Receptor opioide
Os receptores opioides são um grupo de receptores acoplados à proteína G que mediam os efeitos dos opioides endógenos e exógenos. Estes receptores desempenham um papel central na modulação da dor, regulação do humor e comportamentos aditivos. Agonistas e antagonistas dos receptores opioides são amplamente utilizados no manejo da dor e tratamento de dependências, bem como em pesquisas sobre distúrbios neurológicos e psiquiátricos. Na CymitQuimica, oferecemos uma seleção abrangente de moduladores de receptores opioides de alta qualidade para apoiar sua pesquisa em neurobiologia, manejo da dor e terapia de dependência.
Foram encontrados 298 produtos de "Receptor opioide"
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LY2940094 tartrate
CAS:<p>LY-2940094, a nociceptin receptor antagonist, is used potentially for the treatment of major depressive disorder and alcoholism.</p>Fórmula:C26H29ClF2N4O8SCor e Forma:SolidPeso molecular:631.04MCOPPB triHydrochloride
CAS:<p>MCOPPB triHydrochloride (MCOPPB 3HCl) is a nociceptin receptor agonist.</p>Fórmula:C26H43Cl3N4Pureza:99.89% - 99.91%Cor e Forma:SolidPeso molecular:518.01Deltorphin I
CAS:<p>Deltorphin I is an agonist of δ-opioid receptor.</p>Fórmula:C37H52N8O10Pureza:>99.99%Cor e Forma:SolidPeso molecular:768.86Endomorphin 2
CAS:<p>EM-2 reduces sEPSC frequency/amplitude in lamina IX motoneurons; CTOP reverses this. EM-2-IR affects limb muscles via presynaptic/postsynaptic mechanisms.</p>Fórmula:C32H37N5O5Pureza:99.64%Cor e Forma:SolidPeso molecular:571.67EST73502 HCl
CAS:<p>EST73502 is an agonist of μ-opioid receptor(Ki = 64 nM) agonist and an antagonist of σ1 receptor (Ki = 118 nM). EST73502 displays antinociceptive activity.</p>Fórmula:C19H27ClF2N2O2Pureza:99.96%Cor e Forma:SolidPeso molecular:388.88JTC-801
CAS:<p>JTC-801 is a selective opioid receptor-like1 (ORL1) receptor antagonist with IC50 of 94 nM, weakly inhibits receptors δ, κ, and μ.</p>Fórmula:C26H25N3O2·HClPureza:99.27% - 99.59%Cor e Forma:SolidPeso molecular:447.96BMS-986122
CAS:<p>BMS-986122 (BMS 986122) is a positive allosteric modulator of μ-opioid receptors that increases β-arrestin recruitment stimulated by endomorphin 1 in U2OS-OPRM1</p>Fórmula:C16H15BrClNO3S2Pureza:98.42%Cor e Forma:SolidPeso molecular:448.78Sinomenine
CAS:<p>Sinomenine (Kukoline) is a pure alkaloid isolated from the Sinomenium acutum, is utilized in the treatment of rheumatism and arthritis.</p>Fórmula:C19H23NO4Pureza:99.02% - 99.73%Cor e Forma:White PowderPeso molecular:329.39ADL-5747 (HCl)
CAS:<p>ADL-5747, an opioid delta receptor agonist, is used potentially for the treatment of pain.</p>Fórmula:C24H29ClN2O3Cor e Forma:SolidPeso molecular:428.95PZM21
CAS:<p>PZM21 is an effective and selective μ opioid receptor agonist (EC50: 1.8 nM).</p>Fórmula:C19H27N3O2SPureza:99.93% - >99.99%Cor e Forma:SolidPeso molecular:361.5BMS986187
CAS:BMS986187 is a novel Potent and Selective Positive Allosteric Modulators of the delta-Opioid Receptor.Fórmula:C31H34O4Pureza:99.09%Cor e Forma:SolidPeso molecular:470.6GR103545
CAS:<p>GR103545 is a selective agonist of the κ-opioid receptor, which is a radiotracer that can be used as in vivo imaging.</p>Fórmula:C23H29Cl2N3O7Pureza:99.75%Cor e Forma:SolidPeso molecular:530.4LY2795050
CAS:<p>LY2795050 is a novel specific κ-Opioid Receptor antagonist (IC50: 0.72 nM).</p>Fórmula:C23H22ClN3O2Pureza:97.77%Cor e Forma:SolidPeso molecular:407.89DAMGO
CAS:<p>DAMGO (DAGO) is an opioid receptor agonist with the ability to affect the locomotive activity in rodents.</p>Fórmula:C26H35N5O6Pureza:98.83% - 99.92%Cor e Forma:SolidPeso molecular:513.59Adrenorphin 3TFA(88377-68-8(free base))
<p>Adrenorphin 3TFA(88377-68-8(free base)) (Metorphamide) is an agonist of μ-opioid receptor(Ki :12 nM).</p>Fórmula:C50H72N15O15SPureza:>99.99%Cor e Forma:SolidPeso molecular:1326.26[D-Ala2]leucine-enkephalin
CAS:<p>[D-Ala2]-Leucine enkephalin is a delta opioid agonist used to study the signaling pathway of delta opioid receptors.</p>Fórmula:C29H39N5O7Pureza:98.06%Cor e Forma:SolidPeso molecular:569.65Difelikefalin acetate
CAS:Difelikefalin acetate (CR 845 acetate) is a peripherally restricted kappa opioid receptor agonist.Fórmula:C38H57N7O8Pureza:99.55%Cor e Forma:SolidPeso molecular:739.9BAM 22P acetate
<p>BAM 22P acetate is a potent opioid agonist.</p>Fórmula:C132H188N38O33S2Pureza:99.87%Cor e Forma:SoildPeso molecular:2899.27Dynorphin A acetate(80448-90-4 free base)
<p>Dynorphin A acetate is an Endogenous kappa receptor agonist.</p>Fórmula:C101H159N31O25Pureza:99.69%Cor e Forma:SolidPeso molecular:2207.58(D-Ser2)-Leu-Enkephalin-Thr
<p>(D-Ser2)-Leu-Enkephalin-Thr is a delta selective agent of opioid receptor and shows analgesic effects.</p>Fórmula:C33H46N6O10Pureza:94.17%Cor e Forma:SoildPeso molecular:686.75
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