Receptor de Canabinóides
Os receptores de canabinoides são GPCRs que mediam os efeitos dos canabinoides endógenos (endocanabinoides) e dos fitocanabinoides, como aqueles encontrados na cannabis. Os dois principais tipos de receptores de canabinoides, CB1 e CB2, estão envolvidos na regulação de uma ampla gama de processos fisiológicos, incluindo percepção da dor, apetite, humor e função imunológica. Moduladores de receptores de canabinoides têm potencial terapêutico no tratamento de condições como dor crônica, epilepsia e esclerose múltipla. Na CymitQuimica, oferecemos uma ampla gama de moduladores de receptores de canabinoides de alta qualidade para apoiar sua pesquisa em neurofarmacologia, manejo da dor e imunologia.
Foram encontrados 218 produtos de "Receptor de Canabinóides"
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CB1 inverse agonist 2
CAS:CB1 inverse agonist 2, an oral drug, counters CB1 effects, reducing CP55940-induced hypothermia and anorexia in mice.Fórmula:C24H20ClFN2OSCor e Forma:SolidPeso molecular:438.94CB2R agonist 1
CAS:CB2R agonist 1 selectively binds human CB2R, EC50 of 0.56 µM, modulates inflammatory cytokines.Fórmula:C22H32N2OCor e Forma:SolidPeso molecular:340.5LEI 101 hydrochloride
CAS:LEI 101 hydrochloride is potent and selective CB2 partial agonist.Fórmula:C23H26ClFN4O4SCor e Forma:SolidPeso molecular:508.99ANEB-001
CAS:ANEB-001 is an orally active CB1 inhibitor that can be used in studies of acute cannabinoid intoxication.Fórmula:C22H24ClF3N2O2Cor e Forma:SolidPeso molecular:440.89CB1R Allosteric modulator 2
CAS:Compound 18 is a potent CB1R allosteric modulator that acts as a negative modulator (NAM) for CB1R orthosteric ligands.Fórmula:C19H15ClFN3OCor e Forma:SolidPeso molecular:355.79COR 170
CAS:inverse agonist of CB2 receptorsFórmula:C31H36N2O2Pureza:98%Cor e Forma:SolidPeso molecular:468.63CB1/2 agonist 2
CAS:CB1/2 agonist 2 binds tightly to cannabinoid receptors, acting fully on CB1 and inversely on CB2.Fórmula:C26H43NO3Cor e Forma:SolidPeso molecular:417.62PGN36
CAS:PGN36 (Compound 18) is a potent CB2 receptor antagonist with a high affinity (Ki=0.09 μM).Fórmula:C21H23N3O3Cor e Forma:SolidPeso molecular:365.43CB1R Allosteric modulator 1
CAS:CB1R modulator 1 (compound 11), a potent CB1R inhibitor, decreases activity of orthosteric ligands.Fórmula:C24H24ClN3OCor e Forma:SolidPeso molecular:405.92S-777469
CAS:S-777469: Selective CB2 agonist, oral, inhibits itching in mice (Ki: 36 nM). Anti-pruritic.Fórmula:C23H27FN2O4Cor e Forma:SolidPeso molecular:414.47CB2 receptor agonist 3
CAS:GP 2A is a selective agonist of CB2 receptor.Fórmula:C24H23Cl2N3OCor e Forma:SolidPeso molecular:440.36Virodhamine trifluoroacetate
CAS:Virodhamine trifluoroacetate: full GPR55 & CB2 agonist, partial CB1 antagonist, cannabinoid receptor mixed antagonist.Fórmula:C24H38F3NO4Pureza:98%Cor e Forma:SolidPeso molecular:461.56LBP-1
CAS:LBP-1 is a cannabinoid receptor type 1 (CB1) agonist.Fórmula:C23H29ClN6O3Cor e Forma:SolidPeso molecular:472.97MM-22
CAS:biotinylated anandamide analog acts as a probe for visualizing the accumulation and intracellular trafficking of anandamideFórmula:C36H60N4O5SPureza:98%Cor e Forma:SolidPeso molecular:660.95AZD-2207
CAS:AZD-2207 is a cannabinoid receptor CB1 antagonist and highly lipophilic compound for the treatment of type 2 diabetes mellitus and obesity.Fórmula:C25H25Cl2F3N4O4SCor e Forma:SolidPeso molecular:605.46Cannabicitran
CAS:Cannabicitran is a cannabinoid that can decrease rabbits intraocular pressure [1] [2].Fórmula:C21H30O2Cor e Forma:SolidPeso molecular:314.46GAT229
CAS:GAT229 is a CB1 positive modulator, enhancing CB agonist activity without direct activation; influences binding, signaling, and lowers ocular pressure in mice.Fórmula:C22H18N2O2Cor e Forma:SolidPeso molecular:342.39SMM-189
CAS:SMM-189 is a potent and selective CB2 inverse agonist.Fórmula:C19H12Cl2O3Cor e Forma:SolidPeso molecular:359.2CAY10412
CAS:Anandamide (AEA) is an endocannabinoid with neural reuptake. CAY10412, an AEA analog, inhibits this reuptake without binding to CB receptors.Fórmula:C25H36O2SCor e Forma:SolidPeso molecular:400.62KLS-13019
CAS:KLS-13019 is a highly effective and orally active GPR55 receptor antagonist, neuroprotective can reverse chemotherapy-induced peripheral neuropathy (CIPN).Fórmula:C22H29NO3Pureza:>99.99% - >99.99%Cor e Forma:SolidPeso molecular:355.47
