Receptor de Histamina
Os receptores de histamina são GPCRs que mediam os efeitos da histamina, uma amina biogênica envolvida em respostas imunológicas, secreção de ácido gástrico e neurotransmissão. Existem quatro subtipos de receptores de histamina (H1, H2, H3 e H4), cada um desempenhando papéis distintos em reações alérgicas, função gástrica e atividade do sistema nervoso central. Antagonistas dos receptores de histamina são amplamente utilizados no tratamento de alergias, úlceras pépticas e enjoo de movimento. Na CymitQuimica, oferecemos uma seleção abrangente de moduladores de receptores de histamina de alta qualidade para apoiar sua pesquisa em imunologia, gastroenterologia e neurofarmacologia.
Foram encontrados 381 produtos de "Receptor de Histamina"
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Thonzylamine
CAS:<p>Thonzylamine is an antihistamine/anticholinergic, combined with Clofedanol or Phenylephrine for cold, hay fever, or allergy relief.</p>Fórmula:C16H22N4OPureza:99.45%Cor e Forma:SolidPeso molecular:286.37JNJ-5207852
CAS:JNJ-5207852 is a novel, non-imidazole histamine H3 receptor antagonist, with high affinity at the rat (pKi=8.9) and human (pKi=9.24) H3 receptor.Fórmula:C20H32N2OPureza:97.19%Cor e Forma:SolidPeso molecular:316.48LML134
CAS:<p>LML134 (LML-134) is an inverse agonist of Histamine 3 receptor (H3R)(hH3R cAMP and hH3R bdg with Kis of 0.3 nM and 12 nM).</p>Fórmula:C19H29N5O3Pureza:99.36%Cor e Forma:SolidPeso molecular:375.47Triprolidine
CAS:Triprolidine: oral H1 receptor blocker with motor/sensory spinal effects, for allergy research.Fórmula:C19H22N2Cor e Forma:SolidPeso molecular:278.39Pitolisant hydrochloride
CAS:Pitolisant hydrochloride (Ciproxidine) is a potent and selective inverse agonist of the histamine H3 receptor(Ki : 0.16 nM).Fórmula:C17H27Cl2NOPureza:99.72% - 99.91%Cor e Forma:SolidPeso molecular:332.31Pemirolast
CAS:Pemirolast: oral antiallergic, reduces paclitaxel reactions, inhibits neuropeptides, for asthma and conjunctivitis study.Fórmula:C10H8N6OCor e Forma:SolidPeso molecular:228.21Irdabisant hydrochloride
CAS:<p>Irdabisant (CEP-26401) is a selective H3R inverse agonist, BBB-penetrable, with cognition-enhancing effects.</p>Fórmula:C18H24ClN3O2Cor e Forma:SolidPeso molecular:349.86Bromodiphenhydramine hydrochloride
CAS:<p>Bromodiphenhydramine hydrochloride is a new antihistaminic in the control of cutaneous.</p>Fórmula:C17H21BrClNOPureza:97.29%Cor e Forma:SolidPeso molecular:370.71Chlorphenoxamine
CAS:<p>Chlorphenoxamine (Contristamine) is an antihistamine and anticholinergic used as an antipruritic and antiparkinsonian agent.</p>Fórmula:C18H22ClNOPureza:99.44% - 99.85%Cor e Forma:SolidPeso molecular:303.83Zotepine
CAS:<p>Zotepine, an antipsychotic agent, is a potent antagonist of 5-HT2A, 5-HT2C, Histamine H1, α1-adrenergic, and Dopamine D2 receptors, with Kds of 2.6 nM, 3.2 nM,</p>Fórmula:C18H18ClNOSPureza:99.78%Cor e Forma:SolidPeso molecular:331.86Epinastine
CAS:Epinastine (WAL801) is an antihistamine, mast cell stabilizer, and H1 antagonist with anti-allergic properties.Fórmula:C16H15N3Pureza:99.94%Cor e Forma:SolidPeso molecular:249.31GSK189254A
CAS:<p>GSK189254A (GSK189254) is a potent and specific histamine H3 receptor antagonist (pKi values: 9.59-9.90 and 8.51-9.17 for human and rat H3).</p>Fórmula:C21H25N3O2Pureza:98.71% - 99.858%Cor e Forma:SolidPeso molecular:351.44Decloxizine
CAS:Decloxizine is a H1 receptor antagonistFórmula:C21H28N2O2Pureza:99.53%Cor e Forma:White Or Similar To White PowderPeso molecular:340.46Ebastine
CAS:Ebastine (Kestine) (trade names Evastin, Kestine, Ebastel, Aleva) is a non-sedating H1 antihistamine.Fórmula:C32H39NO2Pureza:99.65% - 99.99%Cor e Forma:White To Off-White PowderPeso molecular:469.66Diphenhydramine
CAS:Diphenhydramine (Syntedril): first-gen antihistamine for allergies, antiemetic, antitussive, anticholinergic, sedative, treats drug-induced parkinsonism.Fórmula:C17H21NOPureza:98.07%Cor e Forma:SolidPeso molecular:255.35Acitazanolast
CAS:<p>Acitazanolast (WP-871) is an anti-allergic drug candidate.</p>Fórmula:C9H7N5O3Pureza:98.25%Cor e Forma:SolidPeso molecular:233.18Mequitazine
CAS:Mequitazine (Virginan) is an effective, nonsedative and long-acting histamine H1 antagonist.Fórmula:C20H22N2SPureza:99.98%Cor e Forma:SolidPeso molecular:322.472-Pyridylethylamine dihydrochloride
CAS:2-Pyridylethylamine dihydrochloride is a Histamine H1 receptor agonist.Fórmula:C7H12Cl2N2Pureza:99.42%Cor e Forma:SolidPeso molecular:195.09Samelisant dihydrochloride
CAS:SUVN-G3031: H3 receptor antagonist; may treat cognitive issues, ADHD, epilepsy, sleep, obesity, schizophrenia, eating disorders, pain.Fórmula:C21H33Cl2N3O3Cor e Forma:SolidPeso molecular:446.41Acrivastine
CAS:Acrivastine (Acrivastin) is a short-acting histamine 1 receptor antagonist.Fórmula:C22H24N2O2Pureza:99.73% - >99.99%Cor e Forma:SolidPeso molecular:348.44
