
Receptor adrenérgico
Os receptores adrenérgicos são GPCRs que são ativados por catecolaminas, como adrenalina e noradrenalina. Esses receptores são classificados em subtipos alfa e beta, cada um dos quais desempenha um papel fundamental na regulação da frequência cardíaca, pressão arterial e resposta de luta ou fuga. Moduladores de receptores adrenérgicos são essenciais no tratamento de doenças cardiovasculares, asma e distúrbios de ansiedade. Na CymitQuimica, oferecemos uma ampla gama de moduladores de receptores adrenérgicos de alta qualidade para apoiar sua pesquisa em endocrinologia, farmacologia cardiovascular e resposta ao estresse.
Subcategorias de "Receptor adrenérgico"
Foram encontrados 725 produtos de "Receptor adrenérgico"
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Bucindolol hydrochloride
CAS:Bucindolol, a 4th-gen β-blocker, prevents onset AF; effectiveness varies with β₁/α(2c) genes; best in β₁389 Arg homozygotes.Fórmula:C22H26ClN3O2Cor e Forma:SolidPeso molecular:399.91Phentolamine
CAS:Phentolamine mesylate is an alpha-1 and alpha-2 selective adrenergic receptor antagonistFórmula:C17H19N3OPureza:99.86% - 99.94%Cor e Forma:Crystals SolidPeso molecular:281.35Olodaterol hydrochloride
CAS:<p>Olodaterol hydrochloride (BI-1744 HCl) is a novel, long-acting β2-adrenergic agonist that exerts its pharmacological effect by binding and activating β2-AR.</p>Fórmula:C21H27ClN2O5Pureza:99.11%Cor e Forma:SolidPeso molecular:422.9Glaucine
CAS:<p>Glaucine: antitussive, antioxidative, antiviral, may fight arthritis, boosts IL-10, hinders breast cancer cell spread by inhibiting MMP-9 and NF-κB.</p>Fórmula:C21H25NO4Pureza:99.42% - 99.56%Cor e Forma:SolidPeso molecular:355.43Salbutamol hemisulfate
CAS:Salbutamol hemisulfate (Albuterol Sulfate) is a short-acting β2-adrenergic receptor agonist with an IC50 of 8.93 μM.Fórmula:C13H21NO3H2O4SPureza:99.35%Cor e Forma:White Or Almost White Odourless PowderPeso molecular:576.70Desipramine
CAS:<p>Desipramine: tricyclic antidepressant that blocks norepinephrine reuptake and helps reduce sleep-related pharyngeal collapsibility.</p>Fórmula:C18H22N2Cor e Forma:SolidPeso molecular:266.38Vilanterol trifenatate
CAS:Vilanterol trifenatate is a long-acting agonist of β2-adrenoceptor (β2-AR) with inherent 24-hour activity(β2-AR, β1-AR and β3-AR pEC50s of 10.37, 6.98 and 7.36, respectively)Fórmula:C44H49Cl2NO7Pureza:99.51% - >99.99%Cor e Forma:SolidPeso molecular:774.77Scopine
CAS:Scopine (6,7-Epoxytropine), the metabolite of anisodine, is an α1-adrenergic receptor agonist used in the therapy of acute circulatory shock.Fórmula:C8H13NO2Pureza:99.79% - >99.99%Cor e Forma:SolidPeso molecular:155.19Fluparoxan HCl
CAS:Fluparoxan is a potent α2-adrenergic receptor antagonist (pKB = 7.9) with excellent α2/α1 selectivity (2630 fold).Fórmula:C10H11ClFNO2Cor e Forma:SolidPeso molecular:231.65Dexmedetomidine hydrochloride
CAS:Dexmedetomidine hydrochloride (Precedex) is a potent, selective, orally active α2-adrenoceptor agonist.Cost-effective and quality-assured.Fórmula:C13H16N2·HClPureza:99.94% - 99.94%Cor e Forma:White Or Almost White Crystalline PowderPeso molecular:236.74Phosphorylcholine chloride
CAS:Phosphorylcholine chloride, an antigenic component found on the surface of numerous commensal and pathogenic bacteria inhabiting the upper airway, is integralFórmula:C5H15ClNO4PPureza:99.481% - 99.85%Cor e Forma:SolidPeso molecular:219.6Pimozide
CAS:Pimozide: antipsychotic that blocks type 2 dopamine, alpha-adrenergic, and 5-HT2 receptors, reducing tics and delusions.Fórmula:C28H29F2N3OPureza:99.63% - >99.99%Cor e Forma:SolidPeso molecular:461.55Dobutamine hydrochloride
CAS:<p>Dobutamine hydrochloride (Dobutamine (hydrochloride)) is a catecholamine that acts as a β-adrenergic receptor agonist with potent positive inotropic effects.</p>Fórmula:C18H24ClNO3Pureza:97.15% - 99.94%Cor e Forma:SolidPeso molecular:337.84Levalbuterol tartrate
CAS:Levalbuterol tartrate is a short-acting β2-adrenergic receptor agonist and the R enantiomer of salbutamol.Cost-effective and quality-assured.Fórmula:C17H27NO9Pureza:99.28% - 99.98%Cor e Forma:SolidPeso molecular:389.39Xamoterol
CAS:Xamoterol is a cardiac stimulant.Fórmula:C16H25N3O5Cor e Forma:SolidPeso molecular:339.39Napitane Mesylate
CAS:Napitane Mesylate inhibits norepinephrine transporter and blocks CNS CA uptake as an alpha 2-adrenoceptor antagonist.Fórmula:C23H29NO5SPureza:98%Cor e Forma:SolidPeso molecular:431.55Nomifensine
CAS:Nomifensine ((±)-Nomifensin) is a norepinephrine-dopamine reuptake inhibitor that prevents dopamine reuptake into synaptosomes.Fórmula:C16H18N2Pureza:99.83% - ≥95%Cor e Forma:SolidPeso molecular:238.33Apraclonidine
CAS:Apraclonidine (ALO 2145), an α2/weak α1 agonist, lowers IOP; used as eye drops.Fórmula:C9H10Cl2N4Cor e Forma:SolidPeso molecular:245.11Tulobuterol hydrochloride
CAS:Tulobuterol hydrochloride (Hokunalin) is a long-acting beta2-adrenergic receptor agonist.Fórmula:C12H19Cl2NOPureza:99.24% - >99.99%Cor e Forma:Appearance White Crystalline PowderPeso molecular:264.19Clebopride malate
CAS:Clebopride malate is a dopamine antagonist drug Used to treat functional gastrointestinal disorders such as nausea or vomiting.Fórmula:C24H30ClN3O7Pureza:99.52%Cor e Forma:SolidPeso molecular:507.96
