Receptor opioide
Os receptores opioides são um grupo de receptores acoplados à proteína G que mediam os efeitos dos opioides endógenos e exógenos. Estes receptores desempenham um papel central na modulação da dor, regulação do humor e comportamentos aditivos. Agonistas e antagonistas dos receptores opioides são amplamente utilizados no manejo da dor e tratamento de dependências, bem como em pesquisas sobre distúrbios neurológicos e psiquiátricos. Na CymitQuimica, oferecemos uma seleção abrangente de moduladores de receptores opioides de alta qualidade para apoiar sua pesquisa em neurobiologia, manejo da dor e terapia de dependência.
Foram encontrados 297 produtos de "Receptor opioide"
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Moguisteine
CAS:<p>Moguisteine (BBR-2173) is a new-type peripheral non-narcotic antitussive drug.</p>Fórmula:C16H21NO5SPureza:99.98%Cor e Forma:SolidPeso molecular:339.41Trimebutine maleate
CAS:<p>Trimebutine maleate (Polibutin) is a weak mu-opioid agonist and has antimuscarinic effects.</p>Fórmula:C26H33NO9Pureza:99.76% - 99.98%Cor e Forma:White SolidPeso molecular:503.55Meptazinol hydrochloride
CAS:<p>Meptazinol hydrochloride (Meptazinol HCl) , a unique centrally opioid analgesic, is used as a narcotic antagonist with analgesic properties.</p>Fórmula:C15H23NO·HClPureza:99.75%Cor e Forma:White SolidPeso molecular:269.81Matrine
CAS:<p>Matrine (Vegard), an alkaloid isolated from the Sophora genus, acts as a kappa opioid receptor agonist.</p>Fórmula:C15H24N2OPureza:97.16% - >99.99%Cor e Forma:SolidPeso molecular:248.36CP 866087
CAS:<p>CP 866087 is an opioid receptor antagonist for the study of female sexual dysfunction.</p>Fórmula:C24H30N2O3SPureza:99.22% - 99.74%Cor e Forma:SolidPeso molecular:426.57Naltrexone hydrochloride
CAS:<p>Naltrexone hydrochloride (Naltrexone HCl) is a synthetic opioid antagonist used in the prevention of relapse of opiate addiction and alcoholism.</p>Fórmula:C20H24ClNO4Pureza:98.72% - 99.65%Cor e Forma:White Crystalline PowderPeso molecular:377.862Loperamide hydrochloride
CAS:<p>Loperamide hydrochloride (ADL 2-1294) is a synthetic, piperidine derivative and opioid agonist with antidiarrheal activity.</p>Fórmula:C29H34Cl2N2O2Pureza:99.91% - >99.99%Cor e Forma:Crystals Practically Insoluble In WaterPeso molecular:513.50Alvimopan
CAS:<p>Alvimopan is a potent opioid antagonist targeting gut receptors to reverse opioid effects on motility.</p>Fórmula:C25H32N2O4Pureza:99.47% - 99.78%Cor e Forma:SolidPeso molecular:424.53Samidorphan HCl
CAS:<p>Samidorphan HCl is an orally active and highly potent modulator of the opioid system that binds to μ‐opioid, κ‐opioid, and delta-opioid receptors.</p>Fórmula:C21H27ClN2O4Pureza:96.79% - 97.85%Cor e Forma:SoildPeso molecular:406.9BTRX-335140
CAS:<p>BTRX-335140 (CYM-53093) is a potent and selective orally active κ-opioid receptor (KOR) antagonist with antagonistic activity.Cost-effective and quality-assured.</p>Fórmula:C25H32FN5O2Pureza:98% - 99.89%Cor e Forma:SolidPeso molecular:453.55Apitegromab
CAS:<p>Apitegromab (SRK-015) is a new myostatin inhibitor, an antibody targeting myostatin precursor, which can be used to study neuromuscular diseases including</p>Pureza:95% - 97.59% (SDS-PAGE); 99.78% (SEC-HPLC)Cor e Forma:LiquidSinomenine hydrochloride
CAS:<p>Sinomenine hydrochloride (Kukoline hydrochloride) is extracted from Sinomenium Acutum Rehderett Wilson.</p>Fórmula:C19H24ClNO4Pureza:99.43%Cor e Forma:SolidPeso molecular:365.851LY2940094
CAS:<p>LY2940094 (LY-2940094) decreases ethanol self-administration in animal models.</p>Fórmula:C22H23ClF2N4O2SPureza:99.4%Cor e Forma:SolidPeso molecular:480.96ZT 52656A hydrochloride
CAS:<p>ZT 52656A is a selective agonist of kappa opioid, and used for the prevention or alleviation of pain in the eye.</p>Fórmula:C19H26ClF3N2OPureza:98.78%Cor e Forma:SolidPeso molecular:390.87Nocistatin
CAS:<p>Nocistatin, a neuropeptide, blocks Nociceptin effects and inhibits 5-HT release, acting on an opioid-related receptor.</p>Fórmula:C32H56N10O12Cor e Forma:SolidPeso molecular:772.85SB 205607 dihydrobromide
CAS:<p>non-peptide δ1 opioid receptor agonist</p>Fórmula:C23H24N2OPureza:98%Cor e Forma:SolidPeso molecular:344.45Valorphin
CAS:<p>Valorphin (Valorphin TFAsalt) has opioid analgesic activity, binds to rat mu-opioid receptor, with an IC50 of 14 nM.</p>Fórmula:C44H61N9O11Pureza:98%Cor e Forma:SolidPeso molecular:892.01β-Endorphin (1-27) (human)
CAS:<p>β-Endorphin (1-27) (human) is an opioid antagonist that selectively binds to μ-, δ-, and κ-opioid receptors, with dissociation constants (Kis) of 5.31, 6.17,</p>Fórmula:C139H217N33O40SPureza:98%Cor e Forma:SolidPeso molecular:3022.47CSD-CH2(1,8)-NH2
<p>CSD-CH2(1,8)-NH2 is a selective and competitive kappa-opioid receptor (KOR) antagonist with a K i of 6.8 nM.</p>Fórmula:C76H125N25O15S2Pureza:98%Cor e Forma:SolidPeso molecular:1693.09Adrenorphin
CAS:<p>Adrenorphin (Metorphamide)(3TFA) is an agonist of μ-opioid receptor(Ki :12 nM).</p>Fórmula:C44H69N15O9SPureza:98%Cor e Forma:SolidPeso molecular:984.18N-Phenethylnoroxymorphone
CAS:<p>N-Phenethylnoroxymorphone is an opioid compound that can enhance morphine-induced analgesia in rats. It is used in the research of neurological disorders.</p>Fórmula:C24H25NO4Cor e Forma:SolidPeso molecular:391.46AT-121 hydrochloride
CAS:<p>AT-121 hydrochloride: dual nociception/mu-opioid agonist, Ki 3.67/16.49 nM, safe, non-addictive pain reliever with analgesic effects.</p>Fórmula:C24H39ClN4O3SPureza:97.28% - >99.99%Cor e Forma:SolidPeso molecular:499.11(S,S)-J-113397
CAS:<p>(S,S)-J-113397 is an isomer of J-113397 . J-113397 is an Opioid Receptor antagonist [1] .</p>Fórmula:C24H37N3O2Cor e Forma:SolidPeso molecular:399.57Leumorphin, human
CAS:<p>Leumorphin, human, is a potent agonist of the kappa opioid receptor (κ opioid receptor) and inhibits the contraction of the guinea pig ileum's myenteric plexus-</p>Fórmula:C150H224N42O46Pureza:98%Cor e Forma:SolidPeso molecular:3351.64Dynorphin B (1-9)
CAS:<p>Dynorphin B (1-9), a neuropeptide and the N-terminal cleavage product of dynorphin B, has its formation inhibited by N-ethylmaleimide (NEM), a non-selective</p>Fórmula:C54H78N16O12Pureza:98%Cor e Forma:SolidPeso molecular:1143.3HINT1-IN-1
<p>HINT1-IN-1 (compound 8) is an inhibitor of histidine triad nucleotide-binding protein 1 (HINT1) with a Ki of 1.14 μM. It influences the cross-regulation between μ-opioid receptors (MOR) and NMDA receptors (NMDAR).</p>Fórmula:C23H24N8O5Cor e Forma:SolidPeso molecular:492.49DPDPE
CAS:<p>DPDPE is selective δ-opioid receptor agonist peptide.</p>Fórmula:C30H39N5O7S2Pureza:98%Cor e Forma:SolidPeso molecular:645.79Frakefamide TFA
<p>Frakefamide TFA: potent, peripherally active μ-opioid agonist; doesn't cross blood-brain barrier.</p>Fórmula:C32H35F4N5O7Cor e Forma:SolidPeso molecular:677.64Dermorphin Analog
<p>Dermorphin Analog, a heptapeptide from amphibian skin, binds μ-opioid receptors selectively and strongly.</p>Fórmula:C44H59N11O10Pureza:98%Cor e Forma:SolidPeso molecular:901.43Helianorphin-19
<p>Helianorphin-19: Potent KOR agonist (Ki=25 nM; EC50=45 nM), 200x selective over μ/δ receptors, effective in mouse pain model, non-sedative.</p>Cor e Forma:Liquidβ-Endorphin (1-27) (human) acetate
<p>β-Endorphin (1-27) (human) acetate, existing in the hypophysis cerebri and hypothalamus, exhibits antinociception activity.</p>Fórmula:C141H221N33O42SPureza:96.52%Cor e Forma:SolidPeso molecular:3082.52Trimebutine
CAS:<p>Trimebutine (Mebutin) is a spasmolytic agent that regulates intestinal and colonic motility and relieves abdominal pain with antimuscarinic and weak mu-opioid</p>Fórmula:C22H29NO5Pureza:98.13% - 99.49%Cor e Forma:SolidPeso molecular:387.47CTOP acetate
<p>CTOP acetate is a somatostatin analogue and a μ-opioid receptor antagonist.</p>Fórmula:C52H71N11O13S2Pureza:99.87%Cor e Forma:SoildPeso molecular:1122.32UFP-101 acetate
<p>UFP-101 acetate is a selective and competitive antagonist of the NOP receptor (pKi = 10.24) with >3000-fold selectivity over δ, μ, and κ opioid receptors.</p>Fórmula:C84H142N32O23Pureza:95.92%Cor e Forma:SolidPeso molecular:1968.23β-Endorphin (6-31), human
CAS:<p>β-Endorphin is an endogenous opioid neuropeptide and opioid receptor agonist that preferentially binds to μ-opioid receptors.</p>Fórmula:C131H218N34O40Pureza:98%Cor e Forma:SolidPeso molecular:2909.38LY255582
CAS:<p>LY255582 is a selective centrally active opioid receptor antagonist with high affinity for mu, delta and kappa receptors with Ki of 0.4 nM, 5.2, 2.0 nM,</p>Fórmula:C22H35NO2Pureza:98%Cor e Forma:SolidPeso molecular:345.52Neuropeptide AF (human)
CAS:<p>Neuropeptide AF (93-110), Human is an endogenous antiopioid peptide.</p>Fórmula:C90H132N26O25Pureza:98%Cor e Forma:SolidPeso molecular:1978.17Naldemedine
CAS:<p>Naldemedine (S 297995), developed by Shionogi, is a drug for opioid side effects like constipation. It's well tolerated with minor GI issues.</p>Fórmula:C32H34N4O6Cor e Forma:SolidPeso molecular:570.64(N-Me-Tyr1,N-Me-Arg7,D-Leu-NHEt8)-Dynorphin A (1-8)
CAS:<p>E-2078, known chemically as (N-Me-Tyr1,N-Me-Arg7,D-Leu-NHEt8)-Dynorphin A (1-8), is a stable analog of Dynorphin A (1–8) and functions as a kappa opioid</p>Fórmula:C50H81N15O9Cor e Forma:SolidPeso molecular:1036.27BPR1M97
CAS:<p>BPR1M97 is a mu opioid receptor (MOP) and neuropeptide-orphin FQ (NOP) receptor agonist with blood-brain barrier permeability and potency, with Kis values of 1.</p>Fórmula:C18H18Cl2N2OPureza:98.78% - 99.95%Cor e Forma:SolidPeso molecular:349.25Ac-RYYRIK-NH2
CAS:<p>NOP site high affinity ligand (Ki=1.5 nM); blocks nociceptin effects in rat brain/heart; agonist in vivo, reduces mouse movement.</p>Fórmula:C44H70N14O9Pureza:98%Cor e Forma:SolidPeso molecular:939.12Neuropeptide AF (human) acetate
<p>Neuropeptide AF (human) acetate (Neuropeptide AF (human) acetate (192387-38-5 Free base)) is an anti-opioid neuropeptide, a Neuropeptide AF (human) derivative,</p>Pureza:99.89%Cor e Forma:Soildβ-Endorphin, equine
CAS:<p>Endorphin Beta is A substance produced in the brain, especially in the pituitary gland, Endorphin Beta blocks the sensation of pain.</p>Fórmula:C154H248N42O44SPureza:98%Cor e Forma:SolidPeso molecular:3423.94difelikefalin acetate(1024828-77-0 Free base)
CAS:<p>is a ketone and a building block.</p>Fórmula:C38H57N7O8Pureza:96.94%Cor e Forma:SolidPeso molecular:739.9[D-Ala2]leucine-enkephalin acetate
<p>[D-Ala2]leucine-enkephalin acetate ([D-Ala2]leucine-enkephalin acetate (64963-01-5 free base)) is a delta opioid agonist used to study the signaling pathway of</p>Fórmula:C31H43N5O9Pureza:98%Cor e Forma:SolidPeso molecular:629.65[(pF)Phe4]Nociceptin(1-13)NH2 acetate
<p>[(pF)Phe4]Nociceptin(1-13)NH2 acetate is a selective agonist of NOP receptor with a pKi of 10.68 and a pEC50 of 9.31.</p>Fórmula:C63H103FN22O17Pureza:98.03%Cor e Forma:SolidPeso molecular:1459.63Axelopran
CAS:<p>Axelopran (TD-1211) treats opioid constipation; it's a potent, selective peripheral opioid blocker.</p>Fórmula:C26H39N3O4Cor e Forma:SolidPeso molecular:457.61β-Lipotropin (60-65)
CAS:<p>β-Lipotropin (60-65) (β-LPH (60-65)), an opioid agonist, is a significant [1] opioid peptide.</p>Fórmula:C33H47N9O8SCor e Forma:SolidPeso molecular:729.85Deltorphin acetate
<p>Deltorphin acetate is a substance obtained from the skin secretions of a frog, Phyllomedusa bicolor and shows high selectivity and affinity for δ-opioid</p>Fórmula:C46H66N10O12S2Pureza:98.93%Cor e Forma:SolidPeso molecular:1015.21KOR agonist 5
<p>KOR agonist 5 (Compound 10a) is both a KOR/MOR modulator, exhibiting agonistic effects on KOR and antagonistic effects on MOR. It effectively blocks morphine-induced antinociception and gastrointestinal motility inhibition. KOR agonist 5 is applicable in research related to substance use disorder (SUD).</p>Fórmula:C38H38N2O5Cor e Forma:SolidPeso molecular:602.72Clocinnamox mesylate
CAS:<p>Clocinnamox mesylate: irreversible μ-opioid blocker; Ki: 0.7 nM (mouse μ), 1.9 nM (δ), 5.7 nM (κ).</p>Fórmula:C30H33ClN2O7SCor e Forma:SolidPeso molecular:601.11DALDA TFA
<p>DALDA TFA is a potent, μ-opioid receptor agonist exhibiting high selectivity and an affinity constant (K i) of 1.69 nM.</p>Fórmula:C30H45N9O5·xC2HF3O2Pureza:98%Cor e Forma:SolidPeso molecular:611.74 (free base)Dynorphin B (1-13) (TFA)
<p>Dynorphin B (1-13) TFA acts as an agonist on opioid κ-receptor .</p>Fórmula:C76H116N21F3O19Cor e Forma:SolidPeso molecular:1684.86KOR agonist 4
<p>KOR agonist 4 (compound 39) is an agonist targeting the κ opioid receptor (Kappa Opioid Receptor) and activates G protein signaling. It has an EC50 of 14 nM and an Emax of 83% for binding to GTPγS. This compound demonstrates moderate to high intrinsic clearance in human liver cells and shows selectivity for the κ opioid receptor over the μ (MOR) and δ (DOR) opioid receptors by factors of 60 and 810, respectively. KOR agonist 4 is useful for research into central nervous system (CNS) disorders.</p>Fórmula:C21H25N3Cor e Forma:SolidPeso molecular:319.44β-Endorphin, equine TFA
<p>β-Endorphin, equine TFA, an endogenous opioid peptide, demonstrates high affinity binding to μ/δ opioid receptors and possesses analgesic properties [1] [2] [3</p>Fórmula:C156H249F3N42O46SCor e Forma:SolidPeso molecular:3537.96Akuammicine
CAS:<p>Akuammicine, as an indole alkaloid from Catharanthus roseus, can be used in cancer cell eradication.</p>Fórmula:C20H22N2O2Cor e Forma:SolidPeso molecular:322.408Nociceptin(1-7)
CAS:<p>Bioactive metabolite of nociceptin, antagonist of nociceptin-induced hyperalgesia</p>Fórmula:C31H41N7O9Pureza:98%Cor e Forma:SolidPeso molecular:655.709[(pF)Phe4]Nociceptin(1-13)NH2
CAS:<p>Potent, selective OP4 agonist; pKi=10.68, pEC50=9.80. >8000x selectivity vs other opioid receptors; long-lasting in vivo effects.</p>Fórmula:C61H99FN22O15Pureza:98%Cor e Forma:SolidPeso molecular:1399.6Ac-RYYRWK-NH2 TFA
CAS:<p>Ac-RYYRWK-NH2: potent, specific NOP receptor partial agonist with 0.071 nM affinity; no affinity for μ/κ/δ-opioid receptors.</p>Fórmula:C51H70F3N15O11Cor e Forma:SolidPeso molecular:1126.21ICI 174,864
CAS:<p>Selective δ opioid antagonist. Exhibits partial agonist in vitro activity at δ receptors at high concentrations.</p>Fórmula:C38H53N5O7Pureza:98%Cor e Forma:White SolidPeso molecular:691.87PL-017
CAS:<p>μ opioid receptor agonist; IC50: 5.5 nM (μ), >10,000 nM (δ). Induces reversible analgesia, catalepsy, hyperthermia in rats.</p>Fórmula:C29H37N5O5Pureza:98%Cor e Forma:SolidPeso molecular:535.64[Met5]-Enkephalin, amide
CAS:<p>[Met5]-Enkephalin, amide activates δ and ζ opioid receptors; has multiple forms and varying plasma levels.</p>Fórmula:C27H36N6O6SPureza:98%Cor e Forma:SolidPeso molecular:572.68MT-7716 hydrochloride
CAS:<p>MT-7716 hydrochloride is a selective agonist of non-peptide nociceptin receptor (NOP)</p>Fórmula:C27H29ClN4O2Pureza:98%Cor e Forma:SolidPeso molecular:477N-Acetyl-α-Endorphin
CAS:N-Acetyl-α-Endorphin is a chemical compound consisting of α-Endorphin that has been acetylated at the N-terminal.Fórmula:C79H122N18O27SPureza:98%Cor e Forma:SolidPeso molecular:1787.98PIPE-3297
<p>PIPE-3297 (compound 25) is a selective kappa opioid receptor (KOR) agonist that activates the G protein signaling pathway with an EC50 of 1.1 nM and exhibits low β-arrestin-2 recruitment activity (10%). Additionally, PIPE-3297 promotes myelination and has anti-inflammatory properties.</p>Fórmula:C23H30N2OPeso molecular:350.23581[Nphe1]Nociceptin(1-13)NH2
CAS:<p>Competitive nociceptin receptor antagonist with pKi=8.4; no agonist activity; blocks nociceptin effects in vitro/in vivo.</p>Fórmula:C61H100N22O15Pureza:98%Cor e Forma:SolidPeso molecular:1381.6SNC 80
CAS:<p>SNC 80, a non-peptide δ-opioid agonist (Ki=1.78 nM, IC50=2.73 nM), also targets μ-δ heteromers (EC50=52.8 nM), with analgesic and antidepressant potential.</p>Fórmula:C28H39N3O2Pureza:99.65%Cor e Forma:SolidPeso molecular:449.63[DAla2, DArg6] Dynorphin A, (1-13) (porcine)
CAS:'[DAla2, DArg6] Dynorphin A (1-13) porcine is a potent opioid peptide resistant to enzymatic degradation.'Fórmula:C76H128N24O15Cor e Forma:SolidPeso molecular:1617.98CJ-15208
CAS:<p>CJ-15208: κ-opioid antagonist, IC50: 47 nM kappa, 260 nM mu, 2600 nM delta, reverses asimadoline effects in rabbits (ED50 1.3 µM).</p>Fórmula:C34H35N5O4Cor e Forma:SolidPeso molecular:577.67U-54494A hydrochloride
CAS:<p>U-54494A hydrochloride is a benzamide derivative related to kappa opioid receptor agonists. U-54494A hydrochloride has anticonvulsant activity.</p>Fórmula:C18H25Cl3N2OCor e Forma:SolidPeso molecular:391.76Ac-RYYRWK-NH2
CAS:<p>Selective NOP receptor partial agonist peptide; Ki=0.71 nM; >4000 nM for μ, δ, κ receptors; boosts food intake in vivo.</p>Fórmula:C49H69N15O9Pureza:98%Cor e Forma:SolidPeso molecular:1012.17Gluten Exorphin B5
CAS:<p>Gluten exorphin B5 (GE-B5) is a food-derived opioid peptide identified in digests of wheat gluten.</p>Fórmula:C30H38N6O7Pureza:98%Cor e Forma:SolidPeso molecular:594.66Herkinorin
CAS:<p>Herkinorin: μ-opioid agonist with 100x μ-affinity, 50x less κ-affinity than Salvinorin A, from Salvia divinorum. Semi-synthetic from Salvinorin B.</p>Fórmula:C28H30O8Cor e Forma:SolidPeso molecular:494.53Dermorphin
CAS:<p>Dermorphin is agonist of μ-opioid receptor (MOR) agonist.</p>Fórmula:C40H50N8O10Pureza:98.82%Cor e Forma:SolidPeso molecular:802.87[Nphe1]Nociceptin(1-13)NH2 TFA
<p>[Nphe1]Nociceptin(1-13)NH2 is a selective nociceptin receptor antagonist with potential analgesic properties, pKi=8.4, pA2=6.0.</p>Fórmula:C63H101F3N22O17Cor e Forma:SolidPeso molecular:1495.61Dynorphin B (1-13)
CAS:Dynorphin B (1-13) acts as an agonist on opioid κ-receptor.Fórmula:C74H115N21O17Pureza:98%Cor e Forma:SolidPeso molecular:1570.84β-Endorphin (rat)
CAS:<p>β-Endorphin (β-EP) is an endogenous opioid neuropeptide with diverse biological activities.</p>Fórmula:C157H254N42O44SCor e Forma:SolidPeso molecular:3466.07CTAP
CAS:<p>Potent μ opioid antagonist, IC50 3.5 nM, 1200x selectivity over δ and somatostatin, brain-penetrant, active in vivo.</p>Fórmula:C51H69N13O11S2Pureza:98%Cor e Forma:White Solid/PowderPeso molecular:1104.32Orphanin FQ(1-11)
CAS:<p>Nociceptin peptide fragment (1-11) with potent ORL1/KOR-3 receptor agonism (Ki = 55 nM), no opioid receptor affinity, and analgesic in mice.</p>Fórmula:C49H75N15O14Pureza:98%Cor e Forma:SolidPeso molecular:1098.2Ro 64-6198
CAS:<p>Ro 64-6198: Nonpeptide, selective NOP agonist, high brain uptake, EC50=25.6 nM, 100x NOP>opioid affinity.</p>Fórmula:C26H31N3OPureza:98%Cor e Forma:SolidPeso molecular:401.54β-Naltrexamine dihydrochloride
CAS:<p>β-Naltrexamine dihydrochloride is an orally administered, irreversible opioid receptor antagonist. Its derivatives exhibit optimised subtype selectivity and can be used for pain research.</p>Fórmula:C20H28Cl2N2O3Pureza:95.98%Cor e Forma:SoildPeso molecular:415.35Biphalin TFA
CAS:<p>Biphalin TFA is an opioid peptide analog that penetrates the blood-brain barrier (BBB) and encompasses two active enkephalin pharmacophores.</p>Fórmula:C46H56N10O10·xC2HF3O2Pureza:98%Cor e Forma:SolidPeso molecular:909.00 (free base)CTOP
CAS:<p>Potent μ-receptor antagonist, Ki=0.96nM, ineffective at δ (>10,000nM). Alters behavior in vivo, boosts K+ currents in rat neurons in vitro, μ-independent.</p>Fórmula:C50H67N11O11S2Pureza:98%Cor e Forma:SolidPeso molecular:1062.28Cebranopadol hemicitrate
CAS:<p>Cebranopadol hemicitrate is a NOP and opioid receptor agonist that targets human NOP, MOP, KOP, and δ-opioid peptide (DOP) receptors, with Ki/EC50 values of 0.9 nM/13 nM, 0.7 nM/1.2 nM, 2.6 nM/17 nM, and 18 nM/110 nM, respectively. It is used in studies of acute and chronic pain.</p>Cor e Forma:Solid[DPro10] Dynorphin A (1-11)acetate,porcine
<p>[DPro10] Dynorphin A (1-11)acetate,porcine is a highly potent κ-opioid receptor agonist with a Ki value of 0.13 nM.</p>Fórmula:C65H107N21O15Pureza:99.05%Cor e Forma:SoildPeso molecular:1422.7Nociceptin (1-13), amide
CAS:<p>Nociceptin (1-13), amide is a potent ORL1 (OP4) receptor agonist with a pEC50 of 7.9 for mouse vas deferens and a Ki of 0.75 nM for binding to rat forebrain</p>Fórmula:C61H100N22O15Pureza:98%Cor e Forma:SolidPeso molecular:1381.59UFP-101
CAS:<p>Strong, selective NOP receptor antagonist with pKi=10.24; >3000x selectivity over δ, μ, κ receptors; blocks nociceptin effects.</p>Fórmula:C82H138N32O21Pureza:98%Cor e Forma:SolidPeso molecular:1908.19[Arg14,Lys15]Nociceptin
CAS:<p>Potent NOP agonist (EC50 = 1 nM), >875x selective vs opioid receptors; outperforms nociceptin in vivo, increases pain perception, reduces movement.</p>Fórmula:C82H137N31O22Pureza:98%Cor e Forma:SolidPeso molecular:1909.18N-Desmethyl Loperamide
CAS:<p>N-Desmethyl Loperamide is the major metabolite of loperamide. It is also used as the precusor for radiolabelled loperamide.</p>Fórmula:C28H31ClN2O2Cor e Forma:SolidPeso molecular:463.01MT-7716 free base
CAS:<p>MT-7716: selective NOP agonist, potential in preventing alcohol abuse/relapse.</p>Fórmula:C27H28N4O2Pureza:98%Cor e Forma:SolidPeso molecular:440.54Neurotransmitter Receptor Compound Library
<p>A unique collection of 1513 neurotransmitter receptor compounds, can be used for HTS and HCS screening；</p>Cor e Forma:Odour SolidBAM-22P
CAS:<p>Bovine adrenal medulla docosapeptide (BAM-22P) is a potent opioid agonist, derived from the proenkephalin A gene, which is present in the adrenal medulla.</p>Fórmula:C130H184N38O31S2Pureza:98%Cor e Forma:SolidPeso molecular:2839.22TAN67
CAS:<p>TAN67 is the first effective selective non-peptide delta1 opioid receptor.</p>Fórmula:C23H26Br2N2OCor e Forma:SolidPeso molecular:506.282Boc-ypgflt(O-tbu)
CAS:<p>Boc-ypgflt(O-tbu) is a delta-receptor-selective opioid antagonist.</p>Fórmula:C44H64N6O11Cor e Forma:SolidPeso molecular:853.01N-terminally acetylated Endomorphin-1
<p>N-terminally acetylated Endomorphin-1 is a modified Endomorphin-1.</p>Fórmula:C36H40N6O6Pureza:98%Cor e Forma:SolidPeso molecular:652.74Opioid receptor agonist 1
<p>Opioid receptor agonist1 (Compound 2638-28) is an orally active opioid receptor agonist that shows strong affinity for MOR, DOR, and KOR, with Ki values of 5, 24, and 212 nM, respectively. It exhibits analgesic activity in both the mouse warm water tail-flick model and the acetic acid writhing model.</p>Fórmula:C32H45N5OCor e Forma:SolidPeso molecular:515.73(Rac)-SNC80
CAS:<p>(Rac)-SNC80, a racemic δ-opioid agonist (K i 1.78 nM), shows potential for treating various headache disorders.</p>Fórmula:C28H39N3O2Cor e Forma:SolidPeso molecular:449.63DAMGO (TFA)
CAS:<p>DAMGO is a selective peptide agonist of the µ-opioid receptor .</p>Fórmula:C28H36F3N5O8Pureza:98%Cor e Forma:SolidPeso molecular:627.61Deltorphin
CAS:<p>Deltorphin (Dermenkephalin) is Isolated from the skin of Phyllomedusa Sauvage. It also has an affinity to the opioid receptor.</p>Fórmula:C44H62N10O10S2Pureza:98.96%Cor e Forma:SolidPeso molecular:955.15AP-238
CAS:<p>AP-238 is a novel synthetic opioid (NSO) that acts as an agonist for the μ-opioid receptor (MOR), with an EC50 of 248 nM. Additionally, AP-238 exhibits analgesic properties.</p>Fórmula:C18H26N2OCor e Forma:SolidPeso molecular:286.41
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