
Receptor de Dopamina
Os receptores de dopamina são um grupo de GPCRs que respondem ao neurotransmissor dopamina, desempenhando um papel fundamental na regulação do movimento, motivação, recompensa e várias funções cognitivas. Esses receptores são divididos em famílias semelhantes a D1 e D2, cada uma com funções e perfis farmacológicos distintos. Moduladores de receptores de dopamina são amplamente estudados por suas aplicações no tratamento da doença de Parkinson, esquizofrenia, dependência e outros transtornos neuropsiquiátricos. Na CymitQuimica, oferecemos uma ampla gama de moduladores de receptores de dopamina de alta qualidade para apoiar sua pesquisa em neurociência, saúde mental e sinalização GPCR.
Foram encontrados 407 produtos de "Receptor de Dopamina"
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RBI-257 Maleate
CAS:<p>RBI-257 Maleate is a highly potent selective ligand of dopamine D4 receptor.</p>Fórmula:C25H32IN3O5Cor e Forma:SolidPeso molecular:581.44Quinelorane dihydrochloride
CAS:<p>Dopamine D2 and D3 receptor agonist</p>Fórmula:C14H23ClN4Pureza:98%Cor e Forma:SolidPeso molecular:282.81SKF-83822
CAS:<p>SKF-83822 is an agonist of dopamine D1-like receptor.</p>Fórmula:C20H22ClNO2Pureza:98%Cor e Forma:SolidPeso molecular:343.85BRD5814
CAS:<p>BRD5814 is a highly brain penetrant β-arrestin biased D2R antagonist.</p>Fórmula:C21H23ClF3NO2Cor e Forma:SolidPeso molecular:413.86SB-277011 dihydrochloride
CAS:<p>SB-277011 dihydrochloride: potent, selective D3 antagonist; orally bioavailable; crosses blood-brain barrier; pKi 8.0 for D3 receptor.</p>Fórmula:C28H32Cl2N4OPureza:98%Cor e Forma:SolidPeso molecular:511.49PF2562
CAS:<p>PF2562: Dopamine D1 ligand, agonist/partial agonist. Binds D1 receptor (Ki: 113 nM), active in cAMP assay (EC50: 568 nM).</p>Fórmula:C19H17N5OPureza:98%Cor e Forma:SolidPeso molecular:331.37Odapipam
CAS:<p>Odapipam is a selective and high affinity antagonist of benzazepine dopamine D1 receptor (Kd of 0.18 nM).</p>Fórmula:C19H20ClNO2Pureza:98%Cor e Forma:SolidPeso molecular:329.82Lenperone
CAS:<p>Lenperone is a butyrophenone antipsychotic. Like other major tranquilizers, It has some alpha-adrenergic blocking action and is antiemetic.</p>Fórmula:C22H23F2NO2Cor e Forma:SolidPeso molecular:371.42BAK2-66
CAS:<p>BAK2-66 is a selective antagonist of the dopamine D3 receptor.</p>Fórmula:C23H24Cl2FN3O2Pureza:98%Cor e Forma:SolidPeso molecular:464.36Brl 20596
CAS:<p>Brl 20596 is a central dopamine antagonist in the class of anilide.</p>Fórmula:C20H24ClN3O2Pureza:98%Cor e Forma:SolidPeso molecular:373.88FAUC-3019
CAS:<p>FAUC-3019 is a partial agonist of the dopamine D(4) receptor.</p>Fórmula:C22H24N2OCor e Forma:SolidPeso molecular:332.44Lergotrile
CAS:<p>Lergotrile is used as an enzyme Inhibitor (Prolactin).</p>Fórmula:C17H18ClN3Pureza:98%Cor e Forma:SolidPeso molecular:299.8CJB-090 2HCl
CAS:<p>CJB-090 2HCl is a partial agonist of the dopamine D3 receptor.</p>Fórmula:C26H30Cl4N4OCor e Forma:SolidPeso molecular:556.35Gyki 32887
CAS:<p>Gyki 32887 is a dopamine agonist.</p>Fórmula:C23H28N6O6SPureza:98%Cor e Forma:SolidPeso molecular:516.57Amitifadine free base
CAS:<p>Amitifadine (DOV-21947/EB-1010), an antidepressant SNDRI, curbs binge drinking and negative effects in animals with alcoholism-depression.</p>Fórmula:C11H11Cl2NCor e Forma:SolidPeso molecular:228.12A 69024
CAS:<p>A 69024 is a highly selective antagonist of dopamine D-1 receptor.</p>Fórmula:C20H24BrNO4Pureza:98%Cor e Forma:SolidPeso molecular:422.31Seproxetine HCl
CAS:<p>Seproxetine HCl, a more active enantiomer of N-desmethyl metabolite fluoxetine, works by selectively inhibiting the serotonin uptake carrier.</p>Fórmula:C16H17ClF3NOPureza:98%Cor e Forma:SolidPeso molecular:331.76Lergotrile mesylate
CAS:<p>Lergotrile mesylate, an ergoline derivative, suppresses prolactin in vivo and in vitro.</p>Fórmula:C18H22ClN3O3SCor e Forma:SolidPeso molecular:395.9Bromperidol decanoate
CAS:<p>Bromperidol decanoate is an antipsychotic agent that is utilized for long-term maintenance treatment for schizophrenia.</p>Fórmula:C31H41BrFNO3Cor e Forma:SolidPeso molecular:574.56LY 171859
CAS:<p>LY 171859 is an agonist of D2-receptor.</p>Fórmula:C17H14O5Pureza:98%Cor e Forma:SolidPeso molecular:298.29Nor-SCH-12679 Maleate
CAS:<p>Nor-SCH-12679 Maleate is a D1-dopamine receptor antagonist.</p>Fórmula:C22H25NO6Pureza:98%Cor e Forma:SolidPeso molecular:399.44Clothixamide
CAS:<p>Clothixamide(Clotixamide) is a thioxanthene derivative with antipsychotic activity.</p>Fórmula:C24H28ClN3OSPureza:95.51%Cor e Forma:SolidPeso molecular:442.02CI-943
CAS:<p>CI-943 is a novel potential antipsychotic drug that does not bind to dopamine (DA) receptors and has some developmental neurotoxicity.</p>Fórmula:C12H17N5Pureza:98%Cor e Forma:SolidPeso molecular:231.33'-Fluorobenzylspiperone maleate
CAS:<p>ligand for the D2 receptor</p>Fórmula:C34H35F2N3O6Pureza:98%Cor e Forma:SolidPeso molecular:619.66Butaclamol free base
CAS:<p>Butaclamol is a typical antipsychotic which was never marketed. It also acts as a dopamine receptor antagonist.</p>Fórmula:C25H31NOPureza:98%Cor e Forma:SolidPeso molecular:361.52PD 118440
CAS:<p>PD 118440 is a Dopamine antagonist. PD 118440 is an orally active dopamine (DA) agonists with pronounced central nervous system effects.</p>Fórmula:C11H17N3SPureza:98%Cor e Forma:SolidPeso molecular:223.34Sch 24518
CAS:<p>Sc h24518 is an antagonist of D1 receptor.</p>Fórmula:C16H17BrClNOPureza:98%Cor e Forma:SolidPeso molecular:354.67Dicarbine
CAS:<p>Double carbene blocks dopamine receptors, aiding schizophrenia and alcoholism research; it maintains defense reflexes despite mid-brain stimulation.</p>Fórmula:C13H18N2Pureza:98%Cor e Forma:SolidPeso molecular:202.3L-750,667 Trihydrochloride
CAS:<p>L-750,667 Trihydrochloride is a selective D4 receptor antagonist, reverses the dopamine-induced inhibition of cAMP accumulation in the central nervous system.</p>Fórmula:C18H22Cl3IN4Pureza:99.63%Cor e Forma:SolidPeso molecular:527.666-Chloromelatonin
CAS:<p>6-Chloromelatonin: potent, stable melatonin agonist; binds MT2 receptors (pKi=9.77); could help research sleep disorders.</p>Fórmula:C13H15ClN2O2Pureza:98.01% - 99.25%Cor e Forma:SolidPeso molecular:266.72A-77636
CAS:<p>A-77636 is a potent, selective, and long-acting oral dopamine D1 receptor agonist with an effective concentration (EC50) of 1.1 nM and a corresponding pEC50</p>Fórmula:C20H27NO3Pureza:98%Cor e Forma:SolidPeso molecular:329.43D4R agonist-1
CAS:<p>D4R agonist-1 is a selective and potent D4R partial agonist (Ki:2.2 nM).D4R agonist-1 can be used to study neurological diseases.</p>Fórmula:C19H22N4SPureza:98.44%Cor e Forma:SolidPeso molecular:338.47PG 01037 dihydrochloride
CAS:<p>PG 01037 dihydrochloride (PG-01037 2HCl) is a potent and selective dopamine D3 receptor antagonist with a Ki of 0.7 nM.</p>Fórmula:C26H28Cl4N4OPureza:99.89%Cor e Forma:SolidPeso molecular:554.34SKF83959
CAS:<p>SKF83959: dopamine D1 partial agonist, Ki: D1(1.18 nM), D5(7.56 nM), D2(920 nM), D3(399 nM); improves cognitive function in depression, Alzheimer's.</p>Fórmula:C18H20ClNO2Pureza:98.68%Cor e Forma:SolidPeso molecular:317.81WAY-260022
CAS:<p>WAY-260022 is the norepinephrine transporter inhibitor.</p>Fórmula:C21H31F3N2O2Pureza:97.61% - 99.41%Cor e Forma:SolidPeso molecular:400.48UNC9975
CAS:<p>UNC9975 is a D(2) receptor agonist with antipsychotic activity used in the study of neurologic disorders such as schizophrenia.</p>Fórmula:C23H28Cl2N4O2Pureza:98.78% - 98.78%Cor e Forma:SolidPeso molecular:463.4Fananserin
CAS:<p>Fananserin: Oral 5-HT2A antagonist (Ki=0.37 nM, rat), blocks human D4 receptor (Ki=2.93 nM).</p>Fórmula:C23H24FN3O2SPureza:99.88%Cor e Forma:SolidPeso molecular:425.52PD 168568 dihydrochloride
CAS:<p>PD 168568 dihydrochloride (PD 168568 (dihydrochloride)) is an orally active and selective antagonist of D4 dopamine receptor(Ki of 8.8 nM).</p>Fórmula:C22H29Cl2N3OPureza:99.71%Cor e Forma:SolidPeso molecular:422.39Molindone
CAS:<p>Molindone: antipsychotic for schizophrenia; blocks dopamine, often paired with serotonin; dosage affects error/response rates.</p>Fórmula:C16H24N2O2Pureza:99.37% - 99.46%Cor e Forma:Off-White SolidPeso molecular:276.37Milenperone
CAS:<p>Milenperone (R 34009) is a novel anti-invasive compound for the control of behavioral disorders in patients with epilepsy and alcoholism.</p>Fórmula:C22H23ClFN3O2Pureza:98.09% - 99.84%Cor e Forma:SolidPeso molecular:415.89NGD 94-1
CAS:<p>NGD 94-1 is a D4 receptor antagonist that can be used to study psychiatric disorders such as cognitive impairment.</p>Fórmula:C18H20N6Pureza:99.61%Cor e Forma:SolidPeso molecular:320.39Ordopidine
CAS:<p>Ordopidine (ACR325) is a dopaminergic stabilizer that suppresses psychostimulant-induced hyperactivity disorder and stimulates behavior during inactivity.</p>Fórmula:C14H20FNO2SPureza:99.39%Cor e Forma:SolidPeso molecular:285.38Seridopidine
CAS:<p>Seridopidine (ACR343) is a modulator of dopaminergic activity that is used as an oral therapy for schizophrenia, Parkinson's disease, and Tourette's syndrome.</p>Fórmula:C14H20FNO2SPureza:99.65%Cor e Forma:SolidPeso molecular:285.38GBR 12783 dihydrochloride
CAS:<p>GBR 12783 dihydrochloride inhibits dopamine uptake in rats/mice; IC50s: 1.8/1.2 nM. Enhances memory, boosts hippocampal acetylcholine.</p>Fórmula:C28H34Cl2N2OPureza:98.08%Cor e Forma:SolidPeso molecular:485.497-Hydroxy-DPAT hydrobromide
CAS:<p>7-Hydroxy-DPAT hydrobromide is a D3 dopamine receptor agonist that blocks dopamine reuptake, used in research on neurological diseases.</p>Fórmula:C16H26BrNOPureza:99.73%Cor e Forma:SolidPeso molecular:328.29PF-00217830
CAS:<p>PF-00217830: agonist at serotonin 1A & dopamine D2, antagonist at serotonin 2A, potential schizophrenia study drug.</p>Fórmula:C26H30N4O2Pureza:98.72%Cor e Forma:SolidPeso molecular:430.54MLS1547
CAS:<p>MLS1547 is a potent D2 receptor G protein-biased agonist (Ki=1.2 μM, EC50=0.37 μM in Ca2+ assay).</p>Fórmula:C19H19ClN4OPureza:99.64%Cor e Forma:SolidPeso molecular:354.83CyPPA
CAS:<p>CyPPA enhances SK channels, reducing firing rate and extending apamin-sensitive afterhyperpolarization.</p>Fórmula:C16H23N5Pureza:99.88%Cor e Forma:SolidPeso molecular:285.39Benperidol
CAS:<p>Benperidol (Anquil), a butanone derivative, has antipsychotic effects and blocks D2 receptors; useful in PET scans.</p>Fórmula:C22H24FN3O2Pureza:99.91%Cor e Forma:SolidPeso molecular:381.44Remoxipride hydrochloride
CAS:<p>Remoxipride hydrochloride (Roxiam) is a selective antagonist of D2 receptor with IC50s of 1.57 μM, >100 μM and 42 μM for D2 receptor, D1 receptor and α1-</p>Fórmula:C16H24BrClN2O3Pureza:99.88%Cor e Forma:SolidPeso molecular:407.73
