-15599
CAS:<p>F-15599 is a highly selective G-protein biased 5-HT1A receptor agonist(Ki : 3.4 nM).</p>Fórmula:C19H21ClF2N4OPureza:98.72%Cor e Forma:SolidPeso molecular:394.85Pirenperone
CAS:<p>Pirenperone is a putative 5-HT2 receptor antagonist with the central antiserotonergic and antidopaminergic action.</p>Fórmula:C23H24FN3O2Pureza:99.2%Cor e Forma:SolidPeso molecular:393.457-Amino-4-(trifluoromethyl)coumarin
CAS:<p>7-Amino-4-(trifluoromethyl)coumarin (Coumarin 151) is a 5-Hydroxytryptamine Receptor Subtype 1E (HTR1E) antagonist.</p>Fórmula:C10H6F3NO2Pureza:97.31% - 97.84%Cor e Forma:Yellow PowderPeso molecular:229.16Cariprazine
CAS:<p>Cariprazine (RGH-188) is a novel antipsychotic drug candidate that exhibits high affinity for the D3 (Ki=0.085 nM) and D2 (Ki=0.49 nM) receptors, and moderate</p>Fórmula:C21H32Cl2N4OPureza:99.68% - 99.87%Cor e Forma:SolidPeso molecular:427.41Almotriptan Malate
CAS:<p>Almotriptan Malate (PNU180638), a selective 5-HT1B/1D receptor agonist, is used in the therapy of Migraine attacks in adults.</p>Fórmula:C17H25N3O2S·C4H6O5Pureza:99.95%Cor e Forma:Pale Yellow SolidPeso molecular:469.55Escitalopram Oxalate
CAS:<p>Escitalopram Oxalate ((S)-(+)Citalopram oxalate) is a selective serotonin (5-HT) reuptake inhibitor (SSRI) with Ki of 0.89 nM.</p>Fórmula:C22H23FN2O5Pureza:97.39% - 99.73%Cor e Forma:White SolidPeso molecular:414.43Serotonin hydrochloride
CAS:<p>Serotonin hydrochloride (Serotonin HCl) is an endogenous 5-HT receptor agonist, a monoamine neurotransmitter in the CNS, and a catechol O-methyltransferase (</p>Fórmula:C10H13ClN2OPureza:98.05% - 99.93%Cor e Forma:White To Cream PowderPeso molecular:212.676Azaphen
CAS:<p>Azaphen (Pipofezin hydrochloride) is the reuptake of serotonin inhibitor.with antidepressant action and has sedative effects, suggesting antihistamine activity.</p>Fórmula:C16H21Cl2N5OPureza:97.62%Cor e Forma:SolidPeso molecular:370.28Piboserod
CAS:<p>Piboserod (SB-207266) (SB 207266) is a selective 5-HT(4) receptor antagonist.</p>Fórmula:C22H31N3O2Pureza:97.21% - 99.49%Cor e Forma:SolidPeso molecular:369.5Perospirone
CAS:<p>Perospirone (Lullan) is an antagonist of serotonin 5HT2A receptors and dopamine D2 receptors.</p>Fórmula:C23H30N4O2SPureza:99.23%Cor e Forma:White PowderPeso molecular:426.57SB399885
CAS:<p>SB399885 is a potent, brain-penetrant, oral SR-6 antagonist with 200-fold selectivity for SR-6 receptors.</p>Fórmula:C18H21Cl2N3O4SPureza:98.94%Cor e Forma:SolidPeso molecular:446.35LY334370
CAS:<p>LY334370 is a selective 5-HT1F receptor agonist with a Ki of 1.6 nM</p>Fórmula:C21H22FN3OPureza:99.32%Cor e Forma:SolidPeso molecular:351.42Sevoflurane
CAS:<p>Sevoflurane (Fluoromethyl), a noncompetitive inhibitor of 5-HT3 receptor, acts as a low-soluble inhalation anesthetics.</p>Fórmula:C4H3F7OPureza:98%Cor e Forma:Less Oil Colorless OilPeso molecular:200.05Geissoschizine methyl ether
CAS:<p>Geissoschizine methyl ether: an alkaloid from Uncaria hook, key in Yokukansan, impacts mood and social behavior enhancing serotonin activity.</p>Fórmula:C22H26N2O3Pureza:99.24% - 99.68%Cor e Forma:SolidPeso molecular:366.45Ansofaxine hydrochloride
CAS:<p>Ansofaxine hydrochloride (LY03005) is a serotonin-norepinephrine-dopamine reuptake inhibitor (IC50s: 723, 763 and 491 nM, respectively).</p>Fórmula:C24H32ClNO3Pureza:99.57% - 99.77%Cor e Forma:SolidPeso molecular:417.97Tropisetron
CAS:<p>Tropisetron (ICS 205-930) is an α7-nicotinic receptor agonist and 5-HT3 receptor antagonist with Kis of 6.9 nM and 5.3 nM, respectively.</p>Fórmula:C17H20N2O2Pureza:99.68%Cor e Forma:White SolidPeso molecular:284.35Nelotanserin
CAS:<p>Nelotanserin (APD125): strong 5-HT2A inverse agonist (IC50: 1.7 nM), moderate 5-HT2C (79 nM), weak 5-HT2B (791 nM).</p>Fórmula:C18H15BrF2N4O2Pureza:98.42% - 99.88%Cor e Forma:SolidPeso molecular:437.24Amitriptyline
CAS:<p>Amitriptyline: a tricyclic antidepressant used for depression and neuropathic pain.</p>Fórmula:C20H23NPureza:98.24% - 99.64%Cor e Forma:Crystals SolidPeso molecular:277.4Brexpiprazole HCl
CAS:<p>Brexpiprazole HCl (OPC 34712 dihydrochloride) is a new antipsychotic drug.</p>Fórmula:C25H27N3O2S·xHClPureza:99.05%Cor e Forma:SolidPeso molecular:433.6Sarpogrelate hydrochloride
CAS:<p>Sarpogrelate hydrochloride (MCI-9042), a 5-HT2 antagonist with high affinity (Ki=8.39nM), is used as an anti-platelet for PAD, improving vascular function.</p>Fórmula:C24H32ClNO6Pureza:99.73%Cor e Forma:Colorless LiquidPeso molecular:465.97Lurasidone hydrochloride
CAS:<p>Lurasidone HCl: Atypical antipsychotic, treats schizophrenia & bipolar, affects dopamine, serotonin & adrenergic receptors.</p>Fórmula:C28H36N4O2S·HClPureza:99.51%Cor e Forma:SolidPeso molecular:529.14PRX-07034 hydrochloride
CAS:<p>PRX-07034 hydrochloride is a selective antagonist of 5-HT6 receptor. It has cognition and memory-enhancing properties and decreases body weight in rodents.</p>Fórmula:C21H29Cl2N3O4SPureza:98.5%Cor e Forma:SolidPeso molecular:490.44Clozapine N-Oxide
CAS:<p>View and buy CLOZAPINE N-OXIDE from TargetMol.Clozapine N-oxide is a major metabolite of clozapine also known as DREADDs, technology to modulate synthetic receptors in vivo.Cited in 2 publications.</p>Fórmula:C18H19ClN4OPureza:98.43% - 99.94%Cor e Forma:SolidPeso molecular:342.82Nemifitide acetate(173240-15-8 free base)
<p>Nemifitide acetate, synthetic 5-amino acid antidepressant, has quick effect, mimics MIF.</p>Fórmula:C35H47FN10O8Pureza:97.97%Cor e Forma:SolidPeso molecular:754.85Cinitapride
CAS:<p>Cinitapride (Blaston) treats acid reflux and gastric issues, targeting 5-HT2, 5-HT1, and 5-HT4 receptors.</p>Fórmula:C21H30N4O4Pureza:99.52%Cor e Forma:SolidPeso molecular:402.49Pergolide mesylate
CAS:<p>Pergolide mesylate (LY127809), a dopamine agonist for Parkinson's and hyperprolactinemia, was withdrawn for heart valve risk.</p>Fórmula:C20H30N2O3S2Pureza:99.70%Cor e Forma:White To Off-White SolidPeso molecular:410.59Dasotraline hydrochloride
CAS:<p>Dasotraline hydrochloride, a dopamine, norepinephrine, and serotonin reuptake inhibitor with IC50s: 4, 6, 11 nM.</p>Fórmula:C16H16Cl3NPureza:98.92% - 99.6%Cor e Forma:SolidPeso molecular:328.66L-745870 trihydrochloride
CAS:<p>L-745870 trihydrochloride is a highly potent and selective D4 dopamine receptor antagonist.</p>Fórmula:C18H22Cl4N4Pureza:97.52%Cor e Forma:SolidPeso molecular:436.215-Benzyloxygramine
CAS:<p>5-Benzyloxygramine blocks the Dopamin receptors and antagonizes the effects of 5-HT on the rat uterus and the rabbit ear.</p>Fórmula:C18H20N2OPureza:99.13%Cor e Forma:SolidPeso molecular:280.36N-Desmethylclozapine
CAS:<p>N-Desmethylclozapine: 5-HT2C antagonist (IC50: 7.1 nM), dopamine D4 antagonist, δ-opioid agonist.</p>Fórmula:C17H17ClN4Pureza:97.25% - 99.83%Cor e Forma:Yellow Crystalline SolidPeso molecular:312.8NGB 2904
CAS:<p>NGB 2904 is a potent and selective antagonist of dopamine D3 receptor. NGB2904 potently antagonizes mitogenesis stimulated by quinpirole (IC50 = 6.8 nM).</p>Fórmula:C28H29Cl2N3OPureza:98.79%Cor e Forma:SolidPeso molecular:494.46Chlorprothixene
CAS:<p>Chlorprothixene (Truxal) is a typical antipsychotic drug of the thioxanthene class, which was the first of the series to be synthesized.</p>Fórmula:C18H18ClNSPureza:98.77% - 99.756%Cor e Forma:Pale Yellow Crystals SolidPeso molecular:315.86Piperacetazine
CAS:<p>Piperacetazine (Piperacetazinum), an antipsychotic prodrug, is used forschizophrenia.</p>Fórmula:C24H30N2O2SPureza:99.9% - 99.92%Cor e Forma:SolidPeso molecular:410.57Loxapine
CAS:<p>Loxapine, a dibenzoxazepine antipsychotic, treats schizophrenia by blocking D2/D4 and serotonin receptors. Related to clozapine.</p>Fórmula:C18H18ClN3OPureza:99.88%Cor e Forma:Pale Yellowish Crystals From Petroleum Ether SolidPeso molecular:327.81Brexpiprazole
CAS:<p>Brexpiprazole (OPC-34712) is a partial agonist of human 5-hydroxytryptamine (5-HT) 5-HT1A and dopamine D2 receptors.</p>Fórmula:C25H27N3O2SPureza:99.06% - 99.96%Cor e Forma:SolidPeso molecular:433.57Jatrorrhizine
CAS:<p>Jatrorrhizine (neprotin) is a protoberberine alkaloid isolated from Enantia chlorantha (Annonaceae) and other species.</p>Fórmula:C20H20NO4Pureza:97.18% - 99.06%Cor e Forma:SolidPeso molecular:338.38Urapidil
CAS:<p>Urapidil (Ebrantil), a sympatholytic antihypertensive drug, acts as a 5-HT1A receptor agonist and as an α1-adrenoceptor antagonist.</p>Fórmula:C20H29N5O3Pureza:99.85% - >99.99%Cor e Forma:SolidPeso molecular:387.48RS-127445 hydrochloride
CAS:<p>RS-127445 hydrochloride (MT 500) is a selective, high affinity, orally bioavailable 5-HT2B receptor antagonist(pKi : 9.5).</p>Fórmula:C17H17ClFN3Pureza:99.48%Cor e Forma:SolidPeso molecular:317.79Zacopride hydrochloride
CAS:<p>Zacopride is a highly potent 5-HT3 receptor antagonist (Kd = 0.38 nM) and 5-HT4 receptor agonist (Ki = 373 nM). It also is a selective IK1 channel agonist.</p>Fórmula:C15H20ClN3O2·HClPureza:98.32%Cor e Forma:SolidPeso molecular:346.268-Hydroxy-DPAT hydrobromide
CAS:<p>8-Hydroxy-DPAT hydrobromide (8-OH-DPAT hydrobromide) (8-OH-DPAT hydrobromide) is a potent and selective 5-HT1A agonist with a pIC50 of 8.19.</p>Fórmula:C16H26BrNOPureza:98.90% - 99.09%Cor e Forma:SolidPeso molecular:328.29SB-203186 hydrochloride
CAS:<p>SB 203186 hydrochloride is a potent 5-HT4 receptor antagonist</p>Fórmula:C16H20N2O2·HClPureza:99.64%Cor e Forma:SolidPeso molecular:308.81Myristicin
CAS:<p>Myristicin is a natural spice extract with antibacterial, anti-inflammatory, and hepatoprotective properties, and can induce apoptosis.</p>Fórmula:C11H12O3Pureza:99.828%Cor e Forma:LiquidPeso molecular:192.21Hypidone hydrochloride
CAS:<p>Hypidone hydrochloride (YL0919) is a novel antidepressant candidate with dual activity as a 5-HT1A receptor agonist and a selective serotonin reuptake inhibitor</p>Fórmula:C18H23ClN2O2Pureza:99.82% - 99.93%Cor e Forma:SolidPeso molecular:334.84Vortioxetine
CAS:<p>Vortioxetine (Lu AA 21004) is a serotonergic antidepressant used for major depression disorders.</p>Fórmula:C18H22N2SPureza:99.34% - 99.34%Cor e Forma:SolidPeso molecular:298.45BRL 54443
CAS:<p>BRL 54443 is a potent 5-HT1E/1F receptor agonist (pKi values are 8.7 and 8.9 respectively).</p>Fórmula:C14H18N2OPureza:98.07%Cor e Forma:SolidPeso molecular:230.316-fluoro-DL-Tryptophan
CAS:<p>6-fluoro-DL-Tryptophan is an inhibitor of serotonin (5-HT) synthesis.</p>Fórmula:C11H11FN2O2Pureza:99.25%Cor e Forma:Off-White PowderPeso molecular:222.22Serotonin
CAS:<p>Serotonin (5-hydroxytryptamine) is a monoamine neurotransmitter in the CNS and an endogenous 5-HT receptor agonist. High-Quality, Low-Cost!</p>Fórmula:C10H12N2OPureza:97.47% - 99.92%Cor e Forma:SolidPeso molecular:176.22NAN-190 hydrobromide
CAS:<p>NAN-190 hydrobromide is an antagonist of serotonin receptor 5-HT.</p>Fórmula:C23H28BrN3O3Pureza:95.20%Cor e Forma:SolidPeso molecular:474.39Perospirone hydrochloride
CAS:<p>Perospirone hydrochloride (Perospirone HCl) is an atypical antipsychotic agent for the treatment of schizophrenia.</p>Fórmula:C23H31ClN4O2SPureza:99.37%Cor e Forma:White SolidPeso molecular:4633-AQC
CAS:<p>3-AQC is a competitive antagonist of 5-HT3.</p>Fórmula:C20H21N5O4Pureza:99.45%Cor e Forma:SolidPeso molecular:395.41AVN-101
CAS:<p>AVN-101 is a very potent 5-HT7 receptor antagonist.Cost-effective and quality-assured.</p>Fórmula:C21H25ClN2Pureza:99.61%Cor e Forma:SolidPeso molecular:340.89SCH-23390 hydrochloride
CAS:<p>SCH-23390 hydrochloride (R-(+)-SCH23390 hydrochloride) is an effective dopamine receptor antagonist, and for the D1(Ki=0.2 nM) and D5(Ki=0.3 nM).</p>Fórmula:C17H19Cl2NOPureza:98% - 99.83%Cor e Forma:SolidPeso molecular:324.24Mosapride
CAS:<p>Mosapride (AS-4370) is a selective 5HT4 agonist</p>Fórmula:C21H25ClFN3O3Pureza:99.56%Cor e Forma:White To Off-White Crystalline SolidPeso molecular:421.89Tianeptine sodium salt
CAS:<p>Tianeptine sodium salt 是一种选择性5-HT 摄取促进剂,具有抗抑郁、抗焦虑和神经保护作用,可用于缓解疼痛的研究。</p>Fórmula:C21H24ClN2NaO4SPureza:99.82%Cor e Forma:SolidPeso molecular:458.93Vilazodone Hydrochloride
CAS:<p>Vilazodone Hydrochloride (EMD 68843) , a partial agonist of 5-HT1A receptors and specific serotonin reuptake inhibitor (SSRI), is utilized in treating of the</p>Fórmula:C26H27N5O2·HClPureza:99.56% - >99.99%Cor e Forma:SolidPeso molecular:477.99Xaliproden hydrochloride
CAS:<p>Xaliproden is a compound that mimics the effects of nerve growth factor and is also a serotonin 5-HT1A receptor agonist.</p>Fórmula:C24H23ClF3NPureza:99.99%Cor e Forma:SolidPeso molecular:417.89lumateperone Tosylate
CAS:<p>lumateperone Tosylate (ITI-007) is a 5-HT2A receptor antagonist, a partial agonist of presynaptic D2 receptors and an antagonist of postsynaptic D2 receptors.</p>Fórmula:C31H36FN3O4SPureza:95.83% - 99.95%Cor e Forma:SolidPeso molecular:565.7Cerlapirdine
CAS:<p>Cerlapirdine (PF-05212365), a 5-HT6 receptor antagonist, is in trials for Alzheimer's and schizophrenia cognition issues.</p>Fórmula:C22H23N3O3SPureza:98.77%Cor e Forma:SolidPeso molecular:409.5Cariprazine hydrochloride
CAS:<p>Cariprazine hydrochloride (RGH188 hydrochloride) is an antipsychotic drug, is a D3 and D2 receptor partial agonist((Ki of 0.085 nM and 0.49 nM, respectively)</p>Fórmula:C21H33Cl3N4OPureza:99.78% - >99.99%Cor e Forma:SolidPeso molecular:463.87Lerisetron
CAS:<p>Lerisetron is an antagonist of serotonin type 3 (5-HT3) receptor, with antiemetic activity.</p>Fórmula:C18H20N4Pureza:99.15% - 99.82%Cor e Forma:SolidPeso molecular:292.38Indophagolin
CAS:<p>Indophagolin: autophagy inhibitor, IC50 140 nM; blocks P2X4, P2X1, P2X3 receptors, IC50s 2.71, 2.40, 3.49 μM.</p>Fórmula:C19H15BrClF3N2O3SPureza:99.76%Cor e Forma:SolidPeso molecular:523.75Amperozide
CAS:<p>Amperozide (FG 5606), an atypical antipsychotic, antagonizes 5-HT2A and modulates dopamine activity for schizophrenia treatment.</p>Fórmula:C23H29F2N3OPureza:99.68%Cor e Forma:SolidPeso molecular:401.49Metoclopramide hydrochloride hydrate
CAS:<p>Metoclopramide hydrochloride hydrate (Metoclopramide monohydrochloride monohydrate) is a dopamine D2 antagonist that is a drug used for digestive dysfunction.</p>Fórmula:C14H25Cl2N3O3Pureza:99.33%Cor e Forma:SolidPeso molecular:354.27Eltoprazine hydrochloride
CAS:<p>Eltoprazine hydrochloride (DU 28853 hydrochloride) is a partial agonist at serotonin 5-HT1A, 5-HT1B, and 5-HT2B receptors (Ki value of 40, 52, and 81 nM,</p>Fórmula:C12H17ClN2O2Pureza:99.35%Cor e Forma:SolidPeso molecular:256.73Vortioxetine hydrobromide
CAS:<p>Vortioxetine hydrobromide (Lu AA21004 hydrobromide) is a serotonin (5-HT) modulator and stimulator (SMS), inhibits 5-HT1A/1B/3A/7 receptor and SERT (IC50: 15/33</p>Fórmula:C18H22N2S·HBrPureza:98.85% - 99.98%Cor e Forma:SolidPeso molecular:379.36Azaphen dihydrochloride monohydrate
CAS:<p>Azaphen dihydrochloride monohydrate is a 5-hydroxytryptamine reabsorption inhibitor with antidepressant activity and can be used to study neurological diseases.</p>Fórmula:C16H23Cl2N5O2Pureza:99.85%Cor e Forma:SolidPeso molecular:388.29RS-67333
CAS:<p>RS-67333 is a partial agonist of 5-HT4R with neuroprotective effects.</p>Fórmula:C19H29ClN2O2Pureza:99.24%Cor e Forma:SolidPeso molecular:352.9SB 243213
CAS:<p>SB 243213 is a 5-HT2C receptor antagonist with anxiolytic and antidepressant activity used in schizophrenia and movement disorders.</p>Fórmula:C22H19F3N4O2Pureza:98.78% - 99.86%Cor e Forma:SolidPeso molecular:428.41(S)-Mirtazapine
CAS:<p>(S)-Mirtazapine ((S)-Org3770) is a 5-HT2 receptor antagonist with pro-nociceptive effects that can be used to study depression.</p>Fórmula:C17H19N3Pureza:99.37%Cor e Forma:SolidPeso molecular:265.35Renzapride
CAS:<p>Renzapride (BRL 24924) is a mixed 5-hydroxytryptamine type 4 (5-HT4) agonist and 5-HT3 receptor antagonist used in the study of irritable bowel syndrome.</p>Fórmula:C16H22ClN3O2Pureza:98.97% - 99.09%Cor e Forma:SolidPeso molecular:323.82Ketanserin tartrate
CAS:<p>Ketanserin tartrate (KJK-945 tartrate) is a 5-HT2A receptor and α1-adrenergic receptor antagonist for the study of systemic sclerosis.</p>Fórmula:C26H28FN3O9Pureza:99.68%Cor e Forma:SolidPeso molecular:545.51
