Receptor GNRH
Os receptores do hormônio liberador de gonadotropina (GnRH) são GPCRs que se ligam ao GnRH, um hormônio responsável por regular a liberação do hormônio luteinizante (LH) e do hormônio folículo-estimulante (FSH) pela glândula pituitária. Esses receptores são cruciais para a função reprodutiva e são alvo em terapias para condições como câncer de próstata, endometriose e infertilidade. Agonistas e antagonistas dos receptores de GnRH também são usados em tecnologias de reprodução assistida. Na CymitQuimica, oferecemos uma gama abrangente de moduladores de receptores de GnRH de alta qualidade para apoiar sua pesquisa em saúde reprodutiva, endocrinologia e terapia hormonal.
Foram encontrados 84 produtos de "Receptor GNRH"
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Alarelin Acetate
CAS:Alarelin Acetate is a synthetic GnRH agonist which can directly inhibit proliferation and DNA synthesis of rat GSMC through GnRH receptors.Fórmula:C56H78N16O12Pureza:99.81% - >99.99%Cor e Forma:White PowderPeso molecular:1167.34Ref: TM-T1494
5mg58,00€10mg95,00€25mg115,00€1mL*10mM (DMSO)120,00€50mg156,00€100mg180,00€500mg452,00€Degarelix acetate(214766-78-6 free base)
CAS:Degarelix acetate is a competitive and reversible antagonist of gonadotropin-releasing hormone receptor (GnRHR) .Fórmula:C84H107ClN18O18Pureza:98.66%Cor e Forma:SolidPeso molecular:1692.34(R)-Elagolix
CAS:(R)-Elagolix (NBI-56418) is an orally active, highly selective, short-term potent antagonist of the non-peptide gonadotropin-releasing hormone receptor.Fórmula:C32H30F5N3O5Pureza:99.08%Cor e Forma:SolidPeso molecular:631.59Ref: TM-T11174
5mg50,00€1mL*10mM (DMSO)70,00€10mg75,00€25mg137,00€50mg195,00€100mg306,00€200mg452,00€Abarelix
CAS:Abarelix (PPI 149) is a potent gonadotrophin-releasing hormone (GnRH) antagonist, which is used for prostate cancer treatment.Fórmula:C72H95ClN14O14Pureza:>99.99%Cor e Forma:SolidPeso molecular:1416.06[D-Leu6, Val7]-LH-RH (1-9) Ethyl Amide
[D-Leu6, Val7]-LH-RH (1-9) Ethyl Amide is a LHRH peptide analogue.Fórmula:C58H82N16O12Cor e Forma:SolidPeso molecular:1195.37Onvitrelin ucalontide
CAS:Onvitrelin ucalontide is a LHRH analogue with anticancer effect; halts breast, ovarian, and prostate tumors in mice.Fórmula:C163H243N43O32Cor e Forma:SolidPeso molecular:3316.94Kisspeptin-54(human)
CAS:Endogenous ligand for KISS1 receptor; Ki values: rat 1.80 nM, human 1.45 nM. Inhibits tumor spread, stimulates gonadotropin release.Fórmula:C258H401N79O78Pureza:98%Cor e Forma:SolidPeso molecular:5857.49AG 045572
CAS:AG 045572 is a potent GnRH receptor antagonist that inhibits the GnRH receptor in humans and rats with Ki values of 6.0 nM and 3.8 nM, respectively.AG 045572 isFórmula:C30H37NO5Pureza:99.96%Cor e Forma:SolidPeso molecular:491.62LHRH
CAS:Luteinizing hormone-releasing hormone (LHRH) is a neuropeptide produced in the hypothalamus that plays a pivotal role in regulating reproduction and hasFórmula:C55H74N16O14Pureza:98%Cor e Forma:SolidPeso molecular:1183.27LGnRH-III, lamprey
CAS:GnRH III triggers luteinizing and follicle-stimulating hormone release, part of the conserved GnRH family.Fórmula:C59H74N18O14Pureza:98%Cor e Forma:SolidPeso molecular:1259.33MI 1544
CAS:MI 1544 is a LHRH antagonist.Fórmula:C71H94ClN17O13Cor e Forma:SolidPeso molecular:1429.09Luteinizing Hormone Releasing Hormone (LH-RH), salmon
CAS:LH-RH: a hypothalamus-made pituitary hormone, key in reproductive control.Fórmula:C60H73N15O13Pureza:98%Cor e Forma:SolidPeso molecular:1212.31Phoenixin-14
CAS:Phoenixin-14 (PNX-14), an active endogenous isoform, induces an anxiolytic effect by activating the AHA GnRH system in mice and protects against ischemia/
Fórmula:C75H110N18O20Pureza:98%Cor e Forma:SolidPeso molecular:1583.78RS 18286
CAS:RS 18286 is a LHRH antagonist.Fórmula:C74H101Cl2N17O14Cor e Forma:SolidPeso molecular:1523.6LHRH, Ala(6)-
CAS:LHRH, Ala(6)- is a synthetic luteinizing hormone-releasing hormone agonist agent.Fórmula:C56H77N17O13Cor e Forma:SolidPeso molecular:1196.32Avorelin
CAS:Avorelin, a luteinizing hormone releasing hormone (LH-RH) agonist, is used potentially for the treatment of prostate.Fórmula:C65H85N17O12Pureza:98%Cor e Forma:SolidPeso molecular:1296.48(D-Trp6)-LHRH free acid
CAS:(D-Trp6)-LHRH free acid is a luteinizing hormone-releasing hormone ( LHRH ) agonist [1] .Fórmula:C64H81N17O14Peso molecular:1312.43APTAA-LHRH
CAS:APTAA-LHRH is a gonadorelin antagonist.Fórmula:C69H91Cl2N17O14Pureza:98%Cor e Forma:SolidPeso molecular:1453.47Azaline
CAS:Azaline is a gonadorelin antagonist.Fórmula:C74H106ClN23O12Pureza:98%Cor e Forma:SolidPeso molecular:1545.26Linzagolix choline
CAS:Linzagolix choline is a GnRH antagonist. It can be used to study pain associated with uterine fibroids and endometriosis.Fórmula:C27H28F3N3O8SPureza:99.64%Cor e Forma:SolidPeso molecular:611.59LH-RH (4-10)
CAS:LH-RH (4-10), a heptapeptide from LHRH degradation, is made in macrophages and type II pneumocytes.Fórmula:C33H53N11O9Cor e Forma:SolidPeso molecular:747.84Lamprey LH-RH I
CAS:Lamprey LH-RH I triggers ovulation and raises steroid levels in lamprey, inactive in other species.Fórmula:C58H79N15O15Cor e Forma:SolidPeso molecular:1226.34(D-His(Bzl)6)-LHRH (1-7) (free acid)
CAS:(D-His(Bzl)6)-LHRH (1-7) free acid is a synthetic peptide derived from luteinizing hormone-releasing hormone (LHRH). It achieves enhanced stability and biological activity through the introduction of non-natural amino acid residues at specific positions within the LHRH molecule. This modification extends the drug's half-life in the body, reduces its rate of rapid metabolism and clearance, and subsequently increases its efficacy in inhibiting cell proliferation.Fórmula:C53H62N12O11Peso molecular:1043.13Prolactin-Releasing Peptide (1-31), bovine
Prolactin-Releasing Peptide (1-31), bovine, is a fragment of prolactin-releasing peptide (PrRP).Fórmula:C44H80N14O15Peso molecular:1044.59276Bim 21009
CAS:Bim 21009 is an inhibitor of gonadorelin.Fórmula:C74H92ClN17O13Pureza:98%Cor e Forma:SolidPeso molecular:1463.08[D-Phe2,6, Pro3]-LH-RH
CAS:[D-Phe2,6, Pro3]-LH-RH is a potent antagonist of luteinizing hormone-releasing hormone (LHRH).Fórmula:C59H80N14O13Cor e Forma:SolidPeso molecular:1193.35Human follicular gonadotropin releasing peptide
CAS:Human Follicular Gonadotropin Releasing Peptide (hF-GRP) is a hormonal peptide that, in vitro, can induce the secretion of pituitary luteinizing hormone (LH)Fórmula:C68H94N22O27Cor e Forma:SolidPeso molecular:1651.61Prolactin Releasing Peptide (1-31), human acetate
Prolactin Releasing Peptide (1-31), human (acetate), is a potent GPR10 ligand with high affinity, eliciting prolactin secretion.Fórmula:C162H26N56O44SCor e Forma:SolidPeso molecular:3724.17Prolactin Releasing Peptide (1-31), human
CAS:Human Prolactin Releasing Peptide (1-31) is a potent GPR10 agonist; Ki values are 1.03 nM (human) and 0.33 nM (rat).Fórmula:C160H252N56O42SPureza:98%Cor e Forma:SolidPeso molecular:3664.15Surfagon
CAS:Surfagon is an effective LHRH agonist.Fórmula:C56H78N16O12Pureza:98%Cor e Forma:SolidPeso molecular:1167.34[D-Glp1,D-Phe2,D-Trp3,6]-LH-RH
CAS:[D-Glp1,D-Phe2,D-Trp3,6]-LH-RH is a synthetic LHRH analog and a GnRH receptor antagonist.Fórmula:C67H84N16O13Cor e Forma:SolidPeso molecular:1321.48[Gln8]-C517 (LH-RH), chicken
CAS:[Gln8] LH-RH: Avian hypothalamic peptide; prompts anterior pituitary to release gonadotropins, controlling reproduction.Fórmula:C54H71N15O14Pureza:98%Cor e Forma:SolidPeso molecular:1154.23Fsh receptor-binding inhibitor fragment(bi-10)
CAS:FSH antagonist bi-10 suppresses ovulation, induces follicular atresia, and may help in ovarian cancer by downregulating FSHR/ERβ.Fórmula:C42H67N13O19Cor e Forma:SolidPeso molecular:1058.06Zebrafish Kisspeptin-1
CAS:Zebrafish Kisspeptin-1 is the core sequence of the neuropeptide kisspeptin-1, which plays a crucial role in regulating the release of gonadotropin-releasing hormone (GnRH) and modulating the reproductive system.Fórmula:C58H84N16O15Cor e Forma:SolidPeso molecular:1245.39GnRH Associated Peptide (1-24), human
CAS:GnRH Associated Peptide (GAP) (1-24), human, is the 1-24 fragment of hGAP linked to LH-RH via a 3 amino acid site.Fórmula:C117H190N32O43Cor e Forma:SolidPeso molecular:2732.95LH-RH (7-10)
CAS:LH-RH (7-10), a tetrapeptide, is a key LHRH degradation product found in macrophages and pneumocytes.Fórmula:C19H36N8O4Cor e Forma:SolidPeso molecular:440.54(D-Ser4,D-Ser(tBu)6,Azagly10)-LHRH
CAS:Analog of LHRH, stimulates LH and FSH release, controls reproduction.Fórmula:C59H84N18O14Cor e Forma:SolidPeso molecular:1269.41Kisspeptin-54(human) TFA
Endogenous kisspeptin-54(human) TFA targets KISS1/GPR54 receptors; Ki: 1.81 nM (rat), 1.45 nM (human); inhibits metastasis, boosts gonadotropin.Fórmula:C258H401N79O78·C2HF3O2Cor e Forma:SolidPeso molecular:5971.45sGnRH-A
CAS:sGnRH-A, a salmon GnRH analog, boosts growth hormone and induces ovulation for artificial insemination.Fórmula:C64H83N17O12Cor e Forma:SolidPeso molecular:1282.45Phoenixin-14 TFA
Phoenixin-14 TFA (PNX-14 TFA) is an endogenous neuropeptide that can modulate GnRH receptor expression and exerts anxiolytic effects.Fórmula:C75H110N18O20·xC2HF3O2Pureza:99.11%Cor e Forma:SolidPeso molecular:1583.78 (free base)Kisspeptin 13
CAS:Kisspeptin 13 activates GPR54 & GnRH receptors, boosts memory, and aids in Alzheimer's research.Fórmula:C78H107N21O18Cor e Forma:SolidPeso molecular:1626.81Azaline B
CAS:Azaline B is an antagonist of the gonadotropin-releasing hormone (GnRH), with an IC50 of 1.37 nM. It is utilized in research related to pathologies associated with sex hormones, ovulation induction, and male contraception.Fórmula:C80H102ClN23O12Cor e Forma:SolidPeso molecular:1613.27A 76154
CAS:A 76154 is an antagonist of leutenizing hormone releasing hormone (LHRH).Fórmula:C70H93FN12O12Cor e Forma:SolidPeso molecular:1313.584Wy 43657
CAS:Wy 43657 is a gonadorelin antagonist.Fórmula:C71H86N14O13Pureza:98%Cor e Forma:SolidPeso molecular:1343.554LUF5771
CAS:LUF5771: potent allosteric recLH & Org 43553 inhibitor, partial LH receptor activator with low efficacy.Fórmula:C24H23NO2Cor e Forma:SolidPeso molecular:357.44Lecirelin
CAS:Lecirelin is a synthetic GnRH (gonadotropin releasing hormone) analogue which shows a great efficacy in the treatment of bovine ovarian follicular cysts.Fórmula:C59H84N16O12Cor e Forma:SolidPeso molecular:1209.4Lecirelin acetate(61012-19-9 free base)
Lecirelin acetate is a synthetic GnRH (gonadotropin releasing hormone) analogue which shows a great efficacy in the treatment of bovine ovarian follicular cystsFórmula:C61H88N16O14Pureza:98.1%Cor e Forma:SolidPeso molecular:1269.45Relugolix
CAS:Relugolix (RVT-601) is an orally available, non-peptide gonadotropin-releasing hormone (GnRH or luteinizing hormone-releasing hormone (LHRH)) antagonist, withFórmula:C29H27F2N7O5SPureza:98.64% - 99.97%Cor e Forma:SolidPeso molecular:623.63Ref: TM-T3630
2mg39,00€5mg58,00€1mL*10mM (DMSO)81,00€10mg93,00€25mg167,00€50mg250,00€100mg408,00€200mg585,00€Sufugolix
CAS:Sufugolix (TAK-013) is a potent and orally available luteinizing hormone-releasing hormone LHRH receptor.Fórmula:C36H31F2N5O4SPureza:97.78%Cor e Forma:SolidPeso molecular:667.72Fluorogestone acetate
CAS:FGA (Fluorogestone Acetate, SC9880) is 20-25x more potent than progesterone with high potency and short activity duration.Fórmula:C23H31FO5Pureza:99.47%Cor e Forma:CoaPeso molecular:406.49Ref: TM-T21335
2mg39,00€5mg58,00€1mL*10mM (DMSO)74,00€10mg93,00€25mg167,00€50mg245,00€100mg371,00€200mg494,00€
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