Receptor opioide
Os receptores opioides são um grupo de receptores acoplados à proteína G que mediam os efeitos dos opioides endógenos e exógenos. Estes receptores desempenham um papel central na modulação da dor, regulação do humor e comportamentos aditivos. Agonistas e antagonistas dos receptores opioides são amplamente utilizados no manejo da dor e tratamento de dependências, bem como em pesquisas sobre distúrbios neurológicos e psiquiátricos. Na CymitQuimica, oferecemos uma seleção abrangente de moduladores de receptores opioides de alta qualidade para apoiar sua pesquisa em neurobiologia, manejo da dor e terapia de dependência.
Foram encontrados 298 produtos de "Receptor opioide"
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Trap-101 hydrochloride
CAS:<p>nociceptin/orphanin FQ (NOP) receptor antagonist</p>Fórmula:C24H36ClN3O2Pureza:98%Cor e Forma:SolidPeso molecular:434.02Frakefamide
CAS:<p>Frakefamide: potent analgesic, μ-selective agonist, non-CNS penetrating.</p>Fórmula:C30H34FN5O5Pureza:98%Cor e Forma:SolidPeso molecular:563.62Naloxonazine
CAS:<p>Naloxonazine, a potent, selective opiate mu-1 (μ1) antagonist, also influences leishmania through the modulation of host coding function.</p>Fórmula:C38H42N4O6Cor e Forma:SolidPeso molecular:650.76Deltakephalin
CAS:<p>Deltakephalin is a synthetic, potent specific opiate delta receptors agonist.</p>Fórmula:C34H48N6O10Pureza:98%Cor e Forma:SolidPeso molecular:700.78N-Benzylnaltrindole hydrochloride
CAS:δ2 opioid receptor antagonistFórmula:C33H33ClN2O3Pureza:98%Cor e Forma:SolidPeso molecular:541.08Mu opioid receptor antagonist 7
CAS:<p>Compound 24, also known as Mu opioid receptor antagonist 7, is a potent, centrally-acting µ-opioid receptor (µOR) antagonist with an inhibitory concentration (</p>Fórmula:C22H27ClN2O2Pureza:98%Cor e Forma:SolidPeso molecular:386.91μ opioid receptor agonist 3
CAS:<p>Compound 20, identified as μ opioid receptor agonist 3, is a potent µOR agonist that exhibits an EC50 value of 0.87 nM.</p>Fórmula:C22H28N2O2Pureza:98%Cor e Forma:SolidPeso molecular:352.47ADL-08-0011
CAS:<p>ADL-08-0011 is an metabolite of alvimopan.</p>Fórmula:C23H29NO3Cor e Forma:SolidPeso molecular:367.49CYT-1010
CAS:<p>CYT-1010, a mu-opioid receptor agonist; EC50: β-arrestin, 13.1 nM; cAMP, 0.0053 nM. Extracted from patent WO2013173730A2.</p>Fórmula:C35H40N6O5Pureza:98%Cor e Forma:SolidPeso molecular:624.73ICI 204448
CAS:<p>ICI 204448 is a potent and peripherally selective κ-opioid agonist.</p>Fórmula:C23H26Cl2N2O4Cor e Forma:SolidPeso molecular:465.37Icalcaprant
CAS:<p>Icalcaprant is a kappa-opioid receptor antagonist [1].</p>Fórmula:C23H26N4O3Pureza:98%Cor e Forma:SolidPeso molecular:406.48FK 33-824
CAS:<p>FK 33-824, a stable synthetic analog of methionine enkephalin, reversible with naloxone.</p>Fórmula:C29H41N5O7SPureza:98%Cor e Forma:SolidPeso molecular:603.73R-84760 hydrochloride
CAS:<p>R-84760, a potent κ-opioid receptor agonist, relieves tonic pain via supraspinal/spinal pathways, activating noradrenergic descent.</p>Fórmula:C19H25Cl3N2OSCor e Forma:SolidPeso molecular:435.84Norbinaltorphimine dihydrochloride
CAS:<p>Norbinaltorphimine dihydrochloride is a selective and potent κ opioid receptor antagonist that induces itch-associated responses in mice.</p>Fórmula:C40H45Cl2N3O6Pureza:98.17% - 99.88%Cor e Forma:SolidPeso molecular:734.71Isotodesnitazene
CAS:<p>Isotodesnitazene is an opioid compound that primarily targets the μ-opioid receptor (MOR). It exhibits EC50 values of 34.8 nM and 142 nM for MOR-βarr2 and MOR-mini-Gi, respectively. Isotodesnitazene can be utilized for research in opioid drugs.</p>Fórmula:C23H31N3OCor e Forma:SolidPeso molecular:365.51Riminkefon
CAS:<p>Riminkefon is a kappa opioid receptor agonist .</p>Fórmula:C38H57N7O6Cor e Forma:SolidPeso molecular:707.9Mu opioid receptor antagonist 8
CAS:<p>Muopioid Receptor Antagonist 8 (368) serves as an antagonist to the μ-opioid receptor, significantly inhibiting the activation of Gi induced by met-enkephalin at the µOR.</p>Fórmula:C36H35N3O4SCor e Forma:SolidPeso molecular:605.75Mu opioid receptor antagonist 3
<p>Potent, selective MOR antagonist (compound 26); crosses blood-brain barrier. Ki: 0.24 nM, EC50: 0.54 nM; for studying OUD.</p>Fórmula:C25H28N2O4SCor e Forma:SolidPeso molecular:452.57BU09059
CAS:BU09059 is a potent, selective, short-acting antagonist of the κ-opioid receptor (KOR).Fórmula:C28H37N3O5Pureza:98%Cor e Forma:SolidPeso molecular:495.616β-Naltrexol
CAS:<p>6β-Naltrexol is a peripherally selective opioid antagonist that reduces constipation from opioids while minimizing central nervous system effects.</p>Fórmula:C20H25NO4Pureza:99.933%Cor e Forma:SolidPeso molecular:343.42
