Receptor de Bradicinina
Os receptores de bradicinina são GPCRs que mediam os efeitos da bradicinina, um peptídeo envolvido em respostas inflamatórias, sensação de dor e regulação da pressão arterial. Existem dois principais tipos de receptores de bradicinina, B1 e B2, cada um desempenhando papéis distintos em processos fisiopatológicos. Antagonistas dos receptores de bradicinina são usados no tratamento de condições como angioedema hereditário, dor crônica e hipertensão. Na CymitQuimica, oferecemos uma variedade de moduladores de receptores de bradicinina de alta qualidade para apoiar sua pesquisa em inflamação, manejo da dor e biologia cardiovascular.
Foram encontrados 59 produtos de "Receptor de Bradicinina"
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Anatibant 2HCl
CAS:<p>Anatibant 2HCl is a small molecule bradykinin B2 receptor antagonist for the treatment of neurological disorders and may be used in the study of brain injury.</p>Fórmula:C34H36Cl2N6O5S·2ClHPureza:99.17% - 99.58%Cor e Forma:SoildPeso molecular:784.58[Des-Arg9]-Bradykinin acetate
CAS:<p>[Des-Arg9]-Bradykinin acetate is a selective agonist of Bradykinin B1 receptor.</p>Fórmula:C46H65N11O12Pureza:99.05%Cor e Forma:SolidPeso molecular:964.07Fasitibant chloride
CAS:<p>Fasitibant chloride, a potent B2R blocker, alleviates pain and swelling in arthritis.</p>Fórmula:C36H49Cl3N6O6SCor e Forma:SolidPeso molecular:800.23Icatibant
CAS:<p>Icatibant is a selective and specific antagonist of the bradykinin B2 receptor (IC50 and Ki: 1.07 nM and 0.798 nM respectively).</p>Fórmula:C59H89N19O13SPureza:98%Cor e Forma:White SolidPeso molecular:1304.52[Phe8Ψ(CH-NH)-Arg9]-Bradykinin
CAS:<p>Selective bradykinin B2 receptor agonist that is resistant to carboxypeptidase cleavage.</p>Fórmula:C50H75N15O10Pureza:98%Cor e Forma:SolidPeso molecular:1046.23Bombinakinin M
CAS:<p>Potent, selective bradykinin receptor agonist 50x stronger than bradykinin, contracts guinea pig ileum muscle at EC50 4.0 nM.</p>Fórmula:C100H159N31O24Pureza:98%Cor e Forma:SolidPeso molecular:2179.55Lys-(Des-Arg9,Leu8)-Bradykinin
CAS:<p>Lys-(Des-Arg9,Leu8)-Bradykinin is a selective antagonist of the bradykinin B1 receptor [1].</p>Fórmula:C47H75N13O11Pureza:98%Cor e Forma:SolidPeso molecular:998.18(Hyp³)-Bradykinin acetate
<p>(Hyp³)-Bradykinin acetate is an agonist of bradykinin B2 receptor and stimulates inositol phosphate production in cultured human fibroblasts.</p>Fórmula:C52H77N15O14Pureza:99.46%Cor e Forma:SolidPeso molecular:1136.26Sar-[D-Phe8]-des-Arg9-Bradykinin
CAS:<p>Potent bradykinin B1 agonist, EC50 = 9.02 nM, enzyme resistant, induces hypotension and angiogenesis.</p>Fórmula:C47H66N12O11Pureza:98%Cor e Forma:SolidPeso molecular:975.11[Des-Arg9]-Bradykinin
CAS:<p>[Des-Arg9]-Bradykinin ([Des-Arg9]-Bradykinin(2TFA))(2TFA) is an agonist of Bradykinin (B1) receptor.</p>Fórmula:C44H61N11O10Pureza:98%Cor e Forma:SolidPeso molecular:904.02B-Raf IN 14
CAS:<p>B-Raf IN 14 is a BRAF inhibitor.</p>Fórmula:C15H14BrN5O3SPureza:98.32%Cor e Forma:SolidPeso molecular:424.27Labradimil
CAS:<p>Labradimil, a bradykinin B2 agonist, boosts brain drug delivery and tumor survival rates.</p>Fórmula:C49H75N15O12SPureza:98%Cor e Forma:SolidPeso molecular:1098.29[Des-Arg10]-HOE I40 TFA
<p>[Des-Arg10]-HOE I40 TFA is a potent antagonist of the bradykinin B1 receptor.</p>Fórmula:C53H77N15O12S·xC2HF3O2Cor e Forma:SolidDes-Arg9-[Leu8]-Bradykinin acetate
CAS:<p>Des-Arg9-[Leu8]-Bradykinin acetate is a potent antagonist of the bradykinin receptor 1 (B1R), utilized in renal fibrosis research [1].</p>Fórmula:C43H67N11O12Pureza:98%Cor e Forma:SolidPeso molecular:930.06Bombinakinin M acetate
<p>Bombinakinin M acetate is a potent bradykinin receptor agonist with high selectivity for mammalian arterial smooth muscle bradykinin receptors and is</p>Fórmula:C102H163N31O26Pureza:99.80%Cor e Forma:SolidPeso molecular:2239.58NPC 567 acetate
<p>NPC 567 acetate is a bradykinin B2 antagonist and can be used in studies about the treatment of allergic airway disease.</p>Fórmula:C62H91N19O15Pureza:97.72%Cor e Forma:SolidPeso molecular:1342.5FR190997
CAS:<p>FR190997 is an agonist of bradykinin B2 receptor.</p>Fórmula:C37H33Cl2N5O5Cor e Forma:SolidPeso molecular:698.59Fasitibant chloride hydrochloride
CAS:<p>Fasitibant chloride( MEN16132) is an effective and selective non-peptide antagonist of kinin B2 receptor.</p>Fórmula:C36H50Cl4N6O6SCor e Forma:SolidPeso molecular:836.7Lys-Bradykinin
CAS:<p>Endogenous bradykinin receptor agonist</p>Fórmula:C56H85N17O12Pureza:98%Cor e Forma:SolidPeso molecular:1188.38Zoliprofen
CAS:<p>Zoliprofen: potent, oral NSAID with anti-inflammatory, antipyretic, analgesic effects. Exceeds ibuprofen's efficacy in rats and rabbits.</p>Fórmula:C12H11NO3SPureza:99.62%Cor e Forma:SolidPeso molecular:249.29NPC 567
CAS:<p>NPC 567 is an antagonist of the bradykinin receptor.</p>Fórmula:C60H87N19O13Pureza:98%Cor e Forma:SolidPeso molecular:1282.48L 366811
CAS:<p>L 366811 is a potent oxytocin antagonist.</p>Fórmula:C43H56N8O6Cor e Forma:SolidPeso molecular:780.95FR167344 free base
CAS:<p>FR167344 free base: oral, nonpeptide B2 bradykinin receptor antagonist, high-affinity (IC50: 65 nM), no B1 affinity.</p>Fórmula:C30H28BrCl2N5O4Pureza:98%Cor e Forma:SolidPeso molecular:673.38Bradykinin (1-3)
CAS:<p>Bradykinin (1-3) is a fragment of Bradykinin. Bradykinin is an activates pain receptors.</p>Fórmula:C16H28N6O4Pureza:98%Cor e Forma:SolidPeso molecular:368.43JMV-1645
CAS:<p>JMV-1645 is an effective and selective B(1) bradykinin receptor antagonist.</p>Fórmula:C49H69N13O12SPureza:98%Cor e Forma:SolidPeso molecular:1064.23Lys-[Des-Arg9]Bradykinin TFA
CAS:<p>Lys-[Des-Arg9]Bradykinin TFA: natural kinin, selective B1 agonist; Ki: 0.12 nM (human), 1.7 nM (mouse), 0.23 nM (rabbit); weak on B2 receptors.</p>Fórmula:C54H75F6N13O15Cor e Forma:SolidPeso molecular:1260.24MEN 11270
CAS:<p>B2 bradykinin receptor peptide antagonist, pKi 10.3; improves hypotension, bronchoconstriction; B2-selective over 29 receptors/ion channels.</p>Fórmula:C60H90N20O11SPureza:98%Cor e Forma:SolidPeso molecular:1299.56Methionyl-Lysyl-Bradykinin
CAS:<p>Methionyl-Lysyl-Bradykinin (Met-Lys-Bradykinin), a Bradykinin analogue, is a kinin [1] [2] .</p>Fórmula:C61H94N18O13SCor e Forma:SolidPeso molecular:1319.58Bradykinin (1-7)
CAS:<p>Bradykinin (1-7), an amino-truncated peptide derived from Bradykinin, is a metabolite formed through enzymatic cleavage by endopeptidase.</p>Fórmula:C35H52N10O9Pureza:98%Cor e Forma:White Lyophilized PowderPeso molecular:756.85Bradykinin (1-6)
CAS:<p>Bradykinin (1-6) is a stable, CPY-cleaved metabolite that triggers pain, induces muscle contractions, and activates NO synthetase.</p>Fórmula:C30H45N9O8Pureza:98%Cor e Forma:SolidPeso molecular:659.73Lys-[Des-Arg9]Bradykinin
CAS:<p>Selective bradykinin B1 agonist with Ki 0.12 nM; inactive at B2 (>30,000 nM). Lowers blood pressure, more potent than Des-Arg9-Bradykinin.</p>Fórmula:C50H73N13O11Pureza:98%Cor e Forma:SolidPeso molecular:1032.21Retrobradykinin
CAS:<p>Bradykinin analog nonapeptide. Reverse sequence of Bradykinin. Exhibits no significant kinin activity. Can be used as a negative control.</p>Fórmula:C50H73N15O11Cor e Forma:SolidPeso molecular:1060.228Lys-[Hyp3]-Bradykinin
CAS:<p>Lys-[Hyp3]-Bradykinin, a human urine-derived kinin and bradykinin agonist, is used for inflammation research.</p>Fórmula:C56H85N17O13Cor e Forma:SolidPeso molecular:1204.38Bradykinin (1-5)
CAS:<p>Bradykinin (1-5), a stable metabolite of BK produced by ACE, serves as a marker for in vivo BK generation.</p>Fórmula:C27H40N8O6Cor e Forma:SolidPeso molecular:572.66Sar-[D-Phe8]-des-Arg9-Bradykinin acetate
<p>Sar-[D-Phe8]-des-Arg9-Bradykinin acetate is a potent and selective bradykinin B1 receptor agonist (EC50 = 9.02 nM in rabbit aorta) that is resistant to</p>Fórmula:C49H70N12O13Pureza:99.93%Cor e Forma:SolidPeso molecular:1035.15Icatibant Acetate
CAS:<p>Icatibant Acetate, an antagonist of the bradykinin B2 receptor, is used in the treatment of hereditary angioedema.</p>Fórmula:C61H93N19O15SPureza:99.68%Cor e Forma:SolidPeso molecular:1364.575-Hydroxy-1-methylhydantoin
CAS:<p>5-Hydroxy-1-methylhydantoin (HD-003) is an antioxidant potentially for the treatment of renal failure.</p>Fórmula:C4H6N2O3Pureza:99.99%Cor e Forma:SolidPeso molecular:130.1Bradykinin
CAS:<p>Bradykinin is an inflammatory mediator.</p>Fórmula:C50H73N15O11Pureza:99.68%Cor e Forma:SolidPeso molecular:1060.21Emorfazone
CAS:<p>Emorfazone (PH011085) has an anti-nociceptive effect.</p>Fórmula:C11H17N3O3Pureza:99.89%Cor e Forma:SolidPeso molecular:239.27ELN-441958
CAS:<p>ELN-441958 is a potent, neutral antagonist of B1 receptor, inhibits the binding of the B1 agonist ligand [3H]DAKD to IMR-90 cells with Ki of 0.26 nM.</p>Fórmula:C29H29ClN4O2Pureza:99.88%Cor e Forma:SolidPeso molecular:501.02SSR240612
CAS:<p>SSR240612 is a potent, and orally active specific non-peptide bradykinin B1 receptor antagonist (Kis = 0.48-0.73 and 358-481 nM for B1 and B2 receptors,</p>Fórmula:C42H53ClN4O7SPureza:98.59% - 99.16%Cor e Forma:SolidPeso molecular:793.41Bradykinin (acetate)
CAS:<p>Bradykinin (acetate) is an active peptide that is generated by the kallikrein-kinin system.</p>Fórmula:C52H77N15O13Pureza:>99.99%Cor e Forma:SolidPeso molecular:1120.26Lys-[Des-Arg9]Bradykinin,TFA
<p>Lys-[Des-Arg9]Bradykinin,TFA is Endogenous potent and highly selective bradykinin B1 receptor agonist (Ki values are 0.12 and > 30000 nM at human B1 and B2</p>Fórmula:C54H75F6N13O15Pureza:97.35%Cor e Forma:SolidPeso molecular:1260.24[Des-Arg9]-Bradykinin TFA
CAS:<p>[Des-Arg9]-Bradykinin is an agonist of Bradykinin (B1) receptor that displays selectivity for B1 over B2 receptors.</p>Fórmula:C46H62F3N11O12Pureza:>99.99%Cor e Forma:SolidPeso molecular:1018.05Bradykinin (2-9)
CAS:<p>Bradykinin (2-9) (Des-Arg1-bradykinin) is an amino-truncated peptide compound that is a metabolite of Bradykinin.</p>Fórmula:C44H61N11O10Pureza:>99.99%Cor e Forma:SolidPeso molecular:904.02R715 TFA(185052-09-9 free base)
<p>R715 TFA(185052-09-9 free base) is a potent and selective bradykinin B1 receptor antagonist (pA2 = 8.49).</p>Fórmula:C59H82F3N13O14Pureza:>99.99%Cor e Forma:SolidPeso molecular:1254.36Lys-Bradykinin acetate(342-10-9 free base)
CAS:<p>Lys-Bradykinin acetate is an endogenous bradykinin receptor agonist.</p>Fórmula:C58H89N17O14Pureza:99.86%Cor e Forma:SolidPeso molecular:1248.43Lys-[Des-Arg9]Bradykinin acetate
<p>Lys-[Des-Arg9]Bradykinin acetate is an endogenous potent and highly selective bradykinin B1 receptor agonist (Ki values are 0.12 and > 30000 nM at human B1 and</p>Fórmula:C52H77N13O13Pureza:99.93%Cor e Forma:SolidPeso molecular:1092.27BKM-570
CAS:<p>BKM-570, a bradykinin antagonist, causes impressive growth inhibition of lung and prostate tumors.</p>Fórmula:C34H34Cl2F5N3O3Pureza:98%Cor e Forma:SolidPeso molecular:698.55Anatibant
CAS:<p>Anatibant: a strong non-peptide, inhibits bradykinin B2; lowers brain swelling and damage post-trauma.</p>Fórmula:C34H36Cl2N6O5SPureza:98%Cor e Forma:SolidPeso molecular:711.66Fulimetibant
CAS:<p>Fulimetibant is a bradykinin receptor antagonist.</p>Fórmula:C25H21F4N3O3Cor e Forma:SolidPeso molecular:487.45B 4148
CAS:<p>B 4148 is a bradykinin inhibitor.</p>Fórmula:C62H95N19O14S2Cor e Forma:SolidPeso molecular:1394.67NPC 17731
CAS:<p>NPC 17731 is a bradykinin receptor antagonist.</p>Fórmula:C59H95N19O14Cor e Forma:SolidPeso molecular:1294.5MK-0686
CAS:<p>MK-0686 is an orally available bradykinin B1 receptor antagonist with potential anti-inflammatory activity.</p>Fórmula:C22H19ClF4N2O4Pureza:99.88%Cor e Forma:SolidPeso molecular:486.84Safotibant
CAS:<p>Safotibant (LF-22-0542) is a bradykinin B1 receptor antagonist with anti-inflammatory and analgesic activity for the topical treatment of diabetic macular edema</p>Fórmula:C25H34N4O5SPureza:99.62% - 99.67%Cor e Forma:SolidPeso molecular:502.63NVP-SAA164
CAS:<p>NVP-SAA164 is a nonpeptide bradykinin B1 receptor antagonist agent.</p>Fórmula:C36H45N5O5SPureza:98%Cor e Forma:SolidPeso molecular:659.84FK-3657
CAS:<p>FK-3657 is a non-peptide antagonist of bradykinin (BK)-B2 receptor.</p>Fórmula:C30H27Cl2N5O4Cor e Forma:SolidPeso molecular:592.47Fasitibant
CAS:<p>Fasitibant is a potent and selective nonpeptide kinin B2 receptor antagonist.</p>Fórmula:C36H49Cl2N6O6SCor e Forma:SolidPeso molecular:764.78BI-113823
CAS:<p>BI-113823 is an orally active and selective bradykinin B1 receptor antagonist. It alleviates mechanical hyperalgesia induced by complete Freund's adjuvant in rats. BI-113823 is applicable for research on chronic inflammatory pain.</p>Fórmula:C26H44N4O5SCor e Forma:SolidPeso molecular:524.716
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