
Receptor 5-HT
Os receptores 5-HT, também conhecidos como receptores de serotonina, são um grupo de receptores acoplados à proteína G (GPCRs) que mediam os efeitos da serotonina, um neurotransmissor envolvido na regulação do humor, ansiedade, sono, apetite e outros processos fisiológicos. Esses receptores são divididos em vários subtipos, cada um com funções e propriedades farmacológicas distintas. Moduladores de receptores 5-HT são amplamente estudados por seus papéis no tratamento da depressão, distúrbios de ansiedade e outras condições neuropsiquiátricas. Na CymitQuimica, oferecemos uma variedade de moduladores de receptores 5-HT de alta qualidade para apoiar sua pesquisa em neurofarmacologia, transtornos do humor e sinalização GPCR.
Foram encontrados 1043 produtos para "Receptor 5-HT".
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Ketanserin
CAS:Ketanserin: quinazoline derivative, 5-HT2 receptor antagonist, may lower blood pressure and inhibit blood clots.Fórmula:C22H22FN3O3Pureza:99.19% - 99.73%Cor e Forma:SolidPeso molecular:395.43Azatadine dimaleate
CAS:Azatadine dimaleate (SCH10649) is an inhibitor for histamine(IC50=6.5 nM) and cholinergic(IC50=10 nM).Fórmula:C28H30N2O8Pureza:99.7% - >99.99%Cor e Forma:SolidPeso molecular:522.55Pizotifen
CAS:Pizotifen is a serotonin antagonist with mild anticholinergic effects, used in migraine prevention. Not available in the USA.Fórmula:C19H21NSPureza:99.93%Cor e Forma:White SolidPeso molecular:295.44Lamotrigine
CAS:Lamotrigine (BW430C) is an Anti-epileptic Agent and Mood Stabilizer.Fórmula:C9H7Cl2N5Pureza:99.76% - 99.95%Cor e Forma:White SolidPeso molecular:256.09CP-809101 hydrochloride
CAS:CP-809101 hydrochloride is a potent and selective 5-HT2C receptor agonist (pEC50: 9.96/7.19/6.81 for human 5-HT2C/5-HT2B/5-HT2A receptors).Fórmula:C15H18Cl2N4OPureza:99.5%Cor e Forma:Yellow SolidPeso molecular:341.24Alosetron hydrochloride
CAS:Alosetron hydrochloride (GR 68755), a selective 5-HT3 receptor antagonist, can block the actions of serotonin at 5-HT3 sites in the peripheral nervous system.Fórmula:C17H19ClN4OPureza:99.90%Cor e Forma:Off-White PowderPeso molecular:330.81Trazodone hydrochloride
CAS:Trazodone hydrochloride (Trazodone HCl) is a serotonin uptake inhibitor that is used as an antidepressive agent.Fórmula:C19H23Cl2N5OPureza:99.5% - 99.52%Cor e Forma:SolidPeso molecular:408.33Gevotroline
CAS:Gevotroline, a chemical in palm wine that can be used to treat psychosis, is a 5-HT2 receptor antagonist that can be used to study behavioral disorders.Fórmula:C19H20FN3Pureza:99.45%Cor e Forma:SolidPeso molecular:309.38Agomelatine
CAS:Agomelatine (Valdoxan), like melatonin, boosts mood by targeting melatonin and 5-HT2C receptors.Fórmula:C15H17NO2Pureza:99.92%Cor e Forma:White SolidPeso molecular:243.30Ziprasidone hydrochloride
CAS:Ziprasidone hydrochloride (CP-88059 hydrochloride) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychoticFórmula:C21H22CL2N4OSPureza:97.97% - 99.82%Cor e Forma:White SolidPeso molecular:449.4NEO 376
CAS:NEO 376 (SPI-376) is a selective 5-HT1 receptor, GABA receptor and dopamine receptor modulator, showing anti-psychotic actively.Fórmula:C20H24ClN3OPureza:99.56%Cor e Forma:SolidPeso molecular:357.88Ref: TM-T12207
1mg71,00€5mg133,00€1mL*10mM (DMSO)147,00€10mg205,00€25mg353,00€50mg495,00€100mg665,00€200mg893,00€Ondansetron hydrochloride dihydrate
CAS:Ondansetron hydrochloride dihydrate (GR 38032) is a competitive serotonin type 3 receptor antagonist,which has reported anxiolytic and neuroleptic properties.Fórmula:C18H19N3O·HCl·2H2OPureza:99.92%Cor e Forma:SolidPeso molecular:365.86DREADD agonist 21
CAS:DREADD agonist 21 is a potent agonist of human muscarinic acetylcholine M3 receptors (EC50=1.7 nM).Fórmula:C17H18N4Pureza:99.94%Cor e Forma:White SolidPeso molecular:278.35Ref: TM-T11095L
1mL*10mM (DMSO)34,00€5mg42,00€10mg56,00€25mg94,00€50mg152,00€100mg219,00€200mg314,00€SEP-363856 hydrochloride
CAS:SEP-363856 hydrochloride is an oral, CNS-active psychotropic for schizophrenia with a non-D2/5-HT2A mechanism.Fórmula:C9H14ClNOSPureza:99.86% - 99.99%Cor e Forma:White SolidPeso molecular:219.73Ref: TM-T12899L
1mg66,00€2mg96,00€5mg145,00€1mL*10mM (DMSO)160,00€10mg230,00€25mg404,00€50mg595,00€100mg888,00€500mg1.783,00€Naftidrofuryl oxalate
CAS:Naftidrofuryl oxalate treats peripheral/cerebral vascular issues, boosts cell oxidation, is spasmolytic, and may block 5HT-2 serotonin receptors.Fórmula:C26H35NO7Pureza:97.12% - 99.77%Cor e Forma:White SolidPeso molecular:473.56Naluzotan hydrochloride
CAS:Naluzotan hydrochloride, a hERG K+ blocker (IC50: 3800 nM) and potent 5-HT1A agonist (IC50: ~20 nM, Ki: ~5.1 nM), is used in anxiety and depression studies.Fórmula:C23H39ClN4O3SPureza:99.96%Cor e Forma:SolidPeso molecular:487.1Perphenazine
CAS:Perphenazine (Trilafon) is a phenothiazine derivative and a dopamine antagonist with antiemetic and antipsychotic properties.Fórmula:C21H26ClN3OSPureza:99.3% - 99.99%Cor e Forma:White SolidPeso molecular:403.97Vilazodone
CAS:Vilazodone (SB659746A): an SSRI and 5-HT-1A agonist, boosts serotonin to treat depression and anxiety.Fórmula:C26H27N5O2Pureza:99.61%Cor e Forma:White SolidPeso molecular:441.52Aripiprazole
CAS:Aripiprazole (OPC-14597) is a piperazine/quinolone antipsychotic, partial agonist at 5-HT1A/D2, and antagonist at 5-HT2A.Fórmula:C23H27Cl2N3O2Pureza:99.43% - 99.62%Cor e Forma:White SolidPeso molecular:448.39Aniracetam
CAS:Aniracetam (Ro 13-5057)(Ro 13-5057), a nootropic and neuroprotective drug, selectively modulates the AMPA receptor and nAChR.Fórmula:C12H13NO3Pureza:99.88% - 99.89%Cor e Forma:SolidPeso molecular:219.24
