Receptor 5-HT
Os receptores 5-HT, também conhecidos como receptores de serotonina, são um grupo de receptores acoplados à proteína G (GPCRs) que mediam os efeitos da serotonina, um neurotransmissor envolvido na regulação do humor, ansiedade, sono, apetite e outros processos fisiológicos. Esses receptores são divididos em vários subtipos, cada um com funções e propriedades farmacológicas distintas. Moduladores de receptores 5-HT são amplamente estudados por seus papéis no tratamento da depressão, distúrbios de ansiedade e outras condições neuropsiquiátricas. Na CymitQuimica, oferecemos uma variedade de moduladores de receptores 5-HT de alta qualidade para apoiar sua pesquisa em neurofarmacologia, transtornos do humor e sinalização GPCR.
Foram encontrados 940 produtos de "Receptor 5-HT"
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Altanserin
CAS:<p>Altanserin, a 5-HT2A receptor binder, is tagged with F-18 for brain PET scans.</p>Fórmula:C22H22FN3O2SCor e Forma:SolidPeso molecular:411.49Setiptiline maleate
CAS:<p>Setiptiline maleate is a norepinephrine reuptake inhibitor, 2-adrenergic receptor antagonist, H1 receptor inverse agonist, 5-HT serotonin receptor antagonist.</p>Fórmula:C23H23NO4Pureza:99.94%Cor e Forma:SolidPeso molecular:377.43Eplivanserin (mixture)
CAS:<p>Eplivanserin mixture is a selective serotonin reuptake inhibitor and a 5-HT2A receptor antagonist,</p>Fórmula:C19H21FN2O2Cor e Forma:SolidPeso molecular:328.387SB-269970 hydrochloride
CAS:<p>SB-269970 hydrochloride (SB-269970A) , a hydrochloride salt form of SB-269970, is a 5-HT7 receptor antagonist (pKi of 8.3) and exhibits >50-fold selectivity</p>Fórmula:C18H28N2O3S·HClPureza:98.45%Cor e Forma:SolidPeso molecular:388.95Fluvoxamine
CAS:<p>Fluvoxamine (DU-23000) is a selective, orally available 5-HT and serotonin reuptake inhibitor (SSRI) exhibiting antidepressant effects.</p>Fórmula:C15H21F3N2O2Cor e Forma:SolidPeso molecular:318.33SB-200646A
CAS:<p>SB-200646A: oral 5-HT2B/2C antagonist; higher affinity than 5-HT2A (pKi: 7.5, 6.9 vs 5.2); anxiolytic with in vivo effects.</p>Fórmula:C15H15ClN4OPureza:98%Cor e Forma:SolidPeso molecular:302.76Cefaclor
CAS:<p>Cefaclor (Panoral) is a cephalosporin antibiotic.</p>Fórmula:C15H14ClN3O4SPureza:99.03% - 99.98%Cor e Forma:SolidPeso molecular:367.81(R)-Praziquantel-d11
CAS:<p>(R)-Praziquantel D11 is the deuterium labeled (R)-Praziquantel.</p>Fórmula:C19H24N2O2Pureza:98%Cor e Forma:SolidPeso molecular:323.47Sumatriptan
CAS:<p>Sumatriptan (GR 43175 free base) is a 5-HT1 receptor agonist with anti-inflammatory activity used in acute migraine and acute myocardial infarction.</p>Fórmula:C14H21N3O2SPureza:99.93%Cor e Forma:White To Off-White Crystalline PowderPeso molecular:295.4Aripiprazole (D8)
CAS:<p>Aripiprazole D8 (OPC-14597 D8) is the deuterium-labeled Aripiprazole. Aripiprazole is a human 5-HT1A receptor partial agonist (Ki: 4.2 nM).</p>Fórmula:C23H27Cl2N3O2Pureza:98%Cor e Forma:SolidPeso molecular:456.441-Phenylbiguanide HCl
CAS:<p>Compound PDK0269, as 5-HT3 receptor agonists(3–100 μM, pEC50 5.05±0.06), acutely increased XII (hypoglossal) burst frequency and regularity, and decreased bursts/episode . Phenylbiguanide produced a dose-related (10-500 microM) increase in the release of dopamine (280-2000%). When nomifensine (5 microM) was included in the Ringer solution, the effect of Compound PDK0269 on the release of dopamine was ameliorated or inhibited.</p>Fórmula:C8H12ClN5Pureza:99.31%Cor e Forma:SolidPeso molecular:213.67SB-277011 hydrochloride
CAS:<p>SB-277011 hydrochloride (SB-277011A hydrochloride) is a D3R antagonist, which induces delayed ejaculation in rats.</p>Fórmula:C28H31ClN4OPureza:98.54%Cor e Forma:SolidPeso molecular:475.03Thioridazine
CAS:<p>Thioridazine: an antipsychotic, anti-anxiety drug, blocks dopamine D2, PI3K-Akt-mTOR; halts angiogenesis, kills cancer cells, targets CSCs.</p>Fórmula:C21H26N2S2Cor e Forma:SolidPeso molecular:370.57Clozapine-d8
CAS:<p>Clozapine-d8 is a deuterium-labeled analog of Clozapine, used as an internal standard for mass spectrometric analysis of this atypical antipsychotic.</p>Fórmula:C18H19ClN4Cor e Forma:SolidPeso molecular:334.87Spiroxatrine
CAS:<p>Spiroxatrine (R 5188) is a 5-HT1α and α2-adrenergic dual antagonist with sedative activity for the study of diseases related to the cardiovascular system.</p>Fórmula:C22H25N3O3Pureza:99.94%Cor e Forma:SolidPeso molecular:379.45Ziprasidone D8
CAS:<p>Ziprasidone D8, deuterium-labeled, is a potent antipsychotic, antagonizing 5-HT and dopamine receptors.</p>Fórmula:C21H21ClN4OSPureza:98%Cor e Forma:SolidPeso molecular:420.99Agomelatine-d6
CAS:<p>Agomelatine D6 (S-20098 D6) is a deuterium-labeled Agomelatine. Agomelatine is a specific agonist of MT1 and MT2 receptors.</p>Fórmula:C15H17NO2Pureza:98%Cor e Forma:SolidPeso molecular:249.34Quetiapine-d4 hemifumarate
CAS:<p>Quetiapine D4 hemifumarate is the deuterium labeled Quetiapine hemifumarate. Quetiapine hemifumarate is a agonist of 5-HT receptors and a antagonist of dopamine receptor,with ntidepressant and anxiolytic.</p>Fórmula:C25H29N3O6SPureza:98%Cor e Forma:White SolidPeso molecular:503.61Dehydroaripiprazole
CAS:<p>Dehydroaripiprazole (DM-14857), aripiprazole's active metabolite, is formed by CYP3A4 and CYP2D6, with similar antipsychotic effects.</p>Fórmula:C23H25Cl2N3O2Pureza:98.7%Cor e Forma:SolidPeso molecular:446.37Paliperidone Palmitate
CAS:<p>Paliperidone: atypical antipsychotic, dopamine & serotonin antagonist, affects α1/α2 adrenergic and H1 histamine receptors.</p>Fórmula:C39H57FN4O4Pureza:98%Cor e Forma:SolidPeso molecular:664.89
