HIV Protease

Os inibidores da protease do HIV são uma classe de medicamentos antirretrovirais que têm como alvo específico a enzima protease do vírus da imunodeficiência humana (HIV). Ao inibir esta enzima, esses compostos impedem o vírus de processar suas poliproteínas em proteínas maduras e funcionais, bloqueando assim a produção de novos virions infecciosos. Os inibidores da protease do HIV são um pilar da terapia antirretroviral altamente ativa (HAART) utilizada para o tratamento do HIV/AIDS. Na CymitQuimica, oferecemos uma variedade de inibidores da protease do HIV para apoiar sua pesquisa em tratamento do HIV, resistência a medicamentos e virologia.

Foram encontrados 502 produtos de "HIV Protease"

Pureza (%)

100

produtos por página.

+ Info
Tenofovir alafenamide
CAS:
- 379270-37-8
Tenofovir alafenamide (GS-7340) is a nucleotide reverse transcriptase inhibitor (NRTI) and a novel ester prodrug of the antiretroviral tenofovir.
Fórmula:C₂₁H₂₉N₆O₅P
Pureza:99.68% - 99.81%
Cor e Forma:Solid
Peso molecular:476.47
Ref: TM-T2409
+ Info
Lopinavir
CAS:
- 192725-17-0
Lopinavir (ABT-378) is a peptidomimetic HIV protease inhibitor that retains activity against HIV protease with the Val 82 mutation.
Fórmula:C₃₇H₄₈N₄O₅
Pureza:98% - 99.62%
Cor e Forma:White Crystalline Solid
Peso molecular:628.8
Ref: TM-T1623
+ Info
Darunavir
CAS:
- 206361-99-1
Darunavir (TMC114) is an HIV PROTEASE INHIBITOR that is used in the treatment of AIDS and HIV INFECTIONS.
Fórmula:C₂₇H₃₇N₃O₇S
Pureza:99.67% - 99.76%
Cor e Forma:White Amorphous Solid
Peso molecular:547.66
Ref: TM-T2324
+ Info
Didanosine
CAS:
- 69655-05-6
Didanosine (ddI) is a nucleoside reverse transcriptase inhibitor analog of adenosine (IC50: 0.49 μM).
Fórmula:C₁₀H₁₂N₄O₃
Pureza:99.64%
Cor e Forma:White Crystalline Powder
Peso molecular:236.23
Ref: TM-T2578
+ Info
Raltegravir sodium
CAS:
- 1292804-07-9
Raltegravir (MK 0518) sodium is a potent, orally active HIV integrase (IN) inhibitor.
Fórmula:C₂₀H₂₀FN₆NaO₅
Cor e Forma:Solid
Peso molecular:466.405
Ref: TM-T62983
+ Info
Fosamprenavir sodium
CAS:
- 226700-80-7
Fosamprenavir sodium is an HIV protease inhibitor that is the water soluble prodrug of amprenavir.
Fórmula:C₂₅H₃₄N₃Na₂O₉PS
Cor e Forma:Solid
Peso molecular:629.57
Ref: TM-T69713
+ Info
BMS-707035
CAS:
- 729607-74-3
BMS-707035 is a specific HIV-I integrase (IN) inhibitor with IC50 of 15 nM. Phase 2.
Fórmula:C₁₇H₁₉FN₄O₅S
Pureza:99.78%
Cor e Forma:Solid
Peso molecular:410.42
Ref: TM-T6420
+ Info
TAT
CAS:
- 191936-91-1
TAT peptide (YGRKKRRQRRR), originating from the human immunodeficiency virus-1 (HIV-1) transactivator of transcription (TAT), enhances the solubility and
Fórmula:C₆₄H₁₁₈N₃₂O₁₄
Pureza:>99.99%
Cor e Forma:Solid
Peso molecular:1559.83
Ref: TM-TP1809
+ Info
Temsavir
CAS:
- 701213-36-7
Temsavir (BMS626529) is a novel attachment inhibitor that targets HIV-1 gp120 and prevents its binding to CD4+ T cells.
Fórmula:C₂₄H₂₃N₇O₄
Pureza:99.14%
Cor e Forma:Solid
Peso molecular:473.48
Ref: TM-T4665
+ Info
lavendustin B
CAS:
- 125697-91-8
Lavendustin B inhibits Tyrosine Kinase and HIV-1 integrase-LEDGF/p75 interaction.
Fórmula:C₂₁H₁₉NO₅
Pureza:95.72%
Cor e Forma:Off-White Solid
Peso molecular:365.38
Ref: TM-T4182
+ Info
Raltegravir
CAS:
- 518048-05-0
Raltegravir (MK-0518) is a pyrrolidinone derivative and HIV INTEGRASE INHIBITOR that is used in combination with other ANTI-HIV AGENTS for the treatment of HIV
Fórmula:C₂₀H₂₁FN₆O₅
Pureza:99.86% - >99.99%
Cor e Forma:Solid
Peso molecular:444.42
Ref: TM-T2239L
+ Info
2,4-Dihydroxypyridine
CAS:
- 626-03-9
2,4-Dihydroxypyridine: a pyridine derivative, chelates metals, assesses ion levels, measures enzymatic reactions, and quantifies biomolecules.
Fórmula:C₅H₅NO₂
Pureza:97.79%
Cor e Forma:White To Yellow-Beige Crystals Or
Peso molecular:111.1
Ref: TM-T7963
+ Info
I-XW-053 sodium
CAS:
- 1644644-89-2
I-XW-053 sodium inhibits the replication of a diverse panel of primary HIV-1 isolates in Peripheral blood mononuclear cell with no appreciable cytotoxicity.
Fórmula:C₂₂H₁₆N₂NaO₂
Cor e Forma:Solid
Peso molecular:363.372
Ref: TM-T27642
+ Info
LDC4297 hydrochloride
CAS:
- 2319747-14-1
LDC4297 hydrochloride is a selective and potent CDK7 inhibitor with broad-spectrum antiviral activity, useful for research on viral infections.
Fórmula:C₂₃H₂₉ClN₈O
Cor e Forma:Solid
Peso molecular:468.98
Ref: TM-T72385
+ Info
PTACH
CAS:
- 848354-66-5
PTACH (Cpd 51) (NCH-51) is a SAHA-based inhibitor of human HDAC. It can potently inhibit the growth of various human Y cells (EC50: 1 to 10 μM).
Fórmula:C₂₀H₂₆N₂O₂S₂
Pureza:87.44% - 99.74%
Cor e Forma:Solid
Peso molecular:390.56
Ref: TM-T3199
+ Info
Darunavir Ethanolate
CAS:
- 635728-49-3
Darunavir Ethanolate (UIC 94017) is an HIV PROTEASE INHIBITOR that is used in the treatment of AIDS and HIV INFECTIONS.
Fórmula:C₂₉H₄₃N₃O₈S
Pureza:99.84% - 99.86%
Cor e Forma:Solid
Peso molecular:593.74
Ref: TM-T3335
+ Info
Thiamine disulfide
CAS:
- 67-16-3
Thiamine disulfide (Algoneurina) , also known as thiamin or vitamin B1, is a vitamin found in food and manufactured as a dietary supplement and medication.
Fórmula:C₂₄H₃₄N₈O₄S₂
Pureza:99.81% - 99.81%
Cor e Forma:Coa
Peso molecular:562.71
Ref: TM-T20062
+ Info
PMEDAP
CAS:
- 113852-41-8
PMEDAP is a potent inhibitor of Moloney murine sarcoma virus (MSV)-induced tumor formation and associated mortality and an inhibitor of human immunodeficiency
Fórmula:C₈H₁₃N₆O₄P
Pureza:99.77%
Cor e Forma:Solid
Peso molecular:288.2
Ref: TM-T38514
+ Info
Inosine pranobex
CAS:
- 36703-88-5
Inosine pranobex (Delimmun) has a lot of immunomodulatory effects, including inducing T-lymphocyte differentiation, augmenting macrophage and NK cell functions.
Fórmula:C₅₂H₇₈N₁₀O₁₇
Pureza:99.78% - 99.91%
Cor e Forma:Solid
Peso molecular:1115.23
Ref: TM-T3614
+ Info
IMB-301
CAS:
- 64009-84-3
IMB-301 is a small molecular inhibitor via virtual screening according to the hA3G model.
Fórmula:C₁₉H₁₇Cl₂FN₂O
Pureza:99.72%
Cor e Forma:Solid
Peso molecular:379.26
Ref: TM-T9212