
Receptor de Histamina
Os receptores de histamina são GPCRs que mediam os efeitos da histamina, uma amina biogênica envolvida em respostas imunológicas, secreção de ácido gástrico e neurotransmissão. Existem quatro subtipos de receptores de histamina (H1, H2, H3 e H4), cada um desempenhando papéis distintos em reações alérgicas, função gástrica e atividade do sistema nervoso central. Antagonistas dos receptores de histamina são amplamente utilizados no tratamento de alergias, úlceras pépticas e enjoo de movimento. Na CymitQuimica, oferecemos uma seleção abrangente de moduladores de receptores de histamina de alta qualidade para apoiar sua pesquisa em imunologia, gastroenterologia e neurofarmacologia.
Foram encontrados 385 produtos de "Receptor de Histamina"
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Cetirizine Impurity C
CAS:Cetirizine Impurity C - a metabolite of hydroxyzine, is a long-acting, oral H1-antihistamine.Fórmula:C21H25ClN2O3Cor e Forma:SolidPeso molecular:388.89Vapitadine
CAS:Vapitadine is a non-sedative antihistamine compound that relieves itching caused by atopic dermatitis.Fórmula:C17H20N4OPureza:99.77% - 99.86%Cor e Forma:SoildPeso molecular:296.37Cetirizine Impurity C dihydrochloride
CAS:Cetirizine Impurity C dihydrochloride is a Cetirizine metabolite and long-acting H1-antihistamine.Fórmula:C21H27Cl3N2O3Cor e Forma:SolidPeso molecular:461.81H4R antagonist 3
CAS:H4R antagonist 3 is a novel histamine-4 receptor (H4R) antagonist with an EC50 <10 mM.H4R antagonist 3 has potential inflammatory activity for the study ofFórmula:C19H21ClN4SPureza:98%Cor e Forma:SolidPeso molecular:372.924-Methylhistamine
CAS:<p>4-Methylhistamine serves as a potent agonist for the histamine 4 receptor (H4R), holding promise for research into immune-related diseases, including cancer and</p>Fórmula:C6H11N3Pureza:98%Cor e Forma:SolidPeso molecular:125.17Methimepip dihydrobromide
CAS:Methimepip dihydrobromide is a selective H3R agonist.Fórmula:C10H19Br2N3Cor e Forma:SolidPeso molecular:341.091Alcaftadine carboxylic acid
CAS:Alcaftadine is a novel antihistamine for preventing allergic conjunctivitis.Fórmula:C19H21N3O2Cor e Forma:SolidPeso molecular:323.39Histamine & Melatonin Receptor-Targeted Compound Library
<p>A unique collection of xnum compounds targeting histaminergic receptor and melatonin receptor for high throughput screening (HTS) and high content screening (HCS</p>Cor e Forma:Odour SolidDexchlorpheniramine free base
CAS:Dexchlorpheniramine Maleate, a histamine receptor antagonist, is used to treat urticaria, allergic rhinitis, allergic conjunctivitis and pruritus.Fórmula:C16H19ClN2Pureza:98%Cor e Forma:Oily Liquid SolidPeso molecular:274.79JNJ-10181457 (hydrochloride)
CAS:JNJ-10181457 (hydrochloride) is a non-imidazole H3 receptor antagonist that is brain-penetrating and selective, increasing NE and acetylcholine concentrationsFórmula:C20H30Cl2N2OCor e Forma:SolidPeso molecular:385.37Levocarnitine propionate hydrochloride
CAS:Levocarnitine propionate hydrochloride (ST-261) is used for the treatment of the deterioration of renal function, congestive heart failure, and other diseases.Fórmula:C10H20ClNO4Pureza:90% - 99.77%Cor e Forma:SolidPeso molecular:253.72(S)-Azelastine hydrochloride
CAS:(S)-Azelastine HCl, an antihistamine, reduces H1R, M1R, M3R levels and inhibits HNEpC growth.Fórmula:C22H25Cl2N3OPureza:98%Cor e Forma:SolidPeso molecular:418.363-hydroxy Desloratidine
CAS:3-hydroxy Desloratidine is a major metabolite of desloratadine , a tricyclic antagonist of the histamine H1 receptor.Fórmula:C19H19ClN2OCor e Forma:SolidPeso molecular:326.82(+)-Dropropizine
CAS:(+)-Dropropizine can inhibit histamine receptor, anti-allergic, and reduce a cough by modulation of neuropeptides involved in the cough reflex.Fórmula:C13H20N2O2Pureza:>99.99%Cor e Forma:White Or Off White Crystalline PowderPeso molecular:236.31Cetirizine Impurity D
CAS:Cetirizine Impurity D, an antihistamine derivative, acts as a long-lasting H1-receptor antagonist with antiallergic effects.Fórmula:C30H28Cl2N2Cor e Forma:SolidPeso molecular:487.46Cetirizine methyl ester
CAS:Cetirizine methyl ester is a Cetirizine impurity, a long-acting, oral H1-antihistamine and hydroxyzine metabolite.Fórmula:C22H27ClN2O3Cor e Forma:SolidPeso molecular:402.91AM-0466
CAS:AM-0466 has a wide range of applications in life science related research.Fórmula:C27H19F3N4O4SCor e Forma:SolidPeso molecular:552.52Oxmetidine
CAS:Oxmetidine (SKF 92994) is an H2R antagonist that inhibits transmembrane calcium flux in the cardiovascular system and is used in the study of duodenal ulcers.Fórmula:C19H21N5O3SPureza:99.67%Cor e Forma:SolidPeso molecular:399.47Alimemazine D6
CAS:Alimemazine D6 is a deuterium-labeled Alimemazine. Alimemazine is an antihistamine.Fórmula:C18H22N2SPureza:98%Cor e Forma:SolidPeso molecular:304.48Antazoline phosphate
CAS:Antazoline phosphate: H1 histamine receptor antagonist with anticholinergic effects, eases allergies.Fórmula:C17H22N3O4PPureza:98%Cor e Forma:CoaPeso molecular:363.35
