
Receptor de Histamina
Os receptores de histamina são GPCRs que mediam os efeitos da histamina, uma amina biogênica envolvida em respostas imunológicas, secreção de ácido gástrico e neurotransmissão. Existem quatro subtipos de receptores de histamina (H1, H2, H3 e H4), cada um desempenhando papéis distintos em reações alérgicas, função gástrica e atividade do sistema nervoso central. Antagonistas dos receptores de histamina são amplamente utilizados no tratamento de alergias, úlceras pépticas e enjoo de movimento. Na CymitQuimica, oferecemos uma seleção abrangente de moduladores de receptores de histamina de alta qualidade para apoiar sua pesquisa em imunologia, gastroenterologia e neurofarmacologia.
Foram encontrados 385 produtos de "Receptor de Histamina"
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Hydroxyzine-d8 DiHCl
CAS:Hydroxyzine-d8 DiHCl is a deuterated compound of Hydroxyzine DiHCl. Hydroxyzine DiHCl has a CAS number of 2192-20-3.Fórmula:C21H21D8Cl3N2O2Cor e Forma:SolidPeso molecular:455.88Methaphenilene hydrochloride
CAS:Methaphenilene hydrochloride is an H1 receptor antagonist with antihistaminic and anticholinergic activity, in allergic inflammation and autonomic research.Fórmula:C15H21ClN2SPureza:99.84%Cor e Forma:SolidPeso molecular:296.86Mianserin-d3
CAS:Mianserin-d3 is a deuterated compound of Mianserin. Mianserin has a CAS number of 24219-97-4. Mianserin, an H1 receptor reverse agonist, is a psychoactive compound in the tetracyclic antidepressant (TeCA) treatment family. Mianserin has antidepressant, antianxiety, antiemetic, hypotrophic, hypnotic and antihistamine effects, and can be used as a combination of norepinephrine and specific serotonin to treat depression.Fórmula:C18H17D3N2Cor e Forma:SolidPeso molecular:267.38Proxyfan Oxalate
CAS:Proxyfan Oxalate is a potent antagonist of the histamine H3 receptor (histamine H3 receptor), with Ki values of 2.9 nM for rats and 2.7 nM for humans. Its inhibitory effect on H3 receptors is over 1000 times stronger than its effect on other histamine receptors.Fórmula:C15H18N2O5Cor e Forma:SolidPeso molecular:306.31Amthamine
CAS:Compound AMTHAMINE DIHYDROBROMIDE is a useful organic compound for research related to life sciences.Fórmula:C6H11N3SCor e Forma:SoildPeso molecular:157.24Ciproxifan
CAS:Ciproxifan (FUB-359) is a highly effective and specific histamin H3-receptor antagonist (IC50: 9.2 nM).Fórmula:C16H18N2O2Pureza:98.00%Cor e Forma:SolidPeso molecular:270.33Roxatidine acetate
CAS:Roxatidine acetate: anti-ulcer, blocks histamine, reduces acid. Safer at lower doses.Fórmula:C19H28N2O4Pureza:98%Cor e Forma:White Or Off-White PowderPeso molecular:348.44Lodoxamide tromethamine
CAS:Lodoxamide tromethamine is a mast cell stabilizer with anti-allergic properties and can be used in studies about the treatment of asthma and allergicFórmula:C19H28ClN5O12Pureza:98.8%Cor e Forma:SolidPeso molecular:553.91VUF 8430 dihydrobromide
CAS:histamine H4 receptor full agonistFórmula:C4H12BrN5SPureza:98%Cor e Forma:SolidPeso molecular:242.14BMH-7
CAS:BMH-7 (Histamine H4 receptor antagonist-2) is a p53 activator, demonstrating anti-cancer activity by activating the p53 pathway.Fórmula:C20H21N5OPureza:99.71%Cor e Forma:SolidPeso molecular:347.41Tei 6472
CAS:Tei 6472 is a more hydrophilic form of TEI-1338 which is a novel, selective lipoxygenase inhibitor.Fórmula:C32H39N3O5Pureza:98%Cor e Forma:SolidPeso molecular:545.67Nα-Methylhistamine dihydrochloride
CAS:Nα-Methylhistamine dihydrochloride is a histamine H3 receptor agonist.Fórmula:C6H13Cl2N3Pureza:98%Cor e Forma:SolidPeso molecular:198.094Amthamine dihydrobromide
CAS:H2 agonistFórmula:C6H13Br2N3SPureza:98%Cor e Forma:SolidPeso molecular:319.06Carcainium chloride
CAS:Carcainium chloride (Carcainium (chloride)) is a derivative of Lidocaine and possesses an antitussive effect.Fórmula:C18H22ClN3O2Pureza:99.89%Cor e Forma:SolidPeso molecular:347.84Bavisant dihydrochloride
CAS:Bavisant (JNJ-310010740) is an oral, selective H3 receptor antagonist enhancing wakefulness and cognition.Fórmula:C19H29Cl2N3O2Pureza:98%Cor e Forma:SolidPeso molecular:402.36DA 4643
CAS:DA 4643, a histamine H2-receptor antagonist, binds similarly to mifentidine at the receptor.Fórmula:C12H16Cl2N6SPureza:98%Cor e Forma:SolidPeso molecular:347.26Mequitamium iodide
CAS:Mequitamium iodide is a PAF inhibitor, curbing platelet aggregation and bronchoconstriction without blocking PAF receptors.Fórmula:C21H25IN2SCor e Forma:SolidPeso molecular:464.41Impentamine dihydrobromide
CAS:Impentamine dihydrobromide is a histamine H3 receptor antagonist.Fórmula:C8H17Br2N3Pureza:98%Cor e Forma:SolidPeso molecular:315.05Chloracyzine
CAS:Chloracyzine lowers heart oxygen use, shrinks coronary flow after brief dilation, slightly ups heart rate and arterial pressure.Fórmula:C19H21ClN2OSCor e Forma:SolidPeso molecular:360.9AHR-13268D
CAS:AHR-13268D is a new agent of antiallergic/antihistaminic.Fórmula:C28H29F2NNaO4Pureza:98%Cor e Forma:SolidPeso molecular:504.53
