AChR
Os inibidores do receptor de acetilcolina (AChR) são compostos que bloqueiam a atividade dos receptores de acetilcolina, essenciais para a neurotransmissão nos sistemas nervosos central e periférico. Os AChRs desempenham um papel vital na contração muscular, memória e funções cognitivas. Os inibidores de AChRs são usados para estudar condições como miastenia gravis, doença de Alzheimer e outros distúrbios neurológicos. Ao modular a atividade dos AChRs, esses inibidores podem ajudar a desvendar as complexidades da sinalização colinérgica no cérebro. Na CymitQuimica, oferecemos uma gama de inibidores de AChRs para apoiar sua pesquisa em neurociência, farmacologia e doenças neurodegenerativas.
Foram encontrados 636 produtos de "AChR"
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Telenzepine dihydrochloride
CAS:muscarinic M1 receptor antagonistFórmula:C19H23ClN4O2SPureza:98%Cor e Forma:SolidPeso molecular:406.93Dibucaine hydrochloride
CAS:Dibucaine hydrochloride (Cinchocaine hydrochloride), a long-acting local amide anestheticsis, is usually used for surface anesthesia.Fórmula:C20H30ClN3O2Pureza:99.66%Cor e Forma:White PowderPeso molecular:379.92Solifenacin D5 hydrochloride
CAS:Solifenacin D5 HCl: deuterium-labeled M1, M2, M3 muscarinic receptor antagonist with pKi 7.6, 6.9, 8.0.Fórmula:C23H27ClN2O2Pureza:98%Cor e Forma:SolidPeso molecular:403.96Fipexide hydrochloride
CAS:Fipexide (hydrochloride) is a kind of psychoactive drug of the piperazine class.Fórmula:C20H22Cl2N2O4Cor e Forma:SolidPeso molecular:425.31N6-Methyladenosine 5'-monophosphate disodium salt
CAS:N6-Methyladenosine 5'-monophosphate disodium salt is a glycogen phosphorylase b activator and an inhibitor of adenylate kinase II.Fórmula:C11H14N5Na2O7PPureza:99.36% - 99.36%Cor e Forma:SolidPeso molecular:405.21Cevimeline
CAS:Cevimeline: muscarinic agonist, treats dry mouth & Sjögren's, boosts saliva post-cancer radiotherapy.Fórmula:C10H17NOSCor e Forma:Off-White SolidPeso molecular:199.31Fesoterodine L-mandelate
CAS:Fesoterodine L-mandelate is a efficacious antimuscarinic agent for the overactive bladder (OAB).Fórmula:C34H45NO6Cor e Forma:SolidPeso molecular:563.735YM-58790 hydrochloride
CAS:YM-58790 is a potent M3 muscarinic receptor antagonist(Ki of 15 nM).Fórmula:C27H32ClN3O2Pureza:98%Cor e Forma:SolidPeso molecular:466.02Palmatine hydroxide
CAS:Palmatine hydroxide: oral IDO-1 inhibitor (IC50: 3-157μM), targets WNV protease, has anti-cancer/viral and neuroprotective properties.Fórmula:C21H23NO5Cor e Forma:SolidPeso molecular:369.41β2AR/M-receptor agonist-2
CAS:β2AR/M-receptor agonist-2 is a dual-function compound acting as a muscarinic antagonist and β2 adrenoceptor agonist (MABA).Fórmula:C36H49ClN4O7SCor e Forma:SolidPeso molecular:717.31Dexetimide
CAS:Dexetimide, a muscarinic receptor antagonist, treats neuroleptic-induced parkinsonism.Fórmula:C23H26N2O2Cor e Forma:SolidPeso molecular:362.46Varenicline Hydrochloride
CAS:Varenicline Hydrochloride (CP 526555) is an orally active partial agonist of the α4β2 nicotinic acetylcholine receptor (α4β2 nAChR, IC50 = 250 nM).Fórmula:C13H14ClN3Pureza:99.854%Cor e Forma:SolidPeso molecular:247.72Ref: TM-T23502
1mg38,00€5mg80,00€10mg105,00€25mg192,00€50mg297,00€100mg441,00€200mg646,00€1mL*10mM (DMSO)88,00€Glycerophosphoinositol choline
CAS:Glycerophosphoinositol choline is the salt of choline and glycerophosphoinositol.Fórmula:C14H32NO12PCor e Forma:SolidPeso molecular:437.38Cevimeline hydrochloride
CAS:Cevimeline HCl is a muscarinic agonist enhancing salivary and sweat gland secretion.Fórmula:C10H18ClOSCor e Forma:SolidPeso molecular:235.77(±)-Darifenacin
CAS:(±)-Darifenacin is the racemate of Darifenacin. Darifenacin is a selective antagonist of M3 muscarinic receptor.Fórmula:C28H30N2O2Cor e Forma:SolidPeso molecular:426.55VU0467485
CAS:VU0467485 boosts ACh at M4 receptors (EC50: 26.6 nM rat, 78.8 nM human), selective for M4 over M1/2/3/5.Fórmula:C17H17FN4O2SPureza:98%Cor e Forma:SolidPeso molecular:360.41Clorprenaline
CAS:Clorprenaline is a β-adrenergic receptor agonist that activates adenylate cyclase, relaxation of bronchial smooth muscle cells. anti-inflammatory.Fórmula:C11H16ClNOPureza:98.9%Cor e Forma:SolidPeso molecular:213.7Pirmenol hydrochloride
CAS:Pirmenol hydrochloride functions by inhibiting I_K.ACh through the blockade of muscarinic receptors, demonstrating a potent effect with an IC_50 value of 0.1 μMFórmula:C22H31ClN2OCor e Forma:SolidPeso molecular:374.95NBTGR
CAS:NBTGR is a potent nucleoside transport inhibitor(adenosine uptake ,Ki of 70 nM).Fórmula:C17H18N6O6SPureza:98%Cor e Forma:SolidPeso molecular:434.43Tebanicline dihydrochloride
CAS:Tebanicline dihydrochloride: oral analgesic, nAChR modulator, Ki=37 pM at α4β2 receptors, inhibits cytisine binding.Fórmula:C9H13Cl3N2OCor e Forma:SolidPeso molecular:271.57Ispronicline
CAS:Ispronicline (TC-1734) An orally active, selective, and potent α4β2 nAChR partial agonist with antidepressant, neuroprotective, and long-lasting cognitiveFórmula:C14H22N2OPureza:97.70% - 99.16%Cor e Forma:SolidPeso molecular:234.34Biperiden
CAS:Biperiden is a muscarinic antagonist for Parkinson's and drug-induced extrapyramidal symptoms.Fórmula:C21H29NOPureza:99.65%Cor e Forma:Crystals SolidPeso molecular:311.46SSR180711 hydrochloride
CAS:SSR180711 hydrochloride (SSR-180711A HCl) is an Alpha7 nicotinic acetylcholine partial agonist that can be used to study neurolysis.Fórmula:C14H18BrClN2O2Pureza:99.22%Cor e Forma:SolidPeso molecular:361.66(S)-(+)-Dimethindene maleate
CAS:(S)-(+)-Dimethindene maleate is an orally available, selective muscarinic M2 receptor and histamine H1 receptor antagonist that inhibits muscarinic M1 receptorsFórmula:C24H28N2O4Pureza:99.94%Cor e Forma:SolidPeso molecular:408.49NKH477
CAS:NKH477 (Colforsin dapropate hydrochloride) is a derivative of forskolin with antidepressant activity.Fórmula:C27H44ClNO8Pureza:98% - 98%Cor e Forma:SolidPeso molecular:546.09Sabcomeline hydrochloride
CAS:Sabcomeline is a selective M1 receptor partial agonist.Fórmula:C10H16ClN3OCor e Forma:SolidPeso molecular:229.71Tolterodine
CAS:Tolterodine ((R)-(+)-Tolterodine) is an mACh antagonist used in the treatment of detrusor instability and overactive bladder syndrome.Fórmula:C22H31NOPureza:99.71%Cor e Forma:White Like Or Light Brown Crystalline PowderPeso molecular:325.49NS3861 fumarate
CAS:NS3861 fumarate, a partial α3β4 nAChR agonist, binds α3β2, α4β4, α4β2 with Ki values of 0.62, 25, 7.8, 55 nM.Fórmula:C16H18BrNO4SCor e Forma:SolidPeso molecular:400.29ABT-107
CAS:ABT-107: α7 neuronal receptor agonist; protects rats' brains from 6-OHDA-induced damage.Fórmula:C19H20N4OCor e Forma:SolidPeso molecular:320.396NSC 23766
CAS:NSC 23766 is a Rac1 GTPase inhibitor by targeting GEFs, inhibiting cell proliferation.NSC23766 competitively inhibits M2 mAChR-induced Rac1 activation.Fórmula:C24H35N7Pureza:99.49%Cor e Forma:SolidPeso molecular:421.58DL-Cystine
CAS:DL-Cystine is a cysteine derivative that inhibits endothelial cell proliferation by regulating TGFβ1. a GPR inhibitor and nAChR agonist .Fórmula:C6H12N2O4S2Cor e Forma:SolidPeso molecular:240.3Syn-Ake acetate
CAS:Syn-Ake acetate (Dipeptide diaminobutyroyl benzylamide) is a muscarinic acetylcholine receptor antagonist.Fórmula:C19H29N5O3·2(C2H4O2)Pureza:99.60%Cor e Forma:SolidPeso molecular:495.58Succinylcholine Chloride Dihydrate
CAS:Succinylcholine Chloride Dihydrate (Succinyldicholine dichloride) is a nicotinic AChR agonist and also acts as a depolarizing neuromuscular blocker.
Fórmula:C14H30N2O4·2Cl·2H2OPureza:99.87%Cor e Forma:White SolidPeso molecular:397.34α-Conotoxin MII acetate
α-Conotoxin MII acetate is a 16-amino acid peptide from the venom of the marine snail Conus magus.Fórmula:C69H107N23O24S4Pureza:94.82% - 97.79%Cor e Forma:SolidPeso molecular:1770.99Tebanicline hydrochloride
CAS:Tebanicline hydrochloride (Ebanicline hydrochloride) , is an effective synthetic nicotinic (non-opioid) analgesic drug.Fórmula:C9H12Cl2N2OPureza:91.74% - 98.78%Cor e Forma:SolidPeso molecular:235.11Tosedostat
CAS:Tosedostat (CHR-2797), an oral M1 aminopeptidase inhibitor, turns into CHR-79888, blocks tumor cell proteins, causing cell death.Fórmula:C21H30N2O6Pureza:98.14% - 99.84%Cor e Forma:SolidPeso molecular:406.47KH7
CAS:KH7 is a soluble inhibitor of adenylyl cyclase (sAC)-specific.Fórmula:C17H15BrN4O2SPureza:98.43%Cor e Forma:SolidPeso molecular:419.3Propiverine hydrochloride
CAS:Propiverine is a widely used antimuscarinic drug with a mixed mode of action in the treatment of symptoms associated with overactive bladder (OAB).Fórmula:C23H30ClNO3Pureza:99.93%Cor e Forma:White Crystalling PowerPeso molecular:403.94JHU37152
CAS:JHU37152 is a DREADD agonist; Ki: 1.8 nM at hM3Dq, 8.7 nM at hM4Di; EC50: 5 nM (hM3Dq), 0.5 nM (hM4Di) in HEK-293 cell assays.Fórmula:C19H20ClFN4Pureza:99.72%Cor e Forma:SolidPeso molecular:358.84VU0119498
CAS:VU0119498 is a M1 muscarinic receptor agonist (EC50 = 3.1 μM) and pan mAChR M3, M5 positive allosteric modulator (PAM),and is a neuroprotective agent.Fórmula:C15H10BrNO2Pureza:97.56%Cor e Forma:SolidPeso molecular:316.15Clothianidin
CAS:Clothianidin (TI 435), an insecticide, stimulates nAChR as acetylcholine agonist, not AChE inhibitor.Fórmula:C6H8ClN5O2SPureza:99.71% - 99.87%Cor e Forma:Solid PowderPeso molecular:249.68VU0152100
CAS:VU0152100 is an effective and selective allosteric potentiator of M4 mAChR (EC50: 380 ± 93 nM).Fórmula:C18H19N3O2SPureza:99.56%Cor e Forma:SolidPeso molecular:341.43Ref: TM-T17238
2mg39,00€5mg58,00€10mg92,00€25mg195,00€50mg325,00€100mg522,00€200mg743,00€1mL*10mM (DMSO)64,00€Nitrobenzylthioinosine
CAS:Nitrobenzylthioinosine (NBMPR) is an inhibitor of ENT1 transporter that binds to ENT1 transporter with high affinity.
Fórmula:C17H17N5O6SPureza:99.69% - 99.74%Cor e Forma:Off-White SolidPeso molecular:419.41Anisotropine Methylbromide
CAS:Anisotropine Methylbromide is an anticholinergic agent and has been used for relief of gastrointestinal spasm and for the suppression of gastric acid secretion.Fórmula:C17H32BrNO2Pureza:99.73%Cor e Forma:Crystals From Acetone SolidPeso molecular:362.35VU0467154
CAS:VU0467154 is a positive allosteric modulator of the M4 muscarinic acetylcholine receptor.Fórmula:C17H15F3N4O3S2Pureza:99.51% - 99.53%Cor e Forma:SolidPeso molecular:444.45Ref: TM-T17244
1mg47,00€2mg63,00€5mg92,00€10mg126,00€25mg236,00€50mg400,00€100mg695,00€200mg945,00€1mL*10mM (DMSO)101,00€NS9283
CAS:NS9283, a positive allosteric modulator selective for the α4β2 form, reduces ethanol consumption.
Fórmula:C14H8N4OPureza:99.12%Cor e Forma:SolidPeso molecular:248.24ML380
CAS:ML380 is a highly potent and the first CNS penetrant M5 positive allosteric modulator (PAM).Fórmula:C23H25F3N4O3SPureza:99.69%Cor e Forma:SolidPeso molecular:494.53Ref: TM-T28069
2mg47,00€5mg71,00€10mg113,00€25mg178,00€50mg334,00€100mg500,00€500mg1.099,00€1mL*10mM (DMSO)78,00€Varenicline Tartrate
CAS:Varenicline Tartrate (CP 526555-18) is a benzazepine derivative that functions as an ALPHA4/BETA2 NICOTINIC RECEPTOR partial agonist.
Fórmula:C13H13N3·C4H6O6Pureza:98.23% - 98.32%Cor e Forma:Tan SolidPeso molecular:361.35Isopropamide Iodide
CAS:Isopropamide iodide: long-acting anticholinergic, treats peptic ulcers, GI disorders, Alzheimer's.
Fórmula:C23H33IN2OPureza:99.67%Cor e Forma:SolidPeso molecular:480.43Mc-Val-Ala-PAB
CAS:Mc-Val-Ala-PAB, an effective linker, is utilized in antibody-drug-conjugate (ADC).
Fórmula:C25H34N4O6Pureza:98.34% - 99.24%Cor e Forma:SolidPeso molecular:486.56Nitenpyram
CAS:Nitenpyram (Capstar) is a nicotinic acetylcholine receptor (AchR) agonist, used as veterinary medicine to treat parasites of livestock and pets.Fórmula:C11H15ClN4O2Pureza:99.03%Cor e Forma:Light-Yellow CrystalPeso molecular:270.72Mecamylamine hydrochloride
CAS:Mecamylamine hydrochloride (Mevasin) is a nicotinic antagonist, used as a ganglionic blocker in hypertension.Fórmula:C11H22ClNPureza:99.76% - >99.99%Cor e Forma:White SolidPeso molecular:203.75Solifenacin hydrochloride
CAS:Solifenacin Hcl is a muscarinic receptor antagonist.Fórmula:C23H27ClN2O2Pureza:98%Cor e Forma:SolidPeso molecular:398.93Procyclidine hydrochloride
CAS:Procyclidine hydrochloride ((±)-Procyclidine hydrochlorid) is a potent anticholinergic agent and also have NMDA antagonist properties.Fórmula:C19H30ClNOPureza:99.24% - 99.88%Cor e Forma:Crystals From Petroleum Ether White PowderPeso molecular:323.9Encenicline
CAS:Encenicline (EVP-6124), a selective α7 nAChRs agonist, targets cognitive impairment in schizophrenia and Alzheimer's.Fórmula:C16H17ClN2OSPureza:99.20%Cor e Forma:SolidPeso molecular:320.84Ref: TM-T7193
1mg70,00€5mg133,00€10mg207,00€25mg349,00€50mg495,00€100mg675,00€200mg888,00€1mL*10mM (DMSO)144,00€Sofpironium bromide
CAS:Sofpironium bromide (BBI4000) belongs to a class of drugs called anticholinergics, which exert their effect by blocking the action of acetylcholine.Fórmula:C22H32BrNO5Pureza:98.85%Cor e Forma:SolidPeso molecular:470.4Ref: TM-T28827
1mg74,00€5mg160,00€10mg250,00€25mg452,00€50mg680,00€100mg1.008,00€200mg1.349,00€1mL*10mM (DMSO)165,00€Mecamylamine
CAS:Mecamylamine: oral, noncompetitive nAChR blocker, crosses blood-brain barrier, for neuropsychiatric and hypertension research.Fórmula:C11H21NCor e Forma:SolidPeso molecular:167.29Oxyphencyclimine Hydrochloride
CAS:Oxyphencyclimine Hydrochloride (Ulcociclinina) is a synthetic tertiary amine and antimuscarinic agent with antispasmodic and antisecretory activities.Fórmula:C20H29ClN2O3Pureza:99.55%Cor e Forma:SolidPeso molecular:380.91Pempidine
CAS:Pempidine (1,2,2,6,6-Pentamethylpiperidine) is a nicotinic antagonist, has been used as a ganglionic blocker in the treatment of hypertension.Fórmula:C10H21NPureza:98.18% - 99.28%Cor e Forma:Colorless - Light Yellow Clear LiquidPeso molecular:155.28Propiverine
CAS:Propiverine reduces muscle spasms by limiting calcium influx, targeting bladder smooth muscles, aiding OAB research.Fórmula:C23H29NO3Cor e Forma:SolidPeso molecular:367.48NS 1738
CAS:NS 1738 (NSC-213859) is a positive allosteric modulator of the α7-containing neuronal nicotinic acetylcholine receptors (nAChRs)Fórmula:C14H9Cl2F3N2O2Pureza:99.11%Cor e Forma:SolidPeso molecular:365.13Dinotefuran
CAS:Dinotefuran (MTI-446), a neonicotinoid insecticide, targets pests by blocking their nervous system.Fórmula:C7H14N4O3Pureza:99.89%Cor e Forma:White Crystalline PowderPeso molecular:202.21Dronedarone
CAS:Dronedarone (SR 33589) is an amiodarone analogue which has an effective and promising treatment for Atrial fibrillation.Fórmula:C31H44N2O5SPureza:98.85% - 99.99%Cor e Forma:SolidPeso molecular:556.76EB-3D
CAS:EB-3D is a potent and selective choline kinase alpha 1 (ChoKα1) inhibitor(IC50 : 1 μM).with anti-cancer activity.Fórmula:C30H36Br2N4O2Pureza:99.48%Cor e Forma:SolidPeso molecular:644.4Ref: TM-T7955
1mg92,00€2mg120,00€5mg187,00€10mg274,00€25mg472,00€50mg655,00€100mg924,00€200mg1.225,00€1mL*10mM (DMSO)278,00€Oxyphenonium bromide
CAS:Oxyphenonium bromide is an anticholinergic used to study and treat ulcers and relieve visceral spasms.
Fórmula:C21H34BrNO3Pureza:98.96%Cor e Forma:SolidPeso molecular:428.404MC-Val-Cit-PABC-PNP
CAS:MC-Val-Cit-PABC-PNP, also known as Mc-Val-Cit-PABC-PNP, is a cathepsin cleavable ADC peptide linker.Fórmula:C35H43N7O11Pureza:97.2% - 98.055%Cor e Forma:SolidPeso molecular:737.76Propantheline
CAS:Propantheline: oral muscarinic receptor blocker for smooth muscle issues, hyperhidrosis, and bladder control.Fórmula:C23H30NO3Cor e Forma:SolidPeso molecular:368.49Batefenterol
CAS:Batefenterol (GSK961081) is a muscarinic antagonist and β2-agonist with high affinity (Ki: 1.4/1.3/3.7 nM).Fórmula:C40H42ClN5O7Pureza:97.94% - 98.4%Cor e Forma:SolidPeso molecular:740.24Bestim
CAS:Bestim is an immunomodulatory dipeptide that is synthetic.Fórmula:C16H19N3O5Pureza:99.76%Cor e Forma:SolidPeso molecular:333.34Ref: TM-T25146
1mg88,00€5mg172,00€10mg259,00€25mg425,00€50mg598,00€100mg810,00€200mg1.074,00€1mL*10mM (DMSO)182,00€VU0152099
CAS:VU0152099 is a potent and selective M4 mAChR allosteric potentiator(EC50 = 380 ± 93 nM).Fórmula:C18H17N3O3SPureza:98.46%Cor e Forma:SolidPeso molecular:355.41Adiphenine
CAS:Adiphenine is an inhibitor of nicotinic receptors.Fórmula:C20H25NO2Cor e Forma:SolidPeso molecular:311.42Rivanicline hemioxalate
Rivanicline hemioxalate is a selective α4β2 nicotinic receptor agonist (K i =26 nM), over 1,000x preference to α7 (K i =3.6 μM), with limited side effects.Fórmula:C12H16N2O4Pureza:98%Cor e Forma:SolidPeso molecular:207.23Simufilam dihydrochloride
CAS:Simufilam dihydrochloride is an oral, low-toxic FLNA activator for Alzheimer's research, restoring FLNA structure and function.Fórmula:C15H23Cl2N3OPureza:98.83%Cor e Forma:SolidPeso molecular:332.3Ref: TM-T9172
1mg52,00€5mg90,00€10mg143,00€25mg294,00€50mg380,00€100mg497,00€200mg655,00€1mL*10mM (DMSO)101,00€suvn-911
CAS:suvn-911 is a potent and selective antagonist of neuronal nicotinic acetylcholine α4β2 receptor (Ki = 1.5 nM) with antidepressant activity.Fórmula:C11H14Cl2N2OPureza:98.88%Cor e Forma:SolidPeso molecular:261.15Ref: TM-T9787
1mg67,00€5mg133,00€10mg205,00€25mg339,00€50mg482,00€100mg658,00€200mg888,00€1mL*10mM (DMSO)172,00€Coluracetam
CAS:Coluracetam (MKC-231)(MKC-231) is a Choline Uptake Enhancer.Fórmula:C19H23N3O3Pureza:99.96%Cor e Forma:SolidPeso molecular:341.4Aclidinium bromide
CAS:Aclidinium bromide (LAS-W 330) is a synthetic anticholinergic agent that is used as an inhalant for treatment of acute bronchospasm due to chronic bronchitis.
Fórmula:C26H30NO4S2·BrPureza:99.53% - 99.69%Cor e Forma:SolidPeso molecular:564.55Encenicline hydrochloride
CAS:Encenicline hydrochloride (EVP-6124 hydrochloride) is a new-type partial agonist of α7 neuronal nicotinic acetylcholine receptors (nAChRs).Fórmula:C16H17ClN2OS·HClPureza:98.34% - 99.85%Cor e Forma:SolidPeso molecular:357.3Pempidine HCl
CAS:Pempidine HCl, a nicotinic antagonist and former hypertension treatment, now mainly serves as a lab tool.Fórmula:C10H22ClNCor e Forma:SolidPeso molecular:191.74Piperidolate hydrochloride
CAS:Piperidolate hydrochloride, an antimuscarinic, reduces acetylcholine-induced intestinal spasms in rats and dogs.Fórmula:C21H26ClNO2Pureza:99.5%Cor e Forma:SolidPeso molecular:359.89Batefenterol Succinate
CAS:Batefenterol Succinate is a first-in-class inhaled bifunctional bronchodilator possessing muscarinic receptor antagonist and β2-adrenoceptor agonist properties.Fórmula:C44H48ClN5O11Cor e Forma:SolidPeso molecular:858.34VU0238441
CAS:VU0238441 is agonist of Muscarinic acetylcholine receptor M5 (human) with EC50 of 2.1μM.Fórmula:C16H9ClF3NO2Pureza:100%Cor e Forma:SolidPeso molecular:339.7Benzetimide hydrochloride
CAS:Benzetimide hydrochloride (R4929) is an antagonist of muscarinic acetylcholine receptor.treatment neuroleptic-induced parkinsonism.Fórmula:C23H27ClN2O2Pureza:99.32%Cor e Forma:Off-White PowderPeso molecular:398.93Oxyphencyclimine
CAS:Oxyphencyclimine is a muscarinic receptor antagonist (MRA) anticholinergic drug used to treat peptic ulcers.Fórmula:C20H28N2O3Cor e Forma:SolidPeso molecular:344.45(S)-UFR2709
CAS:(S)-UFR2709, a nAChR competitive antagonist, favors α4β2 over α7, reduces anxiety and alcohol use in rats.Fórmula:C13H17NO2Cor e Forma:SolidPeso molecular:219.284mAChR-IN-1 hydrochloride
CAS:mAChR-IN-1 hydrochloride is a potent muscarinic cholinergic receptor (mAChR) antagonist, with an IC50 of 17 Nm.Fórmula:C23H26ClIN2O2Pureza:99.87%Cor e Forma:SolidPeso molecular:524.82Ref: TM-T5655
1mg40,00€5mg90,00€10mg133,00€25mg227,00€50mg314,00€100mg393,00€200mg520,00€1mL*10mM (DMSO)95,00€Solifenacin
CAS:Solifenacin (YM905 free base) (YM905 free base) is a novel muscarinic receptor antagonist, its pKis for M1, M2 and M3 receptors is of 7.6, 6.9 and 8.0,Fórmula:C23H26N2O2Pureza:99.87%Cor e Forma:SolidPeso molecular:362.46LY2119620
CAS:LY2119620 is a specific, and allosteric agonist of human M2 and M4 muscarinic acetylcholine receptors.Fórmula:C19H24ClN5O3SPureza:99.7%Cor e Forma:SolidPeso molecular:437.94Pirmenol
CAS:Pirmenol is a new antiarrhythmic drugFórmula:C22H30N2OPureza:97.24%Cor e Forma:SolidPeso molecular:338.49VU0357017 hydrochloride
CAS:VU0357017 hydrochloride (ML071 hydrochloride) is highly selective M1 agonists act at an allosteric site to activate the receptor (EC50: 477 ± 172 nM; Pec50: 6.Fórmula:C18H28ClN3O3Pureza:99% - 99.97%Cor e Forma:SolidPeso molecular:369.89Darifenacin
CAS:Darifenacin (UK-88525) is a muscarinic receptor M3 antagonist with anticonvulsant activity and can be used to study urinary incontinence and overactive bladder.Fórmula:C28H30N2O2Pureza:99.78%Cor e Forma:SolidPeso molecular:426.55Ref: TM-T62320
2mg39,00€5mg58,00€10mg93,00€25mg152,00€50mg236,00€100mg356,00€200mg522,00€1mL*10mM (DMSO)64,00€Ilmetropium iodide
CAS:Ilmetropium iodide is a bronchodilator.Fórmula:C20H30INO3Pureza:98.45%Cor e Forma:SolidPeso molecular:459.36BNC210
CAS:BNC210 (IW-2143) is a α7 nAChR negative allosteric modulator. BNC210 has potent activity in animal models of anxiety and depression.Fórmula:C17H23N3O3Pureza:97.05% - >99.99%Cor e Forma:SolidPeso molecular:317.38Brompheniramine
CAS:Brompheniramine, an alkylamine antihistamine, targets H1 receptors (Kd=6.06nM) and has anticholinergic/depressant qualities. Blocks Ca/Na/hERG channels.Fórmula:C16H19BrN2Cor e Forma:SolidPeso molecular:319.24Harman hydrochloride
CAS:Harman hydrochloride triggers CYP1A1 gene via AhR, potentially causing mutations and cancer.Fórmula:C12H11ClN2Pureza:99.35%Cor e Forma:SolidPeso molecular:218.68Ursulcholic acid
CAS:Ursulcholic acid (Ursulcholic) is a water-soluble anticholinergic compound.Fórmula:C24H40O10S2Pureza:98%Cor e Forma:SolidPeso molecular:552.7Nor-benzetimide
CAS:Norbenzetimide, an organic compound, is prepared from benzetimide by catalytic transfer hydrogenolysis.Fórmula:C16H20N2O2Pureza:98.63%Cor e Forma:SolidPeso molecular:272.34Ref: TM-T22380
1mg72,00€5mg136,00€10mg197,00€25mg324,00€50mg452,00€100mg607,00€200mg810,00€1mL*10mM (DMSO)135,00€Nitrocaramiphen hydrochloride
CAS:Nitrocaramiphen hydrochloride is a selective M1 muscarinic antagonist and inhibits binding to sigma sites in brain.Fórmula:C18H27ClN2O4Pureza:99.74%Cor e Forma:SolidPeso molecular:370.87W-84 dibromide
CAS:W-84 dibromide (HDMPPA) is a M2-receptor selective modulator.Fórmula:C32H44Br2N4O4Pureza:95.56%Cor e Forma:SolidPeso molecular:708.52CCMI
CAS:CCMI (AVL-3288) is a potent and selective modulator of α7 nAChR-positive allosteric.Fórmula:C19H15Cl2N3O2Pureza:>99.99%Cor e Forma:SolidPeso molecular:388.25Glycopyrrolate
CAS:Glycopyrrolate: muscarinic antagonist, antispasmodic for GI issues, reduces salivation with anesthesia.Fórmula:C19H28BrNO3Pureza:99.41% - 99.64%Cor e Forma:SolidPeso molecular:398.33
