
Receptor 5-HT
Os receptores 5-HT, também conhecidos como receptores de serotonina, são um grupo de receptores acoplados à proteína G (GPCRs) que mediam os efeitos da serotonina, um neurotransmissor envolvido na regulação do humor, ansiedade, sono, apetite e outros processos fisiológicos. Esses receptores são divididos em vários subtipos, cada um com funções e propriedades farmacológicas distintas. Moduladores de receptores 5-HT são amplamente estudados por seus papéis no tratamento da depressão, distúrbios de ansiedade e outras condições neuropsiquiátricas. Na CymitQuimica, oferecemos uma variedade de moduladores de receptores 5-HT de alta qualidade para apoiar sua pesquisa em neurofarmacologia, transtornos do humor e sinalização GPCR.
Foram encontrados 940 produtos de "Receptor 5-HT"
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PF-4479745
CAS:<p>PF-4479745 ia a potent and selective agonist of 5-HT2C receptor.</p>Fórmula:C17H22N4Pureza:98%Cor e Forma:SolidPeso molecular:282.38Masupirdine mesylate
CAS:<p>Masupirdine mesylate (SUVN-502 mesylate) is a 5-HT6 receptor antagonist.Masupirdine mesylate is used to study neurological disorders such as Alzheimer's disease</p>Fórmula:C23H32BrN3O9S3Pureza:99.57%Cor e Forma:SolidPeso molecular:670.61Ipsapirone
CAS:<p>Ipsapirone is a partial agonist of 5-HT1A receptor and produces an inhibitory effect on 5-HT2 and the α1-adrenergic function at high doses.</p>Fórmula:C19H23N5O3SPureza:99.51%Cor e Forma:SolidPeso molecular:401.48Lidanserin
CAS:<p>Lidanserin is an antagonist of the 5-HT2A and α1-adrenergic receptor.</p>Fórmula:C26H31FN2O4Pureza:98%Cor e Forma:SolidPeso molecular:454.53SB357134
CAS:<p>SB357134 is a potent, selective and orally active antagonist of 5-HT6 receptor and shows nootropic effects in animal studies.</p>Fórmula:C17H18Br2FN3O3SPureza:98%Cor e Forma:SolidPeso molecular:523.21SDZ 205-557 hydrochloride
CAS:<p>5-HT3/5-HT4 receptor antagonist</p>Fórmula:C14H22Cl2N2O3Pureza:98%Cor e Forma:SolidPeso molecular:337.24Levemopamil HCl
CAS:<p>Levemopamil HCl is used as a calcium channel blocker.</p>Fórmula:C23H31ClN2Pureza:98%Cor e Forma:SolidPeso molecular:370.96Iferanserin
CAS:<p>Iferanserin (S-MPEC) is a selective antagonist of the 5-HT receptor (serotonin receptor) with an affinity for 5-HT2A receptors.</p>Fórmula:C23H28N2OCor e Forma:SolidPeso molecular:348.48TIK-301
CAS:<p>TIK-301 is a chlorinated melatonin derivative and a potent, high-affinity, and orally active melatonin MT1 and MT2 receptors agonist (Kis: 0.081 nM and 0.042 nM</p>Fórmula:C14H17ClN2O2Pureza:98%Cor e Forma:SolidPeso molecular:280.75SB 206553 hydrochloride
CAS:<p>SB 206553 hydrochloride is a 5-HT2C inverse agonist and a 5-HT2C/5-HT2B receptor antagonist with anxiolytic activity, useful for studying neurological disorders</p>Fórmula:C17H17ClN4OPureza:99.56%Cor e Forma:SolidPeso molecular:328.8Fonazine
CAS:<p>Forazine (dimethiazide) is a phenothiazine drug used in the treatment of migraine and is a serotonin antagonist and a histamine antagonist.</p>Fórmula:C19H25N3O2S2Cor e Forma:SolidPeso molecular:391.55SB 207710
CAS:<p>SB 207710 is a selective and high affinity antagonist of 5-HT4 receptor.</p>Fórmula:C19H27IN2O4Cor e Forma:SolidPeso molecular:474.33UCSF678
CAS:<p>UCSF678: selective 42 nM partial agonist at 5-HT5AR, fewer off-target effects, and lower assay risks than SB-699551.</p>Fórmula:C15H18N2O2SCor e Forma:SolidPeso molecular:290.38Pridefine
CAS:<p>Pridefine: antidepressant, balances serotonin, dopamine, norepinephrine reuptake, weakly releases them.</p>Fórmula:C19H21NPureza:99.15% - 99.66%Cor e Forma:SolidPeso molecular:263.385-HT4 antagonist 1
CAS:<p>5-HT4 antagonist 1 is an antagonist of 5-HT4 (pKi = 9.6).</p>Fórmula:C23H36N4O5SPureza:99.75%Cor e Forma:SolidPeso molecular:480.62DR-4004
CAS:<p>DR-4004 is a selective serotonin 5-HT7 receptor antagonist.</p>Fórmula:C26H30N2OCor e Forma:SolidPeso molecular:386.53E-3620
CAS:<p>E-3620 is a potent antagonist of the 5-HT3 receptor and can be used to study dyskinesia and gastrointestinal dysfunction.</p>Fórmula:C20H27Cl2N3O2Pureza:98.88% - 98.88%Cor e Forma:SolidPeso molecular:412.35GR 55562 dihydrochloride
CAS:<p>5-HT1B (5-HT1Dβ) silent antagonist</p>Fórmula:C23H27Cl2N3O2Pureza:99.45%Cor e Forma:SolidPeso molecular:448.39S-15535
CAS:<p>S-15535 is a potent, orally active, partial 5-HT1A receptor agonist.</p>Fórmula:C21H24N2O2Pureza:98%Cor e Forma:SolidPeso molecular:336.43T 82
CAS:<p>T 82 is an antagonist of 5-HT3 and inhibitor of acetylcholinesterase (AChE) and used for the treatment of Alzheimer's Disease.</p>Fórmula:C56H62N6O8Pureza:98%Cor e Forma:SolidPeso molecular:947.146SKF-83566 hydrobromide
CAS:<p>D1-like dopamine receptor antagonist</p>Fórmula:C17H19BrClNOPureza:98%Cor e Forma:SolidPeso molecular:368.7OSU 6162 hydrochloride
CAS:<p>Dopamine stabilizer</p>Fórmula:C15H24ClNO2SPureza:98%Cor e Forma:SolidPeso molecular:317.88MS 245 oxalate
CAS:<p>MS 245 oxalate is a 5-HT6 antagonist.</p>Fórmula:C21H24N2O7SPureza:98%Cor e Forma:SolidPeso molecular:448.49MDL 73005EF hydrochloride
CAS:<p>5-HT1A receptor antagonist</p>Fórmula:C20H27ClN2O4Pureza:98%Cor e Forma:SolidPeso molecular:394.89Eplivanserin hemifumarate
CAS:<p>Eplivanserin is an inverse agonist of 5-HT2A.</p>Fórmula:C23H25FN2O6Cor e Forma:SolidPeso molecular:444.45LY 125180
CAS:<p>LY 125180 is a serotonin antagonist.</p>Fórmula:C18H24ClNOPureza:98%Cor e Forma:SolidPeso molecular:305.84EGIS-7625
CAS:<p>EGIS-7625 is a selective and competitive antagonist of 5-HT2B receptor.</p>Fórmula:C18H24Cl2N4O2Pureza:98%Cor e Forma:SolidPeso molecular:399.32Glemanserin
CAS:<p>Glemanserin (MDL11939) is a specific 5-HT2A antagonist with Ki values of 0.54 nM, 2.5 nM and 2.89 nM for rabbit, human and rat 5-HT2A.</p>Fórmula:C20H25NOPureza:99.93%Cor e Forma:SolidPeso molecular:295.42DV 7028 hydrochloride
CAS:<p>DV 7028 hydrochloride is a 5-HT2A receptor antagonist.</p>Fórmula:C21H26ClFN4O3Pureza:98%Cor e Forma:SolidPeso molecular:436.91RS 23597-190 hydrochloride
CAS:<p>RS 23597-190 hydrochloride is a 5-HT4 receptor antagonist.</p>Fórmula:C16H24Cl2N2O3Pureza:98%Cor e Forma:SolidPeso molecular:363.28L-775,606
CAS:<p>L-775,606 is a selective agonist of 5-hydroxytryptamine 1D.</p>Fórmula:C25H29FN6Pureza:98%Cor e Forma:SolidPeso molecular:432.54MK-212
CAS:<p>MK-212 is a 5HT2C agonist; boosts corticosterone and lowers activity at 0.5-1mg/kg; reduces anxiety without affecting movement at 0.1-0.2mg/kg in mice.</p>Fórmula:C8H11ClN4Cor e Forma:SolidPeso molecular:198.655-HT3 antagonist 2
CAS:<p>5-HT3 antagonist 2 is an antagonist of 5-HT3 receptor.</p>Fórmula:C18H21N3OPureza:98%Cor e Forma:SolidPeso molecular:295.385-HT7 receptor ligand 1
CAS:<p>Compound 5c: 5-HT7 receptor ligand, K i = 8 nM, not hepatotoxic, moderate CYP3A4/CYP2D6 interaction.</p>Fórmula:C21H23N7Cor e Forma:SolidPeso molecular:373.45Bopindolol
CAS:<p>Bopindolol: oral β1/β2-ARs antagonist and partial agonist; prodrug of pindolol for hypertension research.</p>Fórmula:C23H28N2O3Cor e Forma:SolidPeso molecular:380.48Ro 60-0175 fumarate
CAS:<p>5-HT2 receptor agonist</p>Fórmula:C15H16ClFN2O4Pureza:98%Cor e Forma:SolidPeso molecular:342.75Deramciclane fumarate
CAS:<p>Deramciclane fumarate is a 5-HT(2A/C) antagonist with putative anxiolytic activity.</p>Fórmula:C24H35NO5Cor e Forma:SolidPeso molecular:417.54PNU-96415E
CAS:<p>dopamine D4 and serotonergic 5-HT2A receptor antagonist</p>Fórmula:C21H27Cl2FN2OPureza:98%Cor e Forma:SolidPeso molecular:413.36Alaproclate (hydrochloride)
CAS:<p>Alaproclate, an SSRI, enhances serotonin and SIRT1, hinders NMDA and K+ currents in neurons, and shows antidepressant-like effects in rats.</p>Fórmula:C13H19Cl2NO2Cor e Forma:SolidPeso molecular:292.2L 646462
CAS:<p>L 646462 is an antidopaminergic agent.</p>Fórmula:C27H27N3O4Pureza:98%Cor e Forma:SolidPeso molecular:457.52RP5063 Hydrochloride
CAS:<p>RP5063 Hydrochloride is a modulator of multimodal serotonin receptors.</p>Fórmula:C22H26Cl3N3O3Pureza:98%Cor e Forma:SolidPeso molecular:486.82Usmarapride
CAS:<p>Usmarapride (SUVN-D4010) is an oral 5-HT4 receptor agonist, crosses BBB, with an EC50 of 44 nM, for Alzheimer's research.</p>Fórmula:C23H31N5O6Cor e Forma:SolidPeso molecular:473.53AP521
CAS:<p>AP521 is an agonist of the human 5-HT1A receptor (IC50: 94 nM).</p>Fórmula:C20H19ClN2O3SPureza:98%Cor e Forma:SolidPeso molecular:402.89Enciprazine
CAS:<p>Enciprazine (D-3112) shows anxiolytic activity, is used to treat anxiety disorders, and can be used to study depression.</p>Fórmula:C23H32N2O6Pureza:98.63%Cor e Forma:SolidPeso molecular:432.51(R)-Praziquantel
CAS:<p>(R)-Praziquantel is an active enantiomer of praziquantel.</p>Fórmula:C19H24N2O2Pureza:98%Cor e Forma:SolidPeso molecular:312.41Org-13011 fumarate
CAS:<p>Org-13011 fumarate1 is an agonist of the 5-HT1A receptor and can be used to study neurological disorders.</p>Fórmula:C22H29F3N4O5Pureza:98.92%Cor e Forma:SolidPeso molecular:486.48F13714 fumarate
CAS:<p>F13714 fumarate is a 5-HT1A receptor-biased agonist.</p>Fórmula:C25H29ClF2N4O5Pureza:98.86%Cor e Forma:SolidPeso molecular:538.97RG-12915
CAS:<p>RG-12915 is a selective antagonist of 5-HT3(IC50 value of 0.16 nM).</p>Fórmula:C20H25ClN2O2Pureza:98%Cor e Forma:SolidPeso molecular:360.88PNU-282987 free base
CAS:<p>PNU-282987 is an α7 nAChR agonist (EC50=154 nM) and a 5-HT3 antagonist (IC50=4541 nM) for nervous system research.</p>Fórmula:C14H17ClN2OPureza:99.64%Cor e Forma:SolidPeso molecular:264.75Lecozotan HCl
CAS:<p>Lecozotan HCl is a selective 5-HT antagonist boosting glutamate and acetylcholine release without causing 5-HT(1A) tolerance.</p>Fórmula:C28H30ClN5O3Pureza:99.04%Cor e Forma:SolidPeso molecular:520.02R 59-022 hydrochloride
CAS:<p>R 59-022 hydrochloride is a 5-HT antagonist, PKC activator, DGK inhibitor (IC50: 2.8 µM), and modulates lipid production in platelets and neutrophils.</p>Fórmula:C27H27ClFN3OSPureza:97.7%Cor e Forma:SolidPeso molecular:496.04RS 42358-197
CAS:<p>RS 42358-197 (RS 25259-007) is a competitive 5-HT3 receptor antagonist.</p>Fórmula:C19H23ClN2OPureza:99.70%Cor e Forma:SolidPeso molecular:330.85DA-6886
CAS:<p>DA-6886 is a 5-HT4 agonist, relaxes rat oesophagus, with 1000x selectivity over hERG channels, pIC50: 4.3.</p>Fórmula:C19H28Cl2N6O2Pureza:99.28% - 99.91%Cor e Forma:SolidPeso molecular:443.37Adoprazine
CAS:<p>Adoprazine (SLV313) is a potential atypical antipsychotic bearing potent D2 receptor antagonist and 5-HT1A receptor agonist properties.</p>Fórmula:C24H24FN3O2Pureza:99.83%Cor e Forma:SolidPeso molecular:405.46Femoxetine hydrochloride
CAS:<p>Femoxetine hydrochloride is a selective 5-hydroxytryptamine reuptake inhibitor used in the study of migraine, depression and eating disorders.</p>Fórmula:C20H26ClNO2Pureza:99.63%Cor e Forma:SolidPeso molecular:347.88Cyamemazine
CAS:<p>Cyamemazine is an antipsychotic compound with sedative and anxiolytic activity.Cyamemazine is a 5-HT3, 5-HT2A, and 5-HT2C receptor antagonist.</p>Fórmula:C19H21N3SPureza:97.01%Cor e Forma:SolidPeso molecular:323.46Masupirdine free base
CAS:<p>Masupirdine free base (SUVN-502 free base) is a 5-HT6 receptor antagonist that can be used to study neurological disorders like Alzheimer's disease.</p>Fórmula:C21H24BrN3O3SPureza:98.36% - 99.65%Cor e Forma:SolidPeso molecular:478.4Landipirdine
CAS:<p>Landipirdine (RO-5025181) is a selective 5-HT6R antagonist for the study of central nervous system disorders such as dementia.</p>Fórmula:C18H19FN2O3SPureza:97.61% - 99.37%Cor e Forma:SolidPeso molecular:362.42Faxeladol
CAS:<p>Faxeladol: adrenergic, serotonin inhibitor & opioid agonist for neurological studies.</p>Fórmula:C15H23NOPureza:98.09% - 98.77%Cor e Forma:SolidPeso molecular:233.35Tedatioxetine
CAS:<p>Tedatioxetine (Lu AA24530) is a serotonin-norepinephrine-dopamine reuptake inhibitor (SNDRI) with antidepressant properties.</p>Fórmula:C18H21NSPureza:99.76% - >99.99%Cor e Forma:SolidPeso molecular:283.43Cianopramine
CAS:<p>Cianopramine (Ro 112465) is a selective 5-hydroxytryptamine uptake inhibitor and a tricyclic antidepressant used in the study of neurological disorders.</p>Fórmula:C20H23N3Pureza:99.92% - 99.92%Cor e Forma:SolidPeso molecular:305.42BL-1020 Mesylate
CAS:<p>BL-1020 Mesylate (CYP-1020 Mesylate) is a GABA A receptor agonist and D2 antagonist used in studies of neurodegeneration.</p>Fórmula:C28H45ClN4O11S4Pureza:>99.99%Cor e Forma:SolidPeso molecular:777.39Viloxazine
CAS:<p>Viloxazine (Viloxazin) (Viloxazin) is a dual-action compound that functions as a norepinephrine reuptake inhibitor and exhibits potent agonistic activity</p>Fórmula:C13H19NO3Pureza:99.67%Cor e Forma:SolidPeso molecular:237.29CP 96021
CAS:<p>"CP 96021 is an antagonist of 5-HT1/2 receptors, with anti-inflammatory and anti-ulcer effects for treating GI tract and asthma."</p>Fórmula:C29H21FN4OSPureza:97.81% - 99.62%Cor e Forma:SoildPeso molecular:492.57Cilansetron
CAS:<p>Cilansetron is an effective and selective 5-HT3 receptor antagonist that can be used for related diseases caused by colitis.</p>Fórmula:C20H21N3OPureza:99.82% - 99.98%Cor e Forma:SolidPeso molecular:319.4E6801
CAS:<p>E6801: selective 5-HT6 agonist for research in dementia, Parkinson's, depression, obesity, epilepsy, anxiety, etc.</p>Fórmula:C17H18ClN5O2S2Pureza:96.32% - 99.53%Cor e Forma:SolidPeso molecular:423.94Ticalopride
CAS:<p>Ticalopride: 5-HT3 agonist for digestive, orofacial, ENT disorders, and bulimia, GERD, IBS research.</p>Fórmula:C14H20ClN3O3Pureza:99.51%Cor e Forma:SolidPeso molecular:313.78SPD-473 citrate
CAS:<p>SPD-473 citrate is an inhibitior of serotonin/dopamine/norepinephrine reuptake.</p>Fórmula:C23H31Cl2NO8SPureza:99.37%Cor e Forma:SolidPeso molecular:552.47Roxindole
CAS:<p>Roxindole: dopamine agonist, serotonin reuptake inhibitor, 5-HT1A agonist, developed for schizophrenia.</p>Fórmula:C23H26N2OPureza:98.03% - 98.93%Cor e Forma:SolidPeso molecular:346.47Aplindore Fumarate
CAS:<p>Aplindore Fumarate (DAB-452), a selective dopamine D2/D3 partial agonist, is used in Parkinson's and schizophrenia research.</p>Fórmula:C22H22N2O7Pureza:>99.99%Cor e Forma:SolidPeso molecular:426.42Nexopamil
CAS:<p>Nexopamil (LU-49938) is a dual calcium channel and 5-HT2A receptor antagonist that inhibits cell contraction and growth.</p>Fórmula:C24H40N2O3Pureza:97.87% - >99.99%Cor e Forma:SolidPeso molecular:404.59ATC 0175 hydrochloride
CAS:<p>ATC 0175 hydrochloride is an orally active melanocyte concentrating hormone 1 receptor antagonist that is potent and selective.</p>Fórmula:C23H26ClF2N5OPureza:99.98%Cor e Forma:SolidPeso molecular:461.93Perphenazine dihydrochloride
CAS:<p>Perphenazine dihydrochloride: Oral dopamine, histamine-1 antagonist; targets D2, D3, 5-HT2A, Alpha-1A; may treat psychiatric disorders, cancer.</p>Fórmula:C21H28Cl3N3OSPureza:99.67%Cor e Forma:SolidPeso molecular:476.89Liafensine
CAS:<p>Liafensine(BMS-820836): Selective inhibitor for serotonin, norepinephrine, dopamine reuptake; targets major depression, CNS disorders.</p>Fórmula:C24H22N4Pureza:99.91%Cor e Forma:SolidPeso molecular:366.46Piromelatine
CAS:<p>Piromelatine is an agonist of melatonin MT1/MT2 receptors, 5-HT1A and 5-HT1D, and an antagonist of 5-HT2B.Piromelatine has antinociceptive activity with</p>Fórmula:C17H16N2O4Pureza:99.89%Cor e Forma:SolidPeso molecular:312.32Litoxetine
CAS:<p>Litoxetine: a selective 5-HT inhibitor & 5-HT3 antagonist, used as an antidepressant with antiemetic effects, Ki=85 nM.</p>Fórmula:C16H19NOPureza:99.47%Cor e Forma:SolidPeso molecular:241.33Lensiprazine
CAS:<p>Lensiprazine (SLV314) is a potent dopamine D(2) receptor antagonist that acts as a serotonin reuptake inhibitor , and can be used to study bipolar disorder and</p>Fórmula:C24H27FN4O2Pureza:98.04%Cor e Forma:SolidPeso molecular:422.5H-9 dihydrochloride
CAS:<p>H-9 dihydrochloride: Strong PKA inhibitor, curbs 5-HT response and EGF signaling, affects pharyngeal function.</p>Fórmula:C11H15Cl2N3O2SPureza:97.3%Cor e Forma:SolidPeso molecular:324.235-HT6/7 antagonist 1
CAS:<p>5-HT6/7 antagonist 1 is a dual 5-HT6/7/2A and D2 receptor antagonist for the study of dementia and Alzheimer's disease.</p>Fórmula:C22H20FN3O3Pureza:98.78% - 99.26%Cor e Forma:SolidPeso molecular:393.41BMY-14802 hydrochloride
CAS:<p>BMY-14802 hydrochloride (BMS 181100 hydrochloride) is a selective antagonist of σ receptor (IC50 = 112 nM) with antipsychotic effects.</p>Fórmula:C18H23ClF2N4OPureza:99.97%Cor e Forma:SolidPeso molecular:384.85Tiospirone
CAS:<p>Tiospirone (BMY 13859-1 free base) is a 5-HT2 receptor antagonist and a dopamine blocker used in the study of neurological disorders such as schizophrenia.</p>Fórmula:C24H32N4O2SPureza:99.74%Cor e Forma:SolidPeso molecular:440.65-HT1A modulator 1
CAS:<p>5-HT1A modulator 1 displays very high affinities for the 5-HT1A, α1-adrenergic receptor, and D2 receptor (IC50s = 2 nM, 10 nM, and 40 nM).</p>Fórmula:C21H25N3O2SPureza:99.68%Cor e Forma:SolidPeso molecular:383.51Pimethixene maleate
CAS:<p>Pimethixene maleate (Pimetixene maleate) is a 5-HT2B receptor antagonist with sedative activity that can be used to study dry cough in children.</p>Fórmula:C23H23NO4SPureza:99.55%Cor e Forma:SolidPeso molecular:409.5Ecopipam
CAS:<p>Ecopipam: orally active, selective dopamine D1/D5 antagonist (Ki: 1.2 nM/2.0 nM). 40x more selective over D2/D4/5-HT/α2a. For schizophrenia, obesity research.</p>Fórmula:C19H20ClNOPureza:99.68%Cor e Forma:SolidPeso molecular:313.82Anpirtoline hydrochloride
CAS:<p>Anpirtoline hydrochloride (D-16949 hydrochloride) is a 5-HT1B receptor agonist and 5-HT3 receptor antagonist used in the study of dyskinesia.</p>Fórmula:C10H14Cl2N2SPureza:>99.99% - >99.99%Cor e Forma:SolidPeso molecular:265.20Ricasetron
CAS:<p>Ricasetron (Brl 46470) is a 5-HT3 receptor antagonist with pro-axonal lysing properties and is used in the study of anxiety disorders and anxiety disorders.</p>Fórmula:C19H27N3OPureza:99.52%Cor e Forma:SolidPeso molecular:313.44Rilapine
CAS:<p>Rilapine (Rilapinum) is an antipsychotic compound that shows high affinity for 5-HT6 receptors and can be used to study neurological disorders.</p>Fórmula:C22H20ClN3Pureza:97.76% - 99.20%Cor e Forma:SolidPeso molecular:361.87Sarizotan HCl
CAS:<p>Sarizotan HCl (EMD 128130 HCl) is a 5-HT1A receptor and dopamine receptor agonist and an hERG channel inhibitor used in Parkinson;s disease research.</p>Fórmula:C22H22ClFN2OPureza:96%Cor e Forma:SolidPeso molecular:384.87Agomelatine hydrochloride
CAS:<p>Agomelatine HCl is a MT1/MT2 receptor agonist (Ki: 0.1-0.27 nM) and a 5-HT2C antagonist (pKi: 6.2-6.4).</p>Fórmula:C15H18ClNO2Pureza:99.57%Cor e Forma:SolidPeso molecular:279.76Fananserin
CAS:<p>Fananserin: Oral 5-HT2A antagonist (Ki=0.37 nM, rat), blocks human D4 receptor (Ki=2.93 nM).</p>Fórmula:C23H24FN3O2SPureza:99.88%Cor e Forma:SolidPeso molecular:425.52Repinotan
CAS:<p>Repinotan (BAY x 3702 free base) is a 5-HT1A receptor agonist used in acute ischemic stroke studies.</p>Fórmula:C21H24N2O4SPureza:99%Cor e Forma:SolidPeso molecular:400.49cis-Urocanic acid
CAS:<p>cis-Urocanic acid ((E)-Urocanic acid) is a 5-HT2A receptor agonist (Kd: 4.6 nM).</p>Fórmula:C6H6N2O2Pureza:99.81%Cor e Forma:SolidPeso molecular:138.12LY 272015 hydrochloride
CAS:<p>LY 272015 hydrochloride is a 5-HT2B receptor antagonist.</p>Fórmula:C21H25ClN2O2Pureza:99.47%Cor e Forma:SolidPeso molecular:372.89Ensaculin
CAS:<p>Ensaculin, a benzopyrone-piperazine compound, enhances memory, protects neurons, and may treat dementia.</p>Fórmula:C26H32N2O5Pureza:99.17% - 99.67%Cor e Forma:SolidPeso molecular:452.54Quinupramine
CAS:<p>Quinupramine: an oral antidepressant targeting the serotonin system; penetrates CNS; doesn’t affect β-adrenergic system.</p>Fórmula:C21H24N2Pureza:99.77%Cor e Forma:SolidPeso molecular:304.43ADR-851 free base
CAS:<p>ADR-851 free base is an antagonist of the HT3 receptor.</p>Fórmula:C14H18ClN3O2Pureza:97.88% - 98.39%Cor e Forma:SolidPeso molecular:295.77ML 10302 hydrochloride
CAS:<p>ML 10302 hydrochloride is a specific agonist 5-HT4 and binds 5-HT receptors with Kis of 1.07 nM and 782 nM for 5-HT4 and 5-HT3.</p>Fórmula:C15H22Cl2N2O3Pureza:99.99%Cor e Forma:SolidPeso molecular:349.25LY266097 hydrochloride
CAS:<p>LY266097 hydrochloride is a 5-HT2 antagonist with pKi of 7.7/9.8/7.6 for 5-HT2A/B/C, used in depression research.</p>Fórmula:C21H24Cl2N2O2Pureza:98.58%Cor e Forma:SolidPeso molecular:407.338-OH-Dpat
CAS:<p>8-OH-Dpat (8-Hydroxy-DPAT) is a serotonin 1A-receptor agonist that is used experimentally to test the effects of serotonin.</p>Fórmula:C16H25NOPureza:98%Cor e Forma:SolidPeso molecular:247.38SB 699551 dihydrochloride
CAS:<p>SB 699551 dihydrochloride is a 5-ht5a receptor antagonist.</p>Fórmula:C34H47Cl2N3OPureza:99.83%Cor e Forma:SolidPeso molecular:584.66
