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Receptor adrenérgico

Receptor adrenérgico

Os receptores adrenérgicos são GPCRs que são ativados por catecolaminas, como adrenalina e noradrenalina. Esses receptores são classificados em subtipos alfa e beta, cada um dos quais desempenha um papel fundamental na regulação da frequência cardíaca, pressão arterial e resposta de luta ou fuga. Moduladores de receptores adrenérgicos são essenciais no tratamento de doenças cardiovasculares, asma e distúrbios de ansiedade. Na CymitQuimica, oferecemos uma ampla gama de moduladores de receptores adrenérgicos de alta qualidade para apoiar sua pesquisa em endocrinologia, farmacologia cardiovascular e resposta ao estresse.

Subcategorias de "Receptor adrenérgico"

Foram encontrados 729 produtos de "Receptor adrenérgico"

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  • Olodaterol hydrochloride

    CAS:
    <p>Olodaterol hydrochloride (BI-1744 HCl) is a novel, long-acting β2-adrenergic agonist that exerts its pharmacological effect by binding and activating β2-AR.</p>
    Fórmula:C21H27ClN2O5
    Pureza:99.11%
    Cor e Forma:Solid
    Peso molecular:422.9

    Ref: TM-T5159

    1mg
    47,00€
    5mg
    87,00€
    10mg
    140,00€
    25mg
    274,00€
    50mg
    439,00€
    100mg
    707,00€
    200mg
    938,00€
  • Glaucine

    CAS:
    <p>Glaucine: antitussive, antioxidative, antiviral, may fight arthritis, boosts IL-10, hinders breast cancer cell spread by inhibiting MMP-9 and NF-κB.</p>
    Fórmula:C21H25NO4
    Pureza:99.42% - 99.56%
    Cor e Forma:Solid
    Peso molecular:355.43

    Ref: TM-T5S2059

    2mg
    42,00€
    5mg
    62,00€
    10mg
    96,00€
    25mg
    145,00€
  • Salbutamol hemisulfate

    CAS:
    Salbutamol hemisulfate (Albuterol Sulfate) is a short-acting β2-adrenergic receptor agonist with an IC50 of 8.93 μM.
    Fórmula:C13H21NO3H2O4S
    Pureza:99.35%
    Cor e Forma:White Or Almost White Odourless Powder
    Peso molecular:576.70

    Ref: TM-T6652

    1g
    93,00€
    200mg
    42,00€
    500mg
    64,00€
  • Desipramine

    CAS:
    <p>Desipramine: tricyclic antidepressant that blocks norepinephrine reuptake and helps reduce sleep-related pharyngeal collapsibility.</p>
    Fórmula:C18H22N2
    Cor e Forma:Solid
    Peso molecular:266.38

    Ref: TM-T60445

    25mg
    2.033,00€
    50mg
    2.645,00€
    100mg
    3.345,00€
  • Vilanterol trifenatate

    CAS:
    Vilanterol trifenatate is a long-acting agonist of β2-adrenoceptor (β2-AR) with inherent 24-hour activity(β2-AR, β1-AR and β3-AR pEC50s of 10.37, 6.98 and 7.36, respectively)
    Fórmula:C44H49Cl2NO7
    Pureza:99.51% - >99.99%
    Cor e Forma:Solid
    Peso molecular:774.77

    Ref: TM-T5134

    1mg
    37,00€
    5mg
    93,00€
    10mg
    124,00€
    25mg
    219,00€
    50mg
    350,00€
    100mg
    505,00€
    1mL*10mM (DMSO)
    106,00€
  • Scopine

    CAS:
    Scopine (6,7-Epoxytropine), the metabolite of anisodine, is an α1-adrenergic receptor agonist used in the therapy of acute circulatory shock.
    Fórmula:C8H13NO2
    Pureza:99.79% - >99.99%
    Cor e Forma:Solid
    Peso molecular:155.19

    Ref: TM-T6662

    5mg
    49,00€
    10mg
    74,00€
    25mg
    114,00€
    50mg
    170,00€
    100mg
    296,00€
    200mg
    442,00€
    500mg
    710,00€
    1mL*10mM (DMSO)
    49,00€
  • Fluparoxan HCl

    CAS:
    Fluparoxan is a potent α2-adrenergic receptor antagonist (pKB = 7.9) with excellent α2/α1 selectivity (2630 fold).
    Fórmula:C10H11ClFNO2
    Cor e Forma:Solid
    Peso molecular:231.65

    Ref: TM-T27340

    25mg
    1.444,00€
    50mg
    1.882,00€
    100mg
    2.375,00€
  • Dexmedetomidine hydrochloride

    CAS:
    Dexmedetomidine hydrochloride (Precedex) is a potent, selective, orally active α2-adrenoceptor agonist.Cost-effective and quality-assured.
    Fórmula:C13H16N2·HCl
    Pureza:99.94% - 99.94%
    Cor e Forma:White Or Almost White Crystalline Powder
    Peso molecular:236.74

    Ref: TM-T6466

    5mg
    42,00€
    10mg
    55,00€
    25mg
    88,00€
    50mg
    159,00€
    100mg
    226,00€
    200mg
    340,00€
    500mg
    563,00€
    1mL*10mM (DMSO)
    50,00€
  • Phosphorylcholine chloride

    CAS:
    Phosphorylcholine chloride, an antigenic component found on the surface of numerous commensal and pathogenic bacteria inhabiting the upper airway, is integral
    Fórmula:C5H15ClNO4P
    Pureza:99.481% - 99.85%
    Cor e Forma:Solid
    Peso molecular:219.6

    Ref: TM-T6105

    1g
    50,00€
    5g
    106,00€
    500mg
    39,00€
  • Pimozide

    CAS:
    Pimozide: antipsychotic that blocks type 2 dopamine, alpha-adrenergic, and 5-HT2 receptors, reducing tics and delusions.
    Fórmula:C28H29F2N3O
    Pureza:99.63% - >99.99%
    Cor e Forma:Solid
    Peso molecular:461.55

    Ref: TM-T2546

    25mg
    37,00€
    50mg
    52,00€
    100mg
    A consultar
    1mL*10mM (DMSO)
    52,00€
  • Idazoxan hydrochloride

    CAS:
    Idazoxan hydrochloride (RX 781094) is a benzodioxane-linked imidazole. It has alpha-2 adrenoceptor antagonist activity.
    Fórmula:C11H12N2O2·HCl
    Pureza:99.42% - 99.84%
    Cor e Forma:Solid
    Peso molecular:240.69

    Ref: TM-T0115

    2mg
    35,00€
    5mg
    52,00€
    10mg
    78,00€
    25mg
    133,00€
    50mg
    187,00€
    100mg
    281,00€
    200mg
    416,00€
    1mL*10mM (DMSO)
    50,00€
  • Xamoterol

    CAS:
    Xamoterol is a cardiac stimulant.
    Fórmula:C16H25N3O5
    Cor e Forma:Solid
    Peso molecular:339.39

    Ref: TM-T35153

    25mg
    1.444,00€
    50mg
    1.882,00€
    100mg
    2.375,00€
  • Napitane Mesylate

    CAS:
    Napitane Mesylate inhibits norepinephrine transporter and blocks CNS CA uptake as an alpha 2-adrenoceptor antagonist.
    Fórmula:C23H29NO5S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:431.55

    Ref: TM-T26363

    25mg
    1.730,00€
    50mg
    2.262,00€
    100mg
    2.945,00€
  • Nomifensine

    CAS:
    Nomifensine ((±)-Nomifensin) is a norepinephrine-dopamine reuptake inhibitor that prevents dopamine reuptake into synaptosomes.
    Fórmula:C16H18N2
    Pureza:99.83% - ≥95%
    Cor e Forma:Solid
    Peso molecular:238.33

    Ref: TM-T7308

    10mg
    35,00€
    25mg
    49,00€
    50mg
    70,00€
    100mg
    104,00€
    1mL*10mM (DMSO)
    35,00€
  • Apraclonidine

    CAS:
    Apraclonidine (ALO 2145), an α2/weak α1 agonist, lowers IOP; used as eye drops.
    Fórmula:C9H10Cl2N4
    Cor e Forma:Solid
    Peso molecular:245.11

    Ref: TM-T60350

    25mg
    1.444,00€
    50mg
    1.882,00€
    100mg
    2.375,00€
  • Tulobuterol hydrochloride

    CAS:
    Tulobuterol hydrochloride (Hokunalin) is a long-acting beta2-adrenergic receptor agonist.
    Fórmula:C12H19Cl2NO
    Pureza:99.24% - >99.99%
    Cor e Forma:Appearance White Crystalline Powder
    Peso molecular:264.19

    Ref: TM-T3277

    500mg
    40,00€
    1mL*10mM (DMSO)
    34,00€
  • Clebopride malate

    CAS:
    Clebopride malate is a dopamine antagonist drug Used to treat functional gastrointestinal disorders such as nausea or vomiting.
    Fórmula:C24H30ClN3O7
    Pureza:99.52%
    Cor e Forma:Solid
    Peso molecular:507.96

    Ref: TM-T7569

    5mg
    35,00€
    10mg
    48,00€
    25mg
    70,00€
    50mg
    96,00€
    100mg
    145,00€
    200mg
    210,00€
    1mL*10mM (DMSO)
    38,00€
  • Piribedil hydrochloride

    CAS:
    Piribedil HCl treats Parkinson's, circulatory issues, aids cancer research; inhibits MLL1; D2/D3 agonist; α2-antagonist. EC50: 0.18 μM.
    Fórmula:C16H19ClN4O2
    Cor e Forma:Solid
    Peso molecular:334.8

    Ref: TM-T61027

    25mg
    1.444,00€
    50mg
    1.882,00€
    100mg
    2.375,00€
  • Naftopidil hydrochloride

    CAS:
    Naftopidil HCl (BM-15275) is a selective alpha1 blocker with Ki: α1a-3.7 nM, α1b-20 nM, α1d-1.2 nM; it also inhibits cell growth.
    Fórmula:C24H29ClN2O3
    Pureza:99.5%
    Cor e Forma:Solid
    Peso molecular:428.95

    Ref: TM-T9220

    1mg
    44,00€
    5mg
    87,00€
    10mg
    117,00€
    25mg
    202,00€
    50mg
    304,00€
    100mg
    437,00€
    200mg
    612,00€
    1mL*10mM (DMSO)
    97,00€
  • Guanabenz Acetate

    CAS:
    Guanabenz Acetate (Wytensin) is a specific agonist of adrenergic receptor.
    Fórmula:C8H8Cl2N4·C2H4O2
    Pureza:99% - 99.66%
    Cor e Forma:White Solid From Acetonitrile White Solid
    Peso molecular:291.13

    Ref: TM-T6522

    1g
    62,00€
    200mg
    35,00€
    500mg
    48,00€
    1mL*10mM (DMSO)
    34,00€