Receptor de adenosina
Os receptores de adenosina são uma classe de GPCRs que respondem ao nucleosídeo endógeno adenosina. Esses receptores estão envolvidos na regulação de vários processos fisiológicos, incluindo função cardiovascular, ciclos de sono-vigília e respostas imunes. Moduladores de receptores de adenosina têm potencial terapêutico no tratamento de condições como arritmias cardíacas, inflamação e doenças neurodegenerativas. Na CymitQuimica, oferecemos uma seleção de moduladores de receptores de adenosina de alta qualidade para apoiar sua pesquisa em biologia cardiovascular, neurociência e imunologia.
Foram encontrados 249 produtos de "Receptor de adenosina"
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Capadenoson
CAS:Capadenoson (BAY 68-4986) is a selective adenosine-A1 receptor agonist.Fórmula:C25H18ClN5O2S2Pureza:98.85% - 99.57%Cor e Forma:SolidPeso molecular:520.03Enprofylline
CAS:Enprofylline (Enprofilina), a bronchodilator, acts primarily as a competitive nonselective phosphodiesterase inhibitor.Fórmula:C8H10N4O2Pureza:98.37%Cor e Forma:SolidPeso molecular:194.19Ref: TM-T21389
2mg42,00€5mg62,00€10mg88,00€25mg141,00€50mg215,00€100mg318,00€200mg442,00€1mL*10mM (DMSO)59,00€Inosine
CAS:Inosine (NSC-20262), an endogenous purine nucleoside produced by the catabolism of adenosine, is an agonist of adenosine receptors A1R and A2AR. Low-Cost!Fórmula:C10H12N4O5Pureza:99.51% - 99.89%Cor e Forma:SolidPeso molecular:268.23Taminadenant mesylate
CAS:Taminadenant (PBF-509/NIR-178) is an oral adenosine A2A receptor antagonist that activates T-cells to target tumor cells.Fórmula:C11H12BrN7O3SCor e Forma:SolidPeso molecular:402.227Preladenant
CAS:Preladenant (SCH-420814) is an orally bioavailable antagonist of the adenosine A2A receptor (Ki: 1.1 nM) and has >1000-fold selectivity over all other adenosineFórmula:C25H29N9O3Pureza:98.02% - 99.68%Cor e Forma:SolidPeso molecular:503.56CPI-444
CAS:CPI-444 (V81444) is an antagonist of the adenosine A2A receptor.It reduces tumor area in mouse model of murine Her2/neu-expressing breast cancer.Fórmula:C20H21N7O3Pureza:98.78%Cor e Forma:SolidPeso molecular:407.43Ref: TM-T7183
2mg34,00€5mg52,00€10mg73,00€25mg128,00€50mg197,00€100mg295,00€200mg442,00€1mL*10mM (DMSO)52,00€Proxyphylline
CAS:Proxyphylline (7-(2-Hydroxypropyl)theophylline) is a dual of adenosine A1/A2a receptor inhibitor and phosphodiesterase (PDE) inhibitor.Fórmula:C10H14N4O3Pureza:99.48%Cor e Forma:SolidPeso molecular:238.24DPCPX
CAS:DPCPX (PD 116948) is an A1 adenosine receptor antagonistFórmula:C16H24N4O2Pureza:99.23% - 99.93%Cor e Forma:White SolidPeso molecular:304.39Tecadenoson
CAS:Tecadenoson (CVT-510) is a selective agonist of A1 adenosine receptor.
Fórmula:C14H19N5O5Pureza:98.83%Cor e Forma:SolidPeso molecular:337.33N6,N6-Dimethyladenosine
CAS:N6,N6-Dimethyladenosine is find in mycobacterium bovis Bacille Calmette-Guérin tRNA.
Fórmula:C12H17N5O4Pureza:98.79%Cor e Forma:White PowderPeso molecular:295.29Nitrobenzylthioinosine
CAS:Nitrobenzylthioinosine (NBMPR) is an inhibitor of ENT1 transporter that binds to ENT1 transporter with high affinity.
Fórmula:C17H17N5O6SPureza:99.69% - 99.74%Cor e Forma:Off-White SolidPeso molecular:419.41Adenosine receptor antagonist 4
CAS:Adenosine receptor antagonist 4 is an adenosine receptor antagonist.Fórmula:C10H13N3Pureza:99.63% - 99.65%Cor e Forma:Off-White PowderPeso molecular:175.235-Iodotubercidin
CAS:5-Iodotubercidin (NSC-113939) is a potent adenosine kinase inhibitor with IC50 of 26 nM.
Fórmula:C11H13IN4O4Pureza:99.98%Cor e Forma:Tan SolidPeso molecular:392.15MIPS521
CAS:MIPS521 ({2-Amino-4-[3,5-bis(trifluoromethyl)phenyl]thiophen-3-yl}(4-chlorophenyl)methanone) is a positive allosteric modulator of the A1R.Fórmula:C19H10ClF6NOSPureza:99.76%Cor e Forma:SolidPeso molecular:449.8Ref: TM-T9330
1mg35,00€2mg50,00€5mg74,00€10mg105,00€25mg178,00€50mg313,00€100mg485,00€1mL*10mM (DMSO)82,00€CCPA
CAS:CCPA (2-chloro-N(6)cyclopentyladenosine) is a potent and selective agonist of adenosine A1 receptorFórmula:C15H20ClN5O4Pureza:99.1%Cor e Forma:Off-White To Light Yellow SolidPeso molecular:369.8Regadenoson
CAS:Regadenoson (CVT-3146) is a selective A2A receptor agonist that increases coronary blood flow with a longer half-life than adenosine.Fórmula:C15H18N8O5Pureza:99.57% - 99.81%Cor e Forma:Off-White SolidPeso molecular:390.35Ref: TM-T2671
2mg47,00€5mg65,00€10mg92,00€25mg173,00€50mg273,00€100mg416,00€500mg935,00€1mL*10mM (DMSO)72,00€1-Ethyl-6-aminouracil
CAS:1-Ethyl-6-aminouracil (6-AMINO-1-ETHYL-1H-PYRIMIDINE-2,4-DIONE) is an intermediate in the synthesis of a series of new substituted Xanthines which have highFórmula:C6H9N3O2Pureza:99.29%Cor e Forma:SolidPeso molecular:155.155'-N-Ethylcarboxamidoadenosine
CAS:NECA, an adenosine receptor agonist, boosts brain extravasation of fluorescein and dextran without affecting the blood-brain barrier.Fórmula:C12H16N6O4Pureza:98.95% - ≥95%Cor e Forma:PowderPeso molecular:308.29VPC171
CAS:VPC171 is a novel adenosine A1 receptor positive allosteric modulator (PAM).Fórmula:C18H12F3NOSPureza:99.78%Cor e Forma:SolidPeso molecular:347.35Ref: TM-T29112
1mg49,00€5mg96,00€10mg124,00€25mg222,00€50mg309,00€100mg439,00€200mg592,00€1mL*10mM (DMSO)88,00€Vipadenant
CAS:Vipadenant (CEB-4520)(BIIB-014) is an adenosine A2a antagonist with Ki of 1.3 nM; less potent for A1(Ki=69 nM).Fórmula:C16H15N7OPureza:97.25% - 97.36%Cor e Forma:SolidPeso molecular:321.34Ref: TM-T2373
2mg35,00€5mg51,00€10mg80,00€25mg131,00€50mg210,00€100mg313,00€200mg445,00€1mL*10mM (DMSO)215,00€
