Receptor de Histamina
Os receptores de histamina são GPCRs que mediam os efeitos da histamina, uma amina biogênica envolvida em respostas imunológicas, secreção de ácido gástrico e neurotransmissão. Existem quatro subtipos de receptores de histamina (H1, H2, H3 e H4), cada um desempenhando papéis distintos em reações alérgicas, função gástrica e atividade do sistema nervoso central. Antagonistas dos receptores de histamina são amplamente utilizados no tratamento de alergias, úlceras pépticas e enjoo de movimento. Na CymitQuimica, oferecemos uma seleção abrangente de moduladores de receptores de histamina de alta qualidade para apoiar sua pesquisa em imunologia, gastroenterologia e neurofarmacologia.
Foram encontrados 390 produtos para "Receptor de Histamina".
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Phenindamine
CAS:Phenindamine (Nu 1504) is an H1-receptor antagonist which is antihistamine[1].Fórmula:C19H19NCor e Forma:SolidPeso molecular:261.36Acreozast
CAS:Acreozast, a histamine release inhibitor, is used potentially for the treatment of asthma and atopic dermatitis.Fórmula:C15H14ClN3O6Cor e Forma:SolidPeso molecular:367.74CP19
CAS:CP19 blocks histamine receptors; inhibits EBOV and MARV with IC50s of 3.4 μM and 29.5 μM, respectively; antiviral [1].Fórmula:C26H30N2O5Cor e Forma:SolidPeso molecular:450.53Phenindamine Tartrate
CAS:Phenindamine Tartrate, an antihistamine and anticholinergic, treats colds and allergies like sneezing and rashes.Fórmula:C23H25NO6Cor e Forma:SolidPeso molecular:411.454INCB38579
CAS:INCB38579: Oral, selective H4 antagonist; crosses brain barrier; IC50s - hH4R: 4.8 nM, mH4R: 42 nM, rH4R: 32 nM; anti-inflammatory and antipruritic.Fórmula:C25H34N6OCor e Forma:SolidPeso molecular:434.58AZD5213
CAS:AZD5213: selective human H3 receptor antagonist, pKi 9.3, for sleep/cognition research.Fórmula:C19H25N3O2Cor e Forma:SolidPeso molecular:327.42Nebidrazine
CAS:Nebidrazine is an alpha-adrenoceptor agonist.Fórmula:C9H8Cl2N6Cor e Forma:SolidPeso molecular:271.11Toreforant
CAS:Toreforant is an effective and selective histamine H4 receptor antagonist (Ki at the human receptor: 8.4 nM).Fórmula:C23H32N6Pureza:98%Cor e Forma:SolidPeso molecular:392.54Carbinoxamine
CAS:Carbinoxamine: antihistamine for hay fever, angioedema, rhinitis, mild urticaria, dermatographism, allergic conjunctivitis; an H1-antagonist.Fórmula:C16H19ClN2OPureza:98%Cor e Forma:SolidPeso molecular:290.79SUN 1334H
CAS:SUN 1334H is a potent, orally active, highly selective antagonist of H1 receptor(Ki of 9.7 nM).Fórmula:C23H28Cl2F2N2O3Pureza:98%Cor e Forma:SolidPeso molecular:489.38H4R antagonist 1
CAS:H4R antagonist 1: selective histamine H4R inhibitor, IC50 27 nM, no affinity for H1R, H2R, H3R.Fórmula:C11H11BrN8Cor e Forma:SolidPeso molecular:335.16Setastine HCl
CAS:Setastine HCl is a potent antagonist of histamine H1-receptor mediated responses.Fórmula:C22H29Cl2NOCor e Forma:SolidPeso molecular:394.38(R)-(-)-α-Methylhistamine dihydrobromide
CAS:(R)-(-)-α-Methylhistamine dihydrobromide is a potent and selective agonist of H3 histamine receptor( Kd of 50.3 nM).Fórmula:C6H13Br2N3Pureza:99.98%Cor e Forma:SolidPeso molecular:287(±)-Tazifylline
CAS:(±)-Tazifylline is a selective and long-acting antagonist of histamine H1 receptor.Fórmula:C23H32N6O3SPureza:99.54%Cor e Forma:SolidPeso molecular:472.6Ref: TM-T10000
1mg140,00€5mg269,00€1mL*10mM (DMSO)350,00€10mg389,00€25mg610,00€50mg820,00€100mg1.063,00€Carcinine
CAS:Carcinine ditrifluoroacetate is a H3 receptor antagonist.Fórmula:C8H14N4OPureza:98%Cor e Forma:SolidPeso molecular:182.22H3R-IN-1 Hydrochloride
CAS:H3R-IN-1 Hydrochloride is an inverse agonist of histamine receptor 3( H3R ) .Fórmula:C19H24ClN3O3Pureza:98%Cor e Forma:SolidPeso molecular:377.86ICI 162,846
CAS:ICI 162,846 is an orally active and potent H2 receptor antagonist that inhibits gastric secretion and may be used in the study of duodenal ulcers.Fórmula:C11H17F3N6OPureza:99.76%Cor e Forma:SolidPeso molecular:306.29Nedocromil
CAS:Nedocromil (FPL 59002) inhibits the action or formation of multiple mediators. Which including histamine, leukotriene C4 (LTC4), and prostaglandin D2 (PGD2).Fórmula:C19H17NO7Pureza:95% - 97.34%Cor e Forma:SolidPeso molecular:371.34Iodophenpropit dihydrobromide
CAS:Iodophenpropit dihydrobromide: selective histamine H3 antagonist, reversible binding, high affinity (KD: 0.32 nM).Fórmula:C15H20BrIN4SPureza:98%Cor e Forma:SolidPeso molecular:495.22PF-03654746 Tosylate
CAS:PF-03654746 Tosylate is selective antagonist of histamine H3 receptor with high brain penetration.Fórmula:C25H32F2N2O4SPureza:98%Cor e Forma:SolidPeso molecular:494.6Hetramine
CAS:Hetramine is a synthetic pyrimidine agent that possesses antihistamine and anti anaphylactic effects.Fórmula:C15H20N4Pureza:98%Cor e Forma:SolidPeso molecular:256.35Fenethazine
CAS:Fenethazine is an effective antihistamine used as an antiallergic drug.Fórmula:C16H18N2SCor e Forma:SolidPeso molecular:270.39HSR-609
CAS:HSR-609, a histamine H1 receptor antagonist, is used potentially for the treatment of allergic rhinitis.Fórmula:C21H21FN2O3Pureza:98%Cor e Forma:SolidPeso molecular:368.4BMH-7
CAS:BMH-7 (Histamine H4 receptor antagonist-2) is a p53 activator, demonstrating anti-cancer activity by activating the p53 pathway.Fórmula:C20H21N5OPureza:99.71%Cor e Forma:SolidPeso molecular:347.41Tei 6472
CAS:Tei 6472 is a more hydrophilic form of TEI-1338 which is a novel, selective lipoxygenase inhibitor.Fórmula:C32H39N3O5Pureza:98%Cor e Forma:SolidPeso molecular:545.67Nα-Methylhistamine dihydrochloride
CAS:Nα-Methylhistamine dihydrochloride is a histamine H3 receptor agonist.Fórmula:C6H13Cl2N3Pureza:98%Cor e Forma:SolidPeso molecular:198.094Amthamine dihydrobromide
CAS:H2 agonistFórmula:C6H13Br2N3SPureza:98%Cor e Forma:SolidPeso molecular:319.06Carcainium chloride
CAS:Carcainium chloride (Carcainium (chloride)) is a derivative of Lidocaine and possesses an antitussive effect.Fórmula:C18H22ClN3O2Pureza:99.89%Cor e Forma:SolidPeso molecular:347.84DA 4643
CAS:DA 4643, a histamine H2-receptor antagonist, binds similarly to mifentidine at the receptor.Fórmula:C12H16Cl2N6SPureza:98%Cor e Forma:SolidPeso molecular:347.26Mequitamium iodide
CAS:Mequitamium iodide is a PAF inhibitor, curbing platelet aggregation and bronchoconstriction without blocking PAF receptors.Fórmula:C21H25IN2SCor e Forma:SolidPeso molecular:464.41Impentamine dihydrobromide
CAS:Impentamine dihydrobromide is a histamine H3 receptor antagonist.Fórmula:C8H17Br2N3Pureza:98%Cor e Forma:SolidPeso molecular:315.05Chloracyzine
CAS:Chloracyzine lowers heart oxygen use, shrinks coronary flow after brief dilation, slightly ups heart rate and arterial pressure.Fórmula:C19H21ClN2OSCor e Forma:SolidPeso molecular:360.9AHR-13268D
CAS:AHR-13268D is a new agent of antiallergic/antihistaminic.Fórmula:C28H29F2NNaO4Pureza:98%Cor e Forma:SolidPeso molecular:504.53AHR-14310C
CAS:AHR-14310C is a long-acting and nonsedating H1-antihistamine.Fórmula:C24H28F2N2O3Pureza:98%Cor e Forma:SolidPeso molecular:430.49NNC-38-1049
CAS:NNC-38-1049 is a novel selective antagonist of histamine H3.Fórmula:C19H25ClN2O2Pureza:98%Cor e Forma:SolidPeso molecular:348.87Embramine
CAS:Embramine, used as an antihistamine and anticholinergic, is a monoethanolamine.Fórmula:C18H22BrNOPureza:98%Cor e Forma:SolidPeso molecular:348.28Linadryl hydrochloride
CAS:Linadryl hydrochloride may have antihistamine activity.Fórmula:C19H24ClNO2Cor e Forma:SolidPeso molecular:333.85Ramixotidine
CAS:Ramixotidine is a competitive antagonist of histamine H2-receptor.Fórmula:C16H21N3O3SPureza:98%Cor e Forma:SolidPeso molecular:335.42Dacemazine hydrochloride
CAS:Dacemazine is a phenothiazine derivative that acts as a histamine antagonist at the H1 subtype. It was also assessed as a possible anticancer drug.Fórmula:C16H17ClN2OSPureza:98%Cor e Forma:SolidPeso molecular:320.84Rocastine
CAS:Rocastine (AHR-11325) is a selective and potent non-sedating H1 receptor antagonist.Fórmula:C13H19N3OSPureza:98.26%Cor e Forma:Yellow OilPeso molecular:265.37H3 receptor-MO-1
CAS:H3 receptor-MO-1 is a potent modulator of the histamine H3 receptor (H3 receptor) and can be used to study neurodegeneration and cognitive disorders.Fórmula:C20H27N3O2Pureza:99.11%Cor e Forma:White SolidPeso molecular:341.45Bamirastine
CAS:Bamirastine inhibits ligand binding to recombinant human histamine H1 receptor (rhH1R) with an IC50 value of 17.3 nM.Bamirastine has an inhibitory effect onFórmula:C31H37N5O3Pureza:96.68%Cor e Forma:Yellow SolidPeso molecular:527.66CP-66948
CAS:CP-66948 is a potent histamine H2 receptor antagonist with inhibitory effect on gastric acid secretion and can be used to protect gastric and intestinal mucosa.Fórmula:C13H20N6SPureza:99.14%Cor e Forma:SolidPeso molecular:292.4PF-03654764
CAS:PF-03654764, an oral H3 receptor blocker, Ki: human 1.2 nM, rat 7.9 nM, used with Fexofenadine for allergic rhinitis.Fórmula:C20H28F2N2OPureza:>99.99%Cor e Forma:Yellow SolidPeso molecular:350.45Lavoltidine
CAS:Lavoltidine (Loxtidine) is potent and selective H2 receptor antagonist, oral and irreversible,inhibits gastric acid secretion, gastroesophageal reflux disease.Fórmula:C19H29N5O2Pureza:98.30% - 98.36%Cor e Forma:White SolidPeso molecular:359.47Propiomazine HCl
CAS:Propiomazine HCl is an analgesia adjunct.Fórmula:C20H25ClN2OSCor e Forma:SolidPeso molecular:376.94JNJ-39220675
CAS:JNJ-39220675, a selective histamine H3 receptor antagonist, reduces the abuse-related effects of alcohol in rats.Fórmula:C21H24FN3O2Pureza:97.77% - 99.89%Cor e Forma:White OilPeso molecular:369.43VUF14862
CAS:VUF14862 is a robust and fatigue-resistant photoswitchable GPCR antagonist.Fórmula:C26H32N4O2Cor e Forma:SolidPeso molecular:432.56Sch 44643
CAS:Sch 44643 is an antagonist of platelet activating factor with oral activity.Fórmula:C25H22ClN3O2Cor e Forma:SolidPeso molecular:431.91Brl 22321
CAS:Brl 22321 is a mast cell stabilizer.Fórmula:C12H9N3O2Cor e Forma:SolidPeso molecular:227.22
