Receptor de Histamina
Os receptores de histamina são GPCRs que mediam os efeitos da histamina, uma amina biogênica envolvida em respostas imunológicas, secreção de ácido gástrico e neurotransmissão. Existem quatro subtipos de receptores de histamina (H1, H2, H3 e H4), cada um desempenhando papéis distintos em reações alérgicas, função gástrica e atividade do sistema nervoso central. Antagonistas dos receptores de histamina são amplamente utilizados no tratamento de alergias, úlceras pépticas e enjoo de movimento. Na CymitQuimica, oferecemos uma seleção abrangente de moduladores de receptores de histamina de alta qualidade para apoiar sua pesquisa em imunologia, gastroenterologia e neurofarmacologia.
Foram encontrados 358 produtos de "Receptor de Histamina"
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Cyproheptadine hydrochloride sesquihydrate
CAS:<p>Cyproheptadine hydrochloride sesquihydrate (Peritol), an antihistamine, is an antagonist of serotonin and histamine2.</p>Fórmula:C21H24ClNOPureza:99.77% - >99.99%Cor e Forma:White To Slightly Yellowish Crystalline SolidPeso molecular:341.88Mepyramine maleate
CAS:<p>Mepyramine maleate is a mild hypnotic, local anesthetic, and H1 histamine antagonist for allergies and colds.</p>Fórmula:C21H27N3O5Pureza:99.51% - 99.7%Cor e Forma:White Crystalline PowderPeso molecular:401.47Promethazine hydrochloride
CAS:<p>Promethazine HCl: First-gen antihistamine, H1 and mACh blocker, affects 5-HT2A/C, D2, α1 receptors.</p>Fórmula:C17H20N2S·HClPureza:99.85%Cor e Forma:Crystals In Water Has A Ph Of 3 5-5 0 (Ntp 1992)Peso molecular:320.88Pimethixene
CAS:<p>Pimethixene (Calmixen) blocks 5-HT1A, 2A/B/C, H1, D2/D4.4 & muscarinic M1/M2 receptors; potent with pKis 7.54-10.44.</p>Fórmula:C19H19NSPureza:97.50%Cor e Forma:SolidPeso molecular:293.43Mifentidine
CAS:<p>Mifentidine (DA 4577) is an orally available H2 receptor antagonist for the study of gastric emptying and experimental gastric and duodenal ulcers.</p>Fórmula:C13H16N4Pureza:98.34% - 99.73%Cor e Forma:SolidPeso molecular:228.29Pheniramine maleate
CAS:<p>Pheniramine maleate (Trimetose), an alkylamine derivative with antihistaminic and vasodilatory properties, binds to histamine H1 receptors.</p>Fórmula:C16H20N2·C4H4O4Pureza:99.85%Cor e Forma:Physical Description White Powder With A Faint Amine-Like Odor Melting Point 107°CPeso molecular:356.42Amitriptyline hydrochloride
CAS:<p>Amitriptyline hydrochloride (Annoyltin) is the hydrochloride salt of the tricyclic dibenzocycloheptadiene amitriptyline with antidepressant and antinociceptive</p>Fórmula:C20H24ClNPureza:97% - 99.94%Cor e Forma:Crystals White To Off-White PowderPeso molecular:313.86Mirtazapine
CAS:<p>Mirtazapine is a unique tetracyclic antidepressant, may cause temporary liver enzyme elevation, and is linked to rare liver injury.</p>Fórmula:C17H19N3Pureza:99.98%Cor e Forma:SolidPeso molecular:265.35Carebastine
CAS:<p>Carebastine, the active metabolite of Ebastine, is an antagonist of the histamine H1 receptor.</p>Fórmula:C32H37NO4Pureza:99.16%Cor e Forma:Off-White SolidPeso molecular:499.64KSK67
CAS:<p>KSK67 is a selective dual antagonist of sigma-2 and histamine H3 receptors with inhibitory effects on H3 receptors, sigma-1, and sigma-2 receptors, with Ki</p>Fórmula:C22H27N3O2Pureza:99.11%Cor e Forma:SoildPeso molecular:365.47Oxmetidine
CAS:<p>Oxmetidine (SKF 92994) is an H2R antagonist that inhibits transmembrane calcium flux in the cardiovascular system and is used in the study of duodenal ulcers.</p>Fórmula:C19H21N5O3SPureza:99.67%Cor e Forma:SolidPeso molecular:399.47Betahistine mesylate
CAS:<p>Betahistine mesylate (Extovyl), an H1 agonist and vasodilator, treats Meniere's disease and vascular headaches; risks with asthma/ulcers.</p>Fórmula:C8H12N2·2(CH4O3S)Pureza:98% - 99.85%Cor e Forma:CoaPeso molecular:328.4Methapyrilene hydrochloride
CAS:<p>Methapyrilene hydrochloride is a biochemical.</p>Fórmula:C14H20ClN3SCor e Forma:Liquid Solution) 5 5 (Ntp 1992)Peso molecular:297.85H4R antagonist 3
CAS:<p>H4R antagonist 3 is a novel histamine-4 receptor (H4R) antagonist with an EC50 <10 mM.H4R antagonist 3 has potential inflammatory activity for the study of</p>Fórmula:C19H21ClN4SPureza:98%Cor e Forma:SolidPeso molecular:372.92Samelisant
CAS:<p>Samelisant (SUVN-G3031), a selective H3 inverse agonist, Ki=8.7/9.8 nM in humans/rats, has anti-narcoleptic properties.</p>Fórmula:C21H31N3O3Pureza:99.59%Cor e Forma:SolidPeso molecular:373.49Sufotidine
CAS:<p>Sufotidine (AH 25352X) is a highly selective competitive H2 receptor antagonist.</p>Fórmula:C20H31N5O3SPureza:99.03% - 99.92%Cor e Forma:SolidPeso molecular:421.56Tecastemizole
CAS:<p>Tecastemizole (R 43512) is a selective antagonist of H1 receptor and a major metabolite of astemizole with anti-inflammatory effects.</p>Fórmula:C19H21FN4Pureza:99.70%Cor e Forma:SolidPeso molecular:324.4Cetirizine D8 dihydrochloride
CAS:<p>Cetirizine D8 dihydrochloride is a deuterated H1-antihistamine with long-acting effects.</p>Fórmula:C21H26Cl2N2O3Pureza:98%Cor e Forma:SolidPeso molecular:433.4Donetidine
CAS:<p>Donetidine is a histamine H2 receptor antagonist used to treat digestive disorders.</p>Fórmula:C20H25N5O3SPureza:99.32%Cor e Forma:SolidPeso molecular:415.51Histamine H4 receptor antagonist-1
CAS:<p>Histamine H4 receptor antagonist-1 is a potent antagonist of the histamine H4 receptor.</p>Fórmula:C30H38N8O2Cor e Forma:SolidPeso molecular:542.68Thioperamide maleate
CAS:<p>Thioperamide maleate (MR-12842 maleate) is an effective and selective antagonist of H3 receptor (Ki = 4.3 nM) for inhibition of [3H]histamine synthesis (Ki = 31</p>Fórmula:C19H28N4O4SPureza:98.48%Cor e Forma:SolidPeso molecular:408.52Levocarnitine propionate hydrochloride
CAS:<p>Levocarnitine propionate hydrochloride (ST-261) is used for the treatment of the deterioration of renal function, congestive heart failure, and other diseases.</p>Fórmula:C10H20ClNO4Pureza:90% - 99.77%Cor e Forma:SolidPeso molecular:253.724-Methylhistamine
CAS:<p>4-Methylhistamine serves as a potent agonist for the histamine 4 receptor (H4R), holding promise for research into immune-related diseases, including cancer and</p>Fórmula:C6H11N3Pureza:98%Cor e Forma:SolidPeso molecular:125.17Neurotransmitter Receptor Compound Library
<p>A unique collection of 1513 neurotransmitter receptor compounds, can be used for HTS and HCS screening；</p>Cor e Forma:Odour SolidDiphenhydramine hydrochloride
CAS:<p>DPH: antihistamine for cough, nausea, itching, allergy, Parkinson's, sleep aid, cold remedy.</p>Fórmula:C17H22ClNOPureza:99.84%Cor e Forma:Taste Ph (5% Aqueous Solution) 4-6 (Ntp 1992)Peso molecular:291.82Oxmetidine FA
<p>Oxmetidine FA is an orally available specific histamine H2 receptor antagonist with antiulcerogenic properties.</p>Fórmula:C20H23N5O5SPureza:97.34%Cor e Forma:SoildPeso molecular:445.49Nizatidine
CAS:<p>Nizatidine (Acinon) is a competitive and reversible histamine H2-receptor antagonist with antacid activity.</p>Fórmula:C12H21N5O2S2Pureza:99.43%Cor e Forma:White To Off-White Crystalline PowderPeso molecular:331.46Bodilisant
CAS:<p>Bodilisant: nanomolar-affinity hH3R ligand, derived from piperidine, with BODIPY fluorophore.</p>Fórmula:C27H34BF2N3OCor e Forma:SolidPeso molecular:465.4Roxatidine
CAS:<p>Roxatidine, a metabolite of Roxatidine acetate, is a H2-receptor antagonist that prevents ulcers and has anti-inflammatory properties.</p>Fórmula:C17H26N2O3Cor e Forma:SolidPeso molecular:306.4Vapitadine
CAS:<p>Vapitadine is a non-sedative antihistamine compound that relieves itching caused by atopic dermatitis.</p>Fórmula:C17H20N4OPureza:99.77% - 99.86%Cor e Forma:SoildPeso molecular:296.37Cetirizine Impurity C
CAS:<p>Cetirizine Impurity C - a metabolite of hydroxyzine, is a long-acting, oral H1-antihistamine.</p>Fórmula:C21H25ClN2O3Cor e Forma:SolidPeso molecular:388.89Dalcotidine
CAS:<p>Dalcotidine (KU 1257), a histamine H2/H9 blocker, inhibits acid secretion; Ki=0.040, KB=0.041, aids ulcer healing, may lower relapse.</p>Fórmula:C18H29N3O2Pureza:99.11%Cor e Forma:SolidPeso molecular:319.44Nα-Methylhistamine FA
<p>Nα-Methylhistamine FA is a histamine H3 receptor agonist</p>Fórmula:C7H13N3O2Pureza:>99.99%Cor e Forma:SolidPeso molecular:171.2Dexchlorpheniramine free base
CAS:<p>Dexchlorpheniramine Maleate, a histamine receptor antagonist, is used to treat urticaria, allergic rhinitis, allergic conjunctivitis and pruritus.</p>Fórmula:C16H19ClN2Pureza:98%Cor e Forma:Oily Liquid SolidPeso molecular:274.79(S)-Azelastine hydrochloride
CAS:<p>(S)-Azelastine HCl, an antihistamine, reduces H1R, M1R, M3R levels and inhibits HNEpC growth.</p>Fórmula:C22H25Cl2N3OPureza:98%Cor e Forma:SolidPeso molecular:418.36Cetirizine Impurity C dihydrochloride
CAS:<p>Cetirizine Impurity C dihydrochloride is a Cetirizine metabolite and long-acting H1-antihistamine.</p>Fórmula:C21H27Cl3N2O3Cor e Forma:SolidPeso molecular:461.81JNJ-10181457 (hydrochloride)
CAS:<p>JNJ-10181457 (hydrochloride) is a non-imidazole H3 receptor antagonist that is brain-penetrating and selective, increasing NE and acetylcholine concentrations</p>Fórmula:C20H30Cl2N2OCor e Forma:SolidPeso molecular:385.37Alcaftadine carboxylic acid
CAS:<p>Alcaftadine is a novel antihistamine for preventing allergic conjunctivitis.</p>Fórmula:C19H21N3O2Cor e Forma:SolidPeso molecular:323.39Cetirizine Impurity D
CAS:<p>Cetirizine Impurity D, an antihistamine derivative, acts as a long-lasting H1-receptor antagonist with antiallergic effects.</p>Fórmula:C30H28Cl2N2Cor e Forma:SolidPeso molecular:487.46Sigma-1 receptor antagonist 5
<p>Sigma-1 receptor antagonist 5 (compound 12), a 4-pyridylpiperidine derivative, exhibits analgesic properties through its antagonistic action on sigma receptors</p>Fórmula:C26H27N3OPureza:98%Cor e Forma:SolidPeso molecular:397.51Cetirizine methyl ester
CAS:<p>Cetirizine methyl ester is a Cetirizine impurity, a long-acting, oral H1-antihistamine and hydroxyzine metabolite.</p>Fórmula:C22H27ClN2O3Cor e Forma:SolidPeso molecular:402.91Conessine hydrobromide
CAS:<p>Conessine hydrobromide is a naturally occurring steroid alkaloid and has been used in traditional herbal medicine as a treatment for amoebic dysentery.</p>Fórmula:C24H41BrN2Cor e Forma:SolidPeso molecular:437.51(+)-Dropropizine
CAS:<p>(+)-Dropropizine can inhibit histamine receptor, anti-allergic, and reduce a cough by modulation of neuropeptides involved in the cough reflex.</p>Fórmula:C13H20N2O2Pureza:>99.99%Cor e Forma:White Or Off White Crystalline PowderPeso molecular:236.31Histamine & Melatonin Receptor-Targeted Compound Library
<p>A unique collection of xnum compounds targeting histaminergic receptor and melatonin receptor for high throughput screening (HTS) and high content screening (HCS</p>Cor e Forma:Odour SolidKSK94 FA
<p>KSK94 FA is a potent histamine H3 receptor antagonist that inhibits H3 receptors and is used in the study of neuropathic pain and obesity.</p>Fórmula:C26H28N4O3Pureza:97.51%Cor e Forma:SoildPeso molecular:444.53Alimemazine D6
CAS:<p>Alimemazine D6 is a deuterium-labeled Alimemazine. Alimemazine is an antihistamine.</p>Fórmula:C18H22N2SPureza:98%Cor e Forma:SolidPeso molecular:304.48Antazoline phosphate
CAS:<p>Antazoline phosphate: H1 histamine receptor antagonist with anticholinergic effects, eases allergies.</p>Fórmula:C17H22N3O4PPureza:98%Cor e Forma:CoaPeso molecular:363.35Hydroxyzine D8
CAS:<p>Hydroxyzine D8, a deuterium-labeled version of Hydroxyzine, acts as a histamine H1-receptor antagonist.</p>Fórmula:C21H27ClN2O2Pureza:98%Cor e Forma:SolidPeso molecular:382.95Cetirizine D8
CAS:<p>Cetirizine D8 is a deuterium-labeled Cetirizine. Cetirizine is a second-generation antihistamine and a long-acting histamine H1-receptor antagonist.</p>Fórmula:C21H25ClN2O3Pureza:98%Cor e Forma:SolidPeso molecular:396.94Diphenylpyraline
CAS:<p>Diphenylpyridine is the first generation antihistamine, which has the anticholinergic effect of diphenylpiperidine.</p>Fórmula:C19H23NOCor e Forma:SolidPeso molecular:281.39
