Receptor de adenosina
Os receptores de adenosina são uma classe de GPCRs que respondem ao nucleosídeo endógeno adenosina. Esses receptores estão envolvidos na regulação de vários processos fisiológicos, incluindo função cardiovascular, ciclos de sono-vigília e respostas imunes. Moduladores de receptores de adenosina têm potencial terapêutico no tratamento de condições como arritmias cardíacas, inflamação e doenças neurodegenerativas. Na CymitQuimica, oferecemos uma seleção de moduladores de receptores de adenosina de alta qualidade para apoiar sua pesquisa em biologia cardiovascular, neurociência e imunologia.
Foram encontrados 242 produtos de "Receptor de adenosina"
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MRS1220
CAS:<p>MRS1220, a selective and potent antagonist for the human A3 adenosine receptor (hA3AR) with a dissociation constant (Ki) of 0.59 nM, exhibits therapeutic</p>Fórmula:C21H14ClN5O2Pureza:98.43%Cor e Forma:SolidPeso molecular:403.82N 0861
CAS:<p>N 0861 is a selective adenosine A1 receptor antagonist that attenuates renal insufficiency during adenosine-controlled hypotension in rats.</p>Fórmula:C13H17N5Pureza:98.78%Cor e Forma:SolidPeso molecular:243.31Selodenoson
CAS:<p>Selodenoson (RG-14202) is a selective adenosine A1 receptor agonist used to slow the heart rate in patients with atrial fibrillation and to treat arrhythmias.</p>Fórmula:C17H24N6O4Pureza:99.52%Cor e Forma:SolidPeso molecular:376.41ISAM-140
CAS:<p>ISAM-140 is a potent and highly selective antagonist of A2B adenosine receptor.</p>Fórmula:C19H19N3O3Pureza:99.51%Cor e Forma:SolidPeso molecular:337.37GW-493838
CAS:<p>GW-493838 is a potent adenosine A1A receptor agonist for the treatment of dyslipidemia and neuropathic pain, with analgesic effects on post-herpetic neuralgia</p>Fórmula:C21H21ClFN7O4Pureza:99.11% - 99.58%Cor e Forma:SolidPeso molecular:489.89GS-9667
CAS:<p>GS-9667, a selective and partial agonist of the A(1) adenosine receptor (AR), represents an effective therapy for Type 2 diabetes (T2DM) and dyslipidemia via</p>Fórmula:C21H24FN5O4SPureza:99.76% - 99.77%Cor e Forma:SolidPeso molecular:461.51A2A receptor antagonist 1
CAS:<p>A2A receptor antagonist 1 (CPI-444 analog) is an antagonist of both adenosine A2A receptor and A1 receptor with Kis of 4 and 264 nM, respectively.</p>Fórmula:C16H12FN5OPureza:99.52% - 99.93%Cor e Forma:SolidPeso molecular:309.3LAS38096
CAS:<p>LAS38096 is an A2B adenosine receptor antagonist (Ki : 17 nM) that is potent, selective and efficient .</p>Fórmula:C17H12N6OPureza:99.18% - 99.95%Cor e Forma:SolidPeso molecular:316.32N6-(2-Phenylethyl)adenosine
CAS:<p>N6-(2-Phenylethyl)adenosine (N6-Phenethyladenosine) is an adenosine derivative and an agonist of adenosine receptors with Ki values of 11.8 nM and 30.1 nM for</p>Fórmula:C18H21N5O4Pureza:99.83%Cor e Forma:SolidPeso molecular:371.392'-MeCCPA
CAS:<p>2'-MeCCPA is an A1AR agonist that inhibits trichothecene-stimulated adenylate cyclase activity and has analgesic activity for the study of HCV.</p>Fórmula:C16H22ClN5O4Pureza:99.93%Cor e Forma:SolidPeso molecular:383.83KI-7
CAS:<p>KI-7 is an adenosine A2B receptor positive allosteric modulator.</p>Fórmula:C23H18N2O2Pureza:98.33%Cor e Forma:SolidPeso molecular:354.4FK-453
CAS:<p>FK-453 is a potent antagonist of non-xanthine adenosine A1 receptor with diuretic and renal vasodilatory activity.</p>Fórmula:C23H25N3O2Pureza:99.44%Cor e Forma:SolidPeso molecular:375.46GP3269
CAS:<p>GP3269 is a selective, potent, orally active human adenosine kinase (AK) inhibitor (IC50: 11 nM) with anticonvulsant effects in rats.</p>Fórmula:C23H21FN4O3Cor e Forma:SolidPeso molecular:420.44PSB-1115 potassium salt
CAS:<p>PSB-1115 potassium salt, a selective A2B Adenosine Receptor antagonist, inhibits the 2,4,6-trinitrobenzenesulfonic acid (TNBS)-induced contraction inhibition of acetylcholine (ACh) [1].</p>Fórmula:C14H13KN4O5SCor e Forma:SolidPeso molecular:388.44MRS3558
CAS:<p>MRS3558 is an agonist of A3 adenosine receptors.</p>Fórmula:C20H20Cl2N6O3Cor e Forma:SolidPeso molecular:463.32ABT-702 hydrochloride
CAS:<p>ABT-702 hydrochloride effectively inhibits adenosine kinase, exhibiting an IC50 value of 1.7 nM [1] [2].</p>Fórmula:C22H20BrClN6OCor e Forma:SolidPeso molecular:499.79KFM19
CAS:<p>KFM19 is a potent and selective adenosine receptor (A1-receptor) antagonist (IC50 : 50 nM) for the study of neurological disorders.</p>Fórmula:C16H22N4O3Pureza:98.62%Cor e Forma:SolidPeso molecular:318.37Neladenoson dalanate
CAS:<p>Neladenoson dalanate (BAY-1067197), an oral Adenosine A1 receptor partial agonist, is safe with good pharmacokinetics for chronic heart disease.</p>Fórmula:C35H34ClN7O4S2Cor e Forma:SolidPeso molecular:716.27Sulmazole
CAS:<p>Sulmazole (AR-L 115-BS) is a small molecule Sulmazole is a small molecule cGMP-PDE inhibitor.Sulmazole is a competitive inhibitor of A1 adenosine receptors.</p>Fórmula:C14H13N3O2SPureza:99.94%Cor e Forma:SolidPeso molecular:287.34Xanthine amine congener
CAS:<p>Xanthine amine congener is an Adenosine receptor antagonist.</p>Fórmula:C21H28N6O4Pureza:99.7%Cor e Forma:SolidPeso molecular:428.48
