Receptor opioide
Os receptores opioides são um grupo de receptores acoplados à proteína G que mediam os efeitos dos opioides endógenos e exógenos. Estes receptores desempenham um papel central na modulação da dor, regulação do humor e comportamentos aditivos. Agonistas e antagonistas dos receptores opioides são amplamente utilizados no manejo da dor e tratamento de dependências, bem como em pesquisas sobre distúrbios neurológicos e psiquiátricos. Na CymitQuimica, oferecemos uma seleção abrangente de moduladores de receptores opioides de alta qualidade para apoiar sua pesquisa em neurobiologia, manejo da dor e terapia de dependência.
Foram encontrados 330 produtos para "Receptor opioide".
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β-Endorphin, equine
CAS:Endorphin Beta is A substance produced in the brain, especially in the pituitary gland, Endorphin Beta blocks the sensation of pain.Fórmula:C154H248N42O44SPureza:98%Cor e Forma:SolidPeso molecular:3423.94KOR agonist 5
KOR agonist 5 (Compound 10a) is both a KOR/MOR modulator, exhibiting agonistic effects on KOR and antagonistic effects on MOR. It effectively blocks morphine-induced antinociception and gastrointestinal motility inhibition. KOR agonist 5 is applicable in research related to substance use disorder (SUD).Fórmula:C38H38N2O5Cor e Forma:SolidPeso molecular:602.72MT-7716 hydrochloride
CAS:MT-7716 hydrochloride is a selective agonist of non-peptide nociceptin receptor (NOP)Fórmula:C27H29ClN4O2Pureza:98%Cor e Forma:SolidPeso molecular:477(S,S)-J-113397
CAS:(S,S)-J-113397 is an isomer of J-113397 . J-113397 is an Opioid Receptor antagonist [1] .Fórmula:C24H37N3O2Cor e Forma:SolidPeso molecular:399.57β-Lipotropin (61-69)
CAS:β-Lipotropin (61-69) is a potent opioid agonist [1] [2] .Fórmula:C45H66N10O15SCor e Forma:SolidPeso molecular:1019.13SB 205607 dihydrobromide
CAS:non-peptide δ1 opioid receptor agonistFórmula:C23H24N2OPureza:98%Cor e Forma:SolidPeso molecular:344.45HINT1-IN-1
HINT1-IN-1 (compound 8) is an inhibitor of histidine triad nucleotide-binding protein 1 (HINT1) with a Ki of 1.14 μM. It influences the cross-regulation between μ-opioid receptors (MOR) and NMDA receptors (NMDAR).Fórmula:C23H24N8O5Cor e Forma:SolidPeso molecular:492.49α-Neoendorphin (1-8)
CAS:α-Neoendorphin (1-8) is a 8-amino acid peptide derived from the N-terminal of α-Neoendorphin.Fórmula:C49H70N12O11Pureza:98%Cor e Forma:SolidPeso molecular:1003.15Deltorphin acetate
Deltorphin acetate is a substance obtained from the skin secretions of a frog, Phyllomedusa bicolor and shows high selectivity and affinity for δ-opioidFórmula:C46H66N10O12S2Pureza:98.93%Cor e Forma:SolidPeso molecular:1015.21Ref: TM-T20166L
1mg175,00€5mg394,00€10mg590,00€25mg1.060,00€50mg1.591,00€100mg2.387,00€200mg3.580,00€[Met5]-Enkephalin, amide
CAS:[Met5]-Enkephalin, amide activates δ and ζ opioid receptors; has multiple forms and varying plasma levels.Fórmula:C27H36N6O6SPureza:98%Cor e Forma:SolidPeso molecular:572.68Neurotransmitter Receptor Compound Library
A unique collection of 1513 neurotransmitter receptor compounds, can be used for HTS and HCS screening；
Cor e Forma:Odour Solid[Leu5]-Enkephalin
CAS:[Leu5]-Enkephalin (Leu-enkephalin) is an endogenous neuropeptide involved in nociception and an agonist of δ-opioid and μ-opioid receptors (Kis = 4.0 and 3.4 nMFórmula:C28H37N5O7Pureza:99.65% - 99.87%Cor e Forma:White SolidPeso molecular:555.62BMS-986121
CAS:BMS-986121 is a selective positive allosteric modulator (PAM) of the μ opioid receptor with analgesic effects.Fórmula:C15H9Cl2N3O2SPureza:99.67%Cor e Forma:Yellow SolidPeso molecular:366.22Porcine dynorphin A(1-13)
CAS:Porcine dynorphin A (1-13) is a potent κ opioid receptor agonist; it's antinociceptive and raises [Ca2+]i in neurons like NMDA.Fórmula:C75H126N24O15Pureza:98%Cor e Forma:SolidPeso molecular:1603.95Asimadoline
CAS:Asimadoline (EMD-61753) is a proprietary small molecule therapeutic, originally discovered by Merck KGaA of Darmstadt, Germany.Fórmula:C27H30N2O2Cor e Forma:SolidPeso molecular:414.54BAN ORL 24 dihydrochloride
CAS:BAN ORL 24 dihydrochloride is a highly potent nociceptin/orphan FQ (N/OFQ) receptor (NOP) antagonist that can be used to study neurological diseases.Fórmula:C27H37Cl2N3O2Pureza:95.03%Cor e Forma:SolidPeso molecular:506.51Loperamide phenyl
CAS:Loperamide phenyl, an impurity detected in Loperamide, is an opioid receptor agonist.Fórmula:C35H37ClN2O2Cor e Forma:SolidPeso molecular:553.14Alvimopan dihydrate (LY246736 dihydrate)
CAS:Alvimopan dihydrate is a potent, oral μ-opioid receptor blocker (IC50 1.7 nM, Ki 0.47 nM) used in postoperative ileus research.Fórmula:C25H36N2O6Cor e Forma:SolidPeso molecular:460.56Endomorphin 2 TFA
CAS:Endomorphin 2 TFA, displays reasonable affinities for kappa3 binding sites, with Ki value between 20 and 30 nM.Fórmula:C34H38F3N5O7Cor e Forma:SolidPeso molecular:685.69Naloxegol oxalate
CAS:Naloxegol oxalate (NKTR-118) is a peripherally-selective opioid antagonist for the treatment of opioid-induced constipation.Fórmula:C36H55NO15Pureza:99.67% - >99.99%Cor e Forma:SolidPeso molecular:741.83
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