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Receptor de adenosina

Receptor de adenosina

Os receptores de adenosina são uma classe de GPCRs que respondem ao nucleosídeo endógeno adenosina. Esses receptores estão envolvidos na regulação de vários processos fisiológicos, incluindo função cardiovascular, ciclos de sono-vigília e respostas imunes. Moduladores de receptores de adenosina têm potencial terapêutico no tratamento de condições como arritmias cardíacas, inflamação e doenças neurodegenerativas. Na CymitQuimica, oferecemos uma seleção de moduladores de receptores de adenosina de alta qualidade para apoiar sua pesquisa em biologia cardiovascular, neurociência e imunologia.

Foram encontrados 249 produtos de "Receptor de adenosina"

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  • Theobromine

    CAS:
    Theobromine (3,7-Dimethylxanthine), a xanthine alkaloid, is used as a bronchodilator and as a vasodilator.
    Fórmula:C7H8N4O2
    Pureza:99.69% - 99.91%
    Cor e Forma:White To Yellow Crystalline Powder
    Peso molecular:180.16

    Ref: TM-T0625

    1g
    47,00€
    500mg
    34,00€
  • 5'-Amino-5'-deoxyadenosine

    CAS:
    5'-Amino-5'-deoxyadenosine (NH2dAdo) is an adenosine kinase inhibitor targeting malignant tumors of the inert lymphatic system with antitumor and anticancer
    Fórmula:C10H14N6O3
    Pureza:99.72%
    Cor e Forma:Solid
    Peso molecular:266.26

    Ref: TM-T21017

    5mg
    101,00€
    10mg
    167,00€
    25mg
    265,00€
    50mg
    404,00€
  • Rolofylline

    CAS:
    Rolofylline (KW-3902) is an adenosine A1 receptor antagonist used to study acute congestive heart failure and renal dysfunction.
    Fórmula:C20H28N4O2
    Pureza:99.53%
    Cor e Forma:Solid
    Peso molecular:356.46

    Ref: TM-T16782

    1mg
    44,00€
    5mg
    86,00€
    10mg
    110,00€
    25mg
    178,00€
    50mg
    264,00€
    100mg
    389,00€
    1mL*10mM (DMSO)
    101,00€
  • Blontuvetmab

    CAS:
    Blontuvetmab (AT 004), a caninized CD20 monoclonal antibody, is utilized in the study of Canine B-cell lymphoma [1].
    Cor e Forma:Liquid

    Ref: TM-T76932

    1mg
    222,00€
    5mg
    582,00€
    10mg
    888,00€
  • Adenosine receptor inhibitor 1

    CAS:
    Potent, selective adenosine receptor blocker with strong affinity, especially A2A (Ki 68.5 nM). Promising for cancer, neurodegeneration study.
    Fórmula:C17H19ClFN5O3
    Cor e Forma:Solid
    Peso molecular:395.82

    Ref: TM-T61850

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • A2AR-agonist-1

    CAS:
    A2AR-agonist-1 targets A2A Receptor/ENT1 for neuroprotection; potent with Ki of 4.39 (A2AR), 3.47 (ENT1).
    Fórmula:C20H22N6O4
    Pureza:99.9%
    Cor e Forma:Solid
    Peso molecular:410.43

    Ref: TM-T10212

    1mg
    90,00€
    2mg
    127,00€
    5mg
    178,00€
    10mg
    269,00€
    25mg
    427,00€
    50mg
    610,00€
    100mg
    820,00€
    500mg
    1.603,00€
    1mL*10mM (DMSO)
    207,00€
  • TC-G 1004

    CAS:
    adenosine A2A receptors antagonist
    Fórmula:C22H27N7O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:421.5

    Ref: TM-T23435

    50mg
    2.970,00€
  • hA2A/hCA XII modulator 1

    CAS:
    Potent hA2AAR antagonist & hCA XII inhibitor; Ki: hA2AAR 6.4 nM, hCA XII 6.2 nM. Possible cancer research use.
    Fórmula:C24H19N7O4S
    Cor e Forma:Solid
    Peso molecular:501.52

    Ref: TM-T63400

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • IHCH-3064

    CAS:
    IHCH-3064: dual-action cancer immunotherapy, A2AR affinity (Ki 2.2 nM), selective HDAC1 inhibitor (IC50 80.2 nM).
    Fórmula:C25H21N9O2
    Cor e Forma:Solid
    Peso molecular:479.49

    Ref: TM-T63151

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • MRS 1334

    CAS:
    antagonist for the human adenosine A3 receptor
    Fórmula:C31H26N2O6
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:522.55

    Ref: TM-T23017

    25mg
    2.232,00€
  • LUF6000

    CAS:
    LUF6000 is an allosteric modulator of the human A3 adenosine receptor (AR).
    Fórmula:C22H20Cl2N4
    Cor e Forma:Solid
    Peso molecular:411.33

    Ref: TM-T15791

    5mg
    294,00€
    25mg
    690,00€
    50mg
    898,00€
    100mg
    1.575,00€
    1mL*10mM (DMSO)
    323,00€
  • A2A/A1 AR antagonist-1

    CAS:
    A2A/A1 AR antagonist-1 is a potent dual antagonist for ischemic stroke research with Ki values of 5.58 nM (A2A) and 24.2 nM (A1).
    Fórmula:C15H12N6O2
    Cor e Forma:Solid
    Peso molecular:308.29

    Ref: TM-T60732

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • LUF 5834

    CAS:
    A2A and A2B adenosine receptor partial agonist
    Fórmula:C17H12N6OS
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:348.38

    Ref: TM-T22937

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • 5'-(N-Cyclopropyl)carboxamidoadenosine

    CAS:
    adenosine A2 receptor agonist
    Fórmula:C13H16N6O4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:320.3

    Ref: TM-T22523

    5mg
    166,00€
    10mg
    305,00€
  • A1AR antagonist 5

    CAS:
    A1AR antagonist 5 (compound 20) is a potent and selective antagonist of A1 adenosine receptor (A1AR) with a pKi of 6.11 and a pIC 50 of 5.83 [1].
    Fórmula:C17H15ClN4O
    Cor e Forma:Solid
    Peso molecular:326.78

    Ref: TM-T60915

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • A1AR antagonist 3

    CAS:
    Compound 13: selective A1AR antagonist, Ki human A1: 9.69 nM, rat A1: 0.529 nM, useful for neurological research.
    Fórmula:C25H20N2O3S
    Cor e Forma:Solid
    Peso molecular:428.5

    Ref: TM-T62348

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • XCC

    CAS:
    XCC is an Adenosine receptor antagonist.
    Fórmula:C19H22N4O5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:386.4

    Ref: TM-T23537

    50mg
    2.422,00€
  • A1AR antagonist 4

    CAS:
    Compound 22: A1AR antagonist, pIC50 5.51, pKi 6.29, potent and selective.
    Fórmula:C23H25N3O2
    Cor e Forma:Solid
    Peso molecular:375.46

    Ref: TM-T61536

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • MRS1097

    CAS:
    MRS1097 is a selective antagonist A3 adenosine receptor.
    Fórmula:C26H27NO4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:417.5

    Ref: TM-T28098

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • MRS-1191

    CAS:
    MRS-1191 is an effective and selective A3 adenosine receptor antagonist (KB: 92 nM, a Ki: 31.4 nM for human A3 receptor and an IC50: 120 nM for CHO cells).
    Fórmula:C31H27NO4
    Cor e Forma:Solid
    Peso molecular:477.55

    Ref: TM-T16134

    25mg
    603,00€
    50mg
    783,00€
    100mg
    1.341,00€
  • Apadenoson

    CAS:
    Apadenoson: potent A2 agonist, A3 inhibitor (IC 45 nM), anti-inflammatory, for neurological research.
    Fórmula:C23H30N6O6
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:486.52

    Ref: TM-T26641

    25mg
    A consultar
    50mg
    A consultar
    100mg
    A consultar
  • Lu AA 47070

    CAS:
    adenosine A2A receptor antagonist
    Fórmula:C17H20F2N3O6PS
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:463.39

    Ref: TM-T22934

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • A1AR antagonist 2

    CAS:
    Compound 18h is a potent A1 adenosine receptor blocker with Ki of 1.49 nM for hA1, 10.2 nM for hA2A, 50.1 nM for hA2B.
    Fórmula:C17H12N4O
    Cor e Forma:Solid
    Peso molecular:288.3

    Ref: TM-T60580

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • A1/A3 AR antagonist 2

    CAS:
    The compound is an a1/a3 adenosine receptor antagonist, which helps to treat (neurological) inflammatory diseases.
    Fórmula:C22H16N2O3S
    Cor e Forma:Solid
    Peso molecular:388.44

    Ref: TM-T61744

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • AB-MECA

    CAS:
    AB-MECA is a high affinity A3 adenosine receptor agonist. It has high affinity for recombinant A1 and A3 receptors.
    Fórmula:C18H21N7O4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:399.4

    Ref: TM-T14082

    1mg
    239,00€
    5mg
    1.018,00€
    10mg
    1.783,00€
  • A2AAR/HDAC-IN-1

    CAS:
    A2AAR/HDAC-IN-1 (compound 14c) is an orally active, balanced A2AAR/HDAC dual inhibitor of A2AAR (Ki: 163.5 nM), HDAC1 (IC50: 145.3 nM). effect.
    Fórmula:C24H21N7O2
    Cor e Forma:Solid
    Peso molecular:439.47

    Ref: TM-T62521

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • LASSBio-1359

    CAS:
    LASSBio-1359 is an adenosine receptor agonist. It acts by inducing relaxation of the corpus cavernosum. It also acts as a novel selective phosphodiesterase.
    Fórmula:C17H18N2O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:298.34

    Ref: TM-T24388

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • PSB 11 hydrochloride

    CAS:
    PSB 11 hydrochloride is a human adenosine A3 receptor antagonist.
    Fórmula:C16H18ClN5O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:331.8

    Ref: TM-T23199

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • Adenosine receptor antagonist 3

    CAS:
    Adenosine receptor antagonist 3 has the potential for cancer disease research which is a potent adenosine receptor antagonist [1].
    Fórmula:C16H14N6S
    Cor e Forma:Solid
    Peso molecular:322.39

    Ref: TM-T60872

    25mg
    858,00€
    50mg
    1.116,00€
    100mg
    1.791,00€
  • Adentri

    CAS:
    Adentri is a novel antagonist of adenosine A1 receptor with unique diuretic activity.
    Fórmula:C18H24N4O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:344.41

    Ref: TM-T26565

    25mg
    1.369,00€
  • A2A receptor antagonist 3

    CAS:
    A2A receptor antagonist 3 (Example 92) is an adenosine A2a receptor antagonist (Ki: 0.4 nM). receptor (Ki: 1467 nM).
    Fórmula:C26H26N6O2
    Cor e Forma:Solid
    Peso molecular:454.52

    Ref: TM-T62797

    25mg
    1.927,00€
    50mg
    2.507,00€
    100mg
    3.168,00€
  • MRS1186

    CAS:
    MRS1186 is an effective and selective antagonist of the human Adenosine A3 receptor (Ki: 7.66 nM).
    Fórmula:C16H12ClN5O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:341.75

    Ref: TM-T16138

    25mg
    1.444,00€
    50mg
    1.882,00€
    100mg
    2.375,00€
  • Adenosine receptor A1 antagonist 5

    CAS:
    1,3-Dipropyl-8-phenylxanthine is an adenosine antagonist, oxypurine, insecticide, and reduces high blood pressure.
    Fórmula:C17H20N4O2
    Pureza:99.97%
    Cor e Forma:Solid
    Peso molecular:312.37

    Ref: TM-T22466

    1mg
    46,00€
    5mg
    94,00€
    10mg
    137,00€
    25mg
    226,00€
    50mg
    324,00€
    100mg
    447,00€
    200mg
    600,00€
  • MRS1177

    CAS:
    MRS1177 is an effective and selective antagonist of the human Adenosine A3 receptor (hA3AR) (Ki: 0.3 nM).
    Fórmula:C20H12ClN5O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:389.79

    Ref: TM-T16137

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • XU1

    CAS:
    XU1(Benzo[c][1,8]naphthyridin-6(5h)-One) is an Aurora protein kinase inhibitor used for the treatment of diseases suitable for inhibition, regulation or
    Fórmula:C12H8N2O
    Pureza:97.81% - 99.59%
    Cor e Forma:Solid
    Peso molecular:196.2

    Ref: TM-T29170

    1mg
    295,00€
    5mg
    705,00€
    10mg
    982,00€
    25mg
    1.485,00€
    50mg
    2.008,00€
    100mg
    2.655,00€
  • HEMADO

    CAS:
    HEMADO is a potent and selective agonist of adenosine A3 receptor (Ki: 1.1 nM at the human A3 subtype).
    Fórmula:C17H23N5O4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:361.4

    Ref: TM-T15468

    1mg
    112,00€
    5mg
    388,00€
  • A1AR antagonist 6

    CAS:
    A1AR antagonist 6 (compound 15) is a potent and selective antagonist of A1 adenosine receptor(A1AR) with a pKi of 7.13 and a pIC 50 of 6.38[1].
    Fórmula:C17H15N3O2
    Cor e Forma:Solid
    Peso molecular:293.32

    Ref: TM-T60615

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • Lu AA41063

    CAS:
    Lu AA41063 is a potent and selective antagonist of the hA2A receptor.
    Fórmula:C16H17F2N3O2S
    Cor e Forma:Solid
    Peso molecular:353.39

    Ref: TM-T24418

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • Neladenoson dalanate HCl

    CAS:
    Neladenoson dalanate HCl is a potent, selective, orally active partial agonist of adenosine A1 receptor (EC50: 0.1 nM).
    Fórmula:C35H35Cl2N7O4S2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:752.73

    Ref: TM-T24526

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • A3AR antagonist 1

    CAS:
    A3AR antagonist 1 is a potent and selective human A3adenosine receptor (AR) antagonist (Ki: 4.63) and has no affinity for the rat A3AR.
    Fórmula:C32H24N4O4S
    Cor e Forma:Solid
    Peso molecular:560.62

    Ref: TM-T63960

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • Adenosine receptor antagonist 2

    CAS:
    Adenosine receptor antagonist 2 is an orally active A2a (IC50: 1 nM), A2b (IC50: 3 nM) adenosine receptor antagonist that exhibits antitumour effects.
    Fórmula:C23H21FN8O
    Cor e Forma:Solid
    Peso molecular:444.46

    Ref: TM-T62611

    25mg
    1.791,00€
    50mg
    3.025,00€
  • CAY10498

    CAS:
    A3 AR antagonist CAY10498, with Ki of 37 nM, is 60-200x selective over A1/A2A receptors; no dedifferentiation effects shown.
    Fórmula:C18H20N6
    Cor e Forma:Solid
    Peso molecular:320.39

    Ref: TM-T37669

    1mg
    712,00€
    5mg
    3.132,00€
    500µg
    386,00€
  • VUF8507

    CAS:
    Vuf8507 is an allosteric regulator of adenosine receptor.
    Fórmula:C21H15N3O
    Cor e Forma:Solid
    Peso molecular:325.36

    Ref: TM-T35086

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • PD 81723

    CAS:
    Allosteric potentiator at the adenosine A1 receptor
    Fórmula:C14H12F3NOS
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:299.31

    Ref: TM-T23130

    10mg
    623,00€
    50mg
    2.565,00€
  • Sipagladenant

    CAS:
    Sipagladenant: oral inverse agonist for A2A adenosine receptor, may aid frontal lobe dysfunction research.
    Fórmula:C20H19N3O4S
    Cor e Forma:Solid
    Peso molecular:397.45

    Ref: TM-T61876

    25mg
    690,00€
    50mg
    895,00€
    100mg
    1.566,00€
  • SCH-202676 HBr

    CAS:
    SCH-202676 HBr is an allosteric agonist. It also an GPCR antagonist.
    Fórmula:C15H13N3S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:267.35

    Ref: TM-T24770

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • A3AR antagonist 2

    CAS:
    A3AR antagonist 2 is a potent antagonist of the human A3 adenosine receptor, exhibiting a Ki value of 4.54 nM.
    Fórmula:C22H16N6O3
    Cor e Forma:Solid
    Peso molecular:412.4

    Ref: TM-T72588

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • TH-162

    CAS:
    TH-162 (R)-PIA is an A1 adenosine receptor agonist with ~100× higher affinity than its (+)-isomer.
    Fórmula:C19H23N5O4
    Cor e Forma:Solid
    Peso molecular:385.42

    Ref: TM-T26266

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • PQ-69

    CAS:
    PQ-69 is a selective adenosine A1 receptor antagonist with inverse agonist activity.
    Fórmula:C20H19FN4O
    Cor e Forma:Solid
    Peso molecular:350.39

    Ref: TM-T28446

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • MRS 1523

    CAS:
    MRS 1523: selective adenosine A3 antagonist, Ki 18.9/113 nM (human/rat), blocks N-type Ca channels & inhibits action potentials in rat DRG neurons.
    Fórmula:C23H29NO3S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:399.55

    Ref: TM-T16135

    1mg
    178,00€
    5mg
    610,00€
  • Inupadenant

    CAS:
    Inupadenant is an orally active, highly selective A2A receptor antagonist. Inupadenant is not brain-penetrant. Inupadenant has potent anti-tumor activity[1].
    Fórmula:C25H26F2N8O4S2
    Cor e Forma:Solid
    Peso molecular:604.65

    Ref: TM-T37014

    25mg
    2.313,00€
  • CAY10680

    CAS:
    CAY10680 inhibits MAO-B (IC50=34.9 nM) & A2A receptors (Ki=39.5 nM), sparing other adenosine types & MAO-A, may treat Parkinson's.
    Fórmula:C18H16N2O2S
    Cor e Forma:Solid
    Peso molecular:324.4

    Ref: TM-T37354

    5mg
    239,00€
    10mg
    421,00€
    25mg
    945,00€
    50mg
    1.701,00€
  • FR-194921

    CAS:
    FR-194921: potent oral adenosine A1 antagonist, improves cognition, reduces anxiety, similar efficacy in humans, rats, mice.
    Fórmula:C23H23N5O
    Cor e Forma:Solid
    Peso molecular:385.46

    Ref: TM-T27379

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • CVT-2759

    CAS:
    CVT-2759, potential A(1)-ADOR partial agonist, could slow ventricular rate without severe cardiac side effects.
    Fórmula:C17H24N6O6
    Cor e Forma:Solid
    Peso molecular:408.41

    Ref: TM-T31119

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • Adenosine receptor inhibitor 2

    CAS:
    Compound 14b is a potent AR inhibitor with dual affinity, stronger for A1 (Ki = 52.2 nM) than A2A (Ki = 167 nM) ARs.
    Fórmula:C17H20BrN5O2
    Cor e Forma:Solid
    Peso molecular:406.28

    Ref: TM-T62018

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • Acefylline piperazine

    CAS:
    Acefylline piperazine, a less toxic theophylline derivative, treats asthma and bronchitis by bronchodilation, stimulating respiration and CNS.
    Fórmula:C9H10N4O4·xC4H10N2
    Cor e Forma:Solid
    Peso molecular:562.54

    Ref: TM-T70097

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • JNJ-40255293

    CAS:
    JNJ-40255293 is an antagonist of adenosine A2A/A1.
    Fórmula:C23H22N4O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:402.45

    Ref: TM-T24209

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • AK-IN-1

    CAS:
    AK-IN-1: competitive adenosine inhibitor, not ATP; inhibits AK 86-89% at 2-10 µM; promising for ischaemia, inflammation, seizure research.
    Fórmula:C22H21N3O4
    Cor e Forma:Solid
    Peso molecular:391.42

    Ref: TM-T73436

    25mg
    A consultar
    50mg
    A consultar
    100mg
    A consultar
  • ATL-801

    CAS:
    ATL-801 is anselective antagonist of A2B receptor with herapeutic activity for colitis.
    Fórmula:C24H25N7O3
    Cor e Forma:Solid
    Peso molecular:459.5

    Ref: TM-T26680

    25mg
    1.504,00€
    50mg
    1.963,00€
    100mg
    2.520,00€
  • Kira8 Hydrochloride

    CAS:
    Kira8 Hydrochloride is a mono-selective IRE1α inhibitor that allosterically attenuates IRE1α RNase activity with an IC50 of 5.9 nM.
    Fórmula:C31H30Cl2N6O3S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:637.58

    Ref: TM-T11762

    5mg
    1.018,00€
  • A2AAR/HDAC-IN-2

    CAS:
    A2AAR/HDAC-IN-2: potent dual A2AAR/HDAC inhib., Ki 10.3 nM, IC50 18.5 nM, anti-tumor potential.
    Fórmula:C23H26N6O4
    Cor e Forma:Solid
    Peso molecular:450.49

    Ref: TM-T62717

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • Theophylline sodium glycinate

    CAS:
    Theophylline sodium glycinate inhibits PDE3, treats asthma/COPD, blocks adenosine receptors, activates HDAC, reduces inflammation and induces apoptosis.
    Fórmula:C9H12N5NaO4
    Cor e Forma:Solid
    Peso molecular:277.216

    Ref: TM-T60511

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • hA2AAR antagonist 1

    CAS:
    Compound 4a, also known as hA2AAR antagonist 1, is a highly selective hA2AAR antagonist with a Ki value of 5 nM. It is useful in the field of immuno-oncology research.
    Fórmula:C15H15N5O
    Cor e Forma:Solid
    Peso molecular:281.31

    Ref: TM-T88549

    25mg
    1.458,00€
    50mg
    1.839,00€
    100mg
    2.322,00€
  • LUF5831

    CAS:
    LUF5831 is an agonist of adenosine A1 receptor.
    Fórmula:C15H12N4O2S
    Cor e Forma:Solid
    Peso molecular:312.35

    Ref: TM-T27861

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • Draflazine

    CAS:
    Draflazine: ENT1 inhibitor, reverses hypersensitivity in CFA and carrageenan-induced hyperalgesia.
    Fórmula:C30H33Cl2F2N5O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:604.52

    Ref: TM-T15167

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • LUF5981

    CAS:
    LUF5981 is a selective agonist of human adenosine A1 receptor.
    Fórmula:C24H23N3
    Cor e Forma:Solid
    Peso molecular:353.46

    Ref: TM-T27862

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • Cirazoline hydrochloride

    CAS:
    Cirazoline hydrochloride is a synthetic competitive full agonist of α1A-AR (Ki 120 nM) and partial agonist at α1B-AR and α1D-AR.
    Fórmula:C13H17ClN2O
    Pureza:99.863%
    Cor e Forma:Solid
    Peso molecular:252.74

    Ref: TM-T14972

    1mg
    60,00€
    5mg
    130,00€
    10mg
    192,00€
    25mg
    324,00€
    50mg
    480,00€
    100mg
    683,00€
    200mg
    888,00€
  • Bamifylline Hydrochloride

    CAS:
    Bamifylline Hydrochloride, an adenosine A1 receptor antagonist, is uesd to treat bronchiectasis and chronic obstructive pulmonary disease.
    Fórmula:C20H28ClN5O3
    Cor e Forma:Solid
    Peso molecular:421.92

    Ref: TM-T26737

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • MRS1067

    CAS:
    MRS1067 is an antagonist of A3 adenosine receptor.
    Fórmula:C19H16Cl2O3
    Cor e Forma:Solid
    Peso molecular:363.23

    Ref: TM-T28097

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • VUF8504

    CAS:
    VUF8504 is a novel ligand of adenosine A3 receptor.
    Fórmula:C22H17N3O2
    Cor e Forma:Solid
    Peso molecular:355.39

    Ref: TM-T29148

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • WRC-0571

    CAS:
    WRC-0571 is a highly potent, selective antagonist of A1 adenosine receptors.
    Fórmula:C17H26N6O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:330.43

    Ref: TM-T29162

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • Naxifylline

    CAS:
    Naxifylline is an A1 adenosine receptor blocker that increases urine and protects kidneys during edema treatment in heart failure.
    Fórmula:C18H24N4O3
    Cor e Forma:Solid
    Peso molecular:344.41

    Ref: TM-T33600

    25mg
    2.043,00€
    50mg
    2.682,00€
    100mg
    3.600,00€
  • CP 66713

    CAS:
    CP-66713 is an adenosine A2 receptor antagonist.
    Fórmula:C15H10ClN5
    Cor e Forma:Solid
    Peso molecular:295.73

    Ref: TM-T31026

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • A2AAR antagonist 1

    CAS:
    Compound 21a, A2AAR antagonist with 20 nM Ki, useful in neurodegenerative disease study.
    Fórmula:C12H8BrN3O
    Cor e Forma:Solid
    Peso molecular:290.12

    Ref: TM-T60591

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • MRE3008F20

    CAS:
    MRE3008F20 is an AA3R antagonist that inhibits Cl-IB-MECA-induced cAMP production and can be used to study glaucoma and asthma.
    Fórmula:C21H20N8O3
    Pureza:97.29%
    Cor e Forma:Solid
    Peso molecular:432.44

    Ref: TM-T16132

    1mg
    66,00€
    2mg
    96,00€
    5mg
    144,00€
    10mg
    205,00€
    25mg
    349,00€
    50mg
    512,00€
  • A2AR-antagonist-1

    CAS:
    Oral A2AR-antagonist-1, IC50 29 nM; anti-tumor, stable in mice (t1/2 86.1 min), boosts T cells, impedes LAG-3/TIM-3.
    Fórmula:C27H25N5O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:451.52

    Ref: TM-T72626

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • VUF 5574

    CAS:
    VUF 5574 is a selective antagonist of adenosine A3 receptor with a Ki of 4.03 nM for the recombinant human receptor.
    Fórmula:C21H17N5O2
    Pureza:99.53%
    Cor e Forma:Solid
    Peso molecular:371.39

    Ref: TM-T23518

    5mg
    58,00€
    10mg
    94,00€
    25mg
    152,00€
    50mg
    210,00€
    100mg
    305,00€
    200mg
    425,00€
  • ST3932

    CAS:
    ST3932 is a ST1535 metabolite, is a adenosine A2A receptor antagonist(Kis of 8 nM and 33 nM for A2A and A1 receptors, respectively).
    Fórmula:C12H16N8O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:288.31

    Ref: TM-T13008

    25mg
    1.504,00€
    50mg
    1.963,00€
    100mg
    2.520,00€
  • N6-Cyclopentyladenosine

    CAS:
    N6-Cyclopentyladenosine (CPA) is a selective agonist of the adenosine A1 receptor and can be used to mimic the action of the adenosine A1 receptor, with Ki's of
    Fórmula:C15H21N5O4
    Pureza:99.95%
    Cor e Forma:Solid
    Peso molecular:335.36

    Ref: TM-T16263

    10mg
    43,00€
    25mg
    69,00€
    50mg
    93,00€
    100mg
    130,00€
    200mg
    178,00€
    1mL*10mM (DMSO)
    33,00€
  • N-[(4-Aminophenyl)methyl]adenosine

    CAS:
    N-[(4-Aminophenyl)methyl]adenosine is an adenosine receptor inhibitor (Ki: 29 nM for Rat ecto-5′-Nucleotidase).
    Fórmula:C17H20N6O4
    Pureza:98.75%
    Cor e Forma:Solid
    Peso molecular:372.38

    Ref: TM-T16166

    1mg
    52,00€
    5mg
    111,00€
    10mg
    166,00€
    25mg
    318,00€
    50mg
    504,00€
    100mg
    803,00€
    1mL*10mM (DMSO)
    141,00€
  • Sonedenoson

    CAS:
    Sonedenoson (MRE0094) is an adenosine A(2A) receptor agonist and potential inhibitor potentially targeting SARS-CoV-2 coronavirus 2;-O-ribose methyltransferase.
    Fórmula:C18H20ClN5O5
    Pureza:99.79%
    Cor e Forma:Solid
    Peso molecular:421.84

    Ref: TM-T34685

    1mg
    264,00€
    5mg
    650,00€
    10mg
    888,00€
    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • KI-7

    CAS:
    KI-7 is an adenosine A2B receptor positive allosteric modulator.
    Fórmula:C23H18N2O2
    Pureza:98.33%
    Cor e Forma:Solid
    Peso molecular:354.4

    Ref: TM-T9238

    2mg
    35,00€
    5mg
    55,00€
    10mg
    95,00€
    25mg
    172,00€
    50mg
    264,00€
    100mg
    399,00€
    200mg
    560,00€
    1mL*10mM (DMSO)
    62,00€
  • Adenosine antagonist-1

    CAS:

    Adenosine antagonist-1 acts as an adenosine A3 receptor (AA3R) antagonist.

    Fórmula:C18H13N7S
    Pureza:99.28% - 99.95%
    Cor e Forma:Solid
    Peso molecular:359.41

    Ref: TM-T10248

    1mg
    48,00€
    5mg
    92,00€
    10mg
    137,00€
    25mg
    210,00€
    50mg
    314,00€
    100mg
    495,00€
    200mg
    705,00€
  • BAY 60-6583

    CAS:
    BAY 60-6583 is a potent, high-affinity adenosine A2B receptor agonist (EC50 = 3 nM) with affinity for A2B receptors that exceeds that for A1, A2A, and A3
    Fórmula:C19H17N5O2S
    Pureza:98.46% - 99.8%
    Cor e Forma:Solid
    Peso molecular:379.44

    Ref: TM-T14506

    1mg
    39,00€
    2mg
    50,00€
    5mg
    84,00€
    10mg
    116,00€
    25mg
    233,00€
    50mg
    376,00€
    100mg
    567,00€
    200mg
    797,00€
    1mL*10mM (DMSO)
    101,00€
  • GW-493838

    CAS:
    GW-493838 is a potent adenosine A1A receptor agonist for the treatment of dyslipidemia and neuropathic pain, with analgesic effects on post-herpetic neuralgia
    Fórmula:C21H21ClFN7O4
    Pureza:99.11% - 99.58%
    Cor e Forma:Solid
    Peso molecular:489.89

    Ref: TM-T27509

    1mg
    143,00€
    5mg
    346,00€
    10mg
    492,00€
    25mg
    740,00€
    50mg
    999,00€
    100mg
    1.350,00€
    500mg
    2.647,00€
    1mL*10mM (DMSO)
    399,00€
  • ST-1535

    CAS:
    ST 1535: potent, oral A2A adenosine receptor antagonist with antiparkinsonian and antitremor effects, promising for Parkinson's research.
    Fórmula:C12H16N8
    Pureza:99.64% - 99.69%
    Cor e Forma:Solid
    Peso molecular:272.31

    Ref: TM-T28861

    1mg
    34,00€
    5mg
    75,00€
    10mg
    92,00€
    25mg
    150,00€
    50mg
    215,00€
    100mg
    321,00€
    1mL*10mM (DMSO)
    75,00€
  • N6-(2-Phenylethyl)adenosine

    CAS:
    N6-(2-Phenylethyl)adenosine (N6-Phenethyladenosine) is an adenosine derivative and an agonist of adenosine receptors with Ki values of 11.8 nM and 30.1 nM for
    Fórmula:C18H21N5O4
    Pureza:99.83%
    Cor e Forma:Solid
    Peso molecular:371.39

    Ref: TM-T12163

    10mg
    33,00€
    25mg
    59,00€
    50mg
    104,00€
    100mg
    177,00€
    200mg
    316,00€
    1mL*10mM (DMSO)
    33,00€
  • A2A receptor antagonist 1

    CAS:
    A2A receptor antagonist 1 (CPI-444 analog) is an antagonist of both adenosine A2A receptor and A1 receptor with Kis of 4 and 264 nM, respectively.
    Fórmula:C16H12FN5O
    Pureza:99.52% - 99.93%
    Cor e Forma:Solid
    Peso molecular:309.3

    Ref: TM-T37792

    2mg
    A consultar
    5mg
    62,00€
    10mg
    87,00€
    25mg
    183,00€
    50mg
    280,00€
    100mg
    416,00€
    200mg
    A consultar
    1mL*10mM (DMSO)
    47,00€
  • N 0861

    CAS:
    N 0861 is a selective adenosine A1 receptor antagonist that attenuates renal insufficiency during adenosine-controlled hypotension in rats.
    Fórmula:C13H17N5
    Pureza:98.78%
    Cor e Forma:Solid
    Peso molecular:243.31

    Ref: TM-T70722

    1mg
    164,00€
    2mg
    234,00€
    5mg
    389,00€
    10mg
    532,00€
    25mg
    820,00€
    50mg
    1.063,00€
    100mg
    1.423,00€
    200mg
    1.945,00€
  • ANR 94

    CAS:
    ANR94 is a potent hAA2AR antagonist (Ki 46 nM) with potential for Parkinson's research.
    Fórmula:C9H13N5O
    Pureza:98.9%
    Cor e Forma:Solid
    Peso molecular:207.23

    Ref: TM-T22031

    5mg
    46,00€
    10mg
    71,00€
    25mg
    130,00€
    50mg
    219,00€
    100mg
    309,00€
    200mg
    434,00€
    1mL*10mM (DMSO)
    46,00€
  • ISAM-140

    CAS:
    ISAM-140 is a potent and highly selective antagonist of A2B adenosine receptor.
    Fórmula:C19H19N3O3
    Pureza:99.51%
    Cor e Forma:Solid
    Peso molecular:337.37

    Ref: TM-T27629

    5mg
    52,00€
    10mg
    69,00€
    25mg
    100,00€
    50mg
    149,00€
    100mg
    207,00€
    1mL*10mM (DMSO)
    52,00€
  • GS-9667

    CAS:
    GS-9667, a selective and partial agonist of the A(1) adenosine receptor (AR), represents an effective therapy for Type 2 diabetes (T2DM) and dyslipidemia via
    Fórmula:C21H24FN5O4S
    Pureza:99.77% - 99.96%
    Cor e Forma:Solid
    Peso molecular:461.51

    Ref: TM-T27439

    1mg
    71,00€
    5mg
    161,00€
    10mg
    215,00€
    25mg
    353,00€
    50mg
    482,00€
    100mg
    665,00€
    200mg
    893,00€
  • APNEA

    CAS:
    APNEA ((2R,3R,4S,5R)-2-[6-[2-(4-aminophenyl)ethylamino]purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol) is a non-selective agonist of adenosine A3 receptor.
    Fórmula:C18H22N6O4
    Pureza:99.88%
    Cor e Forma:Solid
    Peso molecular:386.41

    Ref: TM-T12159

    25mg
    48,00€
    1mL*10mM (DMSO)
    33,00€
  • LAS38096

    CAS:
    LAS38096 is an A2B adenosine receptor antagonist (Ki : 17 nM) that is potent, selective and efficient .
    Fórmula:C17H12N6O
    Pureza:99.18% - 99.95%
    Cor e Forma:Solid
    Peso molecular:316.32

    Ref: TM-T27800

    1mg
    137,00€
    5mg
    314,00€
    10mg
    427,00€
    25mg
    600,00€
    50mg
    798,00€
    100mg
    1.099,00€
    200mg
    1.468,00€
  • Evodenoson

    CAS:
    Evodenoson (ATL313), a potent A2aR agonist, treats eye diseases, tumors, and immune disorders; potential for glaucoma and blood cancer studies.
    Fórmula:C23H29N7O6
    Pureza:99.75% - 99.83%
    Cor e Forma:Solid
    Peso molecular:499.52

    Ref: TM-T31731

    1mg
    225,00€
    5mg
    567,00€
    10mg
    855,00€
    25mg
    1.645,00€
    50mg
    2.215,00€
    100mg
    3.348,00€
  • MRS1220

    CAS:
    MRS1220, a selective and potent antagonist for the human A3 adenosine receptor (hA3AR) with a dissociation constant (Ki) of 0.59 nM, exhibits therapeutic
    Fórmula:C21H14ClN5O2
    Pureza:98.43%
    Cor e Forma:Solid
    Peso molecular:403.82

    Ref: TM-T23016

    1mg
    50,00€
    5mg
    110,00€
    10mg
    168,00€
    25mg
    288,00€
    50mg
    414,00€
    100mg
    583,00€
    500mg
    A consultar
  • 2'-MeCCPA

    CAS:
    2'-MeCCPA is an A1AR agonist that inhibits trichothecene-stimulated adenylate cyclase activity and has analgesic activity for the study of HCV.
    Fórmula:C16H22ClN5O4
    Pureza:99.93%
    Cor e Forma:Solid
    Peso molecular:383.83

    Ref: TM-T22489

    1mg
    35,00€
    5mg
    71,00€
    10mg
    123,00€
    25mg
    197,00€
    50mg
    301,00€
    100mg
    434,00€
    200mg
    615,00€
  • FK-453

    CAS:
    FK-453 is a potent antagonist of non-xanthine adenosine A1 receptor with diuretic and renal vasodilatory activity.
    Fórmula:C23H25N3O2
    Pureza:99.44%
    Cor e Forma:Solid
    Peso molecular:375.46

    Ref: TM-T27323

    1mg
    192,00€
    5mg
    480,00€
    10mg
    690,00€
    25mg
    1.044,00€
    50mg
    1.414,00€
    100mg
    1.908,00€
    200mg
    2.575,00€
  • Selodenoson

    CAS:
    Selodenoson (RG-14202) is a selective adenosine A1 receptor agonist used to slow the heart rate in patients with atrial fibrillation and to treat arrhythmias.
    Fórmula:C17H24N6O4
    Pureza:99.39%
    Cor e Forma:Solid
    Peso molecular:376.41

    Ref: TM-T28748

    1mg
    84,00€
    5mg
    172,00€
    10mg
    254,00€
    25mg
    416,00€
    50mg
    610,00€
    100mg
    872,00€
    200mg
    1.161,00€
  • Neladenoson dalanate

    CAS:
    Neladenoson dalanate (BAY-1067197), an oral Adenosine A1 receptor partial agonist, is safe with good pharmacokinetics for chronic heart disease.
    Fórmula:C35H34ClN7O4S2
    Cor e Forma:Solid
    Peso molecular:716.27

    Ref: TM-T71157

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€