
AChR
Os inibidores do receptor de acetilcolina (AChR) são compostos que bloqueiam a atividade dos receptores de acetilcolina, essenciais para a neurotransmissão nos sistemas nervosos central e periférico. Os AChRs desempenham um papel vital na contração muscular, memória e funções cognitivas. Os inibidores de AChRs são usados para estudar condições como miastenia gravis, doença de Alzheimer e outros distúrbios neurológicos. Ao modular a atividade dos AChRs, esses inibidores podem ajudar a desvendar as complexidades da sinalização colinérgica no cérebro. Na CymitQuimica, oferecemos uma gama de inibidores de AChRs para apoiar sua pesquisa em neurociência, farmacologia e doenças neurodegenerativas.
Foram encontrados 575 produtos de "AChR"
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MC-Val-Cit-PAB
CAS:<p>MC-Val-Cit-PAB: cathepsin-cleavable ADC linker used in FDA-approved brentuximab vedotin.</p>Fórmula:C28H40N6O7Pureza:98.24%Cor e Forma:SolidPeso molecular:572.65Revefenacin
CAS:<p>Revefenacin (TD-4208) is a mAChR antagonist has a high affinity on M3 receptor( Ki : 0.18 nM),and potentially useful for the treatment of respiratory disease.</p>Fórmula:C35H43N5O4Pureza:98.12%Cor e Forma:SolidPeso molecular:597.75Nitrocaramiphen hydrochloride
CAS:<p>Nitrocaramiphen hydrochloride is a selective M1 muscarinic antagonist and inhibits binding to sigma sites in brain.</p>Fórmula:C18H27ClN2O4Pureza:99.74%Cor e Forma:SolidPeso molecular:370.87Piperidolate
CAS:<p>Piperidolate inhibits intestinal cramp induced by acetylcholine</p>Fórmula:C21H25NO2Pureza:98.45%Cor e Forma:SolidPeso molecular:323.43PNU-282987 S enantiomer free base
CAS:<p>PNU-282987 S enantiomer free base is an agonist of α7 nicotinic acetylcholine receptor (α7 nAChR).</p>Fórmula:C14H17ClN2OPureza:99.74%Cor e Forma:SolidPeso molecular:264.75VU 0238429
CAS:<p>VU 0238429 (SCR-1481B1) is positive allosteric modulator of muscarinic acetylcholine receptor subtype 5 (mAChR5 or M5)( EC50 : 1.16 μM).</p>Fórmula:C17H12F3NO4Pureza:>99.99%Cor e Forma:SolidPeso molecular:351.28Glycopyrrolate
CAS:<p>Glycopyrrolate: muscarinic antagonist, antispasmodic for GI issues, reduces salivation with anesthesia.</p>Fórmula:C19H28BrNO3Pureza:99.41% - 99.64%Cor e Forma:SolidPeso molecular:398.33CCMI
CAS:<p>CCMI (AVL-3288) is a potent and selective modulator of α7 nAChR-positive allosteric.</p>Fórmula:C19H15Cl2N3O2Pureza:>99.99%Cor e Forma:SolidPeso molecular:388.25W-84 dibromide
CAS:<p>W-84 dibromide (HDMPPA) is a M2-receptor selective modulator.</p>Fórmula:C32H44Br2N4O4Pureza:95.56%Cor e Forma:SolidPeso molecular:708.52Prifinium bromide
CAS:<p>Prifinium bromide is a quaternary ammon antimuscarinic. It inhibits hyperkinesia of the digestive organs and urinary tract and has a spasmolytic action.</p>Fórmula:C22H28BrNPureza:97.99%Cor e Forma:SolidPeso molecular:386.37Nor-benzetimide
CAS:<p>Norbenzetimide, an organic compound, is prepared from benzetimide by catalytic transfer hydrogenolysis.</p>Fórmula:C16H20N2O2Pureza:98.63%Cor e Forma:SolidPeso molecular:272.34PNU-120596
CAS:<p>PNU-120596 (NSC-216666) is a positive allosteric modulator of α7 nAChR with EC50 of 216 nM.</p>Fórmula:C13H14ClN3O4Pureza:99.82%Cor e Forma:SolidPeso molecular:311.72MC-Val-Cit-PABC-PNP
CAS:<p>MC-Val-Cit-PABC-PNP, also known as Mc-Val-Cit-PABC-PNP, is a cathepsin cleavable ADC peptide linker.</p>Fórmula:C35H43N7O11Pureza:97.2% - 98.055%Cor e Forma:SolidPeso molecular:737.76Blarcamesine
CAS:<p>Blarcamesine (AVex-73) is a muscarinic M1 agonist potentially for the treatment of Alzheimer's disease.</p>Fórmula:C19H23NOPureza:99.87%Cor e Forma:SolidPeso molecular:281.39(S)-UFR2709
CAS:<p>(S)-UFR2709, a nAChR competitive antagonist, favors α4β2 over α7, reduces anxiety and alcohol use in rats.</p>Fórmula:C13H17NO2Cor e Forma:SolidPeso molecular:219.284Mc-Val-Ala-PAB
CAS:<p>Mc-Val-Ala-PAB, an effective linker, is utilized in antibody-drug-conjugate (ADC).</p>Fórmula:C25H34N4O6Pureza:98.34% - 99.24%Cor e Forma:SolidPeso molecular:486.56PHA 568487
CAS:<p>PHA 568487: α-7 nAChR agonist, rapid brain uptake, lessens oxidative stress & neuroinflammation.</p>Fórmula:C20H24N2O7Cor e Forma:SolidPeso molecular:404.419VU0152099
CAS:<p>VU0152099 is a potent and selective M4 mAChR allosteric potentiator(EC50 = 380 ± 93 nM).</p>Fórmula:C18H17N3O3SPureza:98.46%Cor e Forma:SolidPeso molecular:355.41Bestim
CAS:<p>Bestim is an immunomodulatory dipeptide that is synthetic.</p>Fórmula:C16H19N3O5Pureza:99.76%Cor e Forma:SolidPeso molecular:333.34Oxyphenonium bromide
CAS:<p>Oxyphenonium bromide is an anticholinergic used to study and treat ulcers and relieve visceral spasms.</p>Fórmula:C21H34BrNO3Pureza:98.96%Cor e Forma:SolidPeso molecular:428.404Nitrobenzylthioinosine
CAS:<p>Nitrobenzylthioinosine (NBMPR) is an inhibitor of ENT1 transporter that binds to ENT1 transporter with high affinity.</p>Fórmula:C17H17N5O6SPureza:99.69% - 99.74%Cor e Forma:Off-White SolidPeso molecular:419.41Monepantel
CAS:<p>Monepantel (AAD1566) is an organic anthelmintic and an antagonist of nAChRs from roundworms and esophageostomy.</p>Fórmula:C20H13F6N3O2SPureza:99.83%Cor e Forma:White PowderPeso molecular:473.39Velufenacin
CAS:<p>Velufenacin is an antagonist of muscarinic receptor[1].</p>Fórmula:C19H20ClFN2O2Pureza:99.65%Cor e Forma:SolidPeso molecular:362.83Pentoxyverine
CAS:<p>Pentoxyverine (Carbetapentan) is an orally available cough suppressant, an antagonist of muscarinic receptor M1 and an agonist of the σ1 receptor.</p>Fórmula:C20H31NO3Pureza:97.11%Cor e Forma:SolidPeso molecular:333.47Xanomeline tartrate
CAS:<p>Xanomeline tartrate (LY 246708 tartrate) 是 M1和 M4 mAChR 激动剂,具有抗精神病样活性,可改善认知,可用于研究精神分裂症和阿尔茨海默病。</p>Fórmula:C18H29N3O7SPureza:99.19%Cor e Forma:SolidPeso molecular:431.5AF-710B
CAS:<p>AF710B is an enantiomer of AF710. AF-710B is also a sigma and M1 muscarinic receptors agonist.</p>Fórmula:C20H27N3OSPureza:98.62% - 99.89%Cor e Forma:SolidPeso molecular:357.51Mepenzolate Bromide
CAS:<p>Mepenzolate Bromide (Colibantil) is a muscarinic antagonist used to treat gastrointestinal conditions.</p>Fórmula:C21H26BrNO3Pureza:95.73% - 99.21%Cor e Forma:SolidPeso molecular:420.34Pipecuronium bromide
CAS:<p>Pipecuronium bromide (RGH-1106) is an nAChR antagonist that also acts as a non-depolarising steroidal neuromuscular blocker that causes muscle relaxation.</p>Fórmula:C35H62Br2N4O4Pureza:>99.99%Cor e Forma:PowderPeso molecular:762.7Varenicline
CAS:<p>Varenicline (CP 526555) is a selective partial agonist of the α4β2 nAChR and a full agonist of the α3β4 nAChR and α7 nAChR.</p>Fórmula:C13H13N3Pureza:99.76%Cor e Forma:SolidPeso molecular:211.26Atropine hydrobromide
CAS:<p>Atropine hydrobromide is a biochemical.</p>Fórmula:C17H24BrNO3Cor e Forma:SolidPeso molecular:370.28Anatabine dicitrate
<p>Anatabine dicitrate is a tobacco alkaloid that can cross the blood-brain barrier.</p>Fórmula:C22H28N2O14Pureza:98%Cor e Forma:SolidPeso molecular:544.46Pyrantel
CAS:<p>Pyrantel: Nicotinic agonist; causes spastic paralysis in nematodes by depolarizing block.</p>Fórmula:C11H14N2SPureza:98%Cor e Forma:Crystals From Methanol Yellowish Crystalline PowderPeso molecular:206.31Flavoxate
CAS:<p>Flavoxate is an anticholinergic with antimuscarinic effects.</p>Fórmula:C24H25NO4Cor e Forma:SolidPeso molecular:391.46(±)-Atropine-d3 (N-methyl-d3)
CAS:(±)-Atropine-d3 (N-methyl-d3) is a deuterated compound of (±)-Atropine. (±)-Atropine has a CAS number of 51-55-8. Atropine Sulfate is the sulfate salt of atropine, a naturally-occurring alkaloid isolated from the plant Atropa belladonna. Atropine functions as a sympathetic, competitive antagonist of muscarinic cholinergic receptors, thereby abolishing the effects of parasympathetic stimulation.Fórmula:C17H20D3NO3Peso molecular:292.39Oxantel
CAS:<p>Oxantel is a fumarate reductase inhibitor with anthelmintic activity.</p>Fórmula:C13H16N2OPureza:98%Cor e Forma:SolidPeso molecular:216.28Aprofene
CAS:<p>Aprofene blocks acetylcholine receptors, used for peptic ulcers, endarteritis, cholecystitis, and colitis.</p>Fórmula:C21H27NO2Cor e Forma:SolidPeso molecular:325.44Catestatin
CAS:Non-competitive inhibitor of nicotinic receptors; blocks cationic signalling and catecholamine release; stimulates histamine release. IC50 ~200-250nM.Fórmula:C107H173N37O26SPureza:98%Cor e Forma:SolidPeso molecular:2425.84Dianicline dihydrochloride
CAS:<p>Dianicline dihydrochloride is a partial agonist of α4β2 nicotinic acetylcholine receptor. It increases cessation rates in a dose-dependent manner.</p>Fórmula:C13H16N2OPureza:98%Cor e Forma:SolidPeso molecular:216.28Biperiden lactate
CAS:<p>Biperiden lactate is a biochemical.</p>Fórmula:C24H35NO4Cor e Forma:SolidPeso molecular:401.54VU0029767
CAS:<p>VU0029767 is an allosteric enhancer of the M1 muscarinic receptor, capable of modulating the receptor's activity. This compound enhances M1 receptor activity by increasing agonist affinity. However, VU0029767 demonstrates distinct characteristics from other compounds, particularly under varying experimental conditions such as its interaction with mutated M1 receptors and its effects on downstream signaling pathways.</p>Fórmula:C21H21N3O3Cor e Forma:SolidPeso molecular:363.41Azacyclonol hydrochloride
CAS:<p>Azacyclonol hydrochloride can be used in the treatment of chronic schizophrenia.</p>Fórmula:C18H22ClNOCor e Forma:Off White Crystalline PowderPeso molecular:303.83Diphenidol
CAS:<p>Diphenidol, a muscarinic antagonist, is employed as an antivertigo and antiemetic agent.</p>Fórmula:C21H27NOCor e Forma:Needles From Petroleum Ether SolidPeso molecular:309.45Sulindac sulfide
CAS:<p>Sulindac sulfide: NSAID targeting COX-1, inhibits Ras-Raf-1 and gamma-secretase (IC50: 20.2 μM), active sulinic acid metabolite.</p>Fórmula:C20H17FO2SPureza:99.35%Cor e Forma:SolidPeso molecular:340.41N-0861 racemate
CAS:<p>N-0861 racemate is the racemate of N-0861.</p>Fórmula:C13H17N5Pureza:98%Cor e Forma:SolidPeso molecular:243.31Sulfoxaflor
CAS:<p>Sulfoxaflor (GF 2032) is an agonist of nAChR1 and nAChR2 subtypes and a systemic insecticide. Cost-effective and quality-assured.</p>Fórmula:C10H10F3N3OSPureza:99.56%Cor e Forma:SolidPeso molecular:277.27Sch412348
CAS:<p>Sch412348: potent A2A receptor antagonist, Ki=0.6 nM, >1000-fold selectivity vs. other adenosine receptors.</p>Fórmula:C22H21F2N9OPureza:98%Cor e Forma:SolidPeso molecular:465.46SR 16584
CAS:<p>α3β4 nAChR antagonist</p>Fórmula:C17H22N2OPureza:99.84%Cor e Forma:SolidPeso molecular:270.37Tarafenacin
CAS:<p>Tarafenacin is a highly selective M3 muscarinic receptor antagonist (Ki= 0.19 nM), ~200 fold selectivity over the M2 receptor.</p>Fórmula:C21H20F4N2O2Pureza:98%Cor e Forma:SolidPeso molecular:408.39Meseclazone
CAS:<p>Meseclazone has anti-inflammatory, analgesic, and antipyretic activity. Meseclazone shows inhibitory potency of secondary phase ADP aggregation.</p>Fórmula:C11H10ClNO3Pureza:98%Cor e Forma:SolidPeso molecular:239.654-DAMP
CAS:<p>4-DAMP (4-DAMP methiodide) is a selective muscarinic M1 and M3 subtype receptor antagonist used in the study of allergic rhinitis and cardiovascular disease.</p>Fórmula:C21H26INO2Pureza:98%Cor e Forma:SolidPeso molecular:451.34mAChr-in-1
CAS:<p>mAChR-IN-1 is muscarinic cholinergic receptor(mAChR) antagonist (IC50=17 nM).</p>Fórmula:C23H25IN2O2Pureza:98%Cor e Forma:SolidPeso molecular:488.36Darenzepine
CAS:<p>Darenzepine is a muscarinic receptor inhibitor.</p>Fórmula:C21H21N3O2Pureza:99.87%Cor e Forma:SolidPeso molecular:347.41UB 165 fumarate
CAS:<p>UB 165 fumarate is a nAChR agonist, α4β2 partial, α3β2 full, with a 0.27 nM Ki for [3H]-nicotine in rat brain.</p>Fórmula:C17H19ClN2O4Pureza:99.72%Cor e Forma:SolidPeso molecular:350.8CDD0102
CAS:<p>CDD0102 is a potent agonist of M1 Muscarinic receptor.</p>Fórmula:C8H12N4OPureza:98%Cor e Forma:SolidPeso molecular:180.215-Iodo-A-85380 dihydrochloride
CAS:<p>α4β2 and α6β2 nicotinic acetylcholine receptors agonist</p>Fórmula:C9H13Cl2IN2OPureza:98%Cor e Forma:SolidPeso molecular:363.02Dimethyl-W84 (dibromide)
CAS:<p>Dimethyl-W84, selective M2 muscarinic receptor modulator; slows N-methylscopolamine release, EC50=3 nM.</p>Fórmula:C34H48Br2N4O4Cor e Forma:SolidPeso molecular:736.59LY 2087101
CAS:<p>Allosteric potentiator of α7, α4β2 and α4β4 nAChRs</p>Fórmula:C15H11FN2OS2Pureza:98%Cor e Forma:SolidPeso molecular:318.39AR-R 17779 hydrochloride
CAS:<p>AR-R17779 hydrochloride: potent α7 nAChR agonist; K i : 92 nM (α7), 16,000 nM (α4β2); enhances rat cognition; anxiolytic; anti-inflammatory.</p>Fórmula:C9H15ClN2O2Cor e Forma:SolidPeso molecular:218.68Elucaine
CAS:Elucaine is an antagonist of the muscarinic acetylcholine receptor. It has anti-ulcerative activity.Fórmula:C19H23NO2Pureza:98%Cor e Forma:SolidPeso molecular:297.39(R,R)-Glycopyrrolate
CAS:<p>(R,R)-Glycopyrrolate is an agent of anticholinergic, has the ability to reduce the frequency of drooling in vivo with developmental disabilities.</p>Fórmula:C19H28BrNO3Pureza:98%Cor e Forma:SolidPeso molecular:398.34SIB 1508Y maleate
CAS:<p>neuronal nicotinic ACh receptor agonist</p>Fórmula:C16H18N2O4Pureza:98%Cor e Forma:SolidPeso molecular:302.33LRE1
CAS:<p>LRE1 is a specific and allosteric soluble adenylyl cyclase inhibitor.</p>Fórmula:C12H13ClN4SPureza:>99.99%Cor e Forma:SolidPeso molecular:280.78Terodiline
CAS:<p>Terodiline is an orally available selective muscarinic M1 receptor and calcium channel antagonist for the study of diseases caused by abnormal bladder function.</p>Fórmula:C20H27NPureza:98.20% - 99.59%Cor e Forma:SolidPeso molecular:281.44Methacholine bromide
CAS:<p>Methacholine bromide is a potent M3 agonist for diagnosing asthma by identifying bronchial hyperresponsiveness.</p>Fórmula:C8H18BrNO2Cor e Forma:SolidPeso molecular:240.141Nuvenzepine
CAS:<p>Nuvenzepine is an antagonist of mAChR. It has the potential for gastrospasm treatment.</p>Fórmula:C19H20N4O2Pureza:98%Cor e Forma:SolidPeso molecular:336.39DA 4626
CAS:<p>DA 4626 is an H2-receptor antagonist with KB values akin to those in standard assays.</p>Fórmula:C14H18N4Pureza:98%Cor e Forma:SolidPeso molecular:242.32Telenzepine
CAS:<p>Telenzepine is a potent and selective M1 antimuscarinic.</p>Fórmula:C19H22N4O2SPureza:98%Cor e Forma:SolidPeso molecular:370.47AC260584
CAS:AC260584 is an M1 muscarinic receptor allosteric agonist (pEC50: 7.6).Fórmula:C20H29FN2O2Cor e Forma:SolidPeso molecular:348.45Neramexane Mesylate
CAS:<p>Neramexane: NMDA & nicotinic receptor blocker with neuroprotective, antidepressant, and cognitive-enhancing effects.</p>Fórmula:C12H27NO3SPureza:98%Cor e Forma:SolidPeso molecular:265.41Chlorisondamine diiodide
CAS:<p>long lasting nicotinic antagonist</p>Fórmula:C14H20Cl4I2N2Cor e Forma:SolidPeso molecular:611.94ML381
CAS:<p>ML381 is a M5-orthosteric antagonist with a high selectivity of muscarinic subtype.</p>Fórmula:C21H21N3O4Cor e Forma:SolidPeso molecular:379.41ML169
CAS:<p>ML169 is a selective and brain penetrant M1 positive allosteric modulator (PAM).</p>Fórmula:C21H17BrFN3O4SPureza:98%Cor e Forma:SolidPeso molecular:506.34Zamifenacin
CAS:<p>Zamifenacin obviously decreases colonic motility in irritable bowel syndrome. Zamifenacin is an effective gut-selective muscarinic M3 receptor antagonist.</p>Fórmula:C27H29NO3Pureza:98%Cor e Forma:SolidPeso molecular:415.52BNC375
CAS:<p>BNC375 is a α7 nAChRs type I positive allosteric modulator (EC50: 1.9 μM).</p>Fórmula:C19H23ClN2O3SPureza:98%Cor e Forma:SolidPeso molecular:394.92(R,R)-Reboxetine mesylate
CAS:<p>(R,R)-Reboxetine mesylate: Antidepressant, high bioavailability, (R,R) enantiomer, selective for noradrenaline, low toxicity.</p>Fórmula:C20H27NO6SCor e Forma:SolidPeso molecular:409.5M1 ligand 1
CAS:<p>Compound 3b-b: N-desmethyl arecoline derivative, muscarinic M1 ligand, potential PET radiotracer.</p>Fórmula:C20H21NO2Cor e Forma:SolidPeso molecular:307.39Benzatropine
CAS:<p>Benzatropine: Central muscarinic blocker, inhibits dopamine uptake, treats Parkinson's symptoms.</p>Fórmula:C21H25NOPureza:98%Cor e Forma:SolidPeso molecular:307.43Muscarine iodide
CAS:<p>Muscarinic acetylcholine receptor agonist</p>Fórmula:C9H20INO2Pureza:98%Cor e Forma:SolidPeso molecular:301.17Tridihexethyl chloride
CAS:<p>Tridihexethyl is an anticholinergic, antimuscarinic, and antispasmolytic drug, which can be used to treat acquired nystagmus or peptic ulcer disease.</p>Fórmula:C21H36ClNOCor e Forma:SolidPeso molecular:353.97TC 2559 difumarate
CAS:<p>partial agonist of α4β2 nicotinic acetylcholine receptor</p>Fórmula:C12H18N2OC4H404Pureza:98%Cor e Forma:SolidPeso molecular:380.39TC299423
CAS:<p>TC299423 is a novel agonist for nicotinic acetylcholine receptors (nAChRs). TC299423 modestly selectively targets α6β2 subtype.</p>Fórmula:C11H15N3Cor e Forma:SolidPeso molecular:189.26SM-21 maleate
CAS:<p>Increases release of acetylcholine,σ2 antagonist</p>Fórmula:C22H28ClNO7Pureza:98%Cor e Forma:SolidPeso molecular:453.91TC 1698 dihydrochloride
CAS:<p>nicotinic α7 receptor agonist</p>Fórmula:C13H18N2Pureza:98%Cor e Forma:SolidPeso molecular:202.3Beperidium iodide
CAS:<p>Beperidium iodide is a competitive antagonist of the acetylcholine receptor (pA2: 7.93).</p>Fórmula:C23H34IN3O3Cor e Forma:SolidPeso molecular:527.44WIN 62,577
CAS:<p>WIN 62,577 is a allosteric antagonist of mAChR.</p>Fórmula:C29H31N3OPureza:98%Cor e Forma:SolidPeso molecular:437.58Benzamide Derivative 1
CAS:<p>Benzamide Derivative 1 Benzamide derivative with gastrokinetic activity.Benzamide Derivative 1 can be used in the study of gastrointestinal diseases.</p>Fórmula:C22H34ClN3O3Pureza:>99.99%Cor e Forma:SolidPeso molecular:423.98Alvameline
CAS:<p>Alvameline (Lu25-109) is a partial M1 agonist. Alvameline (Lu25-109) also is a M2/M3 antagonist.</p>Fórmula:C9H15N5Pureza:98%Cor e Forma:SolidPeso molecular:193.25Muscarine chloride
CAS:<p>Muscarine chloride is a toxic alkaloid found in Amanita muscaria and other fungi of the Inocybe species.</p>Fórmula:C9H20ClNO2Cor e Forma:SolidPeso molecular:209.71Quifenadine
CAS:<p>Quifenadine, an H1-histamine receptor blocker, has antiarrhythmic properties.</p>Fórmula:C20H23NOPureza:98%Cor e Forma:SolidPeso molecular:293.4DAU 5884 hydrochloride
CAS:<p>muscarinic M3 receptor antagonist</p>Fórmula:C17H22ClN3O3Pureza:98%Cor e Forma:SolidPeso molecular:351.83Nelonicline
CAS:<p>Nelonicline is a selective agonist of neuronal nicotinic receptors.</p>Fórmula:C17H19N3OSPureza:98%Cor e Forma:SolidPeso molecular:313.42BTM-1086
CAS:<p>BTM-1086 is a potent gastric secretory inhibitor and an anti-ulcer agent.</p>Fórmula:C21H25N3OSPureza:98%Cor e Forma:SolidPeso molecular:367.51CP-601932
CAS:<p>CP-601932 (free base) is a selective base α( 4) β( 2) Nicotinic acetylcholine receptor agonist.</p>Fórmula:C12H12F3NCor e Forma:SolidPeso molecular:227.23Eucatropine
CAS:<p>Eucatropine, an anticholinergic agent, acts as a potent inhibitor of the muscarinic acetylcholine receptor (mAChR) with an IC 50 value of 0.583 μM.</p>Fórmula:C17H25NO3Cor e Forma:SolidPeso molecular:291.39Thiochrome
CAS:<p>Thiochrome is a selective enhancer of M4 muscarinic receptor of acetylcholine (ACh) affinity.</p>Fórmula:C12H14N4OSPureza:98%Cor e Forma:SolidPeso molecular:262.33VU0090157
CAS:<p>VU0090157, a novel allosteric potentiators of M1 muscarinic receptor, may provide novel treatments for schizophrenia and Alzheimer's disease.</p>Fórmula:C19H21N3O7Pureza:98%Cor e Forma:SolidPeso molecular:403.39S-(+)-Mecamylamine hydrochloride
CAS:<p>Dexmecamylamine( TC-5214, NIH-11008) is used as a nicotinic channel modulator with antidepressant activity.</p>Fórmula:C11H22ClNCor e Forma:SolidPeso molecular:203.75T761-0184
CAS:<p>T761-0184 is a potent antagonist of α7 nicotinic receptor (nAChR) [1].</p>Fórmula:C16H20FN3OCor e Forma:SolidPeso molecular:289.35Revatropate
CAS:<p>Revatropate, a selective muscarinic antagonist, is an antimuscarinic drug.</p>Fórmula:C19H27NO4SCor e Forma:SolidPeso molecular:365.49Rispenzepine
CAS:<p>Rispenzepine, a novel mAChRs M1/M3 antagonist, treats immune, infections, and respiratory issues.</p>Fórmula:C19H20N4O2Pureza:98%Cor e Forma:SolidPeso molecular:336.39

