Receptor de adenosina
Os receptores de adenosina são uma classe de GPCRs que respondem ao nucleosídeo endógeno adenosina. Esses receptores estão envolvidos na regulação de vários processos fisiológicos, incluindo função cardiovascular, ciclos de sono-vigília e respostas imunes. Moduladores de receptores de adenosina têm potencial terapêutico no tratamento de condições como arritmias cardíacas, inflamação e doenças neurodegenerativas. Na CymitQuimica, oferecemos uma seleção de moduladores de receptores de adenosina de alta qualidade para apoiar sua pesquisa em biologia cardiovascular, neurociência e imunologia.
Foram encontrados 242 produtos de "Receptor de adenosina"
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5'-Amino-5'-deoxyadenosine
CAS:<p>5'-Amino-5'-deoxyadenosine (NH2dAdo) is an adenosine kinase inhibitor targeting malignant tumors of the inert lymphatic system with antitumor and anticancer</p>Fórmula:C10H14N6O3Pureza:95.55%Cor e Forma:SolidPeso molecular:266.26Blontuvetmab
CAS:<p>Blontuvetmab (AT 004), a caninized CD20 monoclonal antibody, is utilized in the study of Canine B-cell lymphoma [1].</p>Cor e Forma:LiquidAdenosine receptor inhibitor 1
CAS:<p>Potent, selective adenosine receptor blocker with strong affinity, especially A2A (Ki 68.5 nM). Promising for cancer, neurodegeneration study.</p>Fórmula:C17H19ClFN5O3Cor e Forma:SolidPeso molecular:395.82A1AR antagonist 2
CAS:<p>Compound 18h is a potent A1 adenosine receptor blocker with Ki of 1.49 nM for hA1, 10.2 nM for hA2A, 50.1 nM for hA2B.</p>Fórmula:C17H12N4OCor e Forma:SolidPeso molecular:288.3TC-G 1004
CAS:<p>adenosine A2A receptors antagonist</p>Fórmula:C22H27N7O2Pureza:98%Cor e Forma:SolidPeso molecular:421.5SCH-202676 HBr
CAS:<p>SCH-202676 HBr is an allosteric agonist. It also an GPCR antagonist.</p>Fórmula:C15H13N3SPureza:98%Cor e Forma:SolidPeso molecular:267.35A2AR-agonist-1
CAS:<p>A2AR-agonist-1 targets A2A Receptor/ENT1 for neuroprotection; potent with Ki of 4.39 (A2AR), 3.47 (ENT1).</p>Fórmula:C20H22N6O4Pureza:99.9%Cor e Forma:SolidPeso molecular:410.43Lu AA 47070
CAS:<p>adenosine A2A receptor antagonist</p>Fórmula:C17H20F2N3O6PSPureza:98%Cor e Forma:SolidPeso molecular:463.39VUF8507
CAS:<p>Vuf8507 is an allosteric regulator of adenosine receptor.</p>Fórmula:C21H15N3OCor e Forma:SolidPeso molecular:325.36Acefylline piperazine
CAS:<p>Acefylline piperazine, a less toxic theophylline derivative, treats asthma and bronchitis by bronchodilation, stimulating respiration and CNS.</p>Fórmula:C9H10N4O4·xC4H10N2Cor e Forma:SolidPeso molecular:562.54CAY10498
CAS:<p>A3 AR antagonist CAY10498, with Ki of 37 nM, is 60-200x selective over A1/A2A receptors; no dedifferentiation effects shown.</p>Fórmula:C18H20N6Cor e Forma:SolidPeso molecular:320.39Apadenoson
CAS:<p>Apadenoson: potent A2 agonist, A3 inhibitor (IC 45 nM), anti-inflammatory, for neurological research.</p>Fórmula:C23H30N6O6Pureza:98%Cor e Forma:SolidPeso molecular:486.52CVT-2759
CAS:<p>CVT-2759, potential A(1)-ADOR partial agonist, could slow ventricular rate without severe cardiac side effects.</p>Fórmula:C17H24N6O6Cor e Forma:SolidPeso molecular:408.41MRS-1191
CAS:<p>MRS-1191 is an effective and selective A3 adenosine receptor antagonist (KB: 92 nM, a Ki: 31.4 nM for human A3 receptor and an IC50: 120 nM for CHO cells).</p>Fórmula:C31H27NO4Cor e Forma:SolidPeso molecular:477.55Adenosine receptor inhibitor 2
CAS:<p>Compound 14b is a potent AR inhibitor with dual affinity, stronger for A1 (Ki = 52.2 nM) than A2A (Ki = 167 nM) ARs.</p>Fórmula:C17H20BrN5O2Cor e Forma:SolidPeso molecular:406.28Inupadenant
CAS:<p>Inupadenant is an orally active, highly selective A2A receptor antagonist. Inupadenant is not brain-penetrant. Inupadenant has potent anti-tumor activity[1].</p>Fórmula:C25H26F2N8O4S2Cor e Forma:SolidPeso molecular:604.65PD 81723
CAS:<p>Allosteric potentiator at the adenosine A1 receptor</p>Fórmula:C14H12F3NOSPureza:98%Cor e Forma:SolidPeso molecular:299.31Sipagladenant
CAS:<p>Sipagladenant: oral inverse agonist for A2A adenosine receptor, may aid frontal lobe dysfunction research.</p>Fórmula:C20H19N3O4SCor e Forma:SolidPeso molecular:397.45Adenosine receptor antagonist 2
CAS:<p>Adenosine receptor antagonist 2 is an orally active A2a (IC50: 1 nM), A2b (IC50: 3 nM) adenosine receptor antagonist that exhibits antitumour effects.</p>Fórmula:C23H21FN8OCor e Forma:SolidPeso molecular:444.46hA2AAR antagonist 1
CAS:<p>Compound 4a, also known as hA2AAR antagonist 1, is a highly selective hA2AAR antagonist with a Ki value of 5 nM. It is useful in the field of immuno-oncology research.</p>Fórmula:C15H15N5OCor e Forma:SolidPeso molecular:281.31
