
Receptor adrenérgico
Os receptores adrenérgicos são GPCRs que são ativados por catecolaminas, como adrenalina e noradrenalina. Esses receptores são classificados em subtipos alfa e beta, cada um dos quais desempenha um papel fundamental na regulação da frequência cardíaca, pressão arterial e resposta de luta ou fuga. Moduladores de receptores adrenérgicos são essenciais no tratamento de doenças cardiovasculares, asma e distúrbios de ansiedade. Na CymitQuimica, oferecemos uma ampla gama de moduladores de receptores adrenérgicos de alta qualidade para apoiar sua pesquisa em endocrinologia, farmacologia cardiovascular e resposta ao estresse.
Subcategorias de "Receptor adrenérgico"
Foram encontrados 742 produtos para "Receptor adrenérgico".
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Detomidine
CAS:Detomidine is a nonnarcotic, synthetic α2-adrenergic agonist. Detomidine produces dose-dependent sedative and analgesic effects.Fórmula:C12H14N2Pureza:98%Cor e Forma:SolidPeso molecular:186.25Tiamenidine hydrochloride
CAS:Tiamenidine hydrochloride is a centrally-acting alpha1 adrenergic receptor antagonist.Fórmula:C8H11Cl2N3SCor e Forma:SolidPeso molecular:252.16Trimethaphan camsylate
CAS:Trimethaphan camsylate is a nicotinic antagonist that has been used as a ganglionic blocker in hypertension.Fórmula:C32H40N2O5S2Cor e Forma:SolidPeso molecular:596.801Org GC 94
CAS:Org GC 94 is a NaSSA antidepressant targeting histamine/serotonin/adrenergic receptors with clinically relevant anxiolytic and sedative effects.Fórmula:C18H20N2OPureza:99.57% - 99.94%Cor e Forma:Yellow SolidPeso molecular:280.36Phenoprolamine Hydrochloride
CAS:Phenoprolamine HCl: α1 blocker with anti-hypertensive, brain, and heart protection; inhibits CYP2D/3A, crosses the blood-brain barrier.Fórmula:C21H30ClNO3Cor e Forma:SolidPeso molecular:379.92(S)-Carvedilol
CAS:(S)-Carvedilol is a non-selective β/α-1 blocker.It exerts protection against the vascular or cardiac toxicity of Doxorubicin (DOX).Fórmula:C24H26N2O4Pureza:98%Cor e Forma:Less Crystalline Solid Colourless Crystalline SolidPeso molecular:406.47Guanadrel Sulfate
CAS:Guanadrel Sulfate, a postganglionic blocker, is stored in neurons via the norepinephrine pump.Fórmula:C10H21N3O6SCor e Forma:SolidPeso molecular:311.35Guanoxabenz
CAS:Guanoxabenz is an α2 adrenergic receptor agonist.Fórmula:C8H8Cl2N4OPureza:98%Cor e Forma:SolidPeso molecular:247.08Pargolol
CAS:Pargolol is a beta adrenergic receptor antagonist.Fórmula:C16H23NO3Cor e Forma:SolidPeso molecular:277.36Ridazolol
CAS:Ridazolol is a vasodilating and cardioselective beta adrenergic blocker.Fórmula:C15H18Cl2N4O3Pureza:99.13%Cor e Forma:White SolidPeso molecular:373.23Colterol (free base)
CAS:Colterol: short-acting β2 agonist; Bitolterol prodrug treats asthma, COPD bronchospasm.Fórmula:C12H19NO3Cor e Forma:SolidPeso molecular:225.28Clonidine
CAS:Clonidine (Kapvay): central alpha-adrenergic agonist, antihypertensive, often combined, not tied to liver issues.Fórmula:C9H9Cl2N3Pureza:99.42% - 99.44%Cor e Forma:White SolidPeso molecular:230.09Fenmetozole HCl
CAS:Fenmetozole HCl is an antagonist of the actions of ethanol. It attenuates the ethanol-induced reduction in cerebellar cyclic guanosine monophosphate content.Fórmula:C10H11Cl3N2OPureza:98%Cor e Forma:SolidPeso molecular:281.57Metaproterenol
CAS:Metaproterenol also has anti-inflammatory activity. Metaproterenol is a direct-acting sympathomimetic and a β2-adrenergic receptor (β2AR) agonist (IC50: 68 nM).Fórmula:C11H17NO3Pureza:98%Cor e Forma:SolidPeso molecular:211.26Tetrahydrozoline nitrate
CAS:Tetrahydrozoline, an imidazoline derivative, is an α-adrenergic agonist for nasal and eye congestion studies.Fórmula:C13H17N3O3Cor e Forma:SolidPeso molecular:263.297Stresson
CAS:Stresson is a beta-blocking agent bunitrolol.Fórmula:C14H21ClN2O2Cor e Forma:SolidPeso molecular:284.78Medroxalol hydrochloride
CAS:Medroxalol hydrochloride is an antihypertensive agent that possesses both alpha and beta-adrenergic antagonistic properties.Fórmula:C20H25ClN2O5Cor e Forma:SolidPeso molecular:408.88Piribedil Maleate
CAS:Piribedil Maleate is a direct agonist of dopamine that acts by showing selectivity for the D3 subtype.Fórmula:C20H22N4O6Pureza:98%Cor e Forma:SolidPeso molecular:414.41Amibegron hydrochloride
CAS:Amibegron hydrochloride is a selective β3AR agonist that increases energy expenditure and fat oxidation by activating β3ARs in brown adipose tissue.Fórmula:C22H27Cl2NO4Pureza:98.83%Cor e Forma:Yellow SolidPeso molecular:440.36Ref: TM-T10302
1mg90,00€5mg215,00€1mL*10mM (DMSO)245,00€10mg318,00€25mg530,00€50mg755,00€100mg1.018,00€Labetalone hydrochloride
CAS:Labetalone hydrochloride, a Labetalol impurity, is an orally active alpha and beta-adrenoceptor blocker.Fórmula:C19H23ClN2O3Pureza:99.58%Cor e Forma:SolidPeso molecular:362.85
