
Antibiótico
Os inibidores de antibióticos são substâncias que interferem na atividade dos antibióticos, frequentemente utilizados para estudar os mecanismos de resistência a antibióticos ou para aumentar a eficácia dos antibióticos existentes. Esses inibidores desempenham um papel crítico na compreensão de como as bactérias evitam o tratamento com antibióticos e no desenvolvimento de estratégias para superar a resistência. Na CymitQuimica, oferecemos uma variedade de inibidores de antibióticos para apoiar sua pesquisa em resistência antimicrobiana, farmacologia e inovação terapêutica.
Foram encontrados 918 produtos de "Antibiótico"
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Chitin synthase inhibitor 4
CAS:<p>Chitin synthase inhibitor 4: a CHS inhibitor with antimicrobial properties, potential fungicide.</p>Fórmula:C20H15FN4OPureza:99.74%Cor e Forma:SolidPeso molecular:346.36SQ109
CAS:<p>SQ109 (NSC-722041) is an effective inhibitor of the trypomastigote form of the parasite (IC50 = 50 nM). SQ109 is an antitubercular agent and targets MmpL3.</p>Fórmula:C22H38N2Pureza:99.70% - 99.91%Cor e Forma:SolidPeso molecular:330.55Ormetoprim
CAS:<p>Ormetoprim (Ro 5-9754), an antibiotic approved for use in the United States, is used to prevent the spread of disease in freshwater aquaculture.</p>Fórmula:C14H18N4O2Pureza:99.92%Cor e Forma:SolidPeso molecular:274.32RMI 10874
CAS:<p>RMI 10874 is a tilorone analogue. Tilorone is an orally bioavailable antiviral agent.</p>Fórmula:C21H26N2O4Pureza:98%Cor e Forma:SolidPeso molecular:370.44SSJ-183
CAS:<p>SSJ-183 is a low-toxicity and orally available and anti-malarial drug with an IC50 = 7.6 nM against P. falciparum and no lethality at doses up to 2000 mg/kg po.</p>Fórmula:C25H22N4OPureza:99.71% - 99.83%Cor e Forma:SolidPeso molecular:394.47Albitiazolium bromide
CAS:<p>Albitiazolium bromide is an antimalarial compound disrupting phosphatidylcholine biosynthesis in Plasmodium, transported via NPP and cation carriers.</p>Fórmula:C24H42BrN2O2S2Pureza:99.743%Cor e Forma:SolidPeso molecular:534.64Linogliride fumarate
CAS:<p>Linogliride fumarate, a guanidine derivative, stimulates insulin release by blocking ATP-sensitive K+ channels, enhancing glucose tolerance.</p>Fórmula:C20H26N4O5Pureza:98%Cor e Forma:SolidPeso molecular:402.451Pyrrofolic acid
CAS:<p>Pyrrofolic acid shows high anti-folate biological activity for S. faecalis.</p>Fórmula:C23H21N7O7Pureza:98%Cor e Forma:SolidPeso molecular:507.46S 863390
CAS:<p>S 863390 is a renin inhibitor.</p>Fórmula:C37H52N6O4Pureza:98%Cor e Forma:SolidPeso molecular:644.85Tunicamine
CAS:<p>Tunicamine is a reversible polyprenol-phosphate inhibitor.</p>Fórmula:C11H21NO9Pureza:98%Cor e Forma:SolidPeso molecular:311.29Chitin synthase inhibitor 2
CAS:<p>Chitin synthase inhibitor 2 (2b) has an IC50 of 0.09 mM, K i 0.12 mM, shows in vitro antimicrobial activity and boosts fluconazole/polyoxin B.</p>Fórmula:C20H19N3O3Cor e Forma:SolidPeso molecular:349.38CRK12-IN-1
CAS:<p>CRK12-IN-1: strong inhibitor of CRK12, kills T.b. brucei & T. congolense (EC50s: 1.3 & 18 nM).</p>Fórmula:C20H26F2N4O3S2Pureza:99.72%Cor e Forma:SolidPeso molecular:472.57BRD-8000.3
CAS:<p>BRD-8000.3 is a narrow-spectrum antimycobacterial targeting EfpA, inhibiting lipid transport in drug-tolerant Mtb and useful in structural and functional.</p>Fórmula:C19H21BrN4OPureza:99.78% - 99.78%Cor e Forma:SolidPeso molecular:401.3Alalevonadifloxacin HCl
CAS:<p>Alalevonadifloxacin HCl is a novel l-alanine ester prodrug of levonadifloxacin.</p>Fórmula:C22H27ClFN3O5Pureza:98%Cor e Forma:SolidPeso molecular:467.92Pafuramidine maleate
CAS:<p>Pafuramidine is an orally bioavailable prodrug of formamidine which was developed for the treatment of human African trypanosomiasis.</p>Fórmula:C24H24N4O7Pureza:98%Cor e Forma:SolidPeso molecular:480.16Exeporfinium chloride
CAS:<p>Exeporfinium chloride(XF-73) is an antimicrobial agent that can weaken bacterial cell walls.</p>Fórmula:C44H50Cl2N6O2Cor e Forma:SolidPeso molecular:765.81Epirubicin
CAS:<p>Epirubicin, a doxorubicin derivative, is an antineoplastic, inhibits topoisomerase, DNA/RNA synthesis, and Foxp3, reducing T cell activity.</p>Fórmula:C27H29NO11Cor e Forma:SolidPeso molecular:543.52Linogliride
CAS:<p>Linogliride: a guanidine derivative, inhibits insulin release, and enhances glucose tolerance by blocking ATP-sensitive K+ channels in pancreatic beta cells.</p>Fórmula:C16H22N4OPureza:98%Cor e Forma:SolidPeso molecular:286.37Verticillin A
CAS:<p>Verticillin A, an apoptosis inducer, inhibits Leiomyosarcoma and Malignant peripheral nerve sheath tumor growth.</p>Fórmula:C30H28N6O6S4Pureza:98%Cor e Forma:SolidPeso molecular:696.84Pentachloropseudilin
CAS:<p>Pentachloropseudilin inhibits Myosin-1 and speeds up TGF-β receptor turnover, suppressing TGF-β activity.</p>Fórmula:C10H4Cl5NOPureza:98.14%Cor e Forma:SolidPeso molecular:331.41
