
Antibiótico
Os inibidores de antibióticos são substâncias que interferem na atividade dos antibióticos, frequentemente utilizados para estudar os mecanismos de resistência a antibióticos ou para aumentar a eficácia dos antibióticos existentes. Esses inibidores desempenham um papel crítico na compreensão de como as bactérias evitam o tratamento com antibióticos e no desenvolvimento de estratégias para superar a resistência. Na CymitQuimica, oferecemos uma variedade de inibidores de antibióticos para apoiar sua pesquisa em resistência antimicrobiana, farmacologia e inovação terapêutica.
Foram encontrados 928 produtos de "Antibiótico"
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Mal-PEG4-VA-PBD
CAS:<p>Mal-PEG4-VA-PBD is a drug-linker conjugate for Antibody-Drug Conjugates (ADCs), comprising the antitumor antibiotic Pyrrolobenzodiazepine (PBD), connected</p>Fórmula:C68H79N9O17Pureza:98%Cor e Forma:SolidPeso molecular:1294.41Saroaspidin B
CAS:<p>Saroaspidin B is a dimeric form of a biphenyl triphenol, characterized as an antibiotic compound.</p>Fórmula:C25H32O8Cor e Forma:SolidPeso molecular:460.52Nikkomycin Z
CAS:Nikkomycin Z (Nikkomycin Z from Streptomyces tendae) is a competitive chitin synthase inhibitor.It inhibitor of the growth of filamentous fungi, insects,Fórmula:C20H25N5O10Pureza:98%Cor e Forma:SolidPeso molecular:495.44Bleomycin Free Base
CAS:<p>Bleomycin Free Base, a glycopeptide antibiotic, halts DNA function and treats solid tumors.</p>Fórmula:C55H84N17O21S3Cor e Forma:SolidPeso molecular:1415.55Clavicoronic acid
CAS:Clavicoronic acid, a β-lactamase inhibitor, boosts penicillin antibiotics against resistant bacteria.Fórmula:C15H18O4Cor e Forma:SolidPeso molecular:262.3Imidocarb dihydrochloride monohydrate
Imidocarb dihydrochloride monohydrate is an effective antiprotozoal agent against the parasite B. bovis (IC50: 87 μg/ml).Fórmula:C19H24Cl2N6O2Cor e Forma:SolidPeso molecular:439.34Pibrozelesin
CAS:Pibrozelesin, a water-soluble duocarmycin B2 derivative, binds AT-rich DNA, blocking replication and inducing cell death.Fórmula:C32H36BrN5O8Cor e Forma:SolidPeso molecular:698.56Streptonigrin (racemate)
CAS:Streptonigrin: aminoquinone antibiotic; antitumor, antibacterial; blocks β-Catenin/Tcf, cytotoxic; alters hamster chromosomes; (-)-isomer, CAS#3930-19-6.Fórmula:C25H22N4O8Cor e Forma:SolidPeso molecular:506.46CRS-3123
CAS:CRS-3123, a methionyl-tRNA synthetase inhibitor, is used potentially for the treatment of enteric infections.Fórmula:C19H19Br2N3O2SPureza:98%Cor e Forma:SolidPeso molecular:513.25Methacycline
CAS:<p>Methacycline, a tetracycline antibiotic, inhibits bacterial protein synthesis and effectively suppresses epithelial-mesenchymal transition (EMT). It blocks EMT in vitro and inhibits fibrogenesis in vivo without directly affecting the TGF-β1Smad signaling pathway. As an antimicrobial agent, Methacycline holds potential for research in pulmonary fibrosis.</p>Fórmula:C22H22N2O8Cor e Forma:SolidPeso molecular:442.42Antifungal agent 113
CAS:Antifungalagent 113 (compound 9a) serves as an effective antifungal and antibacterial agent. It exhibits strong inhibitory activity against both S. aureus and methicillin-resistant S. aureus.Fórmula:C23H20O5Cor e Forma:SolidPeso molecular:376.40Acetomycin
CAS:<p>Acetomycin, a γ-lactone from S. ramulosus, halts HCT-8 colon and L1210 leukemia cell growth.</p>Fórmula:C10H14O5Cor e Forma:SolidPeso molecular:214.22Kinamycin B
CAS:Kinamycin B is an antibacterial agent with anticancer activity.Fórmula:C20H16N2O8Pureza:98%Cor e Forma:SolidPeso molecular:412.35Neocryptolepine-Cl
CAS:<p>Neocryptolepine-Cl (compound Z24) is an inhibitor of Bcthi4, demonstrating excellent antifungal activity against B. cinerea, with an EC50 value of 0.56 μg/mL.</p>Fórmula:C16H11ClN2Cor e Forma:SolidPeso molecular:266.725Mucidin
CAS:<p>Mucidin is an antifungal antibiotic that inhibits electron transfer reactions within the mitochondrial respiratory chain's cytochrome bc1 complex.</p>Fórmula:C16H18O3Peso molecular:258.31Saptomycin E
CAS:<p>Saptomycin E is an antitumor antibiotic.</p>Fórmula:C33H35NO9Cor e Forma:SolidPeso molecular:589.63Spicamycin
CAS:Spicamycin can be used as a potent inducer of differentiation of human myeloid leukemia cells (HL-60) and murine myeloid leukemia cells (M1).Fórmula:C30H51N7O7Cor e Forma:SolidPeso molecular:621.77Chitin synthase inhibitor 1
Potent, selective CHS inhibitor with 0.12 mM IC50; effective against drug-resistant fungi.Fórmula:C22H20ClN3O3Cor e Forma:SolidPeso molecular:409.872-Acetyl-2-decarboxamidotetracycline
CAS:<p>2-Acetyl-2-decarboxamidotetracycline is a tetracycline-class antibiotic. It exhibits a UV absorption spectrum similar to that of tetracycline or 5-oxytetracycline at concentrations above 300 mμ, characteristic of the BCD ring system.</p>Fórmula:C23H25NO8Cor e Forma:SolidPeso molecular:443.45Ganaplacide hydrochloride
CAS:Ganaplacide hydrochloride (KAF156 HCl) is an orally administered imidazopyrimidine antimalarial agent that inhibits Plasmodium PI4K activity.Fórmula:C22H24ClF2N5OPureza:93.97%Cor e Forma:SoildPeso molecular:447.91Sinefungin
CAS:Sinefungin (Adenosyl-Ornithine) is an effective inhibitor of virion mRNA(guanine-7-)-methyltransferase, mRNA(nucleoside-2'-)-methyltransferase, and viralFórmula:C15H23N7O5Pureza:98.12%Cor e Forma:SolidPeso molecular:381.39Swainsonine
CAS:<p>Swainsonine (Tridolgosir) is an alkaloid isolated from Astragalus membranaceus and is a potent and reversible inhibitor of alpha-mannosidase. swainsonine has antitumour activity and induces apoptosis and cell cycle arrest in the G2/M phase.</p>Fórmula:C8H15NO3Pureza:98%Cor e Forma:Lyophilized PowderPeso molecular:173.21Formycin A
CAS:Formycin A shows antitumor and antiviral activities. Formycin A , a purine nucleoside antibiotic, is a potent human immunodeficiency virus type 1 (HIV-1) inhibitor with an EC50 of 10 μM.Fórmula:C10H13N5O4Pureza:98%Cor e Forma:SolidPeso molecular:267.24A 53868A
CAS:<p>A 53868A is an antibiotic, it is isolated from Streptomyces luridus.</p>Fórmula:C11H22N3O5PPureza:98%Cor e Forma:SolidPeso molecular:307.287Nortopixantrone
CAS:<p>Nortopixantrone(BBR 3438) is a novel 9-azacyclophenanthracene pyrazole that shows antitumor activity in a human prostate cancer model.</p>Fórmula:C20H24N6O2Pureza:>99.99%Cor e Forma:SolidPeso molecular:380.44Erythromycylamine
CAS:Erythromycylamine is a useful organic compound for research related to life sciences. The catalog number is T64443 and the CAS number is 26116-56-3.Fórmula:C37H70N2O12Cor e Forma:SolidPeso molecular:734.969DprE1-IN-8
CAS:<p>DprE1-IN-8 is a potent inhibitor of DprE1, exhibiting an IC50 of less than 0.75 μM.</p>Fórmula:C19H12F3N5O4SPureza:98%Cor e Forma:SolidPeso molecular:463.39Ref: TM-T79628
Produto descontinuadoPKUMDL-LTQ-301
CAS:PKUMDL-LTQ-301 is a potent inhibitor of HipA toxin. PKUMDL-LTQ-301 also inhibits E. coli persistence.Fórmula:C30H28N2O4Pureza:98%Cor e Forma:SolidPeso molecular:480.55

