Receptor adrenérgico
Os receptores adrenérgicos são GPCRs que são ativados por catecolaminas, como adrenalina e noradrenalina. Esses receptores são classificados em subtipos alfa e beta, cada um dos quais desempenha um papel fundamental na regulação da frequência cardíaca, pressão arterial e resposta de luta ou fuga. Moduladores de receptores adrenérgicos são essenciais no tratamento de doenças cardiovasculares, asma e distúrbios de ansiedade. Na CymitQuimica, oferecemos uma ampla gama de moduladores de receptores adrenérgicos de alta qualidade para apoiar sua pesquisa em endocrinologia, farmacologia cardiovascular e resposta ao estresse.
Subcategorias de "Receptor adrenérgico"
Foram encontrados 725 produtos de "Receptor adrenérgico"
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Bufuralol
CAS:Bufuralol (Ro 3-4787) is a 尾-adrenergic receptor blocker with a certain degree of sympathomimetic effects and can be used to study cardiovascular diseases.Fórmula:C16H23NO2Pureza:98.26%Cor e Forma:SolidPeso molecular:261.36N-5984 Hydrochloride
CAS:N-5984 Hydrochloride is a beta3-AR agonist.Fórmula:C20H23Cl2NO5Cor e Forma:SolidPeso molecular:428.31Indacaterol xinafoate
CAS:Indacaterol xinafoate is an ultra-long-acting beta-adrenoceptor agonist.Fórmula:C35H36N2O6Cor e Forma:SolidPeso molecular:580.67Prenalterol hydrochloride
CAS:Prenalterol HCl: beta 1-specific agonist; treats acute cardiac failure, shock, low-output post-MI, Shy-Drager syndrome.Fórmula:C12H20ClNO3Cor e Forma:SolidPeso molecular:261.75OPC-28326
CAS:OPC-28326: an α2-adrenergic blocker; dilates blood vessels; inhibits α2A/B/C receptors with Ki 2040/285/55 nM.Fórmula:C26H35N3O2Pureza:99.79%Cor e Forma:SolidPeso molecular:421.58Talibegron hydrochloride
CAS:Talibegron hydrochloride: β3 adrenoceptor agonist, pD2 3.72, relaxes rat arteries, reduces leptin in mice.Fórmula:C18H22ClNO4Pureza:99.82%Cor e Forma:SolidPeso molecular:351.830990CL
CAS:0990CL is an effective heterotrimer Gαi subunit specific inhibitor, which can interact with purified Go± in GDP-bound state, and can block α2AR mediated cAMPFórmula:C21H21N5Pureza:98.99%Cor e Forma:SolidPeso molecular:343.42CGP-20712
CAS:CGP-20712 is a selective β 1-adrenoceptor antagonist with an IC50 of 0.7 nM.Fórmula:C23H25F3N4O5Pureza:99.40% - 99.58%Cor e Forma:SolidPeso molecular:494.46(±)-Prenalterol
CAS:(±)-Prenalterol (H 80/62) is an agonist of beta-2- and beta-1-adrenergic receptors and is used to study chronic congestive heart failure.Fórmula:C12H19NO3Pureza:99.73%Cor e Forma:SolidPeso molecular:225.28Deriglidole
CAS:Deriglidole (SL 86-0715), an alpha2 receptor inhibitor, blocks colistin/Idazoxan but not prazosin/α2-adrenergic receptors.Fórmula:C16H21N3Pureza:98.12% - 99.03%Cor e Forma:SolidPeso molecular:255.36α1 adrenoceptor-MO-1
CAS:α1 adrenoceptor-MO-1 (S enantiomer) has affinity at alpha 1 adrenergic receptor with alphalytic activity and analgesic action.Fórmula:C20H24ClN5OPureza:99.20% - 99.29%Cor e Forma:SolidPeso molecular:385.89Mafoprazine
CAS:Mafoprazine, a phenylpiperazine derivative, exhibits varying affinities for neuronal receptors, primarily exerting its antipsychotic effects through blocking D2 receptors and enhancing α-adrenergic activity. It also increases the activity of dopamine metabolites.Fórmula:C22H28FN3O3Cor e Forma:SolidPeso molecular:401.47Teoprolol
CAS:Teoprolol is a blocker of β-adrenergic receptor.Fórmula:C23H30N6O4Pureza:98%Cor e Forma:SolidPeso molecular:454.52Vibegron
CAS:Vibegron (MK-4618) is an effective and selective Beta 3 adrenergic receptor agonist, used to treat overactive bladder (OAB).Fórmula:C26H28N4O3Cor e Forma:SolidPeso molecular:444.53Nipradolol
CAS:Nipradolol blocks alpha-1-adrenergic receptors, lowers IOP in rabbits, and reduces NA-induced muscle contraction and dog artery vasodilation.Fórmula:C15H22N2O6Cor e Forma:SolidPeso molecular:326.35(±)-Penbutolol
CAS:(±)-Penbutolol ((Rac)-Penbutolol) is the racemic form of Penbutolol. It acts as an orally active β-adrenergic receptor antagonist. (±)-Penbutolol mitigates the tachycardia induced by exercise, reduces the increase in peak expiratory flow rate (PEFR) caused by physical activity, and decreases plasma renin activity (PRA) at rest. The peak plasma concentration of this compound is achieved one hour after oral administration, with a half-life of 4.5 hours, and it is metabolized into active metabolites in the body. This compound is utilized in research related to cardiovascular diseases.Fórmula:C18H29NO2Cor e Forma:SolidPeso molecular:291.43Bometolol Hydrochloride
CAS:Bometolol Hydrochloride is a beta-adrenergic blocking compound used for the treatment of cardiovascular disease.Fórmula:C25H33ClN2O7Pureza:98%Cor e Forma:SolidPeso molecular:508.99AA 497 (Free Base)
CAS:AA 497, a beta-2 agonist, causes relaxation and suppresses Ca spike frequency.Fórmula:C14H21NO3Pureza:98%Cor e Forma:SolidPeso molecular:251.32Metrazoline
CAS:<p>Metrazoline (o-Methyl-tracizoline) acts as a ligand for adrenergic receptors (low affinity) and imidazoline I2 receptors.</p>Fórmula:C14H16N2O4Cor e Forma:SolidPeso molecular:276.288PF-9404C
CAS:PF-9404C: S-S diastereoisomer, beta-blocker with vasodilation, boosts cyclic GMP in rat aorta cells from 3 to 53 pmol/mg protein.Fórmula:C16H25N3O9Pureza:98%Cor e Forma:SolidPeso molecular:403.38
