NMDAR
Os inibidores do receptor N-Metil-D-Aspartato (NMDAR) são compostos que bloqueiam a atividade dos NMDARs, um subtipo de receptores de glutamato que desempenham um papel crucial na plasticidade sináptica, no aprendizado e na memória. A superativação dos NMDARs está implicada na excitotoxicidade, que pode levar a danos neuronais e está associada a condições como AVC, lesão cerebral traumática e doenças neurodegenerativas. Os inibidores de NMDAR são ferramentas essenciais para estudar a excitotoxicidade e desenvolver terapias neuroprotetoras. Na CymitQuimica, oferecemos uma gama de inibidores de NMDAR para apoiar sua pesquisa em função sináptica, neuroproteção e distúrbios cognitivos.
Foram encontrados 28 produtos de "NMDAR"
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Mephenesin
CAS:<p>Mephenesin (Cresoxydiol) is a centrally acting muscle relaxant with a short duration of action.</p>Fórmula:C10H14O3Pureza:99.49%Cor e Forma:SolidPeso molecular:182.22SDZ 220-040 ammonium
<p>SDZ 220-040 ammonium is a competitive glutamate ionotropic receptor NMDA antagonist used in the study of neurological disorders.</p>Fórmula:C16H19Cl2N2O6PPureza:98.47%Cor e Forma:SolidPeso molecular:437.21L-689560
CAS:<p>L-689560, a radiolabeled ligand, studies NMDA receptors, is an antagonist at GluN1 glycine site.</p>Fórmula:C17H15Cl2N3O3Pureza:98%Cor e Forma:SolidPeso molecular:380.23S1R agonist 2
CAS:<p>S1R agonist 2 is a selective S1R agonist with a Ki of 88 nM for S2R and 1.1 nM for S1R and is protective against ROS and NMDA-induced neurotoxicity.</p>Fórmula:C21H27NOPureza:98.85%Cor e Forma:SolidPeso molecular:309.45GluN2B receptor modulator-1
CAS:<p>GluN2B receptor modulator-1 is a selective negative allosteric modulator of NMDA receptor GluN2B subunits (IC50 31 nM), valuable for neuropharmacology studies.</p>Fórmula:C17H15F3N4O2SPureza:99.56%Cor e Forma:SolidPeso molecular:396.39QNZ46
CAS:<p>QNZ46 is a NR2C/NR2D-selective NMDA receptor non-competitive antagonist.</p>Fórmula:C24H17N3O6Pureza:99.65%Cor e Forma:SolidPeso molecular:443.41Flutriafol
CAS:<p>Flutriafol is a pesticide, demethylation inhibitor, and NMDA receptor agonist</p>Fórmula:C16H13F2N3OPureza:98.75%Cor e Forma:SolidPeso molecular:301.29DNQX disodium salt
CAS:<p>DNQX disodium salt is a water-soluble form of selective antagonist of non-NMDA receptor</p>Fórmula:C8H2N4Na2O6Pureza:98.93%Cor e Forma:SolidPeso molecular:296.1Dizocilpine Maleate
CAS:<p>Dizocilpine Maleate (MK 801) is a potent noncompetitive antagonist of the NMDA receptor with Kd of 37.2 nM in rat brain membranes.</p>Fórmula:C20H19NO4Pureza:99% - 99.96%Cor e Forma:White SolidPeso molecular:337.38Rapastinel Trifluoroacetate
CAS:<p>Rapastinel Trifluoroacetate (GLYX-13 Trifluoroacetate) is an NMDA receptor modulator with glycine-site partial agonist properties.</p>Fórmula:C20H32F3N5O8Pureza:99.01% - 99.77%Cor e Forma:SolidPeso molecular:527.49ZL006
CAS:<p>ZL006 is an effective inhibitor of nNOS/PSD-95 interaction. ZL006 also inhibits NMDA receptor-mediated NO synthesis.</p>Fórmula:C14H11Cl2NO4Pureza:98.29%Cor e Forma:SolidPeso molecular:328.15Traxoprodil
CAS:<p>Traxoprodil (CP101606) is a selective NMDA antagonist and protects hippocampal neurons (IC50: 10 nM).</p>Fórmula:C20H25NO3Pureza:99.89%Cor e Forma:SolidPeso molecular:327.42(-)-Dizocilpine maleate
CAS:<p>(-)-Dizocilpine maleate ((-)-MK 801 (Maleate)) is a potent, selective and non-competitive NMDA receptor antagonist with Kd of 37.2 nM in rat brain membranes.</p>Fórmula:C20H19NO4Pureza:>99.99%Cor e Forma:White SolidPeso molecular:337.37Acamprosate
CAS:<p>Acamprosate, alcohol dependence treatment. Affordable Excellence: Reliable Quality You Can Trust</p>Fórmula:C5H11NO4SPureza:98.30%Cor e Forma:SolidPeso molecular:181.21Glypromate acetate(32302-76-4 free base)
<p>Glypromate acetate is a neuroprotective agent, is a weak NMDA receptor agonist.</p>Fórmula:C14H23N3O8Pureza:99.94%Cor e Forma:SolidPeso molecular:361.35Flupirtine maleate
CAS:<p>Flupirtine maleate (Katadolon maleate), a centrally acting non-opioid analgesia, is the salt form of Flupirtine. Flupirtine is an NMDA receptor antagonist.</p>Fórmula:C15H17FN4O2·C4H4O4Pureza:99.5% - 99.9%Cor e Forma:Off-White Crystalline PowderPeso molecular:420.39L-701324
CAS:<p>L-701324 is an NMDA receptor with high affinity and selectivity for the glycine site, used as an orally active and long-acting anticonvulsant.</p>Fórmula:C21H14ClNO3Pureza:98.63% - >99.99%Cor e Forma:SolidPeso molecular:363.79TCN 201
CAS:<p>TCN 201 is a selective antagonist of NMDA receptors containing the NR2A subunit.</p>Fórmula:C21H17ClFN3O4SPureza:98.5%Cor e Forma:SolidPeso molecular:461.89Eliprodil
CAS:<p>Eliprodil (SL-820715), NR2B-NMDA receptor blocker (IC50: 1 uM), less potent on NR2A/NR2C (IC50>100 uM), explored for Parkinson's and movement issues.</p>Fórmula:C20H23ClFNOPureza:99.53% - 99.77%Cor e Forma:SolidPeso molecular:347.85Radiprodil
CAS:<p>Radiprodil (RGH-896) is an oral NMDA NR2B antagonist for potential DPNP neuropathic pain treatment.</p>Fórmula:C21H20FN3O4Pureza:99.74%Cor e Forma:SolidPeso molecular:397.4
