
Receptor de adenosina
Os receptores de adenosina são uma classe de GPCRs que respondem ao nucleosídeo endógeno adenosina. Esses receptores estão envolvidos na regulação de vários processos fisiológicos, incluindo função cardiovascular, ciclos de sono-vigília e respostas imunes. Moduladores de receptores de adenosina têm potencial terapêutico no tratamento de condições como arritmias cardíacas, inflamação e doenças neurodegenerativas. Na CymitQuimica, oferecemos uma seleção de moduladores de receptores de adenosina de alta qualidade para apoiar sua pesquisa em biologia cardiovascular, neurociência e imunologia.
Foram encontrados 242 produtos de "Receptor de adenosina"
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hA2AAR antagonist 1
CAS:<p>Compound 4a, also known as hA2AAR antagonist 1, is a highly selective hA2AAR antagonist with a Ki value of 5 nM. It is useful in the field of immuno-oncology research.</p>Fórmula:C15H15N5OCor e Forma:SolidPeso molecular:281.31LUF5831
CAS:<p>LUF5831 is an agonist of adenosine A1 receptor.</p>Fórmula:C15H12N4O2SCor e Forma:SolidPeso molecular:312.35Draflazine
CAS:<p>Draflazine: ENT1 inhibitor, reverses hypersensitivity in CFA and carrageenan-induced hyperalgesia.</p>Fórmula:C30H33Cl2F2N5O2Pureza:98%Cor e Forma:SolidPeso molecular:604.52LUF5981
CAS:<p>LUF5981 is a selective agonist of human adenosine A1 receptor.</p>Fórmula:C24H23N3Cor e Forma:SolidPeso molecular:353.46Cirazoline hydrochloride
CAS:<p>Cirazoline hydrochloride is a synthetic competitive full agonist of α1A-AR (Ki 120 nM) and partial agonist at α1B-AR and α1D-AR.</p>Fórmula:C13H17ClN2OPureza:99.863%Cor e Forma:SolidPeso molecular:252.74Bamifylline Hydrochloride
CAS:<p>Bamifylline Hydrochloride, an adenosine A1 receptor antagonist, is uesd to treat bronchiectasis and chronic obstructive pulmonary disease.</p>Fórmula:C20H28ClN5O3Cor e Forma:SolidPeso molecular:421.92MRS1067
CAS:<p>MRS1067 is an antagonist of A3 adenosine receptor.</p>Fórmula:C19H16Cl2O3Cor e Forma:SolidPeso molecular:363.23MRE3008F20
CAS:<p>MRE3008F20 is an AA3R antagonist that inhibits Cl-IB-MECA-induced cAMP production and can be used to study glaucoma and asthma.</p>Fórmula:C21H20N8O3Pureza:97.29%Cor e Forma:SolidPeso molecular:432.44A2AR-antagonist-1
CAS:<p>Oral A2AR-antagonist-1, IC50 29 nM; anti-tumor, stable in mice (t1/2 86.1 min), boosts T cells, impedes LAG-3/TIM-3.</p>Fórmula:C27H25N5O2Pureza:98%Cor e Forma:SolidPeso molecular:451.52VUF 5574
CAS:<p>VUF 5574 is a selective antagonist of adenosine A3 receptor with a Ki of 4.03 nM for the recombinant human receptor.</p>Fórmula:C21H17N5O2Pureza:99.53%Cor e Forma:SolidPeso molecular:371.39ST3932
CAS:<p>ST3932 is a ST1535 metabolite, is a adenosine A2A receptor antagonist(Kis of 8 nM and 33 nM for A2A and A1 receptors, respectively).</p>Fórmula:C12H16N8OPureza:98%Cor e Forma:SolidPeso molecular:288.31APNEA
CAS:<p>APNEA ((2R,3R,4S,5R)-2-[6-[2-(4-aminophenyl)ethylamino]purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol) is a non-selective agonist of adenosine A3 receptor.</p>Fórmula:C18H22N6O4Pureza:99.88%Cor e Forma:SolidPeso molecular:386.41N6-Cyclopentyladenosine
CAS:<p>N6-Cyclopentyladenosine (CPA) is a selective agonist of the adenosine A1 receptor and can be used to mimic the action of the adenosine A1 receptor, with Ki's of</p>Fórmula:C15H21N5O4Pureza:99.84%Cor e Forma:SolidPeso molecular:335.36Sonedenoson
CAS:<p>Sonedenoson (MRE0094) is an adenosine A(2A) receptor agonist and potential inhibitor potentially targeting SARS-CoV-2 coronavirus 2;-O-ribose methyltransferase.</p>Fórmula:C18H20ClN5O5Pureza:99.79%Cor e Forma:SolidPeso molecular:421.84Evodenoson
CAS:<p>Evodenoson (ATL313), a potent A2aR agonist, treats eye diseases, tumors, and immune disorders; potential for glaucoma and blood cancer studies.</p>Fórmula:C23H29N7O6Pureza:99.75% - 99.83%Cor e Forma:SolidPeso molecular:499.52N-[(4-Aminophenyl)methyl]adenosine
CAS:<p>N-[(4-Aminophenyl)methyl]adenosine is an adenosine receptor inhibitor (Ki: 29 nM for Rat ecto-5′-Nucleotidase).</p>Fórmula:C17H20N6O4Pureza:98.75%Cor e Forma:SolidPeso molecular:372.38BAY 60-6583
CAS:<p>BAY 60-6583 is a potent, high-affinity adenosine A2B receptor agonist (EC50 = 3 nM) with affinity for A2B receptors that exceeds that for A1, A2A, and A3</p>Fórmula:C19H17N5O2SPureza:98.46% - 99.8%Cor e Forma:SolidPeso molecular:379.44ANR 94
CAS:<p>ANR94 is a potent hAA2AR antagonist (Ki 46 nM) with potential for Parkinson's research.</p>Fórmula:C9H13N5OPureza:98.9%Cor e Forma:SolidPeso molecular:207.23Adenosine antagonist-1
CAS:<p>Adenosine antagonist-1 acts as an adenosine A3 receptor (AA3R) antagonist.</p>Fórmula:C18H13N7SPureza:99.28% - 99.95%Cor e Forma:SolidPeso molecular:359.41ST-1535
CAS:<p>ST 1535: potent, oral A2A adenosine receptor antagonist with antiparkinsonian and antitremor effects, promising for Parkinson's research.</p>Fórmula:C12H16N8Pureza:99.64% - 99.69%Cor e Forma:SolidPeso molecular:272.31
