
Receptor adrenérgico
Os receptores adrenérgicos são GPCRs que são ativados por catecolaminas, como adrenalina e noradrenalina. Esses receptores são classificados em subtipos alfa e beta, cada um dos quais desempenha um papel fundamental na regulação da frequência cardíaca, pressão arterial e resposta de luta ou fuga. Moduladores de receptores adrenérgicos são essenciais no tratamento de doenças cardiovasculares, asma e distúrbios de ansiedade. Na CymitQuimica, oferecemos uma ampla gama de moduladores de receptores adrenérgicos de alta qualidade para apoiar sua pesquisa em endocrinologia, farmacologia cardiovascular e resposta ao estresse.
Subcategorias de "Receptor adrenérgico"
Foram encontrados 645 produtos de "Receptor adrenérgico"
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Procaterol hydrochloride hydrate
CAS:<p>Short-acting β2-adrenergic receptor agonist used to treat asthma.</p>Fórmula:C32H48Cl2N4O7Pureza:99.71% - 99.97%Cor e Forma:SolidPeso molecular:671.65Solabegron HCl
CAS:<p>Solabegron is a β3 adrenergic receptor agonist that also promotes visceral pain relief by releasing somatostatin.</p>Fórmula:C23H24Cl2N2O3Cor e Forma:SolidPeso molecular:447.35Reboxetine
CAS:<p>Reboxetine (Norebox) is an antidepressant drug used in the treatment of clinical depression, panic disorder and ADD/ADHD.</p>Fórmula:C19H23NO3Pureza:98%Cor e Forma:SolidPeso molecular:313.39LY 78335
CAS:<p>LY 78335 (1-(2,3-Dichlorophenyl)ethanamine hydrochloride) is a phenylethanolamine-N-methyltransferase (PNMT) inhibitor.</p>Fórmula:C8H10Cl3NPureza:99.30% - 99.81%Cor e Forma:SolidPeso molecular:226.53Terazosin
CAS:<p>Terazosin: oral α1-blocker, relaxes blood vessels, treats BPH and hypertension.</p>Fórmula:C19H25N5O4Cor e Forma:SolidPeso molecular:387.43Napitane Mesylate
CAS:<p>Napitane Mesylate inhibits norepinephrine transporter and blocks CNS CA uptake as an alpha 2-adrenoceptor antagonist.</p>Fórmula:C23H29NO5SPureza:98%Cor e Forma:SolidPeso molecular:431.55Salmeterol Xinafoate
CAS:<p>Salmeterol Xinafoate (GR 33343X xinafoate) is a long-acting β2-adrenergic receptor agonist with anti-inflammatory effects, used in the treatment of asthma.</p>Fórmula:C36H45NO7Pureza:98% - 98.24%Cor e Forma:White SolidPeso molecular:603.75Fipamezole HCl
CAS:<p>Fipamezole HCl, a α2-adrenoceptor antagonist, is used potentially for the treatment of dyskinesia associated with Parkinson's disease.</p>Fórmula:C14H16ClFN2Cor e Forma:SolidPeso molecular:266.74Nefazodone hydrochloride
CAS:<p>Nefazodone hydrochloride (Serzone) is a serotoninergic modulating antidepressant that is used in therapy of depression, aggressive behavior and panic disorder.</p>Fórmula:C25H33Cl2N5O2Pureza:99% - 99.86%Cor e Forma:White SolidPeso molecular:506.47Parethoxycaine hydrochloride
CAS:<p>Parethoxycaine hydrochloride (2-(diethylamino)ethyl 4-ethoxybenzoate hydrochloride) is an anesthetic[1].</p>Fórmula:C15H24ClNO3Pureza:99.46%Cor e Forma:SolidPeso molecular:301.81ICI 118,551 hydrochloride
CAS:<p>ICI 118,551 hydrochloride (ICI 118551 hydrochloride) is a highly selective β2 adrenergic receptor antagonist (Kis: 0.7, 49.5, and 611 nM for β2, β1, and β3</p>Fórmula:C17H28ClNO2Pureza:99.296% - 99.76%Cor e Forma:SolidPeso molecular:313.86Glaucine
CAS:<p>Glaucine: antitussive, antioxidative, antiviral, may fight arthritis, boosts IL-10, hinders breast cancer cell spread by inhibiting MMP-9 and NF-κB.</p>Fórmula:C21H25NO4Pureza:99.42% - 99.56%Cor e Forma:SolidPeso molecular:355.43Vilanterol trifenatate
CAS:<p>Vilanterol trifenatate is a long-acting agonist of β2-adrenoceptor (β2-AR) with inherent 24-hour activity(β2-AR, β1-AR and β3-AR pEC50s of 10.37, 6.98 and 7.36, respectively)</p>Fórmula:C44H49Cl2NO7Pureza:99.51% - >99.99%Cor e Forma:SolidPeso molecular:774.77Salbutamol hemisulfate
CAS:<p>Salbutamol hemisulfate (Albuterol Sulfate) is a short-acting β2-adrenergic receptor agonist with an IC50 of 8.93 μM.</p>Fórmula:C13H21NO3H2O4SPureza:99.35%Cor e Forma:White Or Almost White Odourless PowderPeso molecular:576.70Fluparoxan HCl
CAS:<p>Fluparoxan is a potent α2-adrenergic receptor antagonist (pKB = 7.9) with excellent α2/α1 selectivity (2630 fold).</p>Fórmula:C10H11ClFNO2Cor e Forma:SolidPeso molecular:231.65Dexmedetomidine hydrochloride
CAS:<p>Dexmedetomidine hydrochloride (Precedex) is a potent, selective, orally active α2-adrenoceptor agonist.Cost-effective and quality-assured.</p>Fórmula:C13H16N2·HClPureza:99.94% - 99.94%Cor e Forma:White Or Almost White Crystalline PowderPeso molecular:236.74Terazosin hydrochloride dihydrate
CAS:<p>Terazosin hydrochloride dihydrate (Heitrin dihydrate) is a selective α1-adrenoceptor antagonist, used for treatment of symptoms of an enlarged prostate (BPH).</p>Fórmula:C19H25N5O4·HCl·2H2OPureza:99.81%Cor e Forma:White Or Off-White Crystalline PowderPeso molecular:459.92Brexpiprazole HCl
CAS:<p>Brexpiprazole HCl (OPC 34712 dihydrochloride) is a new antipsychotic drug.</p>Fórmula:C25H27N3O2S·xHClPureza:99.05%Cor e Forma:SolidPeso molecular:433.6Zotepine
CAS:<p>Zotepine, an antipsychotic agent, is a potent antagonist of 5-HT2A, 5-HT2C, Histamine H1, α1-adrenergic, and Dopamine D2 receptors, with Kds of 2.6 nM, 3.2 nM,</p>Fórmula:C18H18ClNOSPureza:99.78%Cor e Forma:SolidPeso molecular:331.86Tulobuterol hydrochloride
CAS:<p>Tulobuterol hydrochloride (Hokunalin) is a long-acting beta2-adrenergic receptor agonist.</p>Fórmula:C12H19Cl2NOPureza:99.24% - >99.99%Cor e Forma:Appearance White Crystalline PowderPeso molecular:264.19
