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Receptor adrenérgico

Receptor adrenérgico

Os receptores adrenérgicos são GPCRs que são ativados por catecolaminas, como adrenalina e noradrenalina. Esses receptores são classificados em subtipos alfa e beta, cada um dos quais desempenha um papel fundamental na regulação da frequência cardíaca, pressão arterial e resposta de luta ou fuga. Moduladores de receptores adrenérgicos são essenciais no tratamento de doenças cardiovasculares, asma e distúrbios de ansiedade. Na CymitQuimica, oferecemos uma ampla gama de moduladores de receptores adrenérgicos de alta qualidade para apoiar sua pesquisa em endocrinologia, farmacologia cardiovascular e resposta ao estresse.

Subcategorias de "Receptor adrenérgico"

Foram encontrados 645 produtos de "Receptor adrenérgico"

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  • Butanserin

    CAS:
    <p>Butanserin is a 5-hydroxytryptamine S2-antagonist.</p>
    Fórmula:C24H26FN3O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:423.48
  • Methyldopa hydrochloride

    CAS:
    <p>L-(-)-α-Methyldopa HCl: alpha-adrenergic agonist, antihypertensive, inhibits DOPA decarboxylase.</p>
    Fórmula:C10H14ClNO4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:247.68
  • Afurolol Hydrochloride

    CAS:
    <p>Afurolol Hydrochloride (DL 071-IT) is a non-selective β-adrenergic receptor antagonist. DL 071 IT exhibits intrinsic sympathomimetic activity.</p>
    Fórmula:C15H22ClNO4
    Pureza:98.86%
    Cor e Forma:Solid
    Peso molecular:315.79
  • Ulimorelin

    CAS:
    <p>Ulimorelin, ghrelin receptor agonist (EC50: 29 nM, Ki: 16 nM), is a prokinetic and vasorelaxant via α1-adrenoceptor antagonism.</p>
    Fórmula:C30H39FN4O4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:538.65
  • Ronactolol

    CAS:
    <p>Ronactolol is an aminopropanol derivative with beta-adrenoreceptor blocking activity.</p>
    Fórmula:C20H26N2O4
    Cor e Forma:Solid
    Peso molecular:358.43
  • Levobetaxolol

    CAS:
    <p>Levobetaxolol (AL-1577A/Betaxon) is a beta-blocker for ocular hypertension and glaucoma.</p>
    Fórmula:C18H29NO3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:307.43
  • Guanfacine

    CAS:
    <p>Guanfacine is a selective agonist of the α2A receptor.</p>
    Fórmula:C9H9Cl2N3O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:246.09
  • Arnolol

    CAS:
    <p>Arnolol, a beta blocker, slows heart rate, reduces force of beats, lowers blood pressure, and enhances blood flow.</p>
    Fórmula:C14H23NO3
    Cor e Forma:Solid
    Peso molecular:253.34
  • Lubabegron

    CAS:
    <p>Lubabegron(LY488756) is used as an agonist of β3-adrenoreceptor in veterinary.</p>
    Fórmula:C29H29N3O3S
    Cor e Forma:Solid
    Peso molecular:499.62
  • Zolertine HCl

    CAS:
    <p>Zolertine HCl is an antagonist of alpha-Adrenoceptor.</p>
    Fórmula:C13H19ClN6
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:294.78
  • Cirazoline (free base)

    CAS:
    <p>Cirazoline: full α1A agonist, partial α1B/D, nonselective α2 antagonist; potential vasoconstrictor.</p>
    Fórmula:C13H16N2O
    Cor e Forma:Solid
    Peso molecular:216.28
  • ZD 7114 hydrochloride

    CAS:
    <p>β3-adrenoceptor agonist</p>
    Fórmula:C22H31ClN2O6
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:454.94
  • Protokylol

    CAS:
    <p>Protokylol is a β-adrenergic receptor agonist.</p>
    Fórmula:C18H21NO5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:331.36
  • Metazosin

    CAS:
    <p>Metazosin is an antihypertensive agent that replaces 3H-prazosin from its bond to alpha-1 receptors of the cerebral cortex.</p>
    Fórmula:C18H25N5O4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:375.42
  • Piribedil dihydrochloride

    CAS:
    <p>dopamine agonist</p>
    Fórmula:C16H20Cl2N4O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:371.26
  • Todralazine

    CAS:
    <p>Todralazine is an anti-hypertensive agent and acts as a β2AR blocker. It also has an antioxidant and free radical scavenging activity.</p>
    Fórmula:C11H12N4O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:232.24
  • BFE-55

    CAS:
    <p>BFE-55 is derivative of befunolol (a beta-adrenergic partial agonist). BFE-55 interacts with only the high affinity sites in beta-adrenoceptors</p>
    Fórmula:C14H19NO3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:249.31
  • (RS)-Butyryltimolol

    CAS:
    <p>(RS)-Butyryltimolol, a racemic prodrug of Timolol, enhances its corneal absorption and acts as a β-adrenergic blocker.</p>
    Fórmula:C17H30N4O4S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:386.51
  • L-Alprenolol

    CAS:
    <p>L-Alprenolol is a non-selective beta-blocker and a 5-HT1A and 5-HT1B receptor antagonist.</p>
    Fórmula:C15H23NO2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:249.35
  • Centanafadine

    CAS:
    <p>Centanafadine inhibits NE/DA transporters and serotonin transporter (IC50: NE=6 nM, DA=38 nM, 5-HT=83 nM).</p>
    Fórmula:C15H15N
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:209.29
  • S(-)-Bisoprolol

    CAS:
    <p>S(-)-Bisoprolol, a β1-blocker, may aid in researching hypertension and heart diseases.</p>
    Fórmula:C18H31NO4
    Cor e Forma:Solid
    Peso molecular:325.44
  • Spirendolol

    CAS:
    <p>Spirendolol is an antagonist of β adrenergic receptor.</p>
    Fórmula:C21H31NO3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:345.48
  • Epinephrine bitartrate

    CAS:
    <p>L-Epinephrine Bitartrate is alpha- and beta-adrenergic receptor stimulator.</p>
    Fórmula:C13H19NO9
    Pureza:98.6% - 99.07%
    Cor e Forma:White Solid
    Peso molecular:333.3
  • Epanolol

    CAS:
    <p>Epanolol is a potent β-adrenoceptor partial agonist with a greater affinity for β1- than β2-adrenoceptors.</p>
    Fórmula:C20H23N3O4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:369.41
  • Adrenaline sulfate

    CAS:
    <p>Adrenaline sulfate: orally active, α/β-adrenergic agonist, treats anaphylaxis, researched for cardiac arrest.</p>
    Fórmula:C9H15NO7S
    Cor e Forma:Solid
    Peso molecular:281.279
  • Broxaterol

    CAS:
    <p>Broxaterol is a β2 adrenoreceptor agonist. It is part of a class of drugs that affect the smooth muscle receptors in the body.</p>
    Fórmula:C9H15BrN2O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:263.13
  • B-HT 933 dihydrochloride

    CAS:
    <p>Azepexole (B-HT 933) dihydrochloride is an α2-adrenoceptor agonist, pKi: 8.3/α2A, 7.6/α2B, 7.5/α2C; IC50: 78.72 nM for peristalsis inhibition.</p>
    Fórmula:C9H17Cl2N3O
    Cor e Forma:Solid
    Peso molecular:254.16
  • Levobunolol

    CAS:
    <p>Levobunolol is a nonselective beta-blocker. It is used topically to treat glaucoma.</p>
    Fórmula:C17H25NO3
    Cor e Forma:White To Pink Powder
    Peso molecular:291.39
  • Bufetolol

    CAS:
    <p>Bufetolol is an antagonist of beta-adrenoceptor.</p>
    Fórmula:C18H29NO4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:323.43
  • Alprenolol tartrate, (S)-

    CAS:
    <p>Alprenolol tartrate, (S)- is an 5-HT1A antagonist.</p>
    Fórmula:C19H29NO8
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:399.44
  • Guanoxabenz hydrochloride

    CAS:
    <p>Guanoxabenz hydrochloride, α2 adrenergic receptor agonist; Ki: 4000 nM, α2A form Ki: 40 nM.</p>
    Fórmula:C8H9Cl3N4O
    Cor e Forma:Solid
    Peso molecular:283.54
  • Methyldopate hydrochloride

    CAS:
    <p>Methyldopate HCl is an agent of antihypertensive.</p>
    Fórmula:C12H18ClNO4
    Cor e Forma:Solid
    Peso molecular:275.73
  • UK 1745

    CAS:
    <p>UK 1745 is a novel drug of cardiotonic.</p>
    Fórmula:C16H23ClN2O2
    Cor e Forma:Solid
    Peso molecular:310.82
  • Guanethidine

    CAS:
    <p>Guanethidine sulphate, made in 1959, lowers blood pressure by disrupting neurotransmitters in sympathetic nerves.</p>
    Fórmula:C10H22N4
    Cor e Forma:Solid
    Peso molecular:198.31
  • A 55453

    CAS:
    <p>A 55453 is a radiated ionophore used as a reversibl, high-affinity alpha 1-adrenergic receptor probe.</p>
    Fórmula:C25H32N6O3
    Cor e Forma:Solid
    Peso molecular:464.56
  • RS 79948 hydrochloride

    CAS:
    <p>α2-adrenoreceptor antagonist</p>
    Fórmula:C19H29ClN2O3S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:400.96
  • MK761

    CAS:
    <p>MK761 combines β-blocker and vasodilator effects, matching timolol and indololol in efficacy; active in cat heart and rat atria studies.</p>
    Fórmula:C13H19N3O2
    Cor e Forma:Solid
    Peso molecular:249.31
  • Napamezole

    CAS:
    <p>Napamezole: α2 adrenergic receptor antagonist, blocks α1 in rat vas deferens (Kb 135 nM), reverses clonidine effects on twitch height.</p>
    Fórmula:C14H16N2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:212.29
  • Flestolol sulfate

    CAS:
    <p>Flestolol sulfate is an anti-adrenergic beta-receptor.</p>
    Fórmula:C15H24FN3O8S
    Cor e Forma:Solid
    Peso molecular:425.43
  • BMS-466442

    CAS:
    <p>BMS-466442 is the first selective amino acid transporter alanine serine cysteine transporter-1 inhibitor.</p>
    Fórmula:C31H30N4O5
    Cor e Forma:Solid
    Peso molecular:538.59
  • Mabuterol hydrochloride

    CAS:
    <p>Mabuterol hydrochloride is a selective β2 adrenoreceptor agonist. Mabuterol has a specific effect on beta 2-adrenoceptors with no beta 1-stimulation.</p>
    Fórmula:C13H19Cl2F3N2O
    Cor e Forma:Solid
    Peso molecular:347.20
  • Arbutamine hydrochloride

    CAS:
    <p>Arbutamine hydrochloride is a catecholamine which acts as a cardiac stimulant.</p>
    Fórmula:C18H24ClNO4
    Cor e Forma:Solid
    Peso molecular:353.84
  • Fenmetozole

    CAS:
    <p>Fenmetozole is an antagonist of the actions of ethanol.</p>
    Fórmula:C10H10Cl2N2O
    Cor e Forma:Solid
    Peso molecular:245.11
  • CP 59430

    CAS:
    <p>CP 59430 is an azide analogue of prazosin. Prazosin is a highly selective α 1-adrenergic receptor antagonist.</p>
    Fórmula:C21H22N8O3
    Cor e Forma:Solid
    Peso molecular:434.45
  • Clencyclohexerol

    CAS:
    <p>Clencyclohexerol, like clenbuterol, is a β-adrenoceptor agonist with potential in muscle disorders but poses cardiovascular risks at high doses.</p>
    Fórmula:C14H20Cl2N2O2
    Cor e Forma:Solid
    Peso molecular:319.23
  • Dapiprazole

    CAS:
    <p>Dapiprazole, an alpha blocker, is used to reverse mydriasis after eye examination.</p>
    Fórmula:C19H27N5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:325.45
  • BRL 37344 sodium

    CAS:
    <p>BRL 37344 sodium is a specific agonist of the β3-adrenergic receptor. The treatment of BRL 37344 sodium significantly lowers the bodyweight of obese mice.</p>
    Fórmula:C19H22ClNNaO4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:386.83
  • Pronethalol hydrochloride

    CAS:
    <p>β-adrenergic antagonist</p>
    Fórmula:C15H20ClNO
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:265.78
  • Naminterol

    CAS:
    <p>Naminterol is a phenethanolamine derivative is an agonist of β2 adrenoceptor with bronchodilatory properties, and used for treatment of asthma.</p>
    Fórmula:C19H26N2O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:330.42
  • Zenidolol

    CAS:
    <p>Zenidolol (ICI-118551) is a β2 adrenoceptor blocker with K i values: β2 (0.7 nM), β1 (49.5 nM), β3 (611 nM); used in eye disease research.</p>
    Fórmula:C17H27NO2
    Cor e Forma:Solid
    Peso molecular:277.4
  • ONO-2952

    CAS:
    <p>ONO-2952, a selective TSPO antagonist with Ki: 0.33-9.30 nM, may treat irritable bowel syndrome, reducing stress without causing amnesia.</p>
    Fórmula:C22H20ClFN2O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:398.86
  • (-)-S-Timolol

    CAS:
    <p>(-)-S-Timolol is an antagonist of the beta-Adrenergic .</p>
    Fórmula:C13H26N4O4S
    Cor e Forma:Solid
    Peso molecular:334.44
  • Trimazosin

    CAS:
    <p>Trimazosin, a quinazoline derivative and prazosin relative, lowers blood pressure by blocking alpha1-adrenoceptors.</p>
    Fórmula:C20H29N5O6
    Cor e Forma:Solid
    Peso molecular:435.47
  • Primidolol

    CAS:
    <p>Primidolol is a beta adrenergic receptor antagonist and antihypertensive agent.</p>
    Fórmula:C17H23N3O4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:333.38
  • Oxyfedrine

    CAS:
    <p>Oxyfedrine: oral β-adrenoreceptor agonist, vasodilator for cardiovascular research.</p>
    Fórmula:C19H23NO3
    Cor e Forma:Solid
    Peso molecular:313.39
  • Ko-3290

    CAS:
    <p>Ko-3290 is a cardioselective antagonist of β-adrenoceptors known for its antilipolytic effects in animals.</p>
    Fórmula:C19H25N3O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:343.42
  • Imiloxan hydrochloride

    CAS:
    <p>Imiloxan hydrochloride is an α2-adrenoceptor antagonist.</p>
    Fórmula:C14H17ClN2O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:280.75
  • Metrenperone

    CAS:
    <p>Metrenperone is used as a S(2)-receptor blocker.</p>
    Fórmula:C24H26FN3O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:407.48
  • Zinterol hydrochloride

    CAS:
    <p>Zinterol HCl is a selective β2-adrenoceptor agonist.</p>
    Fórmula:C19H27ClN2O4S
    Cor e Forma:Solid
    Peso molecular:414.95
  • Hexoprenaline

    CAS:
    <p>Hexoprenaline is a stimulant of adrenergic beta 2 receptors used as a bronchodilator, antiasthmatic agent, and tocolytic agent.</p>
    Fórmula:C22H32N2O6
    Cor e Forma:Solid
    Peso molecular:420.5
  • Fenmetozole Tosylate

    CAS:
    <p>Fenmetozole Tosylate , acts as an antidepressant drug. is an antagonist of the actions of ethanol, also antagonizes α2-adrenergic receptor,</p>
    Fórmula:C17H18Cl2N2O4S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:417.31
  • Agroclavine

    CAS:
    <p>Agroclavine is a clavine type of ergot alkaloid with D1 dopamine and a-adrenoceptor agonistic properties.</p>
    Fórmula:C16H18N2
    Cor e Forma:Solid
    Peso molecular:238.33
  • ADRA1D receptor antagonist 1 free base

    CAS:
    <p>ADRA1D antagonist blocks bladder contractions; Ki=1.6 nM, IC30=15 nM, useful in overactive bladder research.</p>
    Fórmula:C15H13ClN4O
    Cor e Forma:Solid
    Peso molecular:300.74
  • (E)-Guanabenz

    CAS:
    <p>(E)-Guanabenz is an oral α2-adrenoceptor agonist, antihypertensive, GADD34 inhibitor, and has neuroprotective properties.</p>
    Fórmula:C8H8Cl2N4
    Cor e Forma:Solid
    Peso molecular:231.08
  • Ro 363 hydrochloride

    CAS:
    <p>Ro 363 hydrochloride: selective β1-adrenoceptor agonist, boosts heart contraction, lowers diastolic pressure.</p>
    Fórmula:C19H26ClNO6
    Cor e Forma:Solid
    Peso molecular:399.87
  • Pargolol hydrochloride

    CAS:
    <p>Pargolol hydrochloride is an antagonist of β adrenergic receptor.</p>
    Fórmula:C16H24ClNO3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:313.82
  • Edivoxetine

    CAS:
    <p>Edivoxetine (LY2216684) is a selective norepinephrine reuptake inhibitor for ADHD and depression.</p>
    Fórmula:C18H26FNO4
    Cor e Forma:Solid
    Peso molecular:339.4
  • Medroxalol

    CAS:
    <p>Medroxalol (RMI81968), an oral α- &amp; β-adrenergic blocker, has antihypertensive and vasodilatory effects.</p>
    Fórmula:C20H24N2O5
    Cor e Forma:Solid
    Peso molecular:372.42
  • Povafonidine

    CAS:
    <p>Povafonidine (PGE-6201204), an alpha-2 adrenoreceptor agonist, constricts vessels, reduces congestion for nasal research.</p>
    Fórmula:C11H13N5
    Cor e Forma:Solid
    Peso molecular:215.25
  • MG 1

    CAS:
    <p>MG 1 is a potent alpha-1 adrenergic receptor antagonist.</p>
    Fórmula:C17H25N3O2
    Pureza:98.98% - >99.99%
    Cor e Forma:Solid
    Peso molecular:303.4
  • ZK-90055 hydrochloride

    CAS:
    <p>ZK-90055 hydrochloride is a β2 adrenergic receptor agonist used to study asthma.</p>
    Fórmula:C16H23ClN2O4
    Pureza:99.26%
    Cor e Forma:Solid
    Peso molecular:342.82
  • Thioproperazine

    CAS:
    <p>Thioproperazine (RP 7843) is an orally effective antipsychotic schizophrenia and bipolar disorder, histamine and adrenergic receptor blocker.</p>
    Fórmula:C22H30N4O2S2
    Pureza:99.45%
    Cor e Forma:Solid
    Peso molecular:446.63
  • Guanadrel

    CAS:
    <p>Guanadrel is an antihypertensive agent.</p>
    Fórmula:C10H19N3O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:213.28
  • (E)-Alprenoxime

    CAS:
    <p>(E)-Alprenoxime is the isomer of the Alprenoxime which is a site-activated ocular β-blocker.</p>
    Fórmula:C15H22N2O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:262.35
  • Dexnafenodone Hydrochloride

    CAS:
    <p>Dexnafenodone Hydrochloride is an adrenergic receptor antagonist and serotonin uptake inhibitor.</p>
    Fórmula:C20H24ClNO
    Cor e Forma:Solid
    Peso molecular:329.86
  • LY 87130

    CAS:
    <p>LY 87130 is a phenylethanolamine-N-methyltransferase inhibitor.</p>
    Fórmula:C12H13N
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:171.24
  • Talsupram hydrochloride

    CAS:
    <p>noradrenalin re-uptake inhibitor</p>
    Fórmula:C20H26ClNS
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:347.95
  • RS 52367

    CAS:
    <p>RS 52367 is a beta-adrenergic antagonist.</p>
    Fórmula:C18H34ClN3O3S
    Cor e Forma:Solid
    Peso molecular:408
  • S 12024-2

    CAS:
    <p>S 12024-2 (Dabelotine mesylate) is a new cognitive drug-enhancer.</p>
    Fórmula:C16H26N2O5S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:358.45
  • Flerobuterol

    CAS:
    <p>Flerobuterol is a potential antidepressant agent related to beta-adrenergic agonists.</p>
    Fórmula:C12H18FNO
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:211.28
  • Befunolol HCl

    CAS:
    <p>Befunolol is a beta blocker with intrinsic sympathomimetic activity and also acts as a β adrenoreceptor partial agonist.</p>
    Fórmula:C16H22ClNO4
    Cor e Forma:Solid
    Peso molecular:327.8
  • Flutonidine

    CAS:
    <p>Flutonidine is an agonist of alpha2-Adrenergic receptor.</p>
    Fórmula:C10H12FN3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:193.22
  • S-Nitroso-N-acetylcysteine

    CAS:
    <p>S-Nitroso-N-acetylcysteine inhibits proliferation and survival of multiple MM cells. It acts by the S-nitrosylation-dependent inhibition of STAT3 and NF-κB.</p>
    Fórmula:C5H8N2O4S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:192.19
  • Bremazocine

    CAS:
    <p>Bremazocineis a potent opiate kappa-agonist and centrally acting analgesic.</p>
    Fórmula:C20H29NO2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:315.45
  • RS 15385-197

    CAS:
    <p>RS 15385-197 is a selective alpha 2-adrenoceptor antagonist.</p>
    Fórmula:C18H26N2O3S
    Cor e Forma:Solid
    Peso molecular:350.48
  • Garomefrine HCl

    CAS:
    <p>Garomefrine HCl, a α1A-adrenoceptor agonist, is potential for the treatment of urinary incontinence.</p>
    Fórmula:C9H14ClFN2O3S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:284.73
  • Cafaminol

    CAS:
    <p>Cafaminol (methylcoffanolamine) is a vasoconstrictor and anticatarrhal of the methylxanthine family related to caffeine which is used as a nasal decongestant.</p>
    Fórmula:C11H17N5O3
    Cor e Forma:Solid
    Peso molecular:267.28
  • R 47243

    CAS:
    <p>R 47243 is used as a racemic alpha 2 antagonist.</p>
    Fórmula:C22H25N3O2S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:395.52
  • Burimamide

    CAS:
    <p>Burimamide is an antagonist of histamine. It appears to block both H2 and H3 histamine receptors.</p>
    Fórmula:C9H16N4S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:212.32
  • BE 2254

    CAS:
    <p>BE 2254 is an antagonist of central noradrenergic receptor.</p>
    Fórmula:C19H21NO2
    Cor e Forma:Solid
    Peso molecular:295.38
  • Dabuzalgron HCl

    CAS:
    <p>Dabuzalgron, an adrenoceptor agonist, is used potentially for the treatment of urinary incontinence.</p>
    Fórmula:C12H17Cl2N3O3S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:354.25
  • Butidrine

    CAS:
    <p>Butidrine has an Antiarrhythmic activities.</p>
    Fórmula:C16H25NO
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:247.38
  • Dipiproverine hydrochloride

    CAS:
    <p>Dipiproverine hydrochloride is an antispasmodic alpha-amino acid ester used as an anticholinergic.</p>
    Fórmula:C20H32Cl2N2O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:403.39
  • JTH-601 free base

    CAS:
    <p>JTH-601 free base is an antagonist of alpha 1 adrenergic receptor.</p>
    Fórmula:C24H35NO4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:401.54
  • JNJ-7925476 HCl

    CAS:
    <p>JNJ-7925476 HCl inhibits DAT, NET, SERT; ED(50): DAT 2.4, NET 0.09, SERT 0.18 mg/kg in rats.</p>
    Fórmula:C20H20ClN
    Cor e Forma:Solid
    Peso molecular:309.83
  • L-748328

    CAS:
    <p>L-748328 is a potent and selective antagonist of human beta(3)-adrenergic receptor.</p>
    Fórmula:C23H27N3O6S2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:505.61
  • SKF 86466 hydrochloride

    CAS:
    <p>SKF 86466 hydrochloride is an α2-adrenoceptor antagonist.</p>
    Fórmula:C11H15Cl2N
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:232.15
  • KUL-7211

    CAS:
    <p>KUL-7211 is an β2 and β3 adrenergic receptor agonist. KUL-7211 is a potent ureteral relaxant with a relatively small hypotensive effect.</p>
    Fórmula:C19H23NO5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:345.39
  • Esprolol hydrochloride

    CAS:
    <p>Esprolol is a β-adrenergic receptor antagonist.</p>
    Fórmula:C17H28ClNO4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:345.86
  • Dipiproverine

    CAS:
    <p>Dipiproverine is an alpha-amino acid ester, an antispasmodic compound. It is used as an anticholinergic drug.</p>
    Fórmula:C20H30N2O2
    Cor e Forma:Solid
    Peso molecular:330.46
  • Dihydroalprenolol, (S)-

    CAS:
    <p>Dihydroalprenolol, (S)- is a hydrogenated alprenolol derivative. It acts as a beta-adrenergic blocker.</p>
    Fórmula:C15H25NO2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:251.36
  • Levomoprolol

    CAS:
    <p>Levomoprolol, (S)-enantiomer of the moprololis, is a beta adrenergic antagonist.</p>
    Fórmula:C13H21NO3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:239.31
  • L-771688 dihydrochloride

    CAS:
    <p>L-771688 is an α1A-adrenoceptor antagonist potentially for the treatment of benign prostatic hyperplasia.</p>
    Fórmula:C28H35Cl2F2N5O5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:630.51
  • Levoprotiline

    CAS:
    <p>Levoprotiline, a fast-acting antidepressant, is the R-enantiomer of Oxaprotiline and successor to maprotiline.</p>
    Fórmula:C20H23NO
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:293.4
  • SNAP 5089

    CAS:
    <p>α1A-adrenoceptor antagonist</p>
    Fórmula:C36H40N4O5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:608.73
  • Dilevalol

    CAS:
    <p>Dilevalol, an RR-stereoisomer of labetalol, is a beta-blocker with partial beta 2-agonism and minimal alpha 1-blockade.</p>
    Fórmula:C19H24N2O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:328.41
  • Delequamine HCl

    CAS:
    <p>Delequamine HCl: potent, selective alpha 2-adrenoceptor blocker; pKi 9.45 in rat cortex, pA2 9.72 in guinea-pig ileum.</p>
    Fórmula:C18H27ClN2O3S
    Cor e Forma:Solid
    Peso molecular:386.94
  • Oxaprotiline

    CAS:
    <p>Oxaprotiline: an antidepressant, norepinephrine inhibitor, and H1 blocker; studied in hospital depression but not marketed.</p>
    Fórmula:C20H23NO
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:293.4
  • Zometapine

    CAS:
    <p>Zometapine (CI 716) is an antidepressant compound that is a derivative of pyrazole and diazepine.</p>
    Fórmula:C14H15ClN4
    Pureza:98.87%
    Cor e Forma:Solid
    Peso molecular:274.75
  • Levoprotiline hydrochloride

    CAS:
    <p>Levoprotiline hydrochloride is an antidepressant.</p>
    Fórmula:C20H24ClNO
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:329.86
  • FMS586

    CAS:
    <p>FMS586 is a selective antagonist of neuropeptide Y Y5 receptor with oral activity.</p>
    Fórmula:C24H30N4O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:390.52
  • Tilisolol HCl

    CAS:
    <p>Tilisolol, a nonselective beta-blocker, dilates dog coronary arteries via ATP-sensitive K(+) channels.</p>
    Fórmula:C17H25ClN2O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:340.85
  • (S)-Viloxazine Hydrochloride

    CAS:
    <p>(S)-Viloxazine Hydrochloride is an S-isomer and NRI used as an antidepressant.</p>
    Fórmula:C13H20ClNO3
    Pureza:99.95%
    Cor e Forma:Solid
    Peso molecular:273.76
  • Tranterol hydrochloride

    CAS:
    <p>Tranterol, a β2-adrenergic receptor agonist, is used potentially for the treatment of asthma.</p>
    Fórmula:C13H19Cl2F3N2O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:347.2
  • Pamatolol

    CAS:
    <p>Pamatolol is a selective and potent beta-adrenoceptor antagonist that has not shown sympathomimetic activity in ex vivo experiments.</p>
    Fórmula:C16H26N2O4
    Pureza:>99.99%
    Cor e Forma:Solid
    Peso molecular:310.39
  • Cicloprolol hydrochloride

    CAS:
    <p>Cicloprolol hydrochloride is a new potent and selective beta 1-adrenoceptor antagonist with partial agonist activity for the study of coronary heart disease.</p>
    Fórmula:C18H30ClNO4
    Pureza:97.26%
    Cor e Forma:Solid
    Peso molecular:359.89
  • L-771688

    CAS:
    <p>L-771688 (SNAP 6383) is a novel potent and selective α1A-adrenoceptor antagonist with a Ki value of 0.43±0.02 nM.L-771688 KE is used for the treatment of benign</p>
    Fórmula:C28H33F2N5O5
    Pureza:94.15%
    Cor e Forma:Solid
    Peso molecular:557.59
  • Indanidine

    CAS:
    <p>Indanidine is a highly selective and potent α-adrenergic agonist with antihypertensive activity.Indanidine is an α-adrenergic antagonist that can be used in the</p>
    Fórmula:C11H13N5
    Pureza:>99.99%
    Cor e Forma:Solid
    Peso molecular:215.25
  • TD-5471 hydrochloride

    CAS:
    <p>TD-5471 hydrochloride is a selective and potent long-acting human β2-adrenergic receptor agonist for the treatment of chronic obstructive pulmonary disease (</p>
    Fórmula:C32H32ClN3O4
    Pureza:99.57%
    Cor e Forma:Solid
    Peso molecular:558.07
  • Napitane

    CAS:
    <p>napitane (A 75200) is a novel catecholamine uptake inhibitor with inhibitory effects on α-adrenergic receptors and potential antidepressant activity for the</p>
    Fórmula:C22H25NO2
    Pureza:99.77% - 99.89%
    Cor e Forma:Solid
    Peso molecular:335.44
  • Norfenefrine HCl

    CAS:
    <p>Norfenefrine HCl is an α1-adrenergic receptor agonist, an endogenous neurotransmitter and sympathomimetic drug for hypotension,glycerol adipose.</p>
    Fórmula:C8H12ClNO2
    Pureza:99.44%
    Cor e Forma:Solid
    Peso molecular:189.64
  • KUL-7211 racemate

    CAS:
    <p>KUL 7211, a selective β-adrenoceptor agonist, exists as a racemate, referred to as KUL 7211 racemate, which is the mixture of its enantiomers.</p>
    Fórmula:C19H23NO5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:345.39
  • Ro 363

    CAS:
    <p>RO 363: Potent β1-adrenoceptor agonist, boosts heart contractility, lowers diastolic pressure.</p>
    Fórmula:C19H25NO6
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:363.4
  • Labetalone hydrochloride

    CAS:
    <p>Labetalone hydrochloride, a Labetalol impurity, is an orally active alpha and beta-adrenoceptor blocker.</p>
    Fórmula:C19H23ClN2O3
    Pureza:99.58%
    Cor e Forma:Solid
    Peso molecular:362.85
  • Naphazoline

    CAS:
    <p>Naphazoline (Naphcon-a) is a sympathomimetic compound with marked alpha adrenergic activity.</p>
    Fórmula:C14H14N2
    Pureza:99.79%
    Cor e Forma:White Crystalline Powder Solid
    Peso molecular:210.27
  • Moprolol

    CAS:
    <p>Moprolol ((±)-Moprolol) is a beta-adrenergic receptor antagonist utilized in research pertaining to essential hypertension [1] [2] [3].</p>
    Fórmula:C13H21NO3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:239.31
  • N-Methyldopamine hydrochloride

    CAS:
    <p>N-Methyldopamine hydrochloride (Ephinine hydrochloride) is an α and β agonist, with indirect sympathomimetic effects similar to dopamine.</p>
    Fórmula:C9H14ClNO2
    Cor e Forma:Solid
    Peso molecular:203.67
  • Ancarolol

    CAS:
    <p>Ancarolol is a blocking agent of beta-adrenergic.</p>
    Fórmula:C18H24N2O4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:332.39
  • Rec 15/2615 dihydrochloride

    CAS:
    <p>Rec 15/2615 dihydrochloride is an antagonist of α1B-adrenergic receptor.</p>
    Fórmula:C26H35Cl2N5O5
    Pureza:97.04% - 99.76%
    Cor e Forma:Solid
    Peso molecular:568.49
  • Arbutamine

    CAS:
    <p>Arbutamine (GP 21213) is a β-adrenoceptor agonist with alpha-1-sympathomimetic activity that can be used to study cardiac stress.</p>
    Fórmula:C18H23NO4
    Pureza:95.06%
    Cor e Forma:Solid
    Peso molecular:317.38
  • (S)-(-)-Propranolol hydrochloride

    CAS:
    <p>(S)-(-)-Propranolol hydrochloride 是一种有效的肾上腺素能受体 (β-adrenergic receptor) 拮抗剂,具有抗高血压活性和潜在的抗癌活性,对β1,β2,和β3受体有抑制作用。(S)-(-)-Propranolol hydrochloride 可改善严重烧伤患者的预后,可用于研究酒精症。</p>
    Fórmula:C16H22ClNO2
    Pureza:99.02% - 99.91%
    Cor e Forma:Solid
    Peso molecular:295.8
  • (S)-Terazosin

    CAS:
    <p>(S)-Terazosin is an active S-enantiomer of Terazosin.</p>
    Fórmula:C19H25N5O4
    Cor e Forma:Solid
    Peso molecular:387.43
  • T-0509

    CAS:
    <p>T-0509 is a selective beta 1 receptor agonist that increases inotropy in canine ventricular muscle and selectively down-regulates rat cardiac beta 1-</p>
    Fórmula:C18H23NO5
    Pureza:97.52% - 98.43%
    Cor e Forma:Solid
    Peso molecular:333.38
  • Cyclazosin HCl

    CAS:
    <p>Cyclazosin HCl is an α-adrenergic receptor antagonist that can be used to study non-arteritic ischemic optic neuropathy.</p>
    Fórmula:C23H28ClN5O4
    Pureza:99.10%
    Cor e Forma:Solid
    Peso molecular:473.95
  • Levobunolol hydrochloride

    CAS:
    <p>Levobunolol hydrochloride 是一种非选择性的 β-肾上腺素受体阻滞剂,可用于治疗青光眼和上斜肌肌障碍的研究。</p>
    Fórmula:C17H26ClNO3
    Pureza:98.49% - >99.99%
    Cor e Forma:Solid
    Peso molecular:327.85
  • L748337

    CAS:
    <p>L748337 is a β3-adrenoceptor antagonist that inhibits β3-, β2-, and β1-adrenoceptors and inhibits the protective effects of CL316243.</p>
    Fórmula:C26H31N3O5S
    Pureza:99.67% - >99.99%
    Cor e Forma:Solid
    Peso molecular:497.61
  • ADRA1D receptor antagonist 1 HCl

    CAS:
    <p>ADRA1D receptor antagonist 1 HCl is a selective α1D adrenergic receptor antagonist (Ki: 1.6 nM) with potential antiproliferative activity.</p>
    Fórmula:C15H14Cl2N4O
    Pureza:98.13%
    Cor e Forma:Solid
    Peso molecular:337.2
  • Romifidine

    CAS:
    <p>Romifidine is used as a sedative in veterinary medicine mainly in large animals such as horses. It acts as an agonist at the α2 adrenergic receptor subtype.</p>
    Fórmula:C9H9BrFN3
    Cor e Forma:Solid
    Peso molecular:258.09
  • LY377604

    CAS:
    <p>LY377604 is a human β3-adrenergic receptor agonist (EC50: 2.4 nM) and β1/2-adrenergic receptor antagonist for the study of obesity.</p>
    Fórmula:C31H32N4O4
    Pureza:99.72% - >99.99%
    Cor e Forma:Solid
    Peso molecular:524.61
  • SM-2470

    CAS:
    <p>SM-2470 is an α1-adrenoceptor antagonist with antihypertensive activity and hypocholesterolemic activity that inhibits cholesterol absorption.</p>
    Fórmula:C23H30ClN5O3
    Pureza:98.91%
    Cor e Forma:Solid
    Peso molecular:459.97
  • Falintolol

    CAS:
    <p>Falintolol is a novel beta-adrenergic antagonist with antihypertensive effects and can be used to study glaucoma.</p>
    Fórmula:C12H24N2O2
    Pureza:>99.99% - >99.99%
    Cor e Forma:Solid
    Peso molecular:228.33
  • Bedoradrine sulfate

    CAS:
    <p>Bedoradrine sulfate (MN-221 sulfate) is a novel, highly selective β2-adrenoceptor agonist.Cost-effective and quality-assured.</p>
    Fórmula:C24H32N2O5H2O4S
    Pureza:99.31%
    Cor e Forma:Solid
    Peso molecular:477.56
  • GP2-114

    CAS:
    <p>GP2-114 is a catecholamine motility mimetic that produces current-dependent cardiovascular effects.Cost-effective and quality-assured.</p>
    Fórmula:C19H24N2O4
    Pureza:99.32%
    Cor e Forma:Solid
    Peso molecular:344.4
  • Egis-11150

    CAS:
    <p>Egis-11150 is a potent inhibitor of adrenergic alpha1, alpha2c, 5-HT2a, 5HT7 receptors.</p>
    Fórmula:C19H21ClFN5O2
    Pureza:97.49% - >99.99%
    Cor e Forma:Solid
    Peso molecular:405.85
  • Amosulalol

    CAS:
    <p>Amosulalol is a combined alpha and beta adrenoceptor antagonist.</p>
    Fórmula:C18H24N2O5S
    Pureza:99.5%
    Cor e Forma:Solid
    Peso molecular:380.46
  • CL 316243

    CAS:
    <p>CL316243 is a highly potent selective agonist of β3-adrenoceptor.Cost-effective and quality-assured.</p>
    Fórmula:C20H18ClNNa2O7
    Pureza:98.00% - 99.68%
    Cor e Forma:Solid
    Peso molecular:465.79
  • Midaglizole hydrochloride

    CAS:
    <p>Midaglizole hydrochloride (DG5128) is an α2-adrenoceptor antagonist with 7.4x more affinity than α1-adrenoceptors (pKi=6.28).</p>
    Fórmula:C16H19Cl2N3
    Pureza:99.39% - 99.82%
    Cor e Forma:Solid
    Peso molecular:324.25
  • Soquinolol

    CAS:
    <p>Soquinolol (Soquinolol mucate) is a beta-adrenergic receptor antagonist with weak local anesthetic activity.Soquinolol has good enteral efficacy and a long</p>
    Fórmula:C17H26N2O3
    Pureza:97.48% - 98.63%
    Cor e Forma:Solid
    Peso molecular:306.4
  • Neldazosin

    CAS:
    <p>Neldazosin is used as a potent α1-adrenoceptor antagonist.</p>
    Fórmula:C18H25N5O4
    Pureza:99.74% - 99.76%
    Cor e Forma:Solid
    Peso molecular:375.42
  • Oxyfedrine L-form HCl

    CAS:
    <p>Oxyfedrine L-form HCl (Ildamen) is a partial agonist at beta-adrenergic receptors and acts as a coronary vasodilator and cardiotonic agent.</p>
    Fórmula:C19H24ClNO3
    Pureza:99.5% - 99.57%
    Cor e Forma:Solid
    Peso molecular:349.85
  • JP1302

    CAS:
    <p>JP1302: α2C adrenoceptor antagonist, Kb 16 nM, Ki 28 nM, antidepressant, FACT disruptor, studies: neuropsychiatric, renal issues.</p>
    Fórmula:C24H24N4
    Pureza:99.96%
    Cor e Forma:Solid
    Peso molecular:368.47
  • Ecastolol

    CAS:
    <p>Ecastolol has anti-angina activity and is an adrenergic receptor antagonist.</p>
    Fórmula:C26H33N3O6
    Pureza:99.89%
    Cor e Forma:Solid
    Peso molecular:483.56
  • Nemazoline Free Base

    CAS:
    <p>Nemazoline Free Base: a long-lasting nasal decongestant, better than oxymetazoline, with no systemic effects or toxicity in dogs and rats.</p>
    Fórmula:C10H11Cl2N3
    Pureza:98.06% - 98.83%
    Cor e Forma:Solid
    Peso molecular:244.12
  • Butofilolol

    CAS:
    <p>Butofilolol is a novel beta-blocker with antihypertensive activity and can be used to study hypertension.</p>
    Fórmula:C17H26FNO3
    Pureza:98.96% - >99.99%
    Cor e Forma:Solid
    Peso molecular:311.392
  • Rafabegron

    CAS:
    <p>Rafabegron (TAK677) is a potent and selective β3 adrenergic receptor agonist for the study of diabetes and obesity.</p>
    Fórmula:C21H23ClN2O4
    Pureza:99.21%
    Cor e Forma:Solid
    Peso molecular:402.87
  • Pipoxazole

    CAS:
    <p>Pipoxazole, an adrenergic receptor antagonist, is used potentially for the treatment of depression.</p>
    Fórmula:C14H20N4O
    Pureza:98.58% - 99.53%
    Cor e Forma:Solid
    Peso molecular:260.33
  • Taprizosin

    CAS:
    <p>Taprizosin(UK-338003) is a selective and orally active α1-adrenoceptor antagonist for vasodilatation in the treatment of benign prostatic hyperplasia.</p>
    Fórmula:C25H26N6O4S
    Pureza:96.34% - 99.11%
    Cor e Forma:Solid
    Peso molecular:506.58
  • Milveterol HCl

    CAS:
    <p>Milveterol HCl is a long-acting β(2) -adrenergic receptor agonist for the potential treatment of chronic obstructive pulmonary disease (COPD).</p>
    Fórmula:C25H30ClN3O4
    Pureza:98.2%
    Cor e Forma:Solid
    Peso molecular:471.98
  • (S)-(+)-Niguldipine hydrochloride

    CAS:
    <p>(S)-(+)-Niguldipine hydrochloride is a selective α1A-AR antagonist used in the study of depression and epilepsy.</p>
    Fórmula:C36H40ClN3O6
    Pureza:98.27%
    Cor e Forma:Solid
    Peso molecular:646.17
  • Dabelotine

    CAS:
    <p>Dabelotine (UNII-6RY56RB98P) is an adrenergic agonist used in the study of dementia.</p>
    Fórmula:C15H22N2O2
    Pureza:98.55%
    Cor e Forma:Solid
    Peso molecular:262.35
  • Besipirdine

    CAS:
    <p>Besipirdine (HP 749 free base) is a non-receptor-dependent cholinomimetic compound with alpha-adrenergic activity and cardiovascular activity.</p>
    Fórmula:C16H17N3
    Pureza:97.15% - 98.85%
    Cor e Forma:Solid
    Peso molecular:251.33
  • Palatrigine

    CAS:
    <p>Palatrigine (BW-A 256C) is a compound with angiotensin-converting enzyme inhibitory and beta-adrenergic receptor blocking properties.</p>
    Fórmula:C12H13Cl2N5
    Pureza:98.87%
    Cor e Forma:Solid
    Peso molecular:298.17
  • Bisaramil hydrochloride

    CAS:
    <p>Bisaramil hydrochloride (Bisaramil) is an antiarrhythmic compound that inhibits free radical production.</p>
    Fórmula:C17H24Cl2N2O2
    Pureza:98.64% - 99.48%
    Cor e Forma:Solid
    Peso molecular:359.29
  • Imiloxan

    CAS:
    <p>Imiloxan (RS-21361) is an α2 adrenergic receptor antagonist used in the treatment of major depressive disorder.</p>
    Fórmula:C14H16N2O2
    Pureza:98.13% - 99.8%
    Cor e Forma:Solid
    Peso molecular:244.29
  • ST 91

    CAS:
    <p>ST-91 is an agonist of α2-adrenoceptor with a mixed α-adrenergic receptor type/subtype selection profile.</p>
    Fórmula:C13H20ClN3
    Pureza:99.83%
    Cor e Forma:Solid
    Peso molecular:253.77
  • ORM-10921

    CAS:
    <p>ORM-10921 is an α2C-adrenoceptor antagonist that has shown antipsychotic and antidepressant activity in animal studies.</p>
    Fórmula:C18H23NO2
    Pureza:99.46% - 99.85%
    Cor e Forma:Solid
    Peso molecular:285.38
  • Fipamezole

    CAS:
    <p>Fipamezole is a potent alpha2 adrenergic receptor antagonist that may be useful for studying autonomic dysfunction in Parkinson's disease.</p>
    Fórmula:C14H15FN2
    Pureza:99.32% - >99.99%
    Cor e Forma:Solid
    Peso molecular:230.28
  • Xamoterol hemifumarate

    CAS:
    <p>Xamoterol hemifumarate is a potent and selective β1-adrenoceptor agonist.Xamoterol hemifumarate is a potential compound for the study of the relationship</p>
    Fórmula:C36H54N6O14
    Pureza:99.79%
    Cor e Forma:White Solid
    Peso molecular:794.37
  • Rezatomidine

    CAS:
    <p>Rezatomidine (AGN203818) is a selective antagonist of α2-adrenergic receptor and can be used in studies about chronic pain, including neuropathic pain.</p>
    Fórmula:C13H16N2S
    Pureza:98.34%
    Cor e Forma:Solid
    Peso molecular:232.34
  • Bedoradrine

    CAS:
    <p>Bedoradrine (MN-221) free base is a novel, highly selective β2-adrenoceptor agonist.Cost-effective and quality-assured.</p>
    Fórmula:C24H32N2O5
    Pureza:>99.99%
    Cor e Forma:Solid
    Peso molecular:428.52
  • Vatinoxan hydrochloride

    CAS:
    <p>Vatinoxan hydrochloride is an antagonist of the peripheral α2 adrenergic receptors.</p>
    Fórmula:C20H27ClN4O4S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:454.97
  • Nolomirole HCl

    CAS:
    <p>Nolomirole HCl (CHF 1035) is a novel selective dopamine agonist with oral activity and inhibitory effects on norepinephrine release, which can be used to study</p>
    Fórmula:C19H28ClNO4
    Pureza:99.03% - >99.99%
    Cor e Forma:Solid
    Peso molecular:369.88
  • Abediterol

    CAS:
    <p>Abediterol (LAS100977): potent, long-acting beta-2 agonist for asthma and COPD treatment.</p>
    Fórmula:C25H30F2N2O4
    Cor e Forma:Solid
    Peso molecular:460.51
  • N-5984

    CAS:
    <p>N-5984, a β3-adrenergic receptor agonist, is used potentially for the treatment of obesity, overactive bladder and type 2 diabetes.</p>
    Fórmula:C20H22ClNO5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:391.85
  • 4-hydroxy Nebivolol hydrochloride

    CAS:
    <p>4-Hydroxy Nebivolol, a primary metabolite of Nebivolol, results from the enzymatic hydroxylation of Nebivolol by the cytochrome P450 (CYP) isoform CYP2D6.</p>
    Fórmula:C22H25F2NO5HCl
    Cor e Forma:Solid
    Peso molecular:457.9
  • (-)-Isoproterenol hydrochloride

    CAS:
    <p>(-)-Isoproterenol hydrochloride is used as a β-adrenergic receptor agonist in the treatment of bradycardia and as a bronchodilator.</p>
    Fórmula:C11H17NO3·CIH
    Cor e Forma:Solid
    Peso molecular:247.72
  • BI-167107

    CAS:
    <p>BI-167107 is a high affinity, full agonist that binds to the β2 adrenergic receptor (β2AR, Kd of 84 pM).</p>
    Fórmula:C21H26N2O4
    Cor e Forma:Solid
    Peso molecular:370.44
  • AGN 192836

    CAS:
    <p>AGN 192836 is a potent and selective α2 adrenergic agonist (EC50s: 8.7, 41 and 6.6 nM for α2A, α2B and α2C receptor).</p>
    Fórmula:C12H13N3O2
    Cor e Forma:Solid
    Peso molecular:231.25
  • β3-AR agonist 2

    CAS:
    <p>β3-AR agonist 2 is a potent and selective agonist of β3-adrenergic receptor (β3-AR with an EC50 of 8 nM).</p>
    Fórmula:C27H38N4O7S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:562.68
  • Mefenidil

    CAS:
    <p>Mefenidil (McN-2378), a selective cerebral vasodilator, was shown to increase CBF in healthy brains without stimulating O2 uptake in a dog anesthesia model.</p>
    Fórmula:C12H11N3
    Pureza:98.27%
    Cor e Forma:Solid
    Peso molecular:197.24
  • (±)-N-Methylcoclaurine

    CAS:
    <p>N-Methylcoclaurine (±) acts as a selective antagonist at the α2-adrenoceptor [1].</p>
    Fórmula:C18H21NO3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:299.36
  • Todralazine hydrochloride

    CAS:
    <p>Todralazine hydrochloride, a β2AR blocker with antioxidant properties, is used in hypertension studies.</p>
    Fórmula:C11H13ClN4O2
    Pureza:99.91%
    Cor e Forma:Solid
    Peso molecular:268.7
  • BMS-194449

    CAS:
    <p>BMS-194449 is a full beta 3 agonist.</p>
    Fórmula:C24H24F4N2O6S
    Cor e Forma:Solid
    Peso molecular:544.52
  • Celiprolol hydrochloride

    CAS:
    <p>Celiprolol hydrochloride (Selectrol) is a cardioselective beta-1 adrenergic antagonist that has intrinsic sympathomimetic activity.</p>
    Fórmula:C20H33N3O4·HCl
    Cor e Forma:White Crystalline Solid
    Peso molecular:415.96
  • Bunazosin Hydrochloride

    CAS:
    <p>Bunazosin Hydrochloride (E 1015) is an alpha(1)-adrenoceptor antagonist used as a systemic antihypertensive and an ocular hypotensive drug.</p>
    Fórmula:C19H28ClN5O3
    Pureza:99.12%
    Cor e Forma:Solid
    Peso molecular:409.91
  • BU-E 75

    CAS:
    <p>BU-E 75 is an agonist of the histamine H2.</p>
    Fórmula:C21H24F2N6
    Cor e Forma:Solid
    Peso molecular:398.45
  • β3-AR agonist 1

    CAS:
    <p>β3-AR agonist 1 is a highly selective, and orally available agonist of β3-adrenergic receptor (EC50: 18 nM), being inactive to β1-, β2-, and α1A-AR (β1/β3, β2/</p>
    Fórmula:C22H28N4O4S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:444.55
  • L-796568 free base

    CAS:
    <p>L-796568 is a potent β3 agonist for obesity with 600x selectivity over β1/β2 receptors (EC50: 3.6 nM).</p>
    Fórmula:C31H27F3N4O3S2
    Cor e Forma:Solid
    Peso molecular:624.7
  • RS100329 hydrochloride

    CAS:
    <p>RS 100329 hydrochloride is an antagonist of α1A-adrenergic receptor.</p>
    Fórmula:C20H26ClF3N4O3
    Pureza:99.95%
    Cor e Forma:Solid
    Peso molecular:462.89
  • Bufuralol (hydrochloride)

    CAS:
    <p>Bufuralol hydrochloride is a potent, non-selective, orally active β-blocker with partial agonist effects and a CYP2D6 probe.</p>
    Fórmula:C16H24ClNO2
    Cor e Forma:Solid
    Peso molecular:297.82
  • LK 204-545

    CAS:
    <p>LK 204-545 is a highly selective antagonist of beta1-adrenoceptor.</p>
    Fórmula:C25H32N4O6
    Cor e Forma:Solid
    Peso molecular:484.54
  • NGD9002

    CAS:
    <p>NGD9002 is a novel generation, topology 2 selective corticotropin releasing factor-1 (CRF-1) receptor antagonist agent.</p>
    Fórmula:C20H31N5O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:357.49
  • L-796568 dihydrochloride

    CAS:
    <p>L-796568: potent β3 agonist (EC50 = 3.6 nM), &gt;600-fold selectivity vs β1/β2, good oral bioavailability, long action.</p>
    Fórmula:C31H29Cl2F3N4O3S2
    Cor e Forma:Solid
    Peso molecular:697.62
  • RS 17053 hydrochloride

    CAS:
    <p>RS 17053 hydrochloride: selective α1A adrenoceptor antagonist, pKi 9.1, pA2 9.8.</p>
    Fórmula:C24H30Cl2N2O2
    Pureza:99.27%
    Cor e Forma:Solid
    Peso molecular:449.41
  • Ritodrine

    CAS:
    <p>Ritodrine (DU21220) is a β-adrenergic agonist as well as an effective uterine relaxant that can be used in arrest premature labor research[1] [2].</p>
    Fórmula:C17H21NO3
    Cor e Forma:Solid
    Peso molecular:287.35
  • Binedaline

    CAS:
    <p>Binedaline is a selective norepinephrine reuptake inhibitor with Ki value of 25 nM.</p>
    Fórmula:C19H23N3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:293.41
  • Epinephrine HCl

    CAS:
    <p>Epinephrine HCl is a hormone and neurotransmitter secreted by the adrenal medulla, agonist of α-adrenergic and β-adrenergic receptor.</p>
    Fórmula:C9H14ClNO3
    Pureza:99.48%
    Cor e Forma:Solid
    Peso molecular:219.67
  • Dibenamine hydrochloride

    CAS:
    <p>Dibenamine hydrochloride is a competitive and irreversible blocking agent of the β-adrenergic receptor.</p>
    Fórmula:C16H19Cl2N
    Pureza:96.43%
    Cor e Forma:Oily Liquid Solid
    Peso molecular:296.23
  • AR-08

    CAS:
    <p>AR-08 is a potent α2-adrenergic receptor agonist for the study of ADHD and attention deficit.</p>
    Fórmula:C12H12N6
    Pureza:99.7%
    Cor e Forma:Solid
    Peso molecular:240.26
  • Fiduxosin

    CAS:
    <p>Fiduxosin is a selective and potent α1-adrenoceptor antagonist with inhibitory effects on α1a-adrenoceptor, α1b-adrenoceptor and α1d-adrenoceptor, with Ki</p>
    Fórmula:C30H29N5O4S
    Pureza:99.73%
    Cor e Forma:Solid
    Peso molecular:555.65