Receptor GNRH
Os receptores do hormônio liberador de gonadotropina (GnRH) são GPCRs que se ligam ao GnRH, um hormônio responsável por regular a liberação do hormônio luteinizante (LH) e do hormônio folículo-estimulante (FSH) pela glândula pituitária. Esses receptores são cruciais para a função reprodutiva e são alvo em terapias para condições como câncer de próstata, endometriose e infertilidade. Agonistas e antagonistas dos receptores de GnRH também são usados em tecnologias de reprodução assistida. Na CymitQuimica, oferecemos uma gama abrangente de moduladores de receptores de GnRH de alta qualidade para apoiar sua pesquisa em saúde reprodutiva, endocrinologia e terapia hormonal.
Foram encontrados 84 produtos de "Receptor GNRH"
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Fertirelin
CAS:Fertirelin, or fertirelin acetate, sold under the brand name Ovalyse, is a gonadotropin-releasing hormone agonist (GnRH agonist).Fórmula:C55H76N16O12Pureza:>99.99%Cor e Forma:SolidPeso molecular:1153.29Ref: TM-TP1288
1mg47,00€2mg63,00€5mg96,00€10mg135,00€50mg177,00€100mg264,00€200mg393,00€1mL*10mM (DMSO)170,00€Cetrorelix diacetate
CAS:Cetrorelix diacetate (NS-75A) is is a gonadotropin-releasing hormone antagonist.Fórmula:C74H100ClN17O18Pureza:98.38%Cor e Forma:SolidPeso molecular:1551.17Ref: TM-T5520L
1mg52,00€5mg90,00€10mg150,00€25mg291,00€50mg437,00€100mg642,00€500mg1.359,00€1mL*10mM (DMSO)251,00€Ganirelix Acetate
CAS:Ganirelix Acetate is a gonadotropin-releasing hormone (GnRH) receptor antagonistFórmula:C82H117ClN18O15Pureza:96.05%Cor e Forma:SolidPeso molecular:1630.4LGnRH-III, lamprey acetate(147859-97-0 free base)
LGnRH-III, lamprey acetate is an evolutionarily conserved member of the GnRH family, can stimulate the secretion of gonadotropins, it stimulates the secretionFórmula:C61H78N18O16Pureza:99.66%Cor e Forma:SolidPeso molecular:1319.38Histrelin acetate
CAS:Histrelin acetate is a nonapeptide analog of gonadotropin-releasing hormone (GnRH) with added potency.Fórmula:C68H90N18O14Pureza:99.92%Cor e Forma:SolidPeso molecular:1383.55Deslorelin acetate(57773-65-6 free base)
Deslorelin acetate(57773-65-6 free base) is a gonadotropin releasing hormone super-agonist (GnRH agonist)Fórmula:C66H87N17O14Pureza:99.84%Cor e Forma:SolidPeso molecular:1342.5Buserelin Acetate (57982-77-1 free base)
CAS:Buserelin Acetate (57982-77-1 free base) (Buserelin Acetate) is an agonist of gonadotropin-releasing hormone receptor(GnRHR).Fórmula:C62H90N16O15Pureza:99.31% - 99.78%Cor e Forma:SolidPeso molecular:1299.48Triptorelin acetate(57773-63-4 free base)
CAS:Triptorelin acetate is a GnRH agonist for hormone-responsive cancers, precocious puberty, and assisted reproduction.Fórmula:C66H86N18O15Pureza:99.90%Cor e Forma:White PowderPeso molecular:1371.53Ref: TM-T21410
5mg55,00€10mg82,00€25mg126,00€50mg182,00€100mg273,00€200mg409,00€1mL*10mM (DMSO)123,00€Elagolix sodium
CAS:Elagolix sodium (NBI-56418 sodium) is a GnRH receptor (GnRHR) antagonist ( IC50 and Ki of 0.25 and 3.7 nM, respectively).Fórmula:C32H29F5N3NaO5Pureza:99.71%Cor e Forma:SolidPeso molecular:653.57Ref: TM-T5031
2mg35,00€5mg52,00€10mg80,00€25mg144,00€50mg227,00€100mg359,00€200mg532,00€1mL*10mM (DMSO)74,00€Nafarelin acetate(76932-56-4 free base)
CAS:Nafarelin acetate (76932-56-4) is a GnRH analog that reduces LH and FSH release, used for estrogen-related treatments.Fórmula:C68H87N17O15Pureza:99.98%Cor e Forma:SolidPeso molecular:1382.55Linzagolix
CAS:Linzagolix is a small-molecule, non-peptide, orally active gonadotropin-releasing hormone antagonist (GnRH antagonist) which is under development by KisseiFórmula:C22H15F3N2O7SPureza:99.33%Cor e Forma:SolidPeso molecular:508.42Goserelin acetate
CAS:<p>Goserelin acetate (Fertilan) is a synthetic long-acting agonist of gonadotropin-releasing hormone, used in treatments of cancer.</p>Fórmula:C61H88N18O16Pureza:99.77% - >99.99%Cor e Forma:White Crystalline PowderPeso molecular:1329.46Cetrorelix Acetate
CAS:Cetrorelix Acetate is gonadotropin-releasing hormone (GnRH) receptor antagonist with an IC50 of 1.21 nM.Fórmula:C70H92ClN17O14·xC2H4O2Pureza:97.96%Cor e Forma:SolidPeso molecular:1491.11Fertirelin acetate
CAS:Fertirelin acetate is a gonadotropin-releasing hormone (GnRH) agonist.Fórmula:C55H74N16O13Cor e Forma:SolidPeso molecular:1167.29Argtide
CAS:Argtide is an luteinizing hormone releasing hormone (LHRH) antagonist.Fórmula:C80H104ClN21O14Cor e Forma:SolidPeso molecular:1619.27NBI-42902
CAS:NBI-42902 is a potent GnRH receptor antagonist (Ki=0.56 nm, Kd=0.19 nm), suppressing serum LH in macaques without causing histamine release.Fórmula:C27H24F3N3O3Cor e Forma:SolidPeso molecular:495.49EA-230
CAS:Ea-230 is an immunomodulator that may be used in the treatment of renal failure.Fórmula:C15H27N5O6Cor e Forma:SolidPeso molecular:373.4BAY 1214784
CAS:BAY 1214784: potent, oral hGnRH-R antagonist, reduces LH levels, low variability, good tolerance, may research uterine fibroids.Fórmula:C29H26ClF4N3O5S2Cor e Forma:SolidPeso molecular:672.11Opigolix
CAS:Opigolix is a Gonadotropin-releasing hormone receptor antagonist.Fórmula:C25H19F3N4O5SPureza:98.60% - 98.97%Cor e Forma:SolidPeso molecular:544.5BAY-784
CAS:<p>BAY-784 is a gonadotropin-releasing hormone receptor (GnRH-R) antagonist (IC50s: 21 and 24 nM for human and rat GnRH-R).</p>Fórmula:C29H26ClF4N3O5S2Pureza:98%Cor e Forma:SolidPeso molecular:672.115α-Pregnane-3α,20α-diol
CAS:5α-Pregnane-3α,20α-diol, an active metabolite of progesterone, is synthesized through intermediates 5α-pregnane-20α-ol-3-one and 5α-pregnane-3α-ol-20-one fromFórmula:C21H36O2Cor e Forma:SolidPeso molecular:320.51T 98475
CAS:gonadotropin-releasing hormone (GnRH, LHRH) receptor antagonist,orally activeFórmula:C37H37F2N3O4SPureza:98%Cor e Forma:SolidPeso molecular:657.77BAY-298
CAS:BAY-298: oral LH-R antagonist; IC50: 96nM (hLH), 23nM (rLH), 78nM (cLH); first to lower sex hormones in vivo.Fórmula:C27H21ClFN3O2Pureza:98%Cor e Forma:SolidPeso molecular:473.93DCOIT
CAS:DCOIT, an isothiazolinone derivative, stimulates the synthesis of follicle-stimulating hormone and luteinizing hormone in the brain by activating the gonadotropin-releasing hormone receptor (GnRHR). Additionally, it interferes with G protein-coupled receptors, MAPK, and Ca 2+ signaling pathways [1].Fórmula:C11H17Cl2NOSCor e Forma:SolidPeso molecular:282.22[D-Ala6]-LH-RH
CAS:[D-Ala6]-LH-RH, a Luteinizing-hormone-releasing hormone (LHRH) analogue, functions as a gonadotropin-releasing hormone (GnRH) receptor agonist [1].Fórmula:C56H77N17O13Cor e Forma:SolidPeso molecular:1196.32Abarelix acetate
CAS:Abarelix acetate: synthetic GnRHR antagonist, spikes histamine, lowers LH and testosterone temporarily, used in advanced prostate cancer.Fórmula:C72H95ClN14O14·xC2H4O2Cor e Forma:SolidPeso molecular:1476.14BAY-899
CAS:BAY-899, oral LH-R antagonist, IC50: 185 nM (hLH), 46 nM (rLH), lowers sex hormones in vivo.Fórmula:C25H19F2N5O2Pureza:98%Cor e Forma:SolidPeso molecular:459.45(R)-BAY-899
(R)-BAY-899: R-isomer, selective LH-R antagonist, effective on hLH (IC50: 185 nM) and rLH (IC50: 46 nM), orally active.Fórmula:C25H19F2N5O2Cor e Forma:SolidPeso molecular:459.45GnRH-R antagonist 1
CAS:Compound 21a: Oral GnRH-R antagonist, IC50=0.57 nM, potent against prostate cancer/prevents LH surges.Fórmula:C31H28F5N7O6SPureza:98%Cor e Forma:SolidPeso molecular:721.65GnRH antagonist 2
CAS:GnRH antagonist 2 is a GnRH receptor antagonist, useful for studying endocrine diseases.Fórmula:C28H27F2N9O5Pureza:98.08%Cor e Forma:SolidPeso molecular:607.57Acyline
CAS:Acyline, a GnRH antagonist, suppresses gonadotropins and testosterone in animals and maintains the effect for 2 weeks in men with one dose.Fórmula:C80H102ClN15O14Cor e Forma:SolidPeso molecular:1533.21Merigolix
CAS:Merigolix is a potent gonadotrophin releasing hormone (GnRH) antagonist .Fórmula:C36H35F7N4O6Cor e Forma:SolidPeso molecular:752.68Goserelin acetate(65807-02-5 Free base)
<p>Goserelin acetate （ICI-118630 acetate） is a naturally occurring decapeptide, a GnRH (gonadotropin releasing hormone) agonist that reduces the production of sex hormones (testosterone and estrogen) for the treatment of prostate cancer, breast cancer and endometriosis.</p>Pureza:99.77%Cor e Forma:Odour SolidDimethandrolone Undecanoate
CAS:Dimethandrolone Undecanoate (DMAU) is a novel orally available androgen with progestational activity and is a potential male contraceptive compound.Fórmula:C31H50O3Pureza:99.65% - >99.99%Cor e Forma:SolidPeso molecular:470.73Ref: TM-T27176
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