
Receptor adrenérgico
Os receptores adrenérgicos são GPCRs que são ativados por catecolaminas, como adrenalina e noradrenalina. Esses receptores são classificados em subtipos alfa e beta, cada um dos quais desempenha um papel fundamental na regulação da frequência cardíaca, pressão arterial e resposta de luta ou fuga. Moduladores de receptores adrenérgicos são essenciais no tratamento de doenças cardiovasculares, asma e distúrbios de ansiedade. Na CymitQuimica, oferecemos uma ampla gama de moduladores de receptores adrenérgicos de alta qualidade para apoiar sua pesquisa em endocrinologia, farmacologia cardiovascular e resposta ao estresse.
Subcategorias de "Receptor adrenérgico"
Foram encontrados 645 produtos de "Receptor adrenérgico"
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Amidephrine hydrochloride
CAS:<p>Amidephrine hydrochloride is a biochemical.</p>Fórmula:C10H17ClN2O3SCor e Forma:SolidPeso molecular:280.77Amidephrine
CAS:<p>Amidephrine is an adrenergic agent.</p>Fórmula:C10H16N2O3SCor e Forma:SolidPeso molecular:244.31LY 344864
CAS:<p>LY 344864, a specifc receptor agonist, is an affinity of 6 nM (Ki) at the recently cloned 5-HT1F receptor.</p>Fórmula:C21H22FN3OPureza:98%Cor e Forma:SolidPeso molecular:351.42BW-A 575C
CAS:<p>BW-A 575C is an inhibitor of ACE.</p>Fórmula:C29H43N5O8Pureza:98%Cor e Forma:SolidPeso molecular:589.68Bambuterol
CAS:<p>long acting beta-adrenoceptor agonist</p>Fórmula:C18H29N3O5Pureza:98%Cor e Forma:Off-White PowderPeso molecular:367.44Landiolol
CAS:<p>Landiolol is used as a highly cardioselective ultra short-acting beta-blocker.</p>Fórmula:C25H39N3O8Pureza:98%Cor e Forma:White Crystalline PowderPeso molecular:509.59D2343
CAS:<p>D2343 is an agonist of β2-adrenoceptor. It also is an inhibitor of α1- adrenoceptor.</p>Fórmula:C20H27NO3Pureza:98%Cor e Forma:SolidPeso molecular:329.43Salmefamol
CAS:<p>Salmefamol is a beta-adrenergic agonist. It may also be used as a bronchodilator.</p>Fórmula:C19H25NO4Pureza:99.89%Cor e Forma:SolidPeso molecular:331.41Efaroxan hydrochloride
CAS:<p>Efaroxan hydrochloride a selective, oral α2-adrenoceptor antagonist significantly potentiates adrenaline-induced increases in insulin levels.</p>Fórmula:C13H17ClN2OPureza:98%Cor e Forma:SolidPeso molecular:252.74Protokylol hydrochloride
CAS:<p>Protokylol hydrochloride is a β-adrenergic agonist and bronchodilator, marketed as Asmetil, Caytine, Palison, Ventaire.</p>Fórmula:C18H22ClNO5Cor e Forma:SolidPeso molecular:367.83Clonidine
CAS:<p>Clonidine (Kapvay): central alpha-adrenergic agonist, antihypertensive, often combined, not tied to liver issues.</p>Fórmula:C9H9Cl2N3Pureza:99.42% - 99.44%Cor e Forma:Crystals SolidPeso molecular:230.09BRL 44408 Maleate Salt
CAS:<p>BRL 44408 Maleate is an α2A-adrenoceptor antagonist with antidepressant and analgesic activity.</p>Fórmula:C17H21N3O4Pureza:98.71%Cor e Forma:SolidPeso molecular:331.37Butaxamine
CAS:<p>Butaxamine is a beta-2 selective adrenergic antagonist used mostly in animal and tissue experiments to characterize BETA-2 adrenergic receptors.</p>Fórmula:C15H25NO3Pureza:98%Cor e Forma:SolidPeso molecular:267.36Lusaperidone
CAS:<p>Kaerophyllin ( (-)-Kaerophylin) inhibits hepatic stellate cell activation and inhibits HSC activation to protect against liver cell damage and fibrosis in rats.</p>Fórmula:C22H21N3O2Pureza:99.75%Cor e Forma:SolidPeso molecular:359.42IMTPPE
CAS:<p>IMTPPE inhibits transcriptional activity and protein level of AR in C4-2 prostate cancer cells. It also inhibits AR-target gene expression.</p>Fórmula:C20H27N3O2SCor e Forma:SolidPeso molecular:373.51Abanoquil
CAS:<p>Abanoquil is an antagonist of alpha-1 adrenoceptor.</p>Fórmula:C22H25N3O4Cor e Forma:SolidPeso molecular:395.45Zinterol
CAS:<p>Zinterol is a potent and selective agonist of β2-adrenoceptor. Zinterol increases ICa in a concentration-dependent manner(EC50 of 2.2 nM).</p>Fórmula:C19H26N2O4SPureza:98%Cor e Forma:SolidPeso molecular:378.49Metoprolol fumarate
CAS:<p>Metoprolol fumarate (CGP 2175C): selective β1-blocker with anti-inflammatory, antitumor, anti-angiogenic effects.</p>Fórmula:C34H54N2O10Cor e Forma:SolidPeso molecular:650.8Clenproperol
CAS:<p>Clenproperol is a β2-adrenergic agonist.</p>Fórmula:C11H16Cl2N2OCor e Forma:SolidPeso molecular:263.16Isoetharine
CAS:<p>Isoetharine is a selective agonist of β2-adrenergic receptor used as a bronchodilator for emphysema, bronchitis, and asthma.</p>Fórmula:C13H21NO3Cor e Forma:SolidPeso molecular:239.31Denopamine
CAS:<p>Denopamine is an agonist of 1-Adrenoceptor.</p>Fórmula:C18H23NO4Cor e Forma:SolidPeso molecular:317.38HEAT hydrochloride
CAS:<p>HEAT hydrochloride is an α1-adrenoceptor antagonist.</p>Fórmula:C19H22ClNO2Pureza:98%Cor e Forma:SolidPeso molecular:331.845-Methylurapidil
CAS:<p>5-Methylurapidil is an alpha1A-adrenoceptor antagonist.</p>Fórmula:C21H31N5O3Pureza:98%Cor e Forma:SolidPeso molecular:401.5Tiamenidine
CAS:<p>Tiamenidine is an antagonist of centrally-acting alpha1 adrenergic receptor.</p>Fórmula:C8H10ClN3SPureza:98%Cor e Forma:SolidPeso molecular:215.7RWJ 52353
CAS:<p>α2D adrenergic receptor agonist</p>Fórmula:C11H10N2SPureza:98%Cor e Forma:SolidPeso molecular:202.28Bucumarol (HCl)
CAS:<p>Bucumarol is a beta-adrenergic blocking agent.</p>Fórmula:C17H24ClNO4Cor e Forma:SolidPeso molecular:341.83Tiodazosin
CAS:<p>Tiodazosin is a competitive antagonist of the postsynaptic alpha-adrenergic receptor.</p>Fórmula:C18H21N7O4SPureza:98%Cor e Forma:SolidPeso molecular:431.47A 61603
CAS:<p>Cixutumumab (IMC-A12) is a humanized IgG monoclonal antibody targeting the IGF1R with anticancer activity.</p>Fórmula:C14H20BrN3O3SCor e Forma:SolidPeso molecular:390.3L 640033
CAS:<p>L 640033 is a beta-agonist.</p>Fórmula:C18H25N3OPureza:98%Cor e Forma:SolidPeso molecular:299.41Sulfinalol
CAS:<p>Sulfinalol is a compound that acts as an orally active β-adrenoceptor antagonist and directly induces vasodilation [1].</p>Fórmula:C20H27NO4SCor e Forma:SolidPeso molecular:377.5A-123189
CAS:<p>A-123189 is a potent, alpha1D-selective antagonist.</p>Fórmula:C26H28N4O3SPureza:98%Cor e Forma:SolidPeso molecular:476.59(±)-Befunolol
CAS:<p>(±)-Befunolol is a blocking agent of β-adrenoceptor.</p>Fórmula:C16H21NO4Pureza:98%Cor e Forma:SolidPeso molecular:291.34(R)-Carvedilol
CAS:<p>(R)-Carvedilol is a non-selective blocker of β/α-1. (R)-Carvedilol exerts protection against the vascular or cardiac toxicity of Doxorubicin (DOX).</p>Fórmula:C24H26N2O4Pureza:98%Cor e Forma:SolidPeso molecular:406.47Tropodifene
CAS:<p>Tropodifene is an inhibitor of the α-Adrenergic receptor.</p>Fórmula:C25H29NO4Pureza:98%Cor e Forma:SolidPeso molecular:407.5Falintolol, (Z)-
CAS:<p>Falintolol, (Z)-, is a novel β-adrenergic antagonist compound distinguished by the inclusion of an oxime moiety.</p>Fórmula:C12H24N2O2Pureza:98%Cor e Forma:SolidPeso molecular:228.33Mezilamine
CAS:<p>Mezilamine is an antagonist of dopamine. It also blocks presynaptic but stimulating postsynaptic alpha-adrenoceptors.</p>Fórmula:C11H18ClN5SPureza:98%Cor e Forma:SolidPeso molecular:287.81WB 4101 hydrochloride
CAS:<p>α1A-adrenergic antagonist</p>Fórmula:C19H24ClNO5Pureza:98%Cor e Forma:SolidPeso molecular:381.85L 665871
CAS:<p>L 665871 is used as a beta-agonist. It works as a potential swine growth promoter.</p>Fórmula:C11H19N3OPureza:98%Cor e Forma:SolidPeso molecular:209.29Amibegron hydrochloride
CAS:<p>Amibegron hydrochloride is a selective β3-adrenoceptor agonist (EC50: 3.5 nM for β-adrenoceptor in rat colon). It has anxiolytic and antidepressant activity.</p>Fórmula:C22H27Cl2NO4Cor e Forma:SolidPeso molecular:440.36Tetrahydrozoline nitrate
CAS:<p>Tetrahydrozoline, an imidazoline derivative, is an α-adrenergic agonist for nasal and eye congestion studies.</p>Fórmula:C13H17N3O3Cor e Forma:SolidPeso molecular:263.297Metaproterenol
CAS:<p>Metaproterenol also has anti-inflammatory activity. Metaproterenol is a direct-acting sympathomimetic and a β2-adrenergic receptor (β2AR) agonist (IC50: 68 nM).</p>Fórmula:C11H17NO3Pureza:98%Cor e Forma:SolidPeso molecular:211.26Fenmetozole HCl
CAS:<p>Fenmetozole HCl is an antagonist of the actions of ethanol. It attenuates the ethanol-induced reduction in cerebellar cyclic guanosine monophosphate content.</p>Fórmula:C10H11Cl3N2OPureza:98%Cor e Forma:SolidPeso molecular:281.57Ridazolol
CAS:<p>Ridazolol is a vasodilating and cardioselective beta adrenergic blocker.</p>Fórmula:C15H18Cl2N4O3Pureza:99.05%Cor e Forma:SolidPeso molecular:373.23Guanoxabenz
CAS:<p>Guanoxabenz is an α2 adrenergic receptor agonist.</p>Fórmula:C8H8Cl2N4OPureza:98%Cor e Forma:SolidPeso molecular:247.08(S)-Carvedilol
CAS:<p>(S)-Carvedilol is a non-selective β/α-1 blocker.It exerts protection against the vascular or cardiac toxicity of Doxorubicin (DOX).</p>Fórmula:C24H26N2O4Pureza:98%Cor e Forma:Less Crystalline Solid Colourless Crystalline SolidPeso molecular:406.47Detomidine
CAS:<p>Detomidine is a nonnarcotic, synthetic α2-adrenergic agonist. Detomidine produces dose-dependent sedative and analgesic effects.</p>Fórmula:C12H14N2Pureza:98%Cor e Forma:White Crystalline PowderPeso molecular:186.25SB-226552
CAS:<p>SB-226552 is an aryloxypropanolamine selective beta3AR agonist.</p>Fórmula:C25H36NO5PCor e Forma:SolidPeso molecular:461.53Undecylenoyl phenylalanine
CAS:<p>Undecylenoyl phenylalanine (Sepiwhite msh QD) is a novel depigmenting agent, which possibly acts as an alpha-melanocyte-stimulating hormone antagonist, thus</p>Fórmula:C20H29NO3Pureza:≥98%Cor e Forma:White To Pinkish Solid PowderPeso molecular:331.45L-749372
CAS:<p>L-749372 is the beta 3 adrenergic receptor 3-Pyridyloxypropanolamine agonist.</p>Fórmula:C22H24IN3O4SPureza:98%Cor e Forma:SolidPeso molecular:553.41Midodrine D6 hydrochloride
CAS:<p>Midodrine D6 hydrochloride is a vasopressor/antihypotensive agent.</p>Fórmula:C12H19ClN2O4Pureza:98%Cor e Forma:SolidPeso molecular:296.78
