Receptor 5-HT
Os receptores 5-HT, também conhecidos como receptores de serotonina, são um grupo de receptores acoplados à proteína G (GPCRs) que mediam os efeitos da serotonina, um neurotransmissor envolvido na regulação do humor, ansiedade, sono, apetite e outros processos fisiológicos. Esses receptores são divididos em vários subtipos, cada um com funções e propriedades farmacológicas distintas. Moduladores de receptores 5-HT são amplamente estudados por seus papéis no tratamento da depressão, distúrbios de ansiedade e outras condições neuropsiquiátricas. Na CymitQuimica, oferecemos uma variedade de moduladores de receptores 5-HT de alta qualidade para apoiar sua pesquisa em neurofarmacologia, transtornos do humor e sinalização GPCR.
Foram encontrados 940 produtos de "Receptor 5-HT"
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Tandospirone
CAS:<p>Tandospirone (SM-3997) is a 5-HT1A receptor partial agonist with anxiolytic and antidepressant activity used in the study of central nervous system disorders.</p>Fórmula:C21H29N5O2Pureza:99.94%Cor e Forma:SolidPeso molecular:383.49Setiptiline
CAS:<p>Setiptiline (Org-8282) is a norepinephrine reuptake inhibitor, 2-adrenergic receptor antagonist, H1 receptor inverse agonist with antidepressant activity.</p>Fórmula:C19H19NPureza:98.05% - 98.07%Cor e Forma:SolidPeso molecular:261.36Latrepirdine dihydrochloride
CAS:<p>Latrepirdine dihydrochloride (Dimebolin dihydrochloride) is an orally active, and neuroactive antagonist of multiple drug targets.</p>Fórmula:C21H25N3·2HClPureza:98.45%Cor e Forma:SolidPeso molecular:392.37Rizatriptan
CAS:<p>Rizatriptan (Risatriptan) is a selective 5-hydroxytryptamine 1B/1D receptor agonist used in the study of migraine.</p>Fórmula:C15H19N5Pureza:99.74%Cor e Forma:SolidPeso molecular:269.35(R)-Mirtazapine
CAS:<p>(R)-Mirtazapine ((R)-Org3770) is a 5-HT3 receptor antagonist, a potential analgesic with anti-injury perception properties.</p>Fórmula:C17H19N3Pureza:99.75%Cor e Forma:SolidPeso molecular:265.35Rotigotine
CAS:<p>Rotigotine (1-Naphthalenol, 5,6,7,8-tetrahydro-6-[propyl[2-(2-thienyl)ethyl]amino]-) is an antiparkinson agent and dopamine receptor agonist.</p>Fórmula:C19H25NOSPureza:99.04% - 99.88%Cor e Forma:SolidPeso molecular:315.47LP-533401 hydrochloride
CAS:<p>LP-533401 hydrochloride is a peripheral Tph inhibitor that does not cross the BBB and can be used to study periodontal disease and hepatic steatosis.</p>Fórmula:C27H23ClF4N4O3Pureza:98%Cor e Forma:SolidPeso molecular:562.94Citalopram
CAS:<p>Citalopram (Lu 10-171), a serotonin and 5-HT reuptake inhibitor.Citalopram has antidepressant activity and may be used to study dementia.</p>Fórmula:C20H21FN2OPureza:99.78% - 99.89%Cor e Forma:SolidPeso molecular:324.39WAY-100635 maleate
CAS:<p>WAY-100635 Maleate is a specific and effective 5-HT receptor antagonist (IC50=0.95 nM).</p>Fórmula:C25H34N4O2·xC4H4O4Pureza:>99.99%Cor e Forma:White SolidPeso molecular:538.645Jatrorrhizine chloride
CAS:<p>Jatrorrhizine chloride (Neprotine chloride) is an alkaloid isolated from Rhizoma coptidis with neuroprotective, antimicrobial, and antiplasmodial activities.</p>Fórmula:C20H20ClNO4Pureza:99.79%Cor e Forma:SolidPeso molecular:373.8S1RA
CAS:<p>S1RA (E-52862)(E-52862) is a potent, selective antagonist of the sigma-1 receptor (σ1R, Ki=17 nM), demonstrating significant selectivity over the sigma-2</p>Fórmula:C20H23N3O2Pureza:99.45%Cor e Forma:SolidPeso molecular:337.42Syk Inhibitor II
CAS:<p>Syk inhibitor II, a cell-permeable, ATP-competitive, pyrimidine-carboxamide compound, selectively and reversibly inhibits Syk (IC50 = 41 nM).</p>Fórmula:C14H15F3N6OPureza:97.63%Cor e Forma:SolidPeso molecular:340.3R 59-022
CAS:<p>R 59-022 (DKGI-I) is a DGK inhibitor and a 5-HT Receptor antagonist that blocks filovirus internalization in host cells.</p>Fórmula:C27H26FN3OSPureza:98.55%Cor e Forma:SolidPeso molecular:459.58Cyproheptadine hydrochloride
CAS:<p>Cyproheptadine hydrochloride (Periactin hydrochloride) is a hydrochloride salt form of cyproheptadine which is a histamine receptor antagonist.</p>Fórmula:C21H21N·HClPureza:99.88% - 99.97%Cor e Forma:SolidPeso molecular:323.86Risperidone Mesylate
CAS:<p>Risperidone Mesylate is a selective serotonin 5-HT2 receptor and dopamine D2 receptor blocker.</p>Fórmula:C24H31FN4O5SPureza:98%Cor e Forma:SolidPeso molecular:506.59Escitalopram
CAS:<p>Escitalopram (Seroplex), a serotonin inhibitor for depression, curbs alcohol intake and is favored over tricyclics for tardive dyskinesia.</p>Fórmula:C20H21FN2OPureza:99.82%Cor e Forma:White Or White Crystalline PowderPeso molecular:324.39N-Methyl amisulpride
CAS:<p>N-Methyl amisulpride (Amisulpride impurity H) is a 5-HT7 receptor, D2 receptor, and D3 receptor antagonist used in the study of acute schizophrenia.</p>Fórmula:C18H29N3O4SCor e Forma:SolidPeso molecular:383.51Keto Ziprasidone
CAS:<p>Ziprasidone, an antipsychotic agent, functions as a dual antagonist of 5-HT (serotonin) and dopamine receptors.</p>Fórmula:C21H19ClN4O2SPureza:98%Cor e Forma:SolidPeso molecular:426.92Arazasetron HCl
CAS:<p>Arazasetron is an antiemetic which acts as a 5-HT3 receptor antagonist, pKi = 9.27.</p>Fórmula:C17H20ClN3O3Pureza:98%Cor e Forma:SolidPeso molecular:349.81Brexpiprazole-d8
CAS:<p>Brexpiprazole D8 is a deuterium-modified partial agonist of 5-HT1A and dopamine receptors, with Ki values of 0.12 nM and 0.3 nM respectively.</p>Fórmula:C25H27N3O2SPureza:98%Cor e Forma:SolidPeso molecular:441.62Amitriptyline-d6 Hydrochloride
CAS:<p>Amitriptyline-d6 Hydrochloride is a deuterated compound of Amitriptyline Hydrochloride. Amitriptyline Hydrochloride has a CAS number of 549-18-8. Amitriptyline Hydrochloride is the hydrochloride salt of the tricyclic dibenzocycloheptadiene amitriptyline with antidepressant and antinociceptive activities.</p>Fórmula:C20H18D6ClNCor e Forma:SolidPeso molecular:319.90Mirtazapine D3
CAS:<p>Mirtazapine D3 is a deuterium labeled Mirtazapine. Mirtazapine is an inhibitor of 5-HT receptor .</p>Fórmula:C17H19N3Pureza:98%Cor e Forma:SolidPeso molecular:268.375-Methyltryptamine hydrochloride
CAS:<p>5-Methyltryptamine hydrochloride is a high-affinity 5-HT1C receptor ligand and a partial agonist of 5-HT. 5-Methyltryptamine hydrochloride protects mice subjected to burn, tourniquet and endotoxin shock.</p>Fórmula:C11H15ClN2Pureza:99.45%Cor e Forma:SolidPeso molecular:210.703Penbutolol sulfate
CAS:<p>Penbutolol sulfate ((-)-Terbuclomine) is able to bind to both β2-adrenergic receptor and β1-adrenergic receptor, thus making it a non-selective β blocker.</p>Fórmula:C18H29NO2H2O4SPureza:98.55%Cor e Forma:SolidPeso molecular:340.47Ketanserinol
CAS:<p>Ketanserinol is a metabolite of the antihypertensive drug ketanserin, which blocks 5-HT2 receptors to treat protamine-induced pulmonary hypertension.</p>Fórmula:C22H24FN3O3Cor e Forma:SolidPeso molecular:397.447-Desmethyl-3-hydroxyagomelatine
CAS:<p>7-Desmethyl-3-hydroxyagomelatine, less active than parent drug Agomelatine, is a melatonergic agonist and 5-HT2C antagonist.</p>Fórmula:C14H15NO3Pureza:98%Cor e Forma:SolidPeso molecular:245.27Diclofensine
CAS:<p>Diclofensine (Ro 8-4650) inhibits the uptake of serotonin, noradrenaline and dopamine.</p>Fórmula:C17H17Cl2NOPureza:97.01% - 98.13%Cor e Forma:SolidPeso molecular:322.23Hydroxy ziprasidone
CAS:<p>Hydroxy ziprasidone is an impurity of Ziprasidone. Ziprasidone, an antipsychotic agent, is a 5-HT and dopamine receptor antagonist.</p>Fórmula:C21H21ClN4O2SPureza:98%Cor e Forma:SolidPeso molecular:428.94Pardoprunox
CAS:<p>Pardoprunox (SLV-308) is a partial dopamine D2 agonist and noradrenergic agonist with serotonin 5-HT1A agonist properties.</p>Fórmula:C12H15N3O2Pureza:98%Cor e Forma:SolidPeso molecular:233.27SB 271046 hydrochloride
CAS:<p>SB 271046 hydrochloride (SB 271046A) is selective, orally active 5-HT6 antagonist and is > 200-fold selective over 55 other receptors, enzymes and ion channels.</p>Fórmula:C20H22ClN3O3S2·HClPureza:99.77%Cor e Forma:SolidPeso molecular:488.45Paroxetine hydrochloride hemihydrate
CAS:<p>Paroxetine hydrochloride hemihydrate (Paxil) is an effective and selective serotonin reuptake inhibitor (SSRI).</p>Fórmula:C38H44Cl2F2N2O7Pureza:99.949%Cor e Forma:SolidPeso molecular:749.67Dolasetron Mesylate
CAS:<p>Dolasetron Mesylate (MDL-73147EF) is an antagonist of the 5-HT3 receptor and can be used in research on the treatment of vomiting and nausea following</p>Fórmula:C20H24N2O6SPureza:99.05%Cor e Forma:White PowderPeso molecular:420.48LY 344864
CAS:<p>LY 344864, a specifc receptor agonist, is an affinity of 6 nM (Ki) at the recently cloned 5-HT1F receptor.</p>Fórmula:C21H22FN3OPureza:98%Cor e Forma:SolidPeso molecular:351.42Ampreloxetine
CAS:<p>Ampreloxetine (TD-9855) is a norepinephrine reuptake inhibitor used to study neurological diseases.</p>Fórmula:C18H18F3NOPureza:98%Cor e Forma:SolidPeso molecular:321.342-Methyl-5-HT maleate
CAS:<p>2-Methyl-5-HT maleate, a selective 5-HT3 agonist, shows anti-depressive effects.</p>Fórmula:C15H18N2O5Pureza:98%Cor e Forma:SolidPeso molecular:306.31Ro 04-6790
CAS:<p>Ro 04-6790 is a 5-HT6 receptor antagonist.</p>Fórmula:C12H16N6O2SPureza:98%Cor e Forma:SolidPeso molecular:308.36ST1936
CAS:<p>ST1936 (ST 1936 oxalate) is a 5-HT6 receptor agonist that stimulates cAMP, Ca2+, ERK1/2, and Fyn kinases by fully activating cloned human 5-HT6 receptors.</p>Fórmula:C13H17ClN2Pureza:98%Cor e Forma:SolidPeso molecular:236.74Org37684
CAS:<p>5-HT2 receptors agonist</p>Fórmula:C14H20ClNO2Pureza:98%Cor e Forma:SolidPeso molecular:269.77Donitriptan
CAS:<p>Donitriptan 是一种 5-HT 受体激动剂，对 5-HT1B 和 5-HT1D 的 pKi 分别为 9.4 和 9.3。</p>Fórmula:C23H25N5O2Pureza:98.76%Cor e Forma:SolidPeso molecular:403.48AR-A 2
CAS:<p>AR-A 2, a selective 5-HT1B antagonist; high guinea pig 5-HT1B/1D affinity (Ki: 0.24, 0.47 nM); 10x less for 5-HT1D (Ki: 5 nM).</p>Fórmula:C27H36N4O2Pureza:98%Cor e Forma:SolidPeso molecular:448.6AVN-322
CAS:<p>AVN-322 is a 5-HT6 receptor antagonist. 5-HT6R antagonists improves cognition in animal models of cognitive impairment.</p>Fórmula:C17H20ClN5O2SPureza:>99.99%Cor e Forma:SolidPeso molecular:393.89Alniditan dihydrochloride
CAS:<p>Alniditan dihydrochloride is a potent 5-HT1D agonist and migraine-abortive agent.</p>Fórmula:C17H28Cl2N4OCor e Forma:SolidPeso molecular:375.34Methiothepin maleate
CAS:<p>Methiothepin maleate (Metitepine) is a 5-HT1, 5-HT6, 5-HT7 serotonin receptor antagonist, which blocks serotonin autoreceptors.</p>Fórmula:C24H28N2O4S2Pureza:98%Cor e Forma:SolidPeso molecular:472.62RS 56812 hydrochloride
CAS:<p>5-HT3 partial agonist</p>Fórmula:C18H22ClN3O2Pureza:98.62%Cor e Forma:SolidPeso molecular:347.84AL-37350A
CAS:<p>AL-37350A is a 5-HT2 receptor-selective agonist with ocular hypotensive activity.</p>Fórmula:C14H18N2OCor e Forma:SolidPeso molecular:230.31CUMI-101
CAS:<p>CUMI-101 is an agonist of 5-HT1A receptor.</p>Fórmula:C19H27N5O3Cor e Forma:SolidPeso molecular:373.45Ifoxetine sulfate
CAS:<p>Ifoxetine sulfate, an atypical 5-HT inhibitor, may show unique therapeutic effects and side-effects.</p>Fórmula:C13H19NO2H2O4SPureza:98%Cor e Forma:SolidPeso molecular:270.34WAY 629 hydrochloride
CAS:<p>5-HT2C agonist</p>Fórmula:C15H19ClN2Pureza:98%Cor e Forma:SolidPeso molecular:262.78E55888
CAS:<p>E55888 is a potent and selective full agonist of the 5HT7 serotonin receptor.</p>Fórmula:C16H23N3Cor e Forma:SolidPeso molecular:257.37Etoperidone hydrochloride
CAS:<p>Etoperidone hydrochloride is an antidepressant agent.</p>Fórmula:C19H29Cl2N5OCor e Forma:SolidPeso molecular:414.37
