Receptor de Histamina
Os receptores de histamina são GPCRs que mediam os efeitos da histamina, uma amina biogênica envolvida em respostas imunológicas, secreção de ácido gástrico e neurotransmissão. Existem quatro subtipos de receptores de histamina (H1, H2, H3 e H4), cada um desempenhando papéis distintos em reações alérgicas, função gástrica e atividade do sistema nervoso central. Antagonistas dos receptores de histamina são amplamente utilizados no tratamento de alergias, úlceras pépticas e enjoo de movimento. Na CymitQuimica, oferecemos uma seleção abrangente de moduladores de receptores de histamina de alta qualidade para apoiar sua pesquisa em imunologia, gastroenterologia e neurofarmacologia.
Foram encontrados 358 produtos de "Receptor de Histamina"
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Pirolate
CAS:<p>Pirolate is a receptor of histamine H1.</p>Fórmula:C16H15N3O5Pureza:98%Cor e Forma:SolidPeso molecular:329.31Bepotastine tosylate
CAS:<p>Bepotastine tosylate: Oral 2nd-gen H1 antagonist, inhibits histamine effects on NGF; treats conjunctivitis, urticaria.</p>Fórmula:C28H33ClN2O6SCor e Forma:SolidPeso molecular:561.09VUF-10497
CAS:<p>VUF-10497: H4 receptor inverse agonist, anti-inflammatory in rats, binds human H1 receptor (pKi=7.57).</p>Fórmula:C18H20ClN5SPureza:98%Cor e Forma:SolidPeso molecular:373.9A331440
CAS:<p>A331440 is an modulator of L-histidine and histamine H3 receptor.</p>Fórmula:C22H27N3OCor e Forma:SolidPeso molecular:349.47Phenindamine
CAS:<p>Phenindamine (Nu 1504) is an H1-receptor antagonist which is antihistamine[1].</p>Fórmula:C19H19NCor e Forma:SolidPeso molecular:261.36Acreozast
CAS:<p>Acreozast, a histamine release inhibitor, is used potentially for the treatment of asthma and atopic dermatitis.</p>Fórmula:C15H14ClN3O6Cor e Forma:SolidPeso molecular:367.74CP19
CAS:<p>CP19 blocks histamine receptors; inhibits EBOV and MARV with IC50s of 3.4 μM and 29.5 μM, respectively; antiviral [1].</p>Fórmula:C26H30N2O5Cor e Forma:SolidPeso molecular:450.53Phenindamine Tartrate
CAS:<p>Phenindamine Tartrate, an antihistamine and anticholinergic, treats colds and allergies like sneezing and rashes.</p>Fórmula:C23H25NO6Cor e Forma:SolidPeso molecular:411.454INCB38579
CAS:<p>INCB38579: Oral, selective H4 antagonist; crosses brain barrier; IC50s - hH4R: 4.8 nM, mH4R: 42 nM, rH4R: 32 nM; anti-inflammatory and antipruritic.</p>Fórmula:C25H34N6OCor e Forma:SolidPeso molecular:434.58Thioperamide
CAS:<p>histamine H3 and H4 antagonist/inverse agonist</p>Fórmula:C15H24N4SPureza:98%Cor e Forma:White SolidPeso molecular:292.44VUF 5681 dihydrobromide
CAS:<p>histamine H3 receptor silent antagonist</p>Fórmula:C11H21Br2N3Pureza:98%Cor e Forma:SolidPeso molecular:355.11Carbinoxamine
CAS:<p>Carbinoxamine: antihistamine for hay fever, angioedema, rhinitis, mild urticaria, dermatographism, allergic conjunctivitis; an H1-antagonist.</p>Fórmula:C16H19ClN2OPureza:98%Cor e Forma:LiquidPeso molecular:290.79Nebidrazine
CAS:<p>Nebidrazine is an alpha-adrenoceptor agonist.</p>Fórmula:C9H8Cl2N6Cor e Forma:SolidPeso molecular:271.11Toreforant
CAS:<p>Toreforant is an effective and selective histamine H4 receptor antagonist (Ki at the human receptor: 8.4 nM).</p>Fórmula:C23H32N6Pureza:98%Cor e Forma:SolidPeso molecular:392.54VUF 8430
CAS:<p>VUF 8430 is a selective agonist for the H4 receptor.</p>Fórmula:C4H11N5SPureza:98%Cor e Forma:SolidPeso molecular:161.23UK-9040
CAS:<p>UK-9040 inhibits gastric secretory.</p>Fórmula:C23H31NSPureza:98%Cor e Forma:SolidPeso molecular:353.56SUN 1334H
CAS:<p>SUN 1334H is a potent, orally active, highly selective antagonist of H1 receptor(Ki of 9.7 nM).</p>Fórmula:C23H28Cl2F2N2O3Pureza:98%Cor e Forma:SolidPeso molecular:489.38Adriforant hydrochloride
CAS:<p>Adriforant hydrochloride is an antagonist of histamine H4 receptor.</p>Fórmula:C13H25Cl3N6Pureza:98%Cor e Forma:SolidPeso molecular:371.74Seliforant
CAS:<p>Seliforant is a histamine H4 receptor antagonist.</p>Fórmula:C12H21N5Pureza:98%Cor e Forma:SolidPeso molecular:235.33(R)-(-)-α-Methylhistamine dihydrobromide
CAS:<p>(R)-(-)-α-Methylhistamine dihydrobromide is a potent and selective agonist of H3 histamine receptor( Kd of 50.3 nM).</p>Fórmula:C6H13Br2N3Pureza:98%Cor e Forma:SolidPeso molecular:287Amthamine dihydrobromide
CAS:<p>H2 agonist</p>Fórmula:C6H13Br2N3SPureza:98%Cor e Forma:SolidPeso molecular:319.06Carcainium chloride
CAS:<p>Carcainium chloride (Carcainium (chloride)) is a derivative of Lidocaine and possesses an antitussive effect.</p>Fórmula:C18H22ClN3O2Pureza:99.89%Cor e Forma:SolidPeso molecular:347.84DA 4643
CAS:<p>DA 4643, a histamine H2-receptor antagonist, binds similarly to mifentidine at the receptor.</p>Fórmula:C12H16Cl2N6SPureza:98%Cor e Forma:SolidPeso molecular:347.26Mequitamium iodide
CAS:<p>Mequitamium iodide is a PAF inhibitor, curbing platelet aggregation and bronchoconstriction without blocking PAF receptors.</p>Fórmula:C21H25IN2SCor e Forma:SolidPeso molecular:464.41Impentamine dihydrobromide
CAS:<p>Impentamine dihydrobromide is a histamine H3 receptor antagonist.</p>Fórmula:C8H17Br2N3Pureza:98%Cor e Forma:SolidPeso molecular:315.05Chloracyzine
CAS:<p>Chloracyzine lowers heart oxygen use, shrinks coronary flow after brief dilation, slightly ups heart rate and arterial pressure.</p>Fórmula:C19H21ClN2OSCor e Forma:SolidPeso molecular:360.9AHR-13268D
CAS:<p>AHR-13268D is a new agent of antiallergic/antihistaminic.</p>Fórmula:C28H29F2NNaO4Pureza:98%Cor e Forma:SolidPeso molecular:504.53AHR-14310C
CAS:<p>AHR-14310C is a long-acting and nonsedating H1-antihistamine.</p>Fórmula:C24H28F2N2O3Pureza:98%Cor e Forma:SolidPeso molecular:430.49NNC-38-1049
CAS:<p>NNC-38-1049 is a novel selective antagonist of histamine H3.</p>Fórmula:C19H25ClN2O2Pureza:98%Cor e Forma:SolidPeso molecular:348.87Aplysamine-1
CAS:<p>Aplysamine-1 is an antagonist of histamine H3 receptor.</p>Fórmula:C15H24Br2N2OPureza:98%Cor e Forma:SolidPeso molecular:408.17Linadryl hydrochloride
CAS:<p>Linadryl hydrochloride may have antihistamine activity.</p>Fórmula:C19H24ClNO2Cor e Forma:SolidPeso molecular:333.85Ramixotidine
CAS:<p>Ramixotidine is a competitive antagonist of histamine H2-receptor.</p>Fórmula:C16H21N3O3SPureza:98%Cor e Forma:SolidPeso molecular:335.42JNJ 10191584 maleate
CAS:<p>JNJ 10191584 maleate (VUF6002 maleate) is an orally active and selective antagonist of H4 receptor (Ki = 26 nM).</p>Fórmula:C17H19ClN4O5Pureza:99.37%Cor e Forma:SolidPeso molecular:394.81Dacemazine hydrochloride
CAS:<p>Dacemazine is a phenothiazine derivative that acts as a histamine antagonist at the H1 subtype. It was also assessed as a possible anticancer drug.</p>Fórmula:C16H17ClN2OSPureza:98%Cor e Forma:SolidPeso molecular:320.84Carcinine
CAS:<p>Carcinine ditrifluoroacetate is a H3 receptor antagonist.</p>Fórmula:C8H14N4OPureza:98%Cor e Forma:SolidPeso molecular:182.22Azatadine
CAS:<p>Azatadine is histamine and cholinergic inhibitor (IC50: 6.5 nM and 10 nM, respectively).</p>Fórmula:C20H22N2Pureza:98%Cor e Forma:SolidPeso molecular:290.4H3R-IN-1 Hydrochloride
CAS:<p>H3R-IN-1 Hydrochloride is an inverse agonist of histamine receptor 3( H3R ) .</p>Fórmula:C19H24ClN3O3Pureza:98%Cor e Forma:SolidPeso molecular:377.86Impromidine
CAS:<p>Impromidine is a highly potent and specific agonist of the histamine H2 receptor.</p>Fórmula:C14H23N7SPureza:98%Cor e Forma:SolidPeso molecular:321.44Rocastine
CAS:<p>Rocastine (AHR-11325) is a selective and potent non-sedating H1 receptor antagonist.</p>Fórmula:C13H19N3OSPureza:98.26%Cor e Forma:SolidPeso molecular:265.37H3 receptor-MO-1
CAS:<p>H3 receptor-MO-1 is a potent modulator of the histamine H3 receptor (H3 receptor) and can be used to study neurodegeneration and cognitive disorders.</p>Fórmula:C20H27N3O2Pureza:99.11%Cor e Forma:SolidPeso molecular:341.45Vapitadine dihydrochloride
CAS:<p>Vapitadine dihydrochloride(R-129160 2HCl) is a novel, potent, selective and non-sedating compound with inhibitory effects on histamine H1.</p>Fórmula:C17H22Cl2N4OPureza:98.28% - 99.30%Cor e Forma:SolidPeso molecular:369.29Bamirastine
CAS:<p>Bamirastine inhibits ligand binding to recombinant human histamine H1 receptor (rhH1R) with an IC50 value of 17.3 nM.Bamirastine has an inhibitory effect on</p>Fórmula:C31H37N5O3Pureza:96.68%Cor e Forma:SolidPeso molecular:527.66CP-66948
CAS:<p>CP-66948 is a potent histamine H2 receptor antagonist with inhibitory effect on gastric acid secretion and can be used to protect gastric and intestinal mucosa.</p>Fórmula:C13H20N6SPureza:99.14%Cor e Forma:SolidPeso molecular:292.4PF-03654764
CAS:<p>PF-03654764, an oral H3 receptor blocker, Ki: human 1.2 nM, rat 7.9 nM, used with Fexofenadine for allergic rhinitis.</p>Fórmula:C20H28F2N2OPureza:>99.99%Cor e Forma:SolidPeso molecular:350.45Lavoltidine
CAS:<p>Lavoltidine (Loxtidine) is potent and selective H2 receptor antagonist, oral and irreversible,inhibits gastric acid secretion, gastroesophageal reflux disease.</p>Fórmula:C19H29N5O2Pureza:98.30% - 98.36%Cor e Forma:SolidPeso molecular:359.47UR-PI376
CAS:<p>UR-PI376 is a selective histamine H4 receptor agonist with low H1/H2 activity and moderate H3 affinity.</p>Fórmula:C17H22N6SCor e Forma:SolidPeso molecular:342.46GSK-239512
CAS:<p>GSK-239512 is an antagonist of H3 receptor and can be used in studies about the treatment of cognitive dysfunction in neurodegenerative disorders.</p>Fórmula:C23H27N3O2Pureza:99.62% - 99.74%Cor e Forma:SolidPeso molecular:377.48S-1-Propenyl-L-cysteine
CAS:<p>S-1-Propenyl-L-cysteine, a stereoisomer of S-allyl-l-cysteine, exhibits immunomodulatory effects and has been shown to decrease blood pressure in hypertensive</p>Fórmula:C6H11NO2SPureza:98%Cor e Forma:SolidPeso molecular:161.22ROS 234 dioxalate
CAS:<p>ROS 234 dioxalate is a potent antagonist of H3(pKB of 9.46 for Guinea-pig ileum H3-receptor)</p>Fórmula:C17H19N5O8Pureza:98%Cor e Forma:SolidPeso molecular:421.37Nedocromil
CAS:<p>Nedocromil (FPL 59002) inhibits the action or formation of multiple mediators. Which including histamine, leukotriene C4 (LTC4), and prostaglandin D2 (PGD2).</p>Fórmula:C19H17NO7Pureza:95% - 97.34%Cor e Forma:SolidPeso molecular:371.34
