Receptor opioide
Os receptores opioides são um grupo de receptores acoplados à proteína G que mediam os efeitos dos opioides endógenos e exógenos. Estes receptores desempenham um papel central na modulação da dor, regulação do humor e comportamentos aditivos. Agonistas e antagonistas dos receptores opioides são amplamente utilizados no manejo da dor e tratamento de dependências, bem como em pesquisas sobre distúrbios neurológicos e psiquiátricos. Na CymitQuimica, oferecemos uma seleção abrangente de moduladores de receptores opioides de alta qualidade para apoiar sua pesquisa em neurobiologia, manejo da dor e terapia de dependência.
Foram encontrados 298 produtos de "Receptor opioide"
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BMS986187
CAS:<p>BMS986187 is a novel Potent and Selective Positive Allosteric Modulators of the delta-Opioid Receptor.</p>Fórmula:C31H34O4Pureza:99.09%Cor e Forma:SolidPeso molecular:470.6GR103545
CAS:<p>GR103545 is a selective agonist of the κ-opioid receptor, which is a radiotracer that can be used as in vivo imaging.</p>Fórmula:C23H29Cl2N3O7Pureza:99.75%Cor e Forma:SolidPeso molecular:530.4LY2795050
CAS:<p>LY2795050 is a novel specific κ-Opioid Receptor antagonist (IC50: 0.72 nM).</p>Fórmula:C23H22ClN3O2Pureza:97.77%Cor e Forma:SolidPeso molecular:407.89DAMGO
CAS:<p>DAMGO (DAGO) is an opioid receptor agonist with the ability to affect the locomotive activity in rodents.</p>Fórmula:C26H35N5O6Pureza:98.83% - 99.92%Cor e Forma:SolidPeso molecular:513.59Adrenorphin 3TFA(88377-68-8(free base))
<p>Adrenorphin 3TFA(88377-68-8(free base)) (Metorphamide) is an agonist of μ-opioid receptor(Ki :12 nM).</p>Fórmula:C50H72N15O15SPureza:>99.99%Cor e Forma:SolidPeso molecular:1326.26[D-Ala2]leucine-enkephalin
CAS:<p>[D-Ala2]-Leucine enkephalin is a delta opioid agonist used to study the signaling pathway of delta opioid receptors.</p>Fórmula:C29H39N5O7Pureza:98.06%Cor e Forma:SolidPeso molecular:569.65Difelikefalin acetate
CAS:<p>Difelikefalin acetate (CR 845 acetate) is a peripherally restricted kappa opioid receptor agonist.</p>Fórmula:C38H57N7O8Pureza:99.55%Cor e Forma:SolidPeso molecular:739.9BAM 22P acetate
<p>BAM 22P acetate is a potent opioid agonist.</p>Fórmula:C132H188N38O33S2Pureza:99.87%Cor e Forma:SoildPeso molecular:2899.27Dynorphin A acetate(80448-90-4 free base)
<p>Dynorphin A acetate is an Endogenous kappa receptor agonist.</p>Fórmula:C101H159N31O25Pureza:99.69%Cor e Forma:SolidPeso molecular:2207.58(D-Ser2)-Leu-Enkephalin-Thr
<p>(D-Ser2)-Leu-Enkephalin-Thr is a delta selective agent of opioid receptor and shows analgesic effects.</p>Fórmula:C33H46N6O10Pureza:94.17%Cor e Forma:SoildPeso molecular:686.75Porcine dynorphin A(1-13) acetate
<p>Porcine dynorphin A(1-13) acetate is a potent κ-opioid agonist with antinociceptive properties, increasing [Ca2+]i like NMDA.</p>Fórmula:C77H130N24O17Pureza:99.14%Cor e Forma:SolidPeso molecular:1664Dynorphin B (1-13) acetate(83335-41-5 free base)
<p>Dynorphin B (1-13) acetate acts as an agonist on opioid κ-receptor.</p>Fórmula:C76H119N21O19Pureza:99.72%Cor e Forma:SolidPeso molecular:1630.89CTAP(TFA) (103429-32-9 free base)
<p>CTAP(TFA) (103429-32-9 free base) is a potent, highly selective, and brain-penetrant antagonist of the μ-opioid receptor with IC50 of 3.5 nM.</p>Fórmula:C53H70F3N13O13S2Pureza:99.62%Cor e Forma:SolidPeso molecular:1218.33Nociceptin (1-13) amide TFA
<p>Nociceptin (1-13), amide: ORL1 receptor agonist, pEC50 7.9 (mouse vas deferens), Ki 0.75 nM (rat forebrain binding).</p>Fórmula:C63H101F3N22O17Pureza:97.64%Cor e Forma:SolidPeso molecular:1495.61Ac-RYYRIK-NH2 acetate
<p>Ac-RYYRIK-NH2 acetate is an agonist at nociceptin/orphanin FQ(noc/OFQ) receptors, affecting spontaneous locomotor activity.</p>Fórmula:C46H74N14O11Pureza:99.84%Cor e Forma:SolidPeso molecular:999.17[Met5]-Enkephalin, amide TFA
<p>[Met5]-Enkephalin, amide TFA (5-Methionine-enkephalin amide (TFA)) is a δ opioid receptors agonist as well as putative ζ (zeta) opioid receptors.</p>Fórmula:C29H37F3N6O8SPureza:99.81%Cor e Forma:SolidPeso molecular:686.7Leuphasyl TFA
CAS:<p>Leuphasyl TFA: a long-lasting, degradation-resistant peptide & δ-opioid receptor agonist for signaling research.</p>Fórmula:C31H40F3N5O9Pureza:98.79%Cor e Forma:SolidPeso molecular:683.67Orphanin FQ(1-11) acetate(178249-41-7 free base)
<p>Nociceptin peptide fragment (1-11 aa), potent ORL1/KOR-3 agonist (Ki=55 nM), non-opioid, analgesic in mice.</p>Fórmula:C51H79N15O16Pureza:95.54%Cor e Forma:SolidPeso molecular:1158.26N-terminally acetylated Leu-enkephalin
<p>Leu-enkephalin, an endogenous 5-amino acid peptide, activates opioid receptors; its acetylated form exists.</p>Fórmula:C30H39N5O8Pureza:>99.99%Cor e Forma:SolidPeso molecular:597.66b-Casomorphin (1-3) Acetate
<p>b-Casomorphin (1-3) Acetate is a tri-peptide with an opioid effect.</p>Fórmula:C25H31N3O7Pureza:98.99%Cor e Forma:SolidPeso molecular:485.53Ac-RYYRWK-NH2 acetate
<p>Ac-RYYRWK-NH2 acetate is a potent partial agonist of the nociceptin receptor(NOP), which is the endogenous ORL1 receptor agonist.</p>Fórmula:C51H73N15O11Pureza:98.59%Cor e Forma:SolidPeso molecular:1072.22Hemorphin-7 acetate(152685-85-3 free base)
<p>Hemorphin-7 acetate is a hemorphin peptide, an endogenous opioid peptide derived from the β-chain of hemoglobin.</p>Fórmula:C51H68N12O13Pureza:99.66%Cor e Forma:SolidPeso molecular:1057.16Dynorphin A 1-10 acetate(79994-24-4 free base)
<p>Dynorphin A (1-10) acetate is an endogenous opioid neuropeptide, binds to extracellular loop 2 of the κ-opioid receptor.</p>Fórmula:C59H95N19O14Pureza:99.88%Cor e Forma:SolidPeso molecular:1294.53[Leu5]-Enkephalin, amide acetate
<p>[Leu5]-Enkephalin, amide acetate is a δ opioid receptor agonist.</p>Fórmula:C30H42N6O8Pureza:99.36%Cor e Forma:SolidPeso molecular:614.69Nociceptin (1-7) acetate
<p>Nociceptin (1-7) acetate is a potent agonist of opioid receptor-like 1 (ORL1) receptor.</p>Fórmula:C31H41N7O9Pureza:98.92%Cor e Forma:SoildPeso molecular:655.7AR-M 1000390 hydrochloride
CAS:<p>ARM-390 HCl is a δ-opioid receptor agonist, brain-penetrant, nonpeptidic, prevents hyperalgesia without desensitization. Derived from SNC 80.</p>Fórmula:C23H29ClN2OPureza:98.66%Cor e Forma:SolidPeso molecular:384.94Bisacodyl
CAS:<p>Bisacodyl (Fenilaxan) is a diphenylmethane stimulant laxative used for the treatment of constipation and for bowel evacuation.</p>Fórmula:C22H19NO4Pureza:99.45% - 99.78%Cor e Forma:Smaller Than 50 Microns Predominate White To Off-White Crystalline PowderPeso molecular:361.39BRL 52537 hydrochloride
CAS:<p>BRL 52537 hydrochloride: selective KOR agonist, may protect against ischemic brain injury, used in stroke and heart attack research.</p>Fórmula:C18H25Cl3N2OPureza:99.04%Cor e Forma:SolidPeso molecular:391.76Aticaprant
CAS:<p>Aticaprant (CERC-501) is a potent and centrally-penetrant antagonist of the kappa-opioid receptor (Ki: 0.807 nM).Cost-effective and quality-assured.</p>Fórmula:C26H27FN2O2Pureza:99.53% - 99.93%Cor e Forma:SolidPeso molecular:418.5Deltorphin 2
CAS:<p>Deltorphin 2 ([D-Ala2]-Deltorphin II) is an agonist of δ opioid receptor with an IC50 of 1 nM.</p>Fórmula:C38H54N8O10Pureza:>99.99%Cor e Forma:SolidPeso molecular:782.88BMS986188
CAS:<p>BMS986188 is a novel Potent and Selective Positive Allosteric Modulator of the delta-Opioid Receptor.</p>Fórmula:C30H31BrO4Pureza:98.76%Cor e Forma:SolidPeso molecular:535.47BW-180C
CAS:<p>BW-180C (DADLE) is a prototypical δ-opioid receptor agonist that also displays activity at the μ-opioid receptor. Displays antinociceptive activity in vivo.</p>Fórmula:C29H39N5O7Pureza:>99.99%Cor e Forma:SolidPeso molecular:569.65DAMGO TFA (78123-71-4(Free base))
<p>DAMGO TFA (78123-71-4(Free base)) is a potent and selective agonist of the Mu-opioid receptor.Cost-effective and quality-assured.</p>Fórmula:C28H36F3N5O8Pureza:98.67% - 99.76%Cor e Forma:SolidPeso molecular:627.6Asimadoline hydrochloride
CAS:<p>Asimadoline HCl (EMD-61753) is a kappa-opioid receptor agonist for pruritus and IBS treatment.</p>Fórmula:C27H31ClN2O2Pureza:98.94% - 99.32%Cor e Forma:SolidPeso molecular:451.01Endomorphin 1
CAS:<p>Endomorphin 1 is a high affinity and selective agonist of the μ-opioid receptor and displays reasonable affinities for kappa3 binding sites (Ki: 20~30 nM).</p>Fórmula:C34H38N6O5Pureza:95.92%Cor e Forma:Solid (Solid Powder )Peso molecular:610.7Salvinorin A
CAS:<p>Salvinorin A is a non-nitrogenous κ-opioid selective agonist.</p>Fórmula:C23H28O8Pureza:99.06%Cor e Forma:SolidPeso molecular:432.46GRT2932Q
CAS:<p>GRT2932Q is a nonpeptidic agonist of the opioid receptor-like 1 (ORL1) [1].</p>Fórmula:C25H26ClN3OCor e Forma:SolidPeso molecular:419.95BMS-986124
CAS:<p>BMS-986124 is an allosteric modulator of the μ-Opioid Receptor.</p>Fórmula:C16H15BrClNO3S2Cor e Forma:SolidPeso molecular:448.78DDD028
CAS:<p>DDD-028 is a potential non-opioid and non-cannabinoid analgesic. It was used for treating neuropathic and inflammatory pain.</p>Fórmula:C20H20N2Pureza:98%Cor e Forma:SolidPeso molecular:288.39GSK1521498
CAS:<p>GSK1521498 is a selective antagonist of the μ-opioid receptor (MOR).</p>Fórmula:C24H23F2N4O4PPureza:98%Cor e Forma:SolidPeso molecular:500.43LY 281217
CAS:<p>LY 281217, an organic opioid agonist, can produce analgesic effects in mice.</p>Fórmula:C32H42N4O6Pureza:98%Cor e Forma:SolidPeso molecular:578.7SR8993
CAS:<p>SR8993 is a highly selective, brain-penetrant agonist of the nociceptin receptor.</p>Fórmula:C25H37FN4Pureza:98%Cor e Forma:SolidPeso molecular:412.59ADL-5859 HCl
CAS:<p>ADL-5859 is a delta-opioid receptor agonist.</p>Fórmula:C24H28N2O3Pureza:98%Cor e Forma:SolidPeso molecular:392.49LY 164929
CAS:<p>LY 164929 is a highly selective ligand for the lower affinity [3H]D-Ala2-D-Leu-5-enkephalin binding site.</p>Fórmula:C28H41N5O4Cor e Forma:SolidPeso molecular:511.66GSK1521498 free base
CAS:<p>GSK1521498 free base is an effective and selective μ-opioid receptor antagonist with potential applications in obesity, alcoholism, and drug addiction.</p>Fórmula:C24H20F2N4Pureza:99.85%Cor e Forma:SolidPeso molecular:402.44ML 190
CAS:<p>ML 190 is a potent and selective κ opioid receptor (KOR) antagonist (Ki=129 nM), exhibiting an IC50=150 nM in β-arrestin assays, drug addiction.</p>Fórmula:C27H32N6O3Pureza:99.88%Cor e Forma:SolidPeso molecular:488.58BW 373U86
CAS:<p>BW373U86 (SNC86), a δ-opioid receptor agonist, demonstrates potent activity with an IC50 value of 1.49 nM and has shown to exhibit antidepressant-like effects [</p>Fórmula:C27H37N3O2Cor e Forma:SolidPeso molecular:435.6GSK1521498 free base (hydrochloride)
CAS:<p>GSK1521498 free base (hydrochloride) is a selective antagonist of the μ-opioid receptor (MOR).</p>Fórmula:C24H21ClF2N4Pureza:98%Cor e Forma:SolidPeso molecular:438.9Endomorphin 1 acetate
CAS:<p>Endomorphin 1 acetate is a μ-opioid receptor agonist with antinociceptive and analgesic effects and can be used to study neurological diseases.</p>Fórmula:C36H42N6O7Cor e Forma:SolidPeso molecular:670.75CP-866087
CAS:<p>CP-866087 is a novel, potent and selective mu-opioid receptor antagonist for the study of female sexual dysfunction.</p>Fórmula:C24H28N2O2Pureza:99.56% - >99.99%Cor e Forma:SoildPeso molecular:376.49
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