
Outros inibidores
Esta categoria abrange uma ampla variedade de inibidores que não se encaixam nas classificações padrão, mas que ainda são essenciais para várias pesquisas bioquímicas e farmacológicas. Esses inibidores podem direcionar vias, enzimas e interações moleculares únicas ou menos estudadas, fornecendo ferramentas valiosas para áreas de pesquisa especializadas. Na CymitQuimica, oferecemos uma seleção diversificada de inibidores de alta qualidade que abrangem múltiplos alvos biológicos e disciplinas de pesquisa, permitindo que você explore novas vias terapêuticas e aprofunde sua compreensão de processos biológicos complexos.
Foram encontrados 36533 produtos de "Outros inibidores"
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FOXM1-IN-2
CAS:<p>FOXM1-IN-2, a FOXM1 inhibitor, exhibits antineoplastic activity [1].</p>Fórmula:C48H47F4N7O12SCor e Forma:SolidPeso molecular:1021.99Antibacterial agent 160
CAS:<p>Antibacterial Agent 160 is a potent antibacterial agent that rapidly eradicates bacteria and inhibits the formation of bacterial biofilms.</p>Fórmula:C29H27ClFN3O6Cor e Forma:SolidPeso molecular:567.99SHP2-IN-14
CAS:<p>SHP2-IN-14 (compound 27) is a potent, orally active allosteric inhibitor of SHP2, displaying strong anti-tumor activity with an IC50 of 7 nM.</p>Fórmula:C22H20Cl2N8OCor e Forma:SolidPeso molecular:483.35CYY292
CAS:<p>CYY292 is a chemical compound acting as an inhibitor of PDGFRα, PDGFRβ, FGFR1, -2, and -3, with respective IC50 values of 5.35, 4.6, 28, 28, and 78 nM.</p>Fórmula:C24H28N8OCor e Forma:SolidPeso molecular:444.53ARN 077
CAS:ARN 077 is a selective N-acylethanolamine acid amidase (NAAA) inhibitor (IC50: 7 nM for human NAAA). ARN 077 significantly increases palmitoyl ethanolamine (PEA) levels within the CNS.Fórmula:C16H21NO4Cor e Forma:SolidPeso molecular:291.34MDVN1003
CAS:MDVN1003 inhibits BTK & PI3Kδ in B cells, blocking NHL growth; it kills lymphoma cells, not erythroblasts.Fórmula:C22H20FN7OPureza:98%Cor e Forma:SolidPeso molecular:417.4480-O16B
CAS:<p>80-O16B, an ionizable cationic lipid featuring disulfide bonds, is utilized in the preparation of lipid nanoparticles (LNP) [1].</p>Fórmula:C39H78N2O4S4Cor e Forma:SolidPeso molecular:767.31IDO/Tubulin-IN-2
CAS:<p>IDO/Tubulin-IN-2 inhibits TDO/tubulin, effective on U87, HepG2, A549, HCT-116, LO2 cancer cells; IC50 values 0.036-1.04 μM, boosts antitumor action.</p>Fórmula:C48H40N6O10Cor e Forma:SolidPeso molecular:860.87FAP-IN-2
CAS:<p>FAP-IN-2 is a 99mTc-labeled, isonitrile-containing derivative of a fibroblast activation protein (FAPI) inhibitor suitable for tumor imaging [1].</p>Fórmula:C24H28F2N6O3Cor e Forma:SolidPeso molecular:486.51I-BET282
CAS:<p>BET-IN-1 is a bromodomain inhibitor extracted from patent WO/2013024104A1 (example 2, plC50: 6.0 - 7.0).</p>Fórmula:C25H30N4O4Pureza:98%Cor e Forma:SolidPeso molecular:450.53Sakura 6
CAS:<p>Sakura 6, a synthetic serotonin transporter (SERT)-binding peptide, enhances the interaction between SERT and neuronal nitric oxide synthase.</p>Fórmula:C31H45N5O7Cor e Forma:SolidPeso molecular:599.73RIOK2-IN-2
CAS:<p>RIOK2-IN-2 (8) functions as an inhibitor of RIOK2, exhibiting IC50 values of 3.02 μM in MKN-1 cells and 5.34 μM in MOLT4 cells [1].</p>Fórmula:C27H23F3N6O2Cor e Forma:SolidPeso molecular:520.51LM2I
CAS:<p>LM2I, a derivative of Spinosyn A (SPA), serves both as an argininosuccinate synthase (ASS1) enzyme activator and a tumor inhibitor through direct interaction</p>Fórmula:C47H77N3O11Cor e Forma:SolidPeso molecular:860.13Tauro-Obeticholic Acid sodium
CAS:<p>Tauro-obeticholic acid, a farnesoid X receptor (FXR) agonist and semisynthetic derivative of chenodeoxycholic acid, is an active metabolite of obeticholic acid.</p>Fórmula:C28H48NO6S·NaCor e Forma:SolidPeso molecular:549.74S-72
CAS:<p>S-72 acts as a microtubule polymerization inhibitor, effective in cell-free assays at concentrations of 1, 3, and 10 µM.</p>Fórmula:C20H22N4O3SCor e Forma:SolidPeso molecular:398.50Ref: TM-T83874
Produto descontinuadoImmune cell migration-IN-1
CAS:<p>Immune cell migration-IN-1 (compound 2) serves as a potent inhibitor of immune cell migration, with potential research applications for mitigating conditions</p>Fórmula:C30H25ClN4O6SCor e Forma:SolidPeso molecular:605.06Antitumor agent-136
CAS:<p>Antitumor Agent-136 (Compound 17), a broad-spectrum antitumor agent and NAMPT inhibitor, exhibits potent activity with an IC50 of 9.5 nM. It efficiently lowers intracellular and extracellular NAMPT protein levels via the ubiquitin proteasome pathway, achieving effective tumor inhibition [1].</p>Fórmula:C58H76N10O11S3Cor e Forma:SolidPeso molecular:1185.48DiaFluo
CAS:<p>DiaFluo is a probe for protein S-sulfinylation from cells.</p>Fórmula:C32H32N4O9SCor e Forma:SolidPeso molecular:648.69Ref: TM-T31416
Produto descontinuadoDDO-2213
CAS:<p>DDO-2213 is a potent, orally active inhibitor of the WDR5-MLL1 interaction, demonstrating an IC50 of 29 nM and a Kd of 72.9 nM against WDR5.</p>Fórmula:C24H27ClFN7OCor e Forma:SolidPeso molecular:483.97And1-IN-1
CAS:<p>And1-IN-1, also known as compound III, is a potent inhibitor of And1 [1].</p>Fórmula:C15H11BCl2O2Cor e Forma:SolidPeso molecular:304.96Antitumor photosensitizer-1
CAS:<p>Antitumor Photosensitizer-1 (Compound 8) is a potent photosensitizer with remarkable photodynamic anti-tumor properties and minimal skin photo-toxicity,</p>Fórmula:C42H51N5O6Cor e Forma:SolidPeso molecular:721.88Anti-MI/R injury agent 1
CAS:<p>Anti-MI/R injury agent 1 (compound 18), derived from Panaxatriol, represents an orally administered, potent agent against myocardial ischemia/reperfusion (MI/R</p>Fórmula:C32H49NO6Cor e Forma:SolidPeso molecular:543.73Antitumor photosensitizer-2
CAS:<p>Compound 11, also known as Antitumor Photosensitizer-2, is a potent photosensitizer with remarkable photodynamic anti-tumor properties and minimal skin photo-</p>Fórmula:C40H47N5O7Cor e Forma:SolidPeso molecular:709.83URAT1 inhibitor 5
CAS:<p>URAT1 Inhibitor 5 (compound 16) serves as a powerful inhibitor of URAT1 and is utilized in hyperuricemia research [1].</p>Fórmula:C18H14BrN3O2SCor e Forma:SolidPeso molecular:416.29Azilsartan mepixetil potassium
CAS:<p>Azilsartan medoxomil potassium (QR-01019K), an angiotensin II receptor antagonist, exhibits a potent and sustained antihypertensive effect, along with a more</p>Fórmula:C36H33KN6O8Cor e Forma:SolidPeso molecular:716.78DG026
CAS:DG026 selectively inhibits IRAP, reducing its cross-presentation in dendritic cells without affecting ERAP1.Fórmula:C35H40N3O4PPureza:98%Cor e Forma:SolidPeso molecular:597.68Ifetroban
CAS:<p>Ifetroban is a potent and selective TxA2/PGH2 receptor antagonist.</p>Fórmula:C25H32N2O5Cor e Forma:SolidPeso molecular:440.53ALS-I-41
CAS:ALS-I-41 is a novel, potent and selective antagonist of oxytocin receptor.Fórmula:C30H38FN3O6SPureza:98%Cor e Forma:SolidPeso molecular:587.7Cortivazol
CAS:Cortivazol is an Anti-Inflammatory Drug.Fórmula:C32H38N2O5Pureza:98%Cor e Forma:SolidPeso molecular:530.65Ref: TM-T25271
Produto descontinuadoIfetroban sodium
CAS:<p>Ifetroban sodium (BMS-180291), oral TXA2/PGH2 antagonist for researching heart, stroke, BP, thrombosis.</p>Fórmula:C25H31N2NaO5Cor e Forma:SolidPeso molecular:462.5229,10-Phenanthrenequinone
CAS:<p>9,10-Phenanthrenequinone is an inhibitor of claudin-5/CLDN5, which induces apoptosis via an NO synthase/ROS-dependent mechanism. It also promotes caspase activation and DNA fragmentation while reducing CLDN5 expression and proteasome proteolysis, contributing to endothelial barrier dysfunction.</p>Fórmula:C14H8O2Cor e Forma:SolidPeso molecular:208.21BB-Cl-Amidine hydrochloride
CAS:BB-Cl-Amidine hydrochloride is an inhibitor of peptidylarginine deminase (PAD) [1].Fórmula:C26H27Cl2N5OPureza:98%Cor e Forma:SolidPeso molecular:496.43BPH-628
CAS:<p>BPH-628 is a bioactive chemical.</p>Fórmula:C20H20O7P2Cor e Forma:SolidPeso molecular:434.32

