Receptor de adenosina
Os receptores de adenosina são uma classe de GPCRs que respondem ao nucleosídeo endógeno adenosina. Esses receptores estão envolvidos na regulação de vários processos fisiológicos, incluindo função cardiovascular, ciclos de sono-vigília e respostas imunes. Moduladores de receptores de adenosina têm potencial terapêutico no tratamento de condições como arritmias cardíacas, inflamação e doenças neurodegenerativas. Na CymitQuimica, oferecemos uma seleção de moduladores de receptores de adenosina de alta qualidade para apoiar sua pesquisa em biologia cardiovascular, neurociência e imunologia.
Foram encontrados 249 produtos de "Receptor de adenosina"
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Adenosine receptor agonist 1
Compound 6m, an A3 adenosine receptor (AR) partial agonist, exhibits a K i value of 6.7 nM as an adenosine receptor agonist.Fórmula:C12H14ClN5O2SeCor e Forma:SolidPeso molecular:374.68A3AR modulator 1
MRS8054 is an oral A3 adenosine receptor positive allosteric modulator, enhancing Cl-IB-MECA-induced activity.Fórmula:C23H25IN4Cor e Forma:SolidPeso molecular:484.38N6-Benzyl-5'-ethylcarboxamido adenosine
CAS:N6-Benzyl-5'-ethylcarboxamido adenosine is a selective A3 adenosine receptor agonist.Fórmula:C19H22N6O4Cor e Forma:SolidPeso molecular:398.42Adenosine receptor antagonist 1
CAS:A2aR-selective antagonist with IC50 of 0.29 nM; 14x more selective over A2bR.Fórmula:C22H15ClFN7OCor e Forma:SolidPeso molecular:447.86LUF7690
CAS:LUF7690 (Compound 9), a clickable and covalent affinity-based probe (AfBP) for the human A3 adenosine receptor (hA3AR), facilitates the detection andFórmula:C25H24FN5O6SCor e Forma:SolidPeso molecular:541.55FSCPX
CAS:FSCPX is a potent and selective irreversible antagonist of the A1 adenosine receptor (A1AR), exhibiting low nanomolar binding potency.Fórmula:C23H27FN4O6SPureza:99.4%Cor e Forma:SolidPeso molecular:506.55Ref: TM-T39039
1mg82,00€5mg180,00€10mg271,00€25mg460,00€50mg617,00€100mg825,00€200mg1.108,00€1mL*10mM (DMSO)86,00€Apadenoson TFA
Apadenoson TFA is a potent adenosine A2A receptor (A2AR) agonist that can be used to improve survival in patients infected with SARS.
Fórmula:C25H31F3N6O8Pureza:98.08%Cor e Forma:SoildPeso molecular:600.55PSB 0777 ammonium salt
CAS:adenosine A2A receptor full agonistFórmula:C18H24N6O7S2Pureza:98%Cor e Forma:SolidPeso molecular:500.55Norisoboldine hydrochloride
CAS:Norisoboldine hydrochloride: an oral AhR agonist from Radix Linderae, for Rheumatoid arthritis and Ulcerative colitis research.Fórmula:C18H20ClNO4Cor e Forma:SolidPeso molecular:349.81A2A/A3 AR antagonist-1
A2A/A3 AR antagonist-1 is a dual fluorescent AR ligand with K i of 90 nM (hA2A) & 31.8 nM (hA3).Fórmula:C56H71N15O12S2Cor e Forma:SolidPeso molecular:1210.39GW-328267
CAS:GW-328267 is an agonist of the adenosine A2 receptor.Fórmula:C21H26N10O4Cor e Forma:SolidPeso molecular:482.5MRS-1706
CAS:MRS-1706: Ki of 1.39nM for A2B; selective inverse agonist; also affects A2A, A1, A3.Fórmula:C27H29N5O5Pureza:99.00%Cor e Forma:SolidPeso molecular:503.55Ref: TM-T16136
1mg34,00€5mg74,00€10mg113,00€25mg222,00€50mg356,00€100mg572,00€200mg803,00€1mL*10mM (DMSO)84,00€Xanthine amine congener trihydrochloride
CAS:Xanthine amine congener trihydrochloride: potent adenosine antagonist, reverses effects of N6-cyclohexyladenosine on urine, sodium excretion, heart rate.Fórmula:C21H29ClN6O4Pureza:98.81%Cor e Forma:SolidPeso molecular:464.95ABT-702
CAS:ABT-702 is an orally active, competitive, and reversible non-nucleoside adenosine kinase (AK) inhibitor analgesic and anti-inflammatory.Fórmula:C22H19BrN6OPureza:99.57%Cor e Forma:SoildPeso molecular:463.33Xanthine amine congener dihydrochloride
CAS:XAC dihydrochloride is an Adenosine A1 and A2 receptor antagonist with IC50s of 1.8 nM and 114 nM, also a mouse convulsant.Fórmula:C21H30Cl2N6O4Cor e Forma:SolidPeso molecular:501.41A-286501
CAS:A-286501: Oral adenosine kinase inhibitor, IC50=0.47 nM, reduces pain via non-opioid, non-NSAID ADO receptors.Fórmula:C11H14BrN5O2Pureza:98%Cor e Forma:SolidPeso molecular:328.17Danshenol B
Danshenol B is a natural product that can be used as a reference standard.Fórmula:C22H26O4Cor e Forma:SolidPeso molecular:354.446AR ligand 40
AR ligand 40 (compound 19c) is an Adenosine A1 Receptor ligand with antagonistic activity. It exhibits antiproliferative effects on SW480, SW48, HCT116, K562, MDA-MB-231, and A549 cells, with EC50 values of 7, 10, 12, 13, 15, and 39 μM, respectively.Fórmula:C21H25N5Cor e Forma:SolidPeso molecular:347.211Theophyllol
CAS:Theophyllol (theophylline sodium acetate) can alter calcium levels in subcellular fractions of rat brain cortex.Fórmula:C9H10N4Na2O4Cor e Forma:SolidPeso molecular:284.18LUF6096
CAS:LUF6096 (CF-602) is a potent allosteric enhancer of the adenosine A3 receptor, exhibiting the capability to enhance agonist binding allosterically whileFórmula:C22H21Cl2N3OPureza:99.5%Cor e Forma:SolidPeso molecular:414.33
