
Receptor 5-HT
Os receptores 5-HT, também conhecidos como receptores de serotonina, são um grupo de receptores acoplados à proteína G (GPCRs) que mediam os efeitos da serotonina, um neurotransmissor envolvido na regulação do humor, ansiedade, sono, apetite e outros processos fisiológicos. Esses receptores são divididos em vários subtipos, cada um com funções e propriedades farmacológicas distintas. Moduladores de receptores 5-HT são amplamente estudados por seus papéis no tratamento da depressão, distúrbios de ansiedade e outras condições neuropsiquiátricas. Na CymitQuimica, oferecemos uma variedade de moduladores de receptores 5-HT de alta qualidade para apoiar sua pesquisa em neurofarmacologia, transtornos do humor e sinalização GPCR.
Foram encontrados 1024 produtos de "Receptor 5-HT"
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Agomelatine-d6
CAS:Agomelatine D6 (S-20098 D6) is a deuterium-labeled Agomelatine. Agomelatine is a specific agonist of MT1 and MT2 receptors.Fórmula:C15H17NO2Pureza:98%Cor e Forma:SolidPeso molecular:249.34Quetiapine-d4 hemifumarate
CAS:Quetiapine D4 hemifumarate is the deuterium labeled Quetiapine hemifumarate. Quetiapine hemifumarate is a agonist of 5-HT receptors and a antagonist of dopamine receptor,with ntidepressant and anxiolytic.Fórmula:C25H29N3O6SPureza:98%Cor e Forma:White SolidPeso molecular:503.61Ziprasidone amino acid
CAS:<p>Ziprasidone Impurity C is a byproduct of Ziprasidone, an antipsychotic that blocks 5-HT and dopamine receptors.</p>Fórmula:C21H23ClN4O2SCor e Forma:SolidPeso molecular:430.95Paliperidone Palmitate
CAS:Paliperidone: atypical antipsychotic, dopamine & serotonin antagonist, affects α1/α2 adrenergic and H1 histamine receptors.Fórmula:C39H57FN4O4Pureza:98%Cor e Forma:SolidPeso molecular:664.89Quetiapine-d8 Fumarate
CAS:Quetiapine-d8 Fumarate is a deuterated compound of Quetiapine Fumarate. Quetiapine Fumarate has a CAS number of 111974-72-2. Quetiapine Fumarate, an atypical antipsychotic, is used in the treatment of bipolar I mania, schizophrenia, bipolar II depression, bipolar I depression.Fórmula:C25H21D8N3O6SCor e Forma:SolidPeso molecular:507.63Spiroxatrine
CAS:Spiroxatrine (R 5188) is a 5-HT1α and α2-adrenergic dual antagonist with sedative activity for the study of diseases related to the cardiovascular system.Fórmula:C22H25N3O3Pureza:99.94%Cor e Forma:SolidPeso molecular:379.45Asenapine hydrochloride
CAS:Asenapine hydrochloride (Org 5222 hydrochloride) is an antagonist of 5-hydroxytryptamine, adrenergic, dopamine, and histamine receptors with antipsychotic effects.Fórmula:C17H17Cl2NOCor e Forma:SolidPeso molecular:322.23Levomepromazine
CAS:Levomepromazine (Methotrimeprazine) is a Ca2+ release inducer with antiviral, anti-inflammatory, neuroprotective, sedative, and anti-nociceptive activities.Fórmula:C19H24N2OSPureza:99.15%Cor e Forma:SolidPeso molecular:328.47Clozapine-d8
CAS:Clozapine-d8 is a deuterium-labeled analog of Clozapine, used as an internal standard for mass spectrometric analysis of this atypical antipsychotic.Fórmula:C18H19ClN4Cor e Forma:SolidPeso molecular:334.87Nefazodone
CAS:Nefazodone (Nefadar) is an oral antidepressant that is an antagonist of postsynaptic 5-HT 2A receptors and 5-HT 2C receptors, and SNDRI.Fórmula:C25H32ClN5O2Pureza:99.85%Cor e Forma:White To Off-White Crystalline PowderPeso molecular:470.01Ref: TM-T21451
2mg45,00€5mg64,00€10mg91,00€25mg187,00€50mg291,00€100mg446,00€200mg637,00€1mL*10mM (DMSO)100,00€WAY-100635
CAS:WAY-100635 is a potent 5-HT 1A receptor antagonist pyramidal neuron firing frequency during conditioned reflexes; a dopamine D4 receptor agonist .Fórmula:C25H34N4O2Pureza:98.972%Cor e Forma:SolidPeso molecular:422.56(Rac)-Rotigotine hydrochloride
CAS:(Rac)-Rotigotine hydrochloride is a racemate of Rotigotine. Rotigotine is a full agonist of dopamine receptor, a partial the 5-HT1A receptor agonist.Fórmula:C19H26ClNOSCor e Forma:SolidPeso molecular:351.93Alosetron D3 Hydrochloride
CAS:Alosetron D3 (GR 68755 D3) Hydrochloride is a deuterium-labeled Alosetron. Alosetron is an antagonist of 5HT3-receptor.Fórmula:C17H19ClN4OPureza:98%Cor e Forma:SolidPeso molecular:333.83Cariprazine D6
CAS:<p>Cariprazine D6 (RGH-188 D6) is a deuterium-labeled Cariprazine. Cariprazine is an antipsychotic agent (D3 receptors, Ki: 0.085 nM; D2 receptors, Ki: 0.49 nM).</p>Fórmula:C21H26D6Cl2N4OPureza:98%Cor e Forma:SolidPeso molecular:433.45Vilazodone-d8
CAS:Vilazodone D8 is a deuterium-labeled vilazodone. Vilazodone is a combined inhibitor of serotonin specific reuptake (SSRI) and agonist of 5-HT1A receptor partial.Fórmula:C26H27N5O2Pureza:98%Cor e Forma:SolidPeso molecular:449.57Dehydroaripiprazole
CAS:Dehydroaripiprazole (DM-14857), aripiprazole's active metabolite, is formed by CYP3A4 and CYP2D6, with similar antipsychotic effects.Fórmula:C23H25Cl2N3O2Pureza:98.7%Cor e Forma:SolidPeso molecular:446.37Quetiapine-d8 Hemifumarate
CAS:Quetiapine-d8 Hemifumarate is a deuterated compound of Quetiapine Hemifumarate. Quetiapine Hemifumarate has a CAS number of 111974-72-2. Quetiapine Fumarate, an atypical antipsychotic, is used in the treatment of bipolar I mania, schizophrenia, bipolar II depression, bipolar I depression.Fórmula:C25H21D8N3O6SCor e Forma:SolidPeso molecular:507.63Asenapine
CAS:Asenapine (Org 5222) is a 5-HT receptor, adrenergic receptor, and histamine receptor antagonist with antipsychotic properties for the treatment of schizophreniaFórmula:C17H16ClNOPureza:99.64%Cor e Forma:CoaPeso molecular:285.775-HT3 antagonist 5
CAS:5-HT3 antagonist 5, a quinoxalin-2-carboxamide, blocks 5-HT3 receptors and has antidepressant effects in mice.Fórmula:C16H13N3O2Pureza:99.84%Cor e Forma:SolidPeso molecular:279.295-HT2B antagonist-1
CAS:Orally active 5-HT2B antagonist; IC50 = 33.4 nM; potential for hepatocellular, cardiovascular, GI disease research.Fórmula:C11H14BrN5Pureza:99.965%Cor e Forma:SolidPeso molecular:296.17
