Receptor de Histamina
Os receptores de histamina são GPCRs que mediam os efeitos da histamina, uma amina biogênica envolvida em respostas imunológicas, secreção de ácido gástrico e neurotransmissão. Existem quatro subtipos de receptores de histamina (H1, H2, H3 e H4), cada um desempenhando papéis distintos em reações alérgicas, função gástrica e atividade do sistema nervoso central. Antagonistas dos receptores de histamina são amplamente utilizados no tratamento de alergias, úlceras pépticas e enjoo de movimento. Na CymitQuimica, oferecemos uma seleção abrangente de moduladores de receptores de histamina de alta qualidade para apoiar sua pesquisa em imunologia, gastroenterologia e neurofarmacologia.
Foram encontrados 358 produtos de "Receptor de Histamina"
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Doxylamine succinate
CAS:<p>Doxylamine Succinate is a pyridine derivate histamine H1 antagonist with pronounced sedative properties.</p>Fórmula:C21H28N2O5Pureza:99.61%Cor e Forma:5 1 (Ntp 1992)Peso molecular:388.46Hydroxyzine Pamoate
CAS:<p>Hydroxyzine Pamoate (Bobsule) is a histamine H1 receptor antagonist that is effective in the treatment of chronic urticaria and histamine-mediated pruritus.</p>Fórmula:C44H43ClN2O8Pureza:99.49%Cor e Forma:SolidPeso molecular:763.27Pemirolast potassium
CAS:<p>Pemirolast potassium, a pyrimidinone antiallergic, blocks antigen-induced Ca²⁺ influx in mast cells.</p>Fórmula:C10H7KN6OPureza:98.91% - 99.63%Cor e Forma:Crystals From Dimethylformamide Crystalline SolidPeso molecular:266.31Roxatidine Acetate hydrochloride
CAS:<p>Roxatidine Acetate hydrochloride (HOE 760) is a specific and competitive histamin H2-receptor antagonist. Roxatidine inhibits gastric acid secretion.</p>Fórmula:C19H29ClN2O4Pureza:99.49%Cor e Forma:SolidPeso molecular:384.9Cyproheptadine hydrochloride sesquihydrate
CAS:<p>Cyproheptadine hydrochloride sesquihydrate (Peritol), an antihistamine, is an antagonist of serotonin and histamine2.</p>Fórmula:C21H24ClNOPureza:99.77% - >99.99%Cor e Forma:White To Slightly Yellowish Crystalline SolidPeso molecular:341.88Levocetirizine
CAS:<p>Levocetirizine is a Histamine-1 Receptor Antagonist. The mechanism of action of levocetirizine is as a Histamine H1 Receptor Antagonist.</p>Fórmula:C21H25ClN2O3Pureza:98% - 99.9%Cor e Forma:White PowderPeso molecular:388.89Mifentidine
CAS:<p>Mifentidine (DA 4577) is an orally available H2 receptor antagonist for the study of gastric emptying and experimental gastric and duodenal ulcers.</p>Fórmula:C13H16N4Pureza:98.34% - 99.73%Cor e Forma:SolidPeso molecular:228.29MK-0249 FA
<p>MK-0249 FA is an H3 inverse agonist that can be used to study attention-deficit, hyperactivity disorder and cognitive disorders in adults.</p>Fórmula:C24H26F3N3O4Pureza:99.98%Cor e Forma:SolidPeso molecular:477.48Meclizine dihydrochloride
CAS:<p>Meclizine dihydrochloride (NSC28728) is a histamine H1 antagonist used in the treatment of motion sickness, vertigo, and nausea during pregnancy and radiation</p>Fórmula:C25H27ClN2·2HClPureza:98.05% - 99.79%Cor e Forma:White Slightly Yellowish Crystalline PowderPeso molecular:463.87Mebhydrolin napadisylate
CAS:<p>Mebhydrolin napadisylate (Incidal) is an antihistamine used to relieve allergic symptoms caused by histamine release, including nasal allergies and allergic</p>Fórmula:C19H20N2C10H8O6S2Pureza:99.35% - 99.96%Cor e Forma:White Or Almost White CrystallinePeso molecular:420.52Mizolastine
CAS:<p>Mizolastine (SL 850324), an antihistamine with IC50 of 47 nM, treats allergies like hay fever and hives.</p>Fórmula:C24H25FN6OPureza:98% - 99.75%Cor e Forma:SolidPeso molecular:432.49Terfenadine
CAS:<p>Terfenadine, metabolized to fexofenadine by CYP3A4, is a non-sedative antihistamine targeting H1 receptors.</p>Fórmula:C32H41NO2Pureza:98.76% - 99.75%Cor e Forma:SolidPeso molecular:471.67Doxepin hydrochloride
CAS:<p>Doxepin hydrochloride, a dibenzoxepin tricyclic, blocks monoamine reuptake and has anticholinergic and antihistaminic effects. Mechanism partly unknown.</p>Fórmula:C19H22ClNOPureza:99.65% - 99.91%Cor e Forma:White To Off-White PowderPeso molecular:315.84Promethazine hydrochloride
CAS:<p>Promethazine HCl: First-gen antihistamine, H1 and mACh blocker, affects 5-HT2A/C, D2, α1 receptors.</p>Fórmula:C17H20N2S·HClPureza:99.85%Cor e Forma:Crystals In Water Has A Ph Of 3 5-5 0 (Ntp 1992)Peso molecular:320.88Talastine
CAS:<p>Talastine is an antihistamine compound that can induce an allergic rash.</p>Fórmula:C19H21N3OPureza:98.50% - 99.44%Cor e Forma:SolidPeso molecular:307.39Cinnarizine
CAS:<p>Cinnarizine is a piperazine, blocks H1-receptor & Ca-channels, has vasodilating & antiemetic effects, may cause Parkinson-like symptoms.</p>Fórmula:C26H28N2Pureza:99.94%Cor e Forma:SolidPeso molecular:368.51Carbinoxamine Maleate Salt
CAS:<p>Carbinoxamine Maleate Salt (Lergefin) is an ethanolamine class of H1 antihistamines with mild antimuscarinic and sedative properties.</p>Fórmula:C20H23ClN2O5Pureza:99.97%Cor e Forma:Off-White SolidPeso molecular:406.86Clemastine fumarate
CAS:<p>Clemastine fumarate (Meclastine (fumarate)) is a synthetic ethanolamine with anticholinergic, sedative, and histamine H1 antagonistic properties.</p>Fórmula:C25H30ClNO5Pureza:99.52% - >99.99%Cor e Forma:Colorless To Faintly Yellow Crystalline Powder Appearance White Or Almost White Crystalline PowderPeso molecular:459.97Ranitidine Hydrochloride
CAS:<p>Ranitidine Hydrochloride (AH19065) is a competitive and reversible inhibitor of histamine H2-receptor antagonists with antacid activity.</p>Fórmula:C13H23ClN4O3SPureza:99.30% - 99.49%Cor e Forma:SolidPeso molecular:350.86Orphenadrine hydrochloride
CAS:<p>Orphenadrine hydrochloride (Mephenamin) is a muscarinic antagonist used to treat drug-induced parkinsonism and to relieve pain from muscle spasm.</p>Fórmula:C18H23NO·HClPureza:99.88%Cor e Forma:Liquid About 5 5 Bitter Numbing Taste (Ntp 1992)Peso molecular:305.85
