Receptor opioide
Os receptores opioides são um grupo de receptores acoplados à proteína G que mediam os efeitos dos opioides endógenos e exógenos. Estes receptores desempenham um papel central na modulação da dor, regulação do humor e comportamentos aditivos. Agonistas e antagonistas dos receptores opioides são amplamente utilizados no manejo da dor e tratamento de dependências, bem como em pesquisas sobre distúrbios neurológicos e psiquiátricos. Na CymitQuimica, oferecemos uma seleção abrangente de moduladores de receptores opioides de alta qualidade para apoiar sua pesquisa em neurobiologia, manejo da dor e terapia de dependência.
Foram encontrados 298 produtos de "Receptor opioide"
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β-Naltrexamine dihydrochloride
CAS:<p>β-Naltrexamine dihydrochloride is an orally administered, irreversible opioid receptor antagonist. Its derivatives exhibit optimised subtype selectivity and can be used for pain research.</p>Fórmula:C20H28Cl2N2O3Pureza:95.98%Cor e Forma:SoildPeso molecular:415.35Biphalin TFA
CAS:<p>Biphalin TFA is an opioid peptide analog that penetrates the blood-brain barrier (BBB) and encompasses two active enkephalin pharmacophores.</p>Fórmula:C46H56N10O10·xC2HF3O2Pureza:98%Cor e Forma:SolidPeso molecular:909.00 (free base)CTOP
CAS:<p>Potent μ-receptor antagonist, Ki=0.96nM, ineffective at δ (>10,000nM). Alters behavior in vivo, boosts K+ currents in rat neurons in vitro, μ-independent.</p>Fórmula:C50H67N11O11S2Pureza:98%Cor e Forma:SolidPeso molecular:1062.28Cebranopadol hemicitrate
CAS:<p>Cebranopadol hemicitrate is a NOP and opioid receptor agonist that targets human NOP, MOP, KOP, and δ-opioid peptide (DOP) receptors, with Ki/EC50 values of 0.9 nM/13 nM, 0.7 nM/1.2 nM, 2.6 nM/17 nM, and 18 nM/110 nM, respectively. It is used in studies of acute and chronic pain.</p>Cor e Forma:Solid[DPro10] Dynorphin A (1-11)acetate,porcine
<p>[DPro10] Dynorphin A (1-11)acetate,porcine is a highly potent κ-opioid receptor agonist with a Ki value of 0.13 nM.</p>Fórmula:C65H107N21O15Pureza:99.05%Cor e Forma:SoildPeso molecular:1422.7Nociceptin (1-13), amide
CAS:<p>Nociceptin (1-13), amide is a potent ORL1 (OP4) receptor agonist with a pEC50 of 7.9 for mouse vas deferens and a Ki of 0.75 nM for binding to rat forebrain</p>Fórmula:C61H100N22O15Pureza:98%Cor e Forma:SolidPeso molecular:1381.59UFP-101
CAS:<p>Strong, selective NOP receptor antagonist with pKi=10.24; >3000x selectivity over δ, μ, κ receptors; blocks nociceptin effects.</p>Fórmula:C82H138N32O21Pureza:98%Cor e Forma:SolidPeso molecular:1908.19[Arg14,Lys15]Nociceptin
CAS:<p>Potent NOP agonist (EC50 = 1 nM), >875x selective vs opioid receptors; outperforms nociceptin in vivo, increases pain perception, reduces movement.</p>Fórmula:C82H137N31O22Pureza:98%Cor e Forma:SolidPeso molecular:1909.18N-Desmethyl Loperamide
CAS:<p>N-Desmethyl Loperamide is the major metabolite of loperamide. It is also used as the precusor for radiolabelled loperamide.</p>Fórmula:C28H31ClN2O2Cor e Forma:SolidPeso molecular:463.01MT-7716 free base
CAS:<p>MT-7716: selective NOP agonist, potential in preventing alcohol abuse/relapse.</p>Fórmula:C27H28N4O2Pureza:98%Cor e Forma:SolidPeso molecular:440.54Neurotransmitter Receptor Compound Library
<p>A unique collection of 1513 neurotransmitter receptor compounds, can be used for HTS and HCS screening；</p>Cor e Forma:Odour SolidBAM-22P
CAS:<p>Bovine adrenal medulla docosapeptide (BAM-22P) is a potent opioid agonist, derived from the proenkephalin A gene, which is present in the adrenal medulla.</p>Fórmula:C130H184N38O31S2Pureza:98%Cor e Forma:SolidPeso molecular:2839.22TAN67
CAS:<p>TAN67 is the first effective selective non-peptide delta1 opioid receptor.</p>Fórmula:C23H26Br2N2OCor e Forma:SolidPeso molecular:506.282Boc-ypgflt(O-tbu)
CAS:<p>Boc-ypgflt(O-tbu) is a delta-receptor-selective opioid antagonist.</p>Fórmula:C44H64N6O11Cor e Forma:SolidPeso molecular:853.01N-terminally acetylated Endomorphin-1
<p>N-terminally acetylated Endomorphin-1 is a modified Endomorphin-1.</p>Fórmula:C36H40N6O6Pureza:98%Cor e Forma:SolidPeso molecular:652.74Opioid receptor agonist 1
<p>Opioid receptor agonist1 (Compound 2638-28) is an orally active opioid receptor agonist that shows strong affinity for MOR, DOR, and KOR, with Ki values of 5, 24, and 212 nM, respectively. It exhibits analgesic activity in both the mouse warm water tail-flick model and the acetic acid writhing model.</p>Fórmula:C32H45N5OCor e Forma:SolidPeso molecular:515.73(Rac)-SNC80
CAS:<p>(Rac)-SNC80, a racemic δ-opioid agonist (K i 1.78 nM), shows potential for treating various headache disorders.</p>Fórmula:C28H39N3O2Cor e Forma:SolidPeso molecular:449.63DAMGO (TFA)
CAS:<p>DAMGO is a selective peptide agonist of the µ-opioid receptor .</p>Fórmula:C28H36F3N5O8Pureza:98%Cor e Forma:SolidPeso molecular:627.61Deltorphin
CAS:<p>Deltorphin (Dermenkephalin) is Isolated from the skin of Phyllomedusa Sauvage. It also has an affinity to the opioid receptor.</p>Fórmula:C44H62N10O10S2Pureza:98.96%Cor e Forma:SolidPeso molecular:955.15AP-238
CAS:<p>AP-238 is a novel synthetic opioid (NSO) that acts as an agonist for the μ-opioid receptor (MOR), with an EC50 of 248 nM. Additionally, AP-238 exhibits analgesic properties.</p>Fórmula:C18H26N2OCor e Forma:SolidPeso molecular:286.41
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