Receptor 5-HT
Os receptores 5-HT, também conhecidos como receptores de serotonina, são um grupo de receptores acoplados à proteína G (GPCRs) que mediam os efeitos da serotonina, um neurotransmissor envolvido na regulação do humor, ansiedade, sono, apetite e outros processos fisiológicos. Esses receptores são divididos em vários subtipos, cada um com funções e propriedades farmacológicas distintas. Moduladores de receptores 5-HT são amplamente estudados por seus papéis no tratamento da depressão, distúrbios de ansiedade e outras condições neuropsiquiátricas. Na CymitQuimica, oferecemos uma variedade de moduladores de receptores 5-HT de alta qualidade para apoiar sua pesquisa em neurofarmacologia, transtornos do humor e sinalização GPCR.
Foram encontrados 985 produtos de "Receptor 5-HT"
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Dolasetron
CAS:<p>Dolasetron (MDL-73147)(MDL-73147) is a serotonin 5-HT3 receptor antagonist. Dolasetron is used to treat nausea and vomiting following chemotherapy.</p>Fórmula:C19H20N2O3Pureza:99.84% - 99.86%Cor e Forma:White PowderPeso molecular:324.37AC-90179 HCl
CAS:<p>AC-90179 HCl: selective 5-HT2A inverse agonist, atypical antipsychotic, reduces hallucinogen-induced vasoconstriction.</p>Fórmula:C23H31ClN2O2Pureza:99.71%Cor e Forma:SolidPeso molecular:402.96Almotriptan Malate
CAS:<p>Almotriptan Malate (PNU180638), a selective 5-HT1B/1D receptor agonist, is used in the therapy of Migraine attacks in adults.</p>Fórmula:C17H25N3O2S·C4H6O5Pureza:99.95%Cor e Forma:Pale Yellow SolidPeso molecular:469.55Ritanserin
CAS:Ritanserin (R 55667) is a long-acting, highly potent, relatively selective, orally bioavailable 5-HT2 receptor antagonist.Cost-effective and quality-assured.Fórmula:C27H25F2N3OSPureza:99.77% - 99.89%Cor e Forma:SolidPeso molecular:477.57Opiranserin hydrochloride
CAS:<p>Opiranserin (VVZ-149) hydrochloride is a dual antagonist of glycine transporter type 2 (GlyT2) and serotonin receptor 2A (5HT2A), with IC50s of 0.86 and 1.3 μM</p>Fórmula:C21H35ClN2O5Pureza:99.33%Cor e Forma:SolidPeso molecular:430.97Eltoprazine dihydrochloride
CAS:<p>Eltoprazine dihydrochloride, a drug developed for aggression, is now studied for L-DOPA-induced dyskinesia in Parkinson's.</p>Fórmula:C12H18Cl2N2O2Pureza:99.64%Cor e Forma:SolidPeso molecular:293.19Nefazodone hydrochloride
CAS:<p>Nefazodone hydrochloride (Serzone) is a serotoninergic modulating antidepressant that is used in therapy of depression, aggressive behavior and panic disorder.</p>Fórmula:C25H33Cl2N5O2Pureza:99% - 99.86%Cor e Forma:White SolidPeso molecular:506.477-Amino-4-(trifluoromethyl)coumarin
CAS:7-Amino-4-(trifluoromethyl)coumarin (Coumarin 151) is a 5-Hydroxytryptamine Receptor Subtype 1E (HTR1E) antagonist.Fórmula:C10H6F3NO2Pureza:97.31% - 97.84%Cor e Forma:Yellow PowderPeso molecular:229.16F-15599
CAS:<p>F-15599 is a highly selective G-protein biased 5-HT1A receptor agonist(Ki : 3.4 nM).</p>Fórmula:C19H21ClF2N4OPureza:98.72%Cor e Forma:SolidPeso molecular:394.85Pirenperone
CAS:<p>Pirenperone is a putative 5-HT2 receptor antagonist with the central antiserotonergic and antidopaminergic action.</p>Fórmula:C23H24FN3O2Pureza:99.2%Cor e Forma:SolidPeso molecular:393.45Cariprazine
CAS:<p>Cariprazine (RGH-188) is a novel antipsychotic drug candidate that exhibits high affinity for the D3 (Ki=0.085 nM) and D2 (Ki=0.49 nM) receptors, and moderate</p>Fórmula:C21H32Cl2N4OPureza:99.68% - 99.87%Cor e Forma:SolidPeso molecular:427.41Melperone
CAS:<p>Melperone, a butyrophenone tranquillizer, caused bradycardia in vivo and in vitro.</p>Fórmula:C16H22FNOPureza:98.84%Cor e Forma:SolidPeso molecular:263.35Escitalopram Oxalate
CAS:<p>Escitalopram Oxalate ((S)-(+)Citalopram oxalate) is a selective serotonin (5-HT) reuptake inhibitor (SSRI) with Ki of 0.89 nM.</p>Fórmula:C22H23FN2O5Pureza:97.39% - 99.73%Cor e Forma:White SolidPeso molecular:414.43Lerisetron
CAS:Lerisetron is an antagonist of serotonin type 3 (5-HT3) receptor, with antiemetic activity.Fórmula:C18H20N4Pureza:99.15% - 99.82%Cor e Forma:SolidPeso molecular:292.38Temanogrel hydrochloride
CAS:Temanogrel hydrochloride is a serotonin antagonist and anti-platelet agent.Fórmula:C24H29ClN4O4Cor e Forma:SolidPeso molecular:472.97Naratriptan hydrochloride
CAS:<p>Naratriptan Hydrochloride, a selective 5-HT1 receptor agonist with anti-migraine effect, induces vasoconstriction and reduces inflammation in migraines.</p>Fórmula:C17H25N3O2S·HClPureza:99.17% - 99.93%Cor e Forma:Beige SolidPeso molecular:371.93Renzapride hydrochloride
CAS:Renzapride is a 5-HT3 antagonist and 5-HT4 agonist. Renzapride also functions as a 5-HT2B antagonist and has some affinity for the 5-HT2A and 5-HT2C receptors.Fórmula:C16H23Cl2N3O2Cor e Forma:SolidPeso molecular:360.28Ralmitaront
CAS:<p>Ralmitaront (RO6889450) is a potent, orally active partial agonist of the trace amine-associated receptor 1 (TAAR1).</p>Fórmula:C17H22N4O2Pureza:99.71% - 99.79%Cor e Forma:SolidPeso molecular:314.38Naftopidil dihydrochloride
CAS:<p>Naftopidil dihydrochloride (KT-611 2HCl) is a selective 5-HT1A and α1-adrenergic receptor antagonist with IC50 of 0.1 μM and 0.2 μM, respectively.</p>Fórmula:C24H28N2O3·2HClPureza:99.76%Cor e Forma:White SolidPeso molecular:465.41TG6-10-1
CAS:<p>TG6-10-1 is an EP2 antagonist.</p>Fórmula:C23H23F3N2O4Pureza:99.66% - ≥95%Cor e Forma:SolidPeso molecular:448.43
