Receptor de Bradicinina
Os receptores de bradicinina são GPCRs que mediam os efeitos da bradicinina, um peptídeo envolvido em respostas inflamatórias, sensação de dor e regulação da pressão arterial. Existem dois principais tipos de receptores de bradicinina, B1 e B2, cada um desempenhando papéis distintos em processos fisiopatológicos. Antagonistas dos receptores de bradicinina são usados no tratamento de condições como angioedema hereditário, dor crônica e hipertensão. Na CymitQuimica, oferecemos uma variedade de moduladores de receptores de bradicinina de alta qualidade para apoiar sua pesquisa em inflamação, manejo da dor e biologia cardiovascular.
Foram encontrados 61 produtos de "Receptor de Bradicinina"
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Anatibant 2HCl
CAS:Anatibant 2HCl is a small molecule bradykinin B2 receptor antagonist for the treatment of neurological disorders and may be used in the study of brain injury.Fórmula:C34H36Cl2N6O5S·2ClHPureza:99.17% - 99.2%Cor e Forma:SoildPeso molecular:784.58Fasitibant chloride
CAS:Fasitibant chloride, a potent B2R blocker, alleviates pain and swelling in arthritis.
Fórmula:C36H49Cl3N6O6SCor e Forma:SolidPeso molecular:800.23Methionyl-Lysyl-Bradykinin
CAS:Methionyl-Lysyl-Bradykinin (Met-Lys-Bradykinin), a Bradykinin analogue, is a kinin [1] [2] .Fórmula:C61H94N18O13SCor e Forma:SolidPeso molecular:1319.58Lys-[Des-Arg9]Bradykinin TFA
CAS:Lys-[Des-Arg9]Bradykinin TFA: natural kinin, selective B1 agonist; Ki: 0.12 nM (human), 1.7 nM (mouse), 0.23 nM (rabbit); weak on B2 receptors.Fórmula:C54H75F6N13O15Cor e Forma:SolidPeso molecular:1260.24Icatibant
CAS:Icatibant is a selective and specific antagonist of the bradykinin B2 receptor (IC50 and Ki: 1.07 nM and 0.798 nM respectively).Fórmula:C59H89N19O13SPureza:98%Cor e Forma:White SolidPeso molecular:1304.52[Phe8Ψ(CH-NH)-Arg9]-Bradykinin
CAS:Selective bradykinin B2 receptor agonist that is resistant to carboxypeptidase cleavage.Fórmula:C50H75N15O10Pureza:98%Cor e Forma:SolidPeso molecular:1046.23Bombinakinin M
CAS:Potent, selective bradykinin receptor agonist 50x stronger than bradykinin, contracts guinea pig ileum muscle at EC50 4.0 nM.Fórmula:C100H159N31O24Pureza:98%Cor e Forma:SolidPeso molecular:2179.55Lys-(Des-Arg9,Leu8)-Bradykinin
CAS:Lys-(Des-Arg9,Leu8)-Bradykinin is a selective antagonist of the bradykinin B1 receptor [1].Fórmula:C47H75N13O11Pureza:98%Cor e Forma:SolidPeso molecular:998.18(Hyp³)-Bradykinin acetate
(Hyp³)-Bradykinin acetate is an agonist of bradykinin B2 receptor and stimulates inositol phosphate production in cultured human fibroblasts.Fórmula:C52H77N15O14Pureza:99.46%Cor e Forma:SolidPeso molecular:1136.26Sar-[D-Phe8]-des-Arg9-Bradykinin
CAS:Potent bradykinin B1 agonist, EC50 = 9.02 nM, enzyme resistant, induces hypotension and angiogenesis.Fórmula:C47H66N12O11Pureza:98%Cor e Forma:SolidPeso molecular:975.11Labradimil
CAS:Labradimil, a bradykinin B2 agonist, boosts brain drug delivery and tumor survival rates.Fórmula:C49H75N15O12SPureza:98%Cor e Forma:SolidPeso molecular:1098.29[Des-Arg10]-HOE I40 TFA
[Des-Arg10]-HOE I40 TFA is a potent antagonist of the bradykinin B1 receptor.
Fórmula:C53H77N15O12S·xC2HF3O2Cor e Forma:SolidDes-Arg9-[Leu8]-Bradykinin acetate
CAS:Des-Arg9-[Leu8]-Bradykinin acetate is a potent antagonist of the bradykinin receptor 1 (B1R), utilized in renal fibrosis research [1].Fórmula:C43H67N11O12Pureza:98%Cor e Forma:SolidPeso molecular:930.06Bombinakinin M acetate
Bombinakinin M acetate is a potent bradykinin receptor agonist with high selectivity for mammalian arterial smooth muscle bradykinin receptors and isFórmula:C102H163N31O26Pureza:99.80%Cor e Forma:SolidPeso molecular:2239.58NPC 567 acetate
NPC 567 acetate is a bradykinin B2 antagonist and can be used in studies about the treatment of allergic airway disease.Fórmula:C62H91N19O15Pureza:97.72%Cor e Forma:SolidPeso molecular:1342.5T-kinin
CAS:T-kinin (Ile-Ser-bradykinin) is a bradykinin-containing peptide utilized in inflammation research [1] [2].Fórmula:C59H89N17O14Peso molecular:1260.44Fasitibant chloride hydrochloride
CAS:Fasitibant chloride( MEN16132) is an effective and selective non-peptide antagonist of kinin B2 receptor.Fórmula:C36H50Cl4N6O6SCor e Forma:SolidPeso molecular:836.7Lys-Bradykinin
CAS:Endogenous bradykinin receptor agonistFórmula:C56H85N17O12Pureza:98%Cor e Forma:SolidPeso molecular:1188.38Zoliprofen
CAS:Zoliprofen: potent, oral NSAID with anti-inflammatory, antipyretic, analgesic effects. Exceeds ibuprofen's efficacy in rats and rabbits.Fórmula:C12H11NO3SPureza:99.62%Cor e Forma:SolidPeso molecular:249.29Ref: TM-T68025
1mg80,00€1mL*10mM (DMSO)159,00€5mg167,00€10mg244,00€25mg455,00€50mg622,00€100mg883,00€500mg1.773,00€NPC 567
CAS:NPC 567 is an antagonist of the bradykinin receptor.Fórmula:C60H87N19O13Pureza:98%Cor e Forma:SolidPeso molecular:1282.48Thrombostatin cont-1
CAS:Thrombostatin cont-1, an analogue of the bradykinin metabolite thrombostatin, has been shown to reduce platelet activation in the canine carotid arteryFórmula:C87H142N34O29S2Peso molecular:2192.4FR167344 free base
CAS:FR167344 free base: oral, nonpeptide B2 bradykinin receptor antagonist, high-affinity (IC50: 65 nM), no B1 affinity.Fórmula:C30H28BrCl2N5O4Pureza:98%Cor e Forma:SolidPeso molecular:673.38Bradykinin (1-3)
CAS:Bradykinin (1-3) is a fragment of Bradykinin. Bradykinin is an activates pain receptors.
Fórmula:C16H28N6O4Pureza:98%Cor e Forma:SolidPeso molecular:368.43FR190997
CAS:FR190997 is an agonist of bradykinin B2 receptor.Fórmula:C37H33Cl2N5O5Cor e Forma:SolidPeso molecular:698.59L 366811
CAS:L 366811 is a potent oxytocin antagonist.Fórmula:C43H56N8O6Cor e Forma:SolidPeso molecular:780.95MEN 11270
CAS:B2 bradykinin receptor peptide antagonist, pKi 10.3; improves hypotension, bronchoconstriction; B2-selective over 29 receptors/ion channels.Fórmula:C60H90N20O11SPureza:98%Cor e Forma:SolidPeso molecular:1299.56JMV-1645
CAS:JMV-1645 is an effective and selective B(1) bradykinin receptor antagonist.Fórmula:C49H69N13O12SPureza:98%Cor e Forma:SolidPeso molecular:1064.23Bradykinin (1-7)
CAS:Bradykinin (1-7), an amino-truncated peptide derived from Bradykinin, is a metabolite formed through enzymatic cleavage by endopeptidase.Fórmula:C35H52N10O9Pureza:98%Cor e Forma:White Lyophilized PowderPeso molecular:756.85Bradykinin (1-6)
CAS:Bradykinin (1-6) is a stable, CPY-cleaved metabolite that triggers pain, induces muscle contractions, and activates NO synthetase.Fórmula:C30H45N9O8Pureza:98%Cor e Forma:SolidPeso molecular:659.73Lys-[Des-Arg9]Bradykinin
CAS:Selective bradykinin B1 agonist with Ki 0.12 nM; inactive at B2 (>30,000 nM). Lowers blood pressure, more potent than Des-Arg9-Bradykinin.Fórmula:C50H73N13O11Pureza:98%Cor e Forma:SolidPeso molecular:1032.21Retrobradykinin
CAS:Bradykinin analog nonapeptide. Reverse sequence of Bradykinin. Exhibits no significant kinin activity. Can be used as a negative control.Fórmula:C50H73N15O11Cor e Forma:SolidPeso molecular:1060.228Lys-[Hyp3]-Bradykinin
CAS:Lys-[Hyp3]-Bradykinin, a human urine-derived kinin and bradykinin agonist, is used for inflammation research.Fórmula:C56H85N17O13Cor e Forma:SolidPeso molecular:1204.38[Des-Arg9]-Bradykinin
CAS:[Des-Arg9]-Bradykinin ([Des-Arg9]-Bradykinin(2TFA))(2TFA) is an agonist of Bradykinin (B1) receptor.Fórmula:C44H61N11O10Pureza:98%Cor e Forma:SolidPeso molecular:904.02B-Raf IN 14
CAS:B-Raf IN 14 is a BRAF inhibitor.Fórmula:C15H14BrN5O3SPureza:98.38%Cor e Forma:SolidPeso molecular:424.27[Des-Arg9]-Bradykinin acetate
CAS:[Des-Arg9]-Bradykinin acetate is a selective agonist of Bradykinin B1 receptor.Fórmula:C46H65N11O12Pureza:99.05%Cor e Forma:SolidPeso molecular:964.07Bradykinin (1-5)
CAS:Bradykinin (1-5), a stable metabolite of BK produced by ACE, serves as a marker for in vivo BK generation.Fórmula:C27H40N8O6Cor e Forma:SolidPeso molecular:572.66Sar-[D-Phe8]-des-Arg9-Bradykinin acetate
Sar-[D-Phe8]-des-Arg9-Bradykinin acetate is a potent and selective bradykinin B1 receptor agonist (EC50 = 9.02 nM in rabbit aorta) that is resistant toFórmula:C49H70N12O13Pureza:99.93%Cor e Forma:SolidPeso molecular:1035.15Icatibant Acetate
CAS:Icatibant Acetate, an antagonist of the bradykinin B2 receptor, is used in the treatment of hereditary angioedema.Fórmula:C61H93N19O15SPureza:99.68% - 99.90%Cor e Forma:SolidPeso molecular:1364.57Ref: TM-T22344
1mg66,00€2mg92,00€5mg177,00€10mg281,00€1mL*10mM (DMSO)355,00€25mg475,00€50mg677,00€100mg888,00€5-Hydroxy-1-methylhydantoin
CAS:5-Hydroxy-1-methylhydantoin (HD-003) is an antioxidant potentially for the treatment of renal failure.Fórmula:C4H6N2O3Pureza:99.99%Cor e Forma:SolidPeso molecular:130.1Bradykinin
CAS:Bradykinin is an inflammatory mediator.Fórmula:C50H73N15O11Pureza:99.68%Cor e Forma:SolidPeso molecular:1060.21Emorfazone
CAS:Emorfazone (PH011085) has an anti-nociceptive effect.Fórmula:C11H17N3O3Pureza:99.89%Cor e Forma:SolidPeso molecular:239.27Ref: TM-T9132
1mg84,00€1mL*10mM (DMSO)152,00€5mg168,00€10mg245,00€25mg404,00€50mg567,00€100mg767,00€200mg1.018,00€ELN-441958
CAS:ELN-441958 is a potent, neutral antagonist of B1 receptor, inhibits the binding of the B1 agonist ligand [3H]DAKD to IMR-90 cells with Ki of 0.26 nM.Fórmula:C29H29ClN4O2Pureza:99.88%Cor e Forma:SolidPeso molecular:501.02Ref: TM-T2086
1mg58,00€5mg128,00€1mL*10mM (DMSO)141,00€10mg200,00€25mg339,00€50mg485,00€100mg658,00€200mg889,00€SSR240612
CAS:SSR240612 is a potent, and orally active specific non-peptide bradykinin B1 receptor antagonist (Kis = 0.48-0.73 and 358-481 nM for B1 and B2 receptors,Fórmula:C42H53ClN4O7SPureza:98.59% - 99.16%Cor e Forma:SolidPeso molecular:793.41Ref: TM-T5048
1mg222,00€5mg512,00€1mL*10mM (DMSO)612,00€10mg700,00€25mg982,00€50mg1.333,00€100mg1.783,00€Bradykinin (acetate)
CAS:Bradykinin (acetate) is an active peptide that is generated by the kallikrein-kinin system.Fórmula:C52H77N15O13Pureza:>99.99%Cor e Forma:SolidPeso molecular:1120.26Lys-[Des-Arg9]Bradykinin,TFA
Lys-[Des-Arg9]Bradykinin,TFA is Endogenous potent and highly selective bradykinin B1 receptor agonist (Ki values are 0.12 and > 30000 nM at human B1 and B2Fórmula:C54H75F6N13O15Pureza:97.35%Cor e Forma:SolidPeso molecular:1260.24[Des-Arg9]-Bradykinin TFA
CAS:[Des-Arg9]-Bradykinin is an agonist of Bradykinin (B1) receptor that displays selectivity for B1 over B2 receptors.Fórmula:C46H62F3N11O12Pureza:>99.99%Cor e Forma:SolidPeso molecular:1018.05Bradykinin (2-9)
CAS:Bradykinin (2-9) (Des-Arg1-bradykinin) is an amino-truncated peptide compound that is a metabolite of Bradykinin.Fórmula:C44H61N11O10Pureza:>99.99%Cor e Forma:SolidPeso molecular:904.02Ref: TM-TP1181
1mg39,00€5mg88,00€10mg130,00€1mL*10mM (DMSO)144,00€25mg210,00€50mg313,00€100mg464,00€200mg660,00€R715 TFA(185052-09-9 free base)
R715 TFA(185052-09-9 free base) is a potent and selective bradykinin B1 receptor antagonist (pA2 = 8.49).Fórmula:C59H82F3N13O14Pureza:>99.99%Cor e Forma:SolidPeso molecular:1254.36Lys-Bradykinin acetate(342-10-9 free base)
CAS:Lys-Bradykinin acetate is an endogenous bradykinin receptor agonist.Fórmula:C58H89N17O14Pureza:99.86%Cor e Forma:SolidPeso molecular:1248.43Lys-[Des-Arg9]Bradykinin acetate
Lys-[Des-Arg9]Bradykinin acetate is an endogenous potent and highly selective bradykinin B1 receptor agonist (Ki values are 0.12 and > 30000 nM at human B1 andFórmula:C52H77N13O13Pureza:99.93%Cor e Forma:SolidPeso molecular:1092.27B 4148
CAS:B 4148 is a bradykinin inhibitor.Fórmula:C62H95N19O14S2Cor e Forma:SolidPeso molecular:1394.67NPC 17731
CAS:NPC 17731 is a bradykinin receptor antagonist.Fórmula:C59H95N19O14Cor e Forma:SolidPeso molecular:1294.5BKM-570
CAS:BKM-570, a bradykinin antagonist, causes impressive growth inhibition of lung and prostate tumors.Fórmula:C34H34Cl2F5N3O3Pureza:98%Cor e Forma:SolidPeso molecular:698.55Anatibant
CAS:Anatibant: a strong non-peptide, inhibits bradykinin B2; lowers brain swelling and damage post-trauma.Fórmula:C34H36Cl2N6O5SPureza:98%Cor e Forma:SolidPeso molecular:711.66Fulimetibant
CAS:Fulimetibant is a bradykinin receptor antagonist.Fórmula:C25H21F4N3O3Cor e Forma:SolidPeso molecular:487.45MK-0686
CAS:MK-0686 is an orally available bradykinin B1 receptor antagonist with potential anti-inflammatory activity.Fórmula:C22H19ClF4N2O4Pureza:99.88%Cor e Forma:SolidPeso molecular:486.84Safotibant
CAS:Safotibant (LF-22-0542) is a bradykinin B1 receptor antagonist with anti-inflammatory and analgesic activity for the topical treatment of diabetic macular edemaFórmula:C25H34N4O5SPureza:99.62% - 99.67%Cor e Forma:SolidPeso molecular:502.63NVP-SAA164
CAS:NVP-SAA164 is a nonpeptide bradykinin B1 receptor antagonist agent.Fórmula:C36H45N5O5SPureza:98%Cor e Forma:SolidPeso molecular:659.84FK-3657
CAS:FK-3657 is a non-peptide antagonist of bradykinin (BK)-B2 receptor.Fórmula:C30H27Cl2N5O4Cor e Forma:SolidPeso molecular:592.47BI-113823
CAS:BI-113823 is an orally active and selective bradykinin B1 receptor antagonist. It alleviates mechanical hyperalgesia induced by complete Freund's adjuvant in rats. BI-113823 is applicable for research on chronic inflammatory pain.Fórmula:C26H44N4O5SCor e Forma:SolidPeso molecular:524.716Fasitibant
CAS:Fasitibant is a potent and selective nonpeptide kinin B2 receptor antagonist.Fórmula:C36H49Cl2N6O6SCor e Forma:SolidPeso molecular:764.78
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