Receptor de adenosina
Os receptores de adenosina são uma classe de GPCRs que respondem ao nucleosídeo endógeno adenosina. Esses receptores estão envolvidos na regulação de vários processos fisiológicos, incluindo função cardiovascular, ciclos de sono-vigília e respostas imunes. Moduladores de receptores de adenosina têm potencial terapêutico no tratamento de condições como arritmias cardíacas, inflamação e doenças neurodegenerativas. Na CymitQuimica, oferecemos uma seleção de moduladores de receptores de adenosina de alta qualidade para apoiar sua pesquisa em biologia cardiovascular, neurociência e imunologia.
Foram encontrados 249 produtos de "Receptor de adenosina"
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Amp579 TFA
Amp579 TFA is a novel adenosine A1/A2a receptor agonist that induces acute and delayed preconditioning against myocardial shock in vivo.Fórmula:C24H29ClF3N5O5SPureza:97.91%Cor e Forma:SoildPeso molecular:592.03Pentoxifylline
CAS:Pentoxifylline (PTX) stimulates cytokines, inhibits phosphodiesterase, enhances blood flow, and increases cell flexibility.Fórmula:C13H18N4O3Pureza:99.26% - 99.93%Cor e Forma:SolidPeso molecular:278.31Adenosine 5'-monophosphate monohydrate
CAS:Adenosine 5'-monophosphate monohydrate (5'-AMP) , also known as 5'-adenylic acid, is a nucleotide that is used as a monomer in RNA.
Fórmula:C10H14N5O7P·H2OPureza:97.68% - 98.49%Cor e Forma:White PowderPeso molecular:365.24Ticlopidine hydrochloride
CAS:Ticlopidine hydrochloride (Ticlodix) is an effective inhibitor of platelet aggregation commonly used in the placement of STENTS in CORONARY ARTERIES.Fórmula:C14H15Cl2NSPureza:99.85% - >99.99%Cor e Forma:White PowderPeso molecular:300.25Aminophylline
CAS:Aminophylline (Phyllocontin) is a competitive nonselective phosphodiesterase inhibitor giving a bronchodilatory effect.Fórmula:C7H8O2·C2H8N2Pureza:99.31%Cor e Forma:White Or Slightly Yellowish Granules Or Powder SolidPeso molecular:420.43AB928
CAS:AB928 is an orally bioavailable, selective dual adenosine receptor (A2aR/A2bR) antagonist. It has immunomodulatory activity[1].Fórmula:C23H22N8OPureza:98.09% - >99.99%Cor e Forma:SolidPeso molecular:426.47Ref: TM-T14078
1mg52,00€5mg117,00€10mg187,00€25mg369,00€50mg437,00€100mg628,00€1mL*10mM (DMSO)127,00€YT 146
CAS:YT 146 is a biochemical.Fórmula:C18H25N5O4Pureza:98.81% - 99.25%Cor e Forma:SolidPeso molecular:375.42CGS 15943
CAS:CGS 15943 is an orally bioavailable non-xanthine antagonist of Adenosine Receptor.Fórmula:C13H8ClN5OPureza:97.4%Cor e Forma:SolidPeso molecular:285.69Ref: TM-T14944
2mg34,00€5mg50,00€10mg82,00€25mg147,00€50mg222,00€100mg334,00€200mg494,00€1mL*10mM (DMSO)55,00€Doxofylline
CAS:Doxofylline (Doxophylline) is a methylxanthine derivative with the presence of a dioxolane group in position 7.Fórmula:C11H14N4O4Pureza:99.958% - >99.99%Cor e Forma:SolidPeso molecular:266.25Theophylline
CAS:Theophylline (1,3-Dimethylxanthine) is a methyl xanthine derivative from tea with diuretic, smooth muscle relaxant, bronchial dilation, cardiac and centralFórmula:C7H8N4O2Pureza:99.65% - 99.98%Cor e Forma:White Solid PowderPeso molecular:180.16DPTN dihydrochloride
CAS:DPTN dihydrochloride is a potent and selective A3AR antagonist with Ki values of 1.65, 9.61 and 8.53 nM in human, mouse and rat, respectively.Fórmula:C22H20Cl2N4OSPureza:99.95%Cor e Forma:SoildPeso molecular:459.39Quercetin-3'-o-phosphate TEA
Quercetin-3'-o-phosphate TEA (Quercetin 3'-phosphate TEA) is an adenosine A receptor antagonist that can be used to prevent and treat metabolic disorders.Fórmula:C21H26NO10PPureza:97.04%Cor e Forma:SoildPeso molecular:483.41Adenosine A1 receptor activator T62
CAS:Adenosine A1 receptor activator T62 is an allosteric enhancer of adenosine A1 receptor, and it produces antinociception in animal models of acute pain and alsoFórmula:C15H14ClNOSPureza:97.83%Cor e Forma:SolidPeso molecular:291.8Ref: TM-T14127
1mg64,00€5mg126,00€10mg180,00€25mg290,00€50mg396,00€100mg537,00€200mg712,00€1mL*10mM (DMSO)187,00€Theophylline monohydrate
CAS:Theophylline monohydrate (Quibron) appears to inhibit phosphodiesterase and prostaglandin production, regulate calcium flux and intracellular calciumFórmula:C7H8N4O2·H2OPureza:99.78%Cor e Forma:SolidPeso molecular:198.18N6-Ethyladenosine
CAS:N6-Ethyladenosine is an adenosine derivative, acts as an agonist of Adenosine receptor(hA1AR and hA3AR with Kis of 4.9 and 4.7 nM , respectively).Fórmula:C12H17N5O4Pureza:99.96%Cor e Forma:SolidPeso molecular:295.29Pamabrom
CAS:Pamabrom is a diuretic for premenstrual and menstrual bloating, swelling, and fullness.Fórmula:C11H18BrN5O3Pureza:99.84% - >99.99%Cor e Forma:CoaPeso molecular:348.2N6-Cyclohexyladenosine
CAS:N6-Cyclohexyladenosine (CHA) is a selective agonist of A1 receptor with EC50 of 8.2 Nm.Fórmula:C16H23N5O4Pureza:99.92% - 99.98%Cor e Forma:SolidPeso molecular:349.38Diphylline
CAS:Diphylline is a bronchodilator with mild vasodilator and diuretic properties, used for asthma, bronchitis, and emphysema.Fórmula:C10H14N4O4Pureza:98.54%Cor e Forma:Crystals From Alcohol SolidPeso molecular:254.24Acefylline
CAS:Acefylline (Theophylline-7-acetic acid), a stimulant drug of the xanthine chemical class, acts as an adenosine receptor antagonist.Fórmula:C9H10N4O4Pureza:99.57%Cor e Forma:White Crystalline SolidPeso molecular:238.2A3AR agonist 1
A3AR Agonist 1 (Compound 12), with a Ki of 25.8 nM, is a potent A3 adenosine receptor (A3AR) agonist that promotes β-arrestin2 recruitment with an effectiveFórmula:C28H34N6O6Pureza:98%Cor e Forma:SolidPeso molecular:550.61Adenosine receptor agonist 1
Compound 6m, an A3 adenosine receptor (AR) partial agonist, exhibits a K i value of 6.7 nM as an adenosine receptor agonist.Fórmula:C12H14ClN5O2SeCor e Forma:SolidPeso molecular:374.68A3AR agonist 2
Compound 19, a selective A3 Adenosine Receptor (A3AR) agonist (K i : 22.1 nM), effectively stimulates β-arrestin2 recruitment with an EC 50 value of 4.36 nM.Fórmula:C34H34N6O6Pureza:98%Cor e Forma:SolidPeso molecular:622.67Xanthine amine congener dihydrochloride
CAS:XAC dihydrochloride is an Adenosine A1 and A2 receptor antagonist with IC50s of 1.8 nM and 114 nM, also a mouse convulsant.Fórmula:C21H30Cl2N6O4Cor e Forma:SolidPeso molecular:501.41LUF6096
CAS:LUF6096 (CF-602) is a potent allosteric enhancer of the adenosine A3 receptor, exhibiting the capability to enhance agonist binding allosterically whileFórmula:C22H21Cl2N3OPureza:99.5%Cor e Forma:SolidPeso molecular:414.33ABT-702
CAS:ABT-702 is an orally active, competitive, and reversible non-nucleoside adenosine kinase (AK) inhibitor analgesic and anti-inflammatory.Fórmula:C22H19BrN6OPureza:99.57%Cor e Forma:SoildPeso molecular:463.33FSCPX
CAS:FSCPX is a potent and selective irreversible antagonist of the A1 adenosine receptor (A1AR), exhibiting low nanomolar binding potency.Fórmula:C23H27FN4O6SPureza:99.4%Cor e Forma:SolidPeso molecular:506.55Ref: TM-T39039
1mg82,00€5mg180,00€10mg271,00€25mg460,00€50mg617,00€100mg825,00€200mg1.108,00€1mL*10mM (DMSO)86,00€Norisoboldine hydrochloride
CAS:Norisoboldine hydrochloride: an oral AhR agonist from Radix Linderae, for Rheumatoid arthritis and Ulcerative colitis research.Fórmula:C18H20ClNO4Cor e Forma:SolidPeso molecular:349.818-Chloro caffeine
CAS:8-Chloro caffeine binds to adenosine receptors with a Ki of 30 µM. It enhances UV-induced chromosomal aberrations in the Cl-I type Chinese hamster embryo lung cells. 8-Chloro caffeine is a derivative of the methylxanthine alkaloid caffeine.Fórmula:C8H9ClN4O2Cor e Forma:SolidPeso molecular:228.64hA3AR agonist 2
hA3AR agonist 2 is a potent activator of A3AR, with a Ki value of 3.5 nM.Fórmula:C11H14ClN5O2SCor e Forma:SolidPeso molecular:315.78PSB 0777 ammonium hydrate
PSB 0777 ammonium hydrate is a potent and selective adenosine A2A receptor full agonist, exhibiting K i values of 44.4 nM for rat A2A receptors and 360 nM forFórmula:C18H20N5O7S2·NH4·75H2OPureza:98%Cor e Forma:SolidPeso molecular:532.09AR ligand 40
AR ligand 40 (compound 19c) is an Adenosine A1 Receptor ligand with antagonistic activity. It exhibits antiproliferative effects on SW480, SW48, HCT116, K562, MDA-MB-231, and A549 cells, with EC50 values of 7, 10, 12, 13, 15, and 39 μM, respectively.Fórmula:C21H25N5Cor e Forma:SolidPeso molecular:347.211PSB 0777 ammonium salt
CAS:adenosine A2A receptor full agonistFórmula:C18H24N6O7S2Pureza:98%Cor e Forma:SolidPeso molecular:500.55MRS-1706
CAS:MRS-1706: Ki of 1.39nM for A2B; selective inverse agonist; also affects A2A, A1, A3.Fórmula:C27H29N5O5Pureza:99.00%Cor e Forma:SolidPeso molecular:503.55Ref: TM-T16136
1mg34,00€5mg74,00€10mg113,00€25mg222,00€50mg356,00€100mg572,00€200mg803,00€1mL*10mM (DMSO)84,00€A3AR modulator 1
MRS8054 is an oral A3 adenosine receptor positive allosteric modulator, enhancing Cl-IB-MECA-induced activity.Fórmula:C23H25IN4Cor e Forma:SolidPeso molecular:484.38GW-328267
CAS:GW-328267 is an agonist of the adenosine A2 receptor.Fórmula:C21H26N10O4Cor e Forma:SolidPeso molecular:482.5Xanthine amine congener trihydrochloride
CAS:Xanthine amine congener trihydrochloride: potent adenosine antagonist, reverses effects of N6-cyclohexyladenosine on urine, sodium excretion, heart rate.Fórmula:C21H29ClN6O4Pureza:98.81%Cor e Forma:SolidPeso molecular:464.95Danshenol B
Danshenol B is a natural product that can be used as a reference standard.Fórmula:C22H26O4Cor e Forma:SolidPeso molecular:354.446A-286501
CAS:A-286501: Oral adenosine kinase inhibitor, IC50=0.47 nM, reduces pain via non-opioid, non-NSAID ADO receptors.Fórmula:C11H14BrN5O2Pureza:98%Cor e Forma:SolidPeso molecular:328.17Theophyllol
CAS:Theophyllol (theophylline sodium acetate) can alter calcium levels in subcellular fractions of rat brain cortex.Fórmula:C9H10N4Na2O4Cor e Forma:SolidPeso molecular:284.18Adenosine receptor antagonist 1
CAS:A2aR-selective antagonist with IC50 of 0.29 nM; 14x more selective over A2bR.Fórmula:C22H15ClFN7OCor e Forma:SolidPeso molecular:447.863F6-9G5
3F6-9G5 is a humanized monoclonal antibody targeting AA2AR/Adenosine A2aR, used in neurodegenerative disease research.Pureza:>95%Cor e Forma:Odour LiquidPeso molecular:146.66 kDaN6-Benzyl-5'-ethylcarboxamido adenosine
CAS:N6-Benzyl-5'-ethylcarboxamido adenosine is a selective A3 adenosine receptor agonist.Fórmula:C19H22N6O4Cor e Forma:SolidPeso molecular:398.42Heterobivalent ligand-1
Heterobivalent ligand-1 targets A2A-D2 receptor heteromer with affinity: Kd for A2A=2.1 nM, D2=0.13 nM.Fórmula:C86H115FN16O21Cor e Forma:SolidPeso molecular:1727.93LUF7690
CAS:LUF7690 (Compound 9), a clickable and covalent affinity-based probe (AfBP) for the human A3 adenosine receptor (hA3AR), facilitates the detection andFórmula:C25H24FN5O6SCor e Forma:SolidPeso molecular:541.55Apadenoson TFA
Apadenoson TFA is a potent adenosine A2A receptor (A2AR) agonist that can be used to improve survival in patients infected with SARS.
Fórmula:C25H31F3N6O8Pureza:98.08%Cor e Forma:SoildPeso molecular:600.55A2A/A3 AR antagonist-1
A2A/A3 AR antagonist-1 is a dual fluorescent AR ligand with K i of 90 nM (hA2A) & 31.8 nM (hA3).Fórmula:C56H71N15O12S2Cor e Forma:SolidPeso molecular:1210.39GR79236
CAS:GR79236 is an effective and selective adenosine A1 receptor agonist (Ki: 3.1 nM) that has analgesic and anti-inflammatory actions.Fórmula:C15H21N5O5Cor e Forma:SolidPeso molecular:351.36(Rac)-Mirabegron-d5
CAS:(Rac)-Mirabegron D5 is a deuterium labeled (Rac)-Mirabegron. Mirabegron is a selective agonist of β3-adrenoceptor.Fórmula:C21H24N4O2SPureza:98%Cor e Forma:SolidPeso molecular:401.54LAS101057
CAS:LAS101057 is a novel orally available and potent and selective A2B receptor antagonist for the study of asthma.Fórmula:C18H14FN5OPureza:99.03% - >99.99%Cor e Forma:SolidPeso molecular:335.34Theophylline-d6
CAS:Theophylline-d6, an internal standard for theophylline quantification in GC/LC-MS, relaxes bronchial muscles and treats asthma/COPD.Fórmula:C7H2D6N4O2Cor e Forma:SolidPeso molecular:186.2
