AChR
Os inibidores do receptor de acetilcolina (AChR) são compostos que bloqueiam a atividade dos receptores de acetilcolina, essenciais para a neurotransmissão nos sistemas nervosos central e periférico. Os AChRs desempenham um papel vital na contração muscular, memória e funções cognitivas. Os inibidores de AChRs são usados para estudar condições como miastenia gravis, doença de Alzheimer e outros distúrbios neurológicos. Ao modular a atividade dos AChRs, esses inibidores podem ajudar a desvendar as complexidades da sinalização colinérgica no cérebro. Na CymitQuimica, oferecemos uma gama de inibidores de AChRs para apoiar sua pesquisa em neurociência, farmacologia e doenças neurodegenerativas.
Foram encontrados 619 produtos de "AChR"
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Dronedarone
CAS:Dronedarone (SR 33589) is an amiodarone analogue which has an effective and promising treatment for Atrial fibrillation.Fórmula:C31H44N2O5SPureza:98.85% - 99.99%Cor e Forma:SolidPeso molecular:556.76Pempidine
CAS:Pempidine (1,2,2,6,6-Pentamethylpiperidine) is a nicotinic antagonist, has been used as a ganglionic blocker in the treatment of hypertension.Fórmula:C10H21NPureza:98.18% - 99.28%Cor e Forma:Colorless - Light Yellow Clear LiquidPeso molecular:155.28Dinotefuran
CAS:Dinotefuran (MTI-446), a neonicotinoid insecticide, targets pests by blocking their nervous system.Fórmula:C7H14N4O3Pureza:99.89%Cor e Forma:White Crystalline PowderPeso molecular:202.21Sofpironium bromide
CAS:Sofpironium bromide (BBI4000) belongs to a class of drugs called anticholinergics, which exert their effect by blocking the action of acetylcholine.Fórmula:C22H32BrNO5Pureza:98.85%Cor e Forma:SolidPeso molecular:470.4Simufilam dihydrochloride
CAS:Simufilam dihydrochloride is an oral, low-toxic FLNA activator for Alzheimer's research, restoring FLNA structure and function.Fórmula:C15H23Cl2N3OPureza:98.83%Cor e Forma:SolidPeso molecular:332.3Varenicline Tartrate
CAS:<p>Varenicline Tartrate (CP 526555-18) is a benzazepine derivative that functions as an ALPHA4/BETA2 NICOTINIC RECEPTOR partial agonist.</p>Fórmula:C13H13N3·C4H6O6Pureza:98.23% - 98.32%Cor e Forma:Tan SolidPeso molecular:361.35JHU37152
CAS:JHU37152 is a DREADD agonist; Ki: 1.8 nM at hM3Dq, 8.7 nM at hM4Di; EC50: 5 nM (hM3Dq), 0.5 nM (hM4Di) in HEK-293 cell assays.Fórmula:C19H20ClFN4Pureza:99.72%Cor e Forma:SolidPeso molecular:358.84Clothianidin
CAS:Clothianidin (TI 435), an insecticide, stimulates nAChR as acetylcholine agonist, not AChE inhibitor.Fórmula:C6H8ClN5O2SPureza:99.71% - 99.87%Cor e Forma:Solid PowderPeso molecular:249.68Syn-Ake acetate
CAS:Syn-Ake acetate (Dipeptide diaminobutyroyl benzylamide) is a muscarinic acetylcholine receptor antagonist.Fórmula:C19H29N5O3·2(C2H4O2)Pureza:99.60%Cor e Forma:SolidPeso molecular:495.58α-Conotoxin MII acetate
α-Conotoxin MII acetate is a 16-amino acid peptide from the venom of the marine snail Conus magus.Fórmula:C69H107N23O24S4Pureza:94.82% - 97.79%Cor e Forma:SolidPeso molecular:1770.99VU0357017 hydrochloride
CAS:VU0357017 hydrochloride (ML071 hydrochloride) is highly selective M1 agonists act at an allosteric site to activate the receptor (EC50: 477 ± 172 nM; Pec50: 6.Fórmula:C18H28ClN3O3Pureza:99% - 99.97%Cor e Forma:SolidPeso molecular:369.89Piperidolate hydrochloride
CAS:Piperidolate hydrochloride, an antimuscarinic, reduces acetylcholine-induced intestinal spasms in rats and dogs.Fórmula:C21H26ClNO2Pureza:99.5%Cor e Forma:SolidPeso molecular:359.89KH7
CAS:KH7 is a soluble inhibitor of adenylyl cyclase (sAC)-specific.Fórmula:C17H15BrN4O2SPureza:98.43%Cor e Forma:SolidPeso molecular:419.3Batefenterol
CAS:Batefenterol (GSK961081) is a muscarinic antagonist and β2-agonist with high affinity (Ki: 1.4/1.3/3.7 nM).Fórmula:C40H42ClN5O7Pureza:97.94% - 98.4%Cor e Forma:SolidPeso molecular:740.24Anisotropine Methylbromide
CAS:Anisotropine Methylbromide is an anticholinergic agent and has been used for relief of gastrointestinal spasm and for the suppression of gastric acid secretion.Fórmula:C17H32BrNO2Pureza:99.73%Cor e Forma:Crystals From Acetone SolidPeso molecular:362.35Cyclodrine hydrochloride
CAS:Cyclodrine hydrochloride is a dual cholinergic muscarinic receptor (mAChR) and nicotinic receptor (nAChR) antagonist that can be used in the study ofFórmula:C19H30ClNO3Pureza:98.59%Cor e Forma:SolidPeso molecular:355.9Umeclidinium bromide
CAS:Umeclidinium bromide (GSK573719A) is a novel mAChR antagonist.Fórmula:C29H34BrNO2Pureza:98.4% - 99.89%Cor e Forma:SolidPeso molecular:508.49PSEM 89S TFA
CAS:<p>PSEM 89S TFA is a brain-penetrant and selective ion channels agonist, and is orthogonally selective for Q79G and L141F, respectively.</p>Fórmula:C18H23F3N2O5Pureza:99.9%Cor e Forma:SolidPeso molecular:404.38PHA 568487 free base
CAS:<p>PHA 568487 free base, an α7 nicotinic receptor agonist, designed to reduce bioactivation and improve in vivo tolerability.</p>Fórmula:C16H20N2O3Pureza:99.74%Cor e Forma:SolidPeso molecular:288.34Blarcamesine
CAS:<p>Blarcamesine (AVex-73) is a muscarinic M1 agonist potentially for the treatment of Alzheimer's disease.</p>Fórmula:C19H23NOPureza:99.87%Cor e Forma:SolidPeso molecular:281.39
