AChR
Os inibidores do receptor de acetilcolina (AChR) são compostos que bloqueiam a atividade dos receptores de acetilcolina, essenciais para a neurotransmissão nos sistemas nervosos central e periférico. Os AChRs desempenham um papel vital na contração muscular, memória e funções cognitivas. Os inibidores de AChRs são usados para estudar condições como miastenia gravis, doença de Alzheimer e outros distúrbios neurológicos. Ao modular a atividade dos AChRs, esses inibidores podem ajudar a desvendar as complexidades da sinalização colinérgica no cérebro. Na CymitQuimica, oferecemos uma gama de inibidores de AChRs para apoiar sua pesquisa em neurociência, farmacologia e doenças neurodegenerativas.
Foram encontrados 612 produtos de "AChR"
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Coluracetam
CAS:Coluracetam (MKC-231)(MKC-231) is a Choline Uptake Enhancer.Fórmula:C19H23N3O3Pureza:99.96%Cor e Forma:SolidPeso molecular:341.4Aclidinium bromide
CAS:<p>Aclidinium bromide (LAS-W 330) is a synthetic anticholinergic agent that is used as an inhalant for treatment of acute bronchospasm due to chronic bronchitis.</p>Fórmula:C26H30NO4S2·BrPureza:99.53% - 99.69%Cor e Forma:SolidPeso molecular:564.55Encenicline hydrochloride
CAS:Encenicline hydrochloride (EVP-6124 hydrochloride) is a new-type partial agonist of α7 neuronal nicotinic acetylcholine receptors (nAChRs).Fórmula:C16H17ClN2OS·HClPureza:98.34% - 99.85%Cor e Forma:SolidPeso molecular:357.3suvn-911
CAS:suvn-911 is a potent and selective antagonist of neuronal nicotinic acetylcholine α4β2 receptor (Ki = 1.5 nM) with antidepressant activity.Fórmula:C11H14Cl2N2OPureza:98.88%Cor e Forma:SolidPeso molecular:261.15α-Conotoxin MII acetate
α-Conotoxin MII acetate is a 16-amino acid peptide from the venom of the marine snail Conus magus.Fórmula:C69H107N23O24S4Pureza:94.82% - 97.79%Cor e Forma:SolidPeso molecular:1770.99BNC210
CAS:<p>BNC210 (IW-2143) is a α7 nAChR negative allosteric modulator. BNC210 has potent activity in animal models of anxiety and depression.</p>Fórmula:C17H23N3O3Pureza:97.05% - >99.99%Cor e Forma:SolidPeso molecular:317.38(S)-UFR2709
CAS:(S)-UFR2709, a nAChR competitive antagonist, favors α4β2 over α7, reduces anxiety and alcohol use in rats.Fórmula:C13H17NO2Cor e Forma:SolidPeso molecular:219.284Oxyphencyclimine
CAS:Oxyphencyclimine is a muscarinic receptor antagonist (MRA) anticholinergic drug used to treat peptic ulcers.Fórmula:C20H28N2O3Cor e Forma:SolidPeso molecular:344.45mAChR-IN-1 hydrochloride
CAS:mAChR-IN-1 hydrochloride is a potent muscarinic cholinergic receptor (mAChR) antagonist, with an IC50 of 17 Nm.Fórmula:C23H26ClIN2O2Pureza:99.87%Cor e Forma:SolidPeso molecular:524.82Benzetimide hydrochloride
CAS:<p>Benzetimide hydrochloride (R4929) is an antagonist of muscarinic acetylcholine receptor.treatment neuroleptic-induced parkinsonism.</p>Fórmula:C23H27ClN2O2Pureza:99.32%Cor e Forma:Off-White PowderPeso molecular:398.93Pirmenol
CAS:Pirmenol is a new antiarrhythmic drugFórmula:C22H30N2OPureza:97.24%Cor e Forma:SolidPeso molecular:338.49LY2119620
CAS:LY2119620 is a specific, and allosteric agonist of human M2 and M4 muscarinic acetylcholine receptors.Fórmula:C19H24ClN5O3SPureza:99.7%Cor e Forma:SolidPeso molecular:437.94Ilmetropium iodide
CAS:<p>Ilmetropium iodide is a bronchodilator.</p>Fórmula:C20H30INO3Pureza:98.45%Cor e Forma:SolidPeso molecular:459.36Darifenacin
CAS:Darifenacin (UK-88525) is a muscarinic receptor M3 antagonist with anticonvulsant activity and can be used to study urinary incontinence and overactive bladder.Fórmula:C28H30N2O2Pureza:99.78%Cor e Forma:SolidPeso molecular:426.55Brompheniramine
CAS:<p>Brompheniramine, an alkylamine antihistamine, targets H1 receptors (Kd=6.06nM) and has anticholinergic/depressant qualities. Blocks Ca/Na/hERG channels.</p>Fórmula:C16H19BrN2Cor e Forma:SolidPeso molecular:319.24DMAB-anabaseine dihydrochloride
CAS:<p>DMAB-anabaseine dihydrochloride (N,N-dimethyl-4-[(E)-(6-pyridin-3-yl-3,4-dihydro-2H-pyridin-5-ylidene)methyl]aniline;dihydrochloride) is an α7-containing</p>Fórmula:C19H23Cl2N3Pureza:99.91%Cor e Forma:SolidPeso molecular:364.31Ethyl (triphenylphosphoranylidene) acetate
CAS:<p>Ethyl (triphenylphosphoranylidene) acetate ((Carbethoxymethylene)triphenylphosphorane) may act as an cholinesterase inhibitor that inhibits AChE and BChE.</p>Fórmula:C22H21O2PPureza:97.985%Cor e Forma:White Or Slight Yellow PowderPeso molecular:348.37Nor-benzetimide
CAS:Norbenzetimide, an organic compound, is prepared from benzetimide by catalytic transfer hydrogenolysis.Fórmula:C16H20N2O2Pureza:98.63%Cor e Forma:SolidPeso molecular:272.34Ursulcholic acid
CAS:Ursulcholic acid (Ursulcholic) is a water-soluble anticholinergic compound.Fórmula:C24H40O10S2Pureza:98%Cor e Forma:SolidPeso molecular:552.7W-84 dibromide
CAS:<p>W-84 dibromide (HDMPPA) is a M2-receptor selective modulator.</p>Fórmula:C32H44Br2N4O4Pureza:95.56%Cor e Forma:SolidPeso molecular:708.52
